amiloride has been researched along with phenylamil in 89 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 14 (15.73) | 18.7374 |
1990's | 30 (33.71) | 18.2507 |
2000's | 17 (19.10) | 29.6817 |
2010's | 24 (26.97) | 24.3611 |
2020's | 4 (4.49) | 2.80 |
Authors | Studies |
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Astakhova, N; Boucher, RC; Geiss, WB; Hirsh, AJ; Johnson, MR; Molino, BF; Sargent, BJ; Smith, RT; Swenson, BD; Usyatinsky, A; Wyle, MJ; Zamurs, A; Zhang, J | 1 |
Bianchi, G; Ferrandi, M; Ferrari, P; Hanozet, GM; Parenti, P | 1 |
Hannam, V; O'Brodovich, H; Rafii, B | 1 |
Lazdunski, M; Van Renterghem, C | 1 |
Armstrong, J; Bourke, JR; Cragoe, EJ; Huxham, GJ; Manley, SW; Matainaho, T | 1 |
Abel, KC; Bourke, JR; Brown, L; Cragoe, EJ; Manley, SW | 1 |
Atsumi, T; Cragoe, EJ; Imae, Y; Sugiyama, S | 1 |
Cragoe, EJ; Erickson, RP; Schiffman, SS; Suggs, MS | 1 |
Barbry, P; Champe, M; Champigny, G; Chassande, O; Frelin, C; Lingueglia, E; Maes, P; Munemitsu, S; Tartar, A; Ullrich, A | 1 |
Cragoe, EJ; Simchowitz, L | 1 |
Cragoe, EJ; Garvin, JL; Mandel, LJ; Simon, SA | 2 |
Barbry, P; Cragoe, EJ; Frelin, C; Lazdunski, M; Vigne, P | 1 |
Barbry, P; Chassande, O; Cragoe, EJ; Ellory, C; Frelin, C; Lazdunski, M; Vigne, P | 1 |
Barbry, P; Champigny, G; Frelin, C; Lazdunski, M; Marsault, R; Vigne, P | 1 |
Cragoe, EJ; Oyarzabal, H; Potter, GD; Sellin, JH | 1 |
Barbry, P; Chassande, O; Duval, D; Frelin, C; Lazdunski, M; Rousseau, B | 1 |
Barbry, P; Champigny, G; Gerard, C; Lazdunski, M; Mauchamp, J; Verrier, B | 1 |
Cragoe, EJ; Oyarzabal, H; Sellin, JH | 1 |
Asher, C; Cragoe, EJ; Garty, H; Moran, A | 1 |
Barbry, P; Chassande, O; Frelin, C; Lazdunski, M; Vigne, P | 1 |
Benos, DJ; Bridges, RJ; Cragoe, EJ; Frizzell, RA | 1 |
Cragoe, EJ; Ehrenfeld, J; Harvey, BJ | 1 |
Bennington, JB; Cragoe, EJ; Knauf, PA; Lannigan, DA | 1 |
Dubinsky, WP; Sellin, JH | 1 |
Guggino, WB; Li, XJ; Snyder, SH; Xu, RH | 1 |
Bose, R; Guia, A; Leblanc, N | 1 |
Frelin, C; van Renterghem, C | 1 |
Baldwin, ML; Brasitus, TA; Cragoe, EJ; Dudeja, PK; Harig, JM; Ramaswamy, K | 1 |
Baker, M; Barbry, P; Chassande, O; Lazdunski, M; Novotny, WF | 1 |
Cragoe, EJ; Dubinsky, WP; Hall, A; Sellin, JH | 1 |
Asher, C; Barbry, P; Clauss, W; Cragoe, E; Garty, H; Goldstein, O | 1 |
Armstrong, JW; Bourke, JR; Cragoe, EJ; Huxham, GJ; Manley, SW; Yap, AS | 1 |
Betz, AL; Ennis, SR; Ren, XD | 1 |
Bose, D; Bose, R; Chau, T; Guia, A | 1 |
Homma, M; Imae, Y; Kawagishi, I; Kudo, S; Magariyama, Y; Muramoto, K; Sugiyama, S | 1 |
Homma, M; Imae, Y; Imagawa, M; Kawagishi, I; McCarter, L | 1 |
Atsumi, T; Homma, M; Kawagishi, I; Kojima, S; Kudo, S; Muramoto, K | 1 |
Blank, U; Clauss, W; Hofmann, T; Lindemann, H; Münker, G; Rückes, C; Weber, W | 1 |
Boucher, RC; Hofmann, T; Knowles, MR; Lindemann, H; Rückes, C; Stutts, MJ; Weber, WM; Ziersch, A | 1 |
Asai, Y; Atsumi, T; Homma, M; Kawagishi, I; Kojima, S | 1 |
Abdulnour-Nakhoul, S; Bor, S; Imeryuz, N; Orlando, RC | 1 |
Jaques, S; Kim, YK; McCarter, LL | 1 |
Martens, H; Schultheiss, G | 1 |
Bury, NR; Wood, CM | 1 |
Estrela, RC; Ponte, CG; Suarez-Kurtz, G | 1 |
Homma, M; Sato, K | 1 |
Alrefai, WA; Dudeja, PK; Gill, RK; Joshi, V; Ramaswamy, K; Tyagi, S | 1 |
Grosell, M; Wood, CM | 1 |
Galvez, F; Goss, GG; Hawkings, GS; Reid, SD | 1 |
Kita-Tsukamoto, K; Kogure, K; Nishino, T; Wada, M; Yao, K | 1 |
Abraham, WM; Boucher, RC; Hirsh, AJ; Hopkins, S; Paradiso, AM; Sabater, JR; Smith, RT; Zamurs, A | 1 |
Burke, J; Handy, RD | 1 |
Brown, S; Dunbar, M; Hughes, C; Klinck, J; Nichols, J; Playle, RC; Winter, A | 1 |
Diecke, FP; Fischbarg, J | 1 |
Chifflet, S; Grasso, S; Hernández, JA | 1 |
Gilmour, KM; Patel, M; Rogers, JT; Wood, CM | 1 |
Goss, GG; Parks, SK; Tresguerres, M | 1 |
Grosell, M; Nadella, SR; Wood, CM | 1 |
Davies, BS; Kim, WK; Parhami, F; Park, KW; Tontonoz, P; Waki, H; Young, SG | 1 |
Araki, M; Inui, T; Kubota, T; Miyamoto, M; Mori, Y; Nimura, Y; Takenaka, H; Watanabe, M | 1 |
Choi, SP; Park, KM; Park, KW; Tontonoz, P; Waki, H | 1 |
Chan, MC; Hata, A; Hickman, T; Hill, NS; Kang, H; Lagna, G; Mecker, SV; Nguyen, PH; Weisman, AS | 1 |
Auer, S; Ibañez-Tallon, I; Santos-Torres, J; Ślimak, MA | 1 |
Del Duca, O; Donini, A; Galperin, V; Nasirian, A | 1 |
Brix, KV; Grosell, M | 1 |
Ashe, KM; Kan, HM; Laurencin, CT; Lo, KW; Ulery, BD | 1 |
Kan, HM; Laurencin, CT; Lo, KW | 1 |
Kim, JG; Kwon, JH; Park, HC; Son, KM; Yang, HC; Zhu, T | 1 |
Brauner, CJ; Wood, CM; Zimmer, AM | 1 |
Defoirdt, T; Yang, Q | 1 |
Nadella, SR; Ng, A; Patel, D; Wood, CM | 1 |
Aghaloo, T; Bezouglaia, O; Cui, ZK; Fan, J; Fartash, A; Guo, M; Im, CS; Lee, JY; Lee, M; Nguyen, J; Wu, BM | 1 |
Fliegel, L; Goss, GG; Guffey, SC | 1 |
Aghaloo, TL; Bezouglaia, O; Cui, ZK; Fan, J; Fartash, A; Guo, M; Im, CS; Kim, S; Lee, M; Patel, N; Wang, CY; Wu, BM | 1 |
Aractingi, S; Desposito, D; Farman, N; Jaisser, F; Maubec, E; Nassar, D; Nguyen, VT; Waeckel, L | 1 |
Gonzales, EB; Snell, HD | 1 |
Kim, WK; Park, KW; Regassa, A | 1 |
Aghaloo, TL; Cui, ZK; Fan, J; Guo, M; Im, CS; Kim, S; Lee, M; Pi-Anfruns, J; Wu, BM | 1 |
Hong, C; Kang, MK; Kim, RH; Lee, C; Park, NH; Phung, S; Shin, KH; Song, M; Stevenson, RG; Yi, JK | 1 |
Leyva-Jimenez, H; Moncada, K; Park, KW; Price, TR; Tontonoz, P; Walzem, RL | 1 |
El-Fiqi, A; Kim, HW; Lee, JH; Mandakhbayar, N | 1 |
Aghaloo, TL; Cui, ZK; Fan, J; Guo, M; Im, DCS; Kim, S; Lee, M; Pi-Anfruns, J; Wu, BM | 1 |
Baker, MAB; Clark, J; Ishida, T; Ito, R; Matzke, NJ; Sowa, Y | 1 |
Bagheri, F; Fink, T; Jahed, V; Lambertsen Larsen, K; Vasheghani-Farahani, E; Zarrabi, A | 1 |
Hu, J; Liu, Y; Sun, H | 1 |
Liu, Y; Miszuk, JM; Pan, Y; Sun, H; Yao, Q | 1 |
Fong, H; Hong, Z; Hu, J; Liang, Z; Miszuk, J; Sanyour, H; Sun, H | 1 |
Atyabi, F; Damoogh, S; Dinarvand, R; Farokhi, M; Gholami, M; Motasadizadeh, H; Mottaghitalab, F; Tavakoli, M | 1 |
89 other study(ies) available for amiloride and phenylamil
Article | Year |
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Design, synthesis, and structure-activity relationships of novel 2-substituted pyrazinoylguanidine epithelial sodium channel blockers: drugs for cystic fibrosis and chronic bronchitis.
Topics: Animals; Bronchi; Bronchitis, Chronic; Combinatorial Chemistry Techniques; Cystic Fibrosis; Dogs; Epithelial Sodium Channels; Guanidines; Models, Molecular; Pyrazines; Respiratory Mucosa; Sodium Channel Blockers; Sodium Channels; Stereoisomerism; Structure-Activity Relationship; Tissue Culture Techniques | 2006 |
Effect of amiloride analogues on sodium transport in renal brush border membrane vesicles from Milan hypertensive rats.
Topics: Amiloride; Animals; Biological Transport, Active; Hypertension; Kidney; Membrane Potentials; Microvilli; Rats; Rats, Mutant Strains; Sodium | 1992 |
Sodium channel but neither Na(+)-H+ nor Na-glucose symport inhibitors slow neonatal lung water clearance.
Topics: Amiloride; Animals; Animals, Newborn; Body Water; Carrier Proteins; Electricity; Guinea Pigs; Lung; Monosaccharide Transport Proteins; Phlorhizin; Sodium Channels; Sodium-Hydrogen Exchangers | 1991 |
A new non-voltage-dependent, epithelial-like Na+ channel in vascular smooth muscle cells.
Topics: Amiloride; Animals; Aorta; Cell Line; Epithelium; Kinetics; Muscle, Smooth, Vascular; Portal Vein; Sodium Channels | 1991 |
Bidirectional ion transport in thyroid: secretion of anions by monolayer cultures that absorb sodium.
Topics: Absorption; Amiloride; Animals; Anions; Bicarbonates; Biological Transport; Bumetanide; Cells, Cultured; Chlorides; Cytological Techniques; Dinoprostone; Drug Resistance; Electrophysiology; Epithelial Cells; Epithelium; Ions; Sodium; Thyroid Gland | 1992 |
Amiloride analogues induce responses in isolated rat cardiovascular tissues by inhibition of Na+/Ca2+ exchange.
Topics: Amiloride; Animals; Calcium; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Heart Rate; In Vitro Techniques; Myocardial Contraction; Rats; Sodium; Vasodilation | 1991 |
Specific inhibition of the Na(+)-driven flagellar motors of alkalophilic Bacillus strains by the amiloride analog phenamil.
Topics: Amiloride; Aminoisobutyric Acids; Bacillus; Cell Membrane; Cell Movement; Drug Resistance, Microbial; Flagella; Hydrogen-Ion Concentration; Kinetics; Membrane Potentials; Sodium; Sodium Channels | 1990 |
Inhibition of taste responses to Na+ salts by epithelial Na+ channel blockers in gerbil.
Topics: Amiloride; Animals; Electrophysiology; Epithelium; Female; Gerbillinae; Sodium; Sodium Channels; Taste | 1990 |
Human kidney amiloride-binding protein: cDNA structure and functional expression.
Topics: Amiloride; Amine Oxidase (Copper-Containing); Amino Acid Sequence; Animals; Base Sequence; Carrier Proteins; Cell Line; Cell Membrane; Cloning, Molecular; DNA; Gene Library; Humans; Kinetics; Molecular Sequence Data; Oligonucleotide Probes; Peptide Mapping; Recombinant Proteins; RNA, Messenger; Sequence Homology, Nucleic Acid; Swine; Transfection | 1990 |
Polyvalent cations inhibit human neutrophil chemotaxis by interfering with the polymerization of actin.
Topics: Actins; Amiloride; Calcium; Cations; Chemotaxis, Leukocyte; Humans; In Vitro Techniques; Kinetics; Macromolecular Substances; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Nickel | 1990 |
Phenamil: an irreversible inhibitor of sodium channels in the toad urinary bladder.
Topics: Amiloride; Animals; Binding, Competitive; Bufo marinus; Cell Membrane Permeability; Chemical Phenomena; Chemistry; Drug Interactions; Drug Synergism; Ion Channels; Kinetics; Mucous Membrane; Sodium; Urinary Bladder | 1985 |
[3H]phenamil, a radiolabelled diuretic for the analysis of the amiloride-sensitive Na+ channels in kidney membranes.
Topics: Amiloride; Animals; Binding Sites; Dose-Response Relationship, Drug; Epithelium; In Vitro Techniques; Ion Channels; Kidney; Sodium; Swine; Tritium | 1986 |
Binding of 3H-phenamil, an irreversible amiloride analog, to toad urinary bladder: effects of aldosterone and vasopressin.
Topics: Aldosterone; Amiloride; Animals; Bufo marinus; In Vitro Techniques; Ion Channels; Kinetics; Urinary Bladder; Vasopressins | 1986 |
Purification and subunit structure of the [3H]phenamil receptor associated with the renal apical Na+ channel.
Topics: Amiloride; Animals; Binding Sites; Cell Membrane; Chromatography, Affinity; Chromatography, Ion Exchange; Epithelium; Ion Channels; Kidney Tubules; Kidney Tubules, Distal; Molecular Weight; Receptors, Drug; Sodium Channels; Swine | 1987 |
A new type of amiloride-sensitive cationic channel in endothelial cells of brain microvessels.
Topics: Amiloride; Animals; Binding Sites; Blood-Brain Barrier; Cattle; Electric Conductivity; Endothelium, Vascular; In Vitro Techniques; Ion Channels; Potassium; Sodium | 1989 |
Phenamil inhibits electrogenic sodium absorption in rabbit ileum.
Topics: Amiloride; Animals; Chlorides; Ileum; In Vitro Techniques; Intestinal Absorption; Male; Ouabain; Rabbits; Sