Page last updated: 2024-08-21

amiloride and quinine

amiloride has been researched along with quinine in 35 studies

Research

Studies (35)

TimeframeStudies, this research(%)All Research%
pre-19906 (17.14)18.7374
1990's15 (42.86)18.2507
2000's7 (20.00)29.6817
2010's7 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Avdeef, A; Tam, KY1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Anagnostopoulos, T; Belachgar, F; Discala, F; Hulin, P; Planelles, G1
Gusev, GP; Sherstobitov, AO; Skulskii, IA1
Cornet, M; Delpire, E; Gilles, R1
Brierley, GP; Jung, DW1
Forstner, G; Forstner, J; Marcon, MA; McCool, D1
Boyer, JL; Corasanti, JG; Gleeson, D1
Abramcheck, FJ; Helman, SI; Van Driessche, W1
Brierley, GP; Davis, MH; Jung, DW1
Graf, J; Haddad, P1
Hoffmann, EK; Kramhøft, B; Lambert, IH1
Levinson, C; Smith, TC1
Persechini, PM; Soldati, L1
Diaz, J; Muallem, S; Xu, X; Zhao, H1
Bendayan, R; Lo, B; Silverman, M1
Anderson, PA; Schetz, JA1
Beauchamp, GK; Breslin, PA1
Bieda, M; Copenhagen, DR; Dixon, DB; Takahashi, K1
Boutellier, S; Lutz, TA; Rossi, R; Scharrer, E; Seebacher, MC; Sutter, DA1
Harada, S; Kasahara, Y; Yamaguchi, K; Yamamoto, T1
Ossebaard, CA; Polet, IA; Smith, DV1
Marunaka, Y; Niisato, N; O'Brodovich, H; Post, M; Tanswell, AK1
Lundy, RF; Norgren, R1
Bittinger, F; Brockerhoff, P; Deutsch, C; Kilbinger, H; Kirkpatrick, CJ; Roth, E; Wessler, I1
Chiba, T; Marcus, DC1
Hanafusa, T; Hosoi, K; Min, KY; Mori, H; Nakahari, T; Shiima, C1
Delay, ER; Kondoh, T1
Drucker, DJ; Inoue, M; Iwata, S; Margolskee, RF; Ninomiya, Y; Shigemura, N; Takai, S; Yanagawa, Y; Yasumatsu, K; Yoshida, R1
He, L; Kumarhia, D; McCluskey, LP1

Reviews

2 review(s) available for amiloride and quinine

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

33 other study(ies) available for amiloride and quinine

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
How well can the Caco-2/Madin-Darby canine kidney models predict effective human jejunal permeability?
    Journal of medicinal chemistry, 2010, May-13, Volume: 53, Issue:9

    Topics: Animals; Disease Models, Animal; Dogs; Humans; Jejunal Diseases; Kidney Diseases; Models, Biological; Permeability; Porosity; Regression Analysis

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Barium- or quinine-induced depolarization activates K+, Na+ and cationic conductances in frog proximal tubular cells.
    The Journal of physiology, 1992, Volume: 448

    Topics: Amiloride; Animals; Barium; Kidney Tubules, Proximal; Membrane Potentials; Methazolamide; Potassium; Potassium Channels; Quinine; Rana ridibunda; Sodium; Sodium-Potassium-Exchanging ATPase

1992
Potassium transport in lamprey (Lampetra fluviatilis) erythrocytes: evidence for K+ channels.
    Comparative biochemistry and physiology. Comparative physiology, 1992, Volume: 101, Issue:3

    Topics: Amiloride; Animals; Barium; Biological Transport; Calcium; Erythrocytes; Lampreys; Magnesium Chloride; Potassium; Potassium Channels; Quinine; Rubidium Radioisotopes; Sodium; Sucrose; Tea

1992
Volume regulation in rat pheochromocytoma cultured cells submitted to hypoosmotic conditions.
    Archives internationales de physiologie, de biochimie et de biophysique, 1991, Volume: 99, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adrenal Gland Neoplasms; Amiloride; Animals; Colforsin; Hypotonic Solutions; Kinetics; Pheochromocytoma; Potassium Chloride; Quinine; Rats; Rubidium Radioisotopes; Sodium Chloride; Trifluoperazine; Tumor Cells, Cultured

1991
Kinetic properties of the K+/H+ antiport of heart mitochondria.
    Biochemistry, 1990, Jan-16, Volume: 29, Issue:2

    Topics: Amiloride; Animals; Biological Transport; Calcimycin; Carrier Proteins; Cations, Monovalent; Cattle; Choline; Dicyclohexylcarbodiimide; Fluoresceins; Fluorescent Dyes; Hydrogen-Ion Concentration; Hypotonic Solutions; Kinetics; Magnesium; Mitochondria, Heart; Potassium; Potassium-Hydrogen Antiporters; Quinine

1990
Inhibition of mucin secretion in a colonic adenocarcinoma cell line by DIDS and potassium channel blockers.
    Biochimica et biophysica acta, 1990, Apr-09, Volume: 1052, Issue:1

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adenocarcinoma; Amiloride; Barium; Barium Compounds; Calcimycin; Cell Line; Chlorides; Colonic Neoplasms; Furosemide; Humans; Kinetics; Mucins; Ouabain; Potassium Channels; Quinine; Stilbenes; Tetraethylammonium; Tetraethylammonium Compounds; Tumor Cells, Cultured; Vasoactive Intestinal Peptide

1990
Effects of osmotic stresses on isolated rat hepatocytes. I. Ionic mechanisms of cell volume regulation.
    The American journal of physiology, 1990, Volume: 258, Issue:2 Pt 1

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Animals; Barium; Bicarbonates; Bumetanide; Cells, Cultured; Chlorides; Hypertonic Solutions; Hypotonic Solutions; Kinetics; Liver; Male; Osmolar Concentration; Potassium Chloride; Quinine; Rats; Rats, Inbred Strains; Sodium Chloride

1990
Autoregulation of apical membrane Na+ permeability of tight epithelia. Noise analysis with amiloride and CGS 4270.
    The Journal of general physiology, 1985, Volume: 85, Issue:4

    Topics: Amiloride; Animals; Cell Membrane Permeability; Electricity; Epithelium; Homeostasis; Ion Channels; Physiology; Pyrazines; Quinidine; Quinine; Rana pipiens; Skin; Sodium

1985
Intravesicular pH changes in submitochondrial particles induced by monovalent cations: relationship to the Na+/H+ and K+/H+ antiporters.
    Archives of biochemistry and biophysics, 1988, Aug-01, Volume: 264, Issue:2

    Topics: Amiloride; Animals; Calcimycin; Calcium; Carrier Proteins; Cations, Monovalent; Cattle; Dextrans; Dicyclohexylcarbodiimide; Fluorescein-5-isothiocyanate; Fluoresceins; Fluorescent Dyes; Hydrogen-Ion Concentration; Lithium; Magnesium; Mitochondria, Heart; Potassium; Potassium-Hydrogen Antiporters; Quinine; Sodium; Sodium-Hydrogen Exchangers; Spectrometry, Fluorescence; Submitochondrial Particles; Valinomycin

1988
Volume-regulatory K+ fluxes in the isolated perfused rat liver: characterization by ion transport inhibitors.
    The American journal of physiology, 1989, Volume: 257, Issue:3 Pt 1

    Topics: Amiloride; Animals; Barium; Biological Transport; Carrier Proteins; Cell Membrane Permeability; Hypertonic Solutions; Ions; Liver; Male; Osmolar Concentration; Ouabain; Perfusion; Potassium; Quinine; Rats; Rats, Inbred Strains; Sodium-Hydrogen Exchangers

1989
Na+/H+ exchange in Ehrlich ascites tumor cells: activation by cytoplasmic acidification and by treatment with cupric sulphate.
    The Journal of membrane biology, 1988, Volume: 102, Issue:1

    Topics: Amiloride; Animals; Carcinoma, Ehrlich Tumor; Carrier Proteins; Cell Membrane; Copper; Copper Sulfate; Cytoplasm; Hydrogen-Ion Concentration; Kinetics; Mice; Pimozide; Quinine; Sodium-Hydrogen Exchangers

1988
Quinine inhibits multiple Na+ and K+ transport mechanisms in Ehrlich ascites tumor cells.
    Biochimica et biophysica acta, 1989, Jan-16, Volume: 978, Issue:1

    Topics: Adenosine Triphosphate; Amiloride; Animals; Biological Transport; Calcium; Carcinoma, Ehrlich Tumor; Furosemide; Male; Membrane Potentials; Mice; Mice, Inbred ICR; Ouabain; Potassium; Potassium Channels; Propranolol; Quinine; Sodium

1989
Depolarization of macrophage polykaryons in the absence of external sodium induces a cyclic stimulation of a calcium-activated potassium conductance.
    Biochimica et biophysica acta, 1988, Dec-09, Volume: 972, Issue:3

    Topics: Amiloride; Animals; Calcium; Cell Nucleus; Electric Conductivity; Electric Stimulation; Gallopamil; Hydrogen-Ion Concentration; Kinetics; Macrophages; Membrane Potentials; Mice; Mice, Inbred AKR; Mice, Inbred C3H; Potassium Channels; Quinine; Sodium

1988
Regulation of [Na+]i in resting and stimulated submandibular salivary ducts.
    The Journal of biological chemistry, 1995, Aug-18, Volume: 270, Issue:33

    Topics: Amiloride; Animals; Barium Compounds; Carbachol; Ion Transport; Male; Ouabain; Quinidine; Quinine; Rats; Sodium; Submandibular Gland; Tetraethylammonium; Tetraethylammonium Compounds

1995
Characterization of cimetidine transport in LLCPK1 cells.
    Journal of the American Society of Nephrology : JASN, 1994, Volume: 5, Issue:1

    Topics: Amiloride; Animals; Anti-Bacterial Agents; Azides; Biological Transport; Carrier Proteins; Cell Line; Cimetidine; Guanidine; Guanidines; Kidney; Macrolides; Microscopy, Fluorescence; Models, Biological; Niacinamide; Proton-Translocating ATPases; Quinidine; Quinine; Sodium Azide; Sodium-Hydrogen Exchangers; Swine; Tetraethylammonium; Tetraethylammonium Compounds

1994
Pharmacology of the high-affinity apamin receptor in rabbit heart.
    Cardiovascular research, 1995, Volume: 30, Issue:5

    Topics: Amiloride; Animals; Apamin; Calcium Channels; Cell Membrane; Chlorides; Dihydropyridines; Dose-Response Relationship, Drug; Filtration; Hydrogen-Ion Concentration; Iodine Radioisotopes; Methods; Myocardium; Potassium Channels; Protein Binding; Quinine; Rabbits; Scorpion Venoms; Temperature

1995
Suppression of bitterness by sodium: variation among bitter taste stimuli.
    Chemical senses, 1995, Volume: 20, Issue:6

    Topics: Adult; Amiloride; Anions; Caffeine; Cations; Drug Interactions; Humans; Lithium Chloride; Magnesium Sulfate; Potassium Chloride; Quinine; Sodium; Sodium Chloride; Taste; Urea

1995
Quinine, intracellular pH and modulation of hemi-gap junctions in catfish horizontal cells.
    Vision research, 1996, Volume: 36, Issue:24

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Animals; Catfishes; Cobalt; Electric Conductivity; Electrophysiology; Gap Junctions; Hydrogen-Ion Concentration; Patch-Clamp Techniques; Quinine; Retina

1996
Hyperpolarization of hepatocytes by 2,5-AM: implications for hepatic control of food intake.
    The American journal of physiology, 1997, Volume: 272, Issue:3 Pt 2

    Topics: Amiloride; Animals; Apamin; Appetite; Azepines; Barium; Bicarbonates; Chlorides; Female; Flufenamic Acid; Glyburide; Homeostasis; In Vitro Techniques; Liver; Male; Mannitol; Membrane Potentials; Mice; Mice, Inbred ICR; Ouabain; Potassium Channel Blockers; Potassium Channels; Quinine; Rats; Rats, Sprague-Dawley; Sodium

1997
Different characteristics of gustatory responses between the greater superficial petrosal and chorda tympani nerves in the rat.
    Chemical senses, 1997, Volume: 22, Issue:2

    Topics: Amiloride; Animals; Chorda Tympani Nerve; Electrophysiology; Expectorants; Hydrochloric Acid; Male; Muscle Relaxants, Central; Palate, Soft; Quinine; Rats; Rats, Sprague-Dawley; Saccharin; Sodium Acetate; Sodium Chloride; Sucrose; Taste; Tongue

1997
Amiloride effects on taste quality: comparison of single and multiple response category procedures.
    Chemical senses, 1997, Volume: 22, Issue:3

    Topics: Amiloride; Humans; Hydrochloric Acid; Lithium Chloride; Quinine; Sodium; Taste

1997
Roles of Ca2+ and protein tyrosine kinase in insulin action on cell volume via Na+ and K+ channels and Na+/K+/2Cl- cotransporter in fetal rat alveolar type II pneumocyte.
    The Journal of membrane biology, 1999, Mar-01, Volume: 168, Issue:1

    Topics: Amiloride; Animals; Bumetanide; Calcium; Calcium-Transporting ATPases; Carrier Proteins; Cell Size; Chelating Agents; Egtazic Acid; Enzyme Inhibitors; Female; Humans; Infant, Newborn; Insulin; Phenols; Phosphorylation; Potassium Channels; Pregnancy; Pregnancy in Diabetics; Protein Processing, Post-Translational; Protein-Tyrosine Kinases; Pulmonary Alveoli; Quinine; Rats; Rats, Wistar; Receptor, Insulin; Respiratory Distress Syndrome, Newborn; Signal Transduction; Sodium Channels; Sodium-Potassium-Chloride Symporters; Thapsigargin

1999
Pontine gustatory activity is altered by electrical stimulation in the central nucleus of the amygdala.
    Journal of neurophysiology, 2001, Volume: 85, Issue:2

    Topics: Amiloride; Amygdala; Animals; Brain Mapping; Citric Acid; Drug Combinations; Electric Stimulation; Electrophysiology; Male; Neural Inhibition; Neurons, Afferent; Pons; Quinine; Rats; Rats, Sprague-Dawley; Sodium Chloride; Taste; Tongue

2001
Release of non-neuronal acetylcholine from the isolated human placenta is mediated by organic cation transporters.
    British journal of pharmacology, 2001, Volume: 134, Issue:5

    Topics: Acetylcholine; Amiloride; Cimetidine; Corticosterone; DNA, Antisense; Dose-Response Relationship, Drug; Female; Guanidine; Humans; In Vitro Techniques; Norepinephrine; Organic Cation Transport Proteins; Organic Cation Transporter 1; Organic Cation Transporter 2; Piperidines; Placenta; Pregnancy; Procaine; Quinine; Time Factors; Verapamil

2001
Basolateral K+ conductance establishes driving force for cation absorption by outer sulcus epithelial cells.
    The Journal of membrane biology, 2001, Nov-15, Volume: 184, Issue:2

    Topics: Absorption; Amiloride; Animals; Barium; Cations, Monovalent; Electric Conductivity; Enzyme Inhibitors; Epithelial Cells; Gerbillinae; Lidocaine; Membrane Potentials; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Quinine; Sodium-Potassium-Exchanging ATPase

2001
Terbutaline-induced triphasic changes in volume of rat alveolar type II cells: the role of cAMP.
    The Japanese journal of physiology, 2002, Volume: 52, Issue:6

    Topics: Adrenergic beta-Agonists; Amiloride; Animals; Calcium; Cell Size; Cells, Cultured; Colforsin; Cyclic AMP; Ionomycin; Male; Microscopy, Video; Potassium Channels; Pulmonary Alveoli; Quinine; Rats; Rats, Wistar; Sodium Channels; Terbutaline; Thapsigargin

2002
Dried bonito dashi: taste qualities evaluated using conditioned taste aversion methods in wild-type and T1R1 knockout mice.
    Chemical senses, 2015, Volume: 40, Issue:2

    Topics: Amiloride; Amino Acids; Animals; Avoidance Learning; Citric Acid; Conditioning, Classical; Cooking; Dose-Response Relationship, Drug; Food; Glutamic Acid; Hydrogen-Ion Concentration; Inosine Monophosphate; Lactic Acid; Male; Mice, Inbred C57BL; Mice, Knockout; Quinine; Receptors, G-Protein-Coupled; Sodium Glutamate; Sucrose; Taste Perception

2015
Glucagon-like peptide-1 is specifically involved in sweet taste transmission.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2015, Volume: 29, Issue:6

    Topics: Amiloride; Animals; Chorda Tympani Nerve; Enzyme-Linked Immunosorbent Assay; Exenatide; Glucagon-Like Peptide 1; Glucagon-Like Peptide-1 Receptor; Hydrochloric Acid; Mice, Inbred C57BL; Mice, Knockout; Mice, Transgenic; Microscopy, Confocal; Neurons; Peptides; Quinine; Receptors, Glucagon; Saccharin; Signal Transduction; Sodium Chloride; Sucrose; Taste; Taste Buds; Venoms

2015
Inflammatory stimuli acutely modulate peripheral taste function.
    Journal of neurophysiology, 2016, 06-01, Volume: 115, Issue:6

    Topics: Amiloride; Analgesics, Non-Narcotic; Analysis of Variance; Animals; Body Weight; Capsaicin; Chorda Tympani Nerve; Dose-Response Relationship, Drug; Epithelial Sodium Channel Blockers; Female; Functional Laterality; Interleukin-6; Lipopolysaccharides; Quinine; Rats; Sensory Receptor Cells; Sodium; Sodium Acetate; Sodium Chloride; Taste Buds; Tomography Scanners, X-Ray Computed; Tumor Necrosis Factor-alpha

2016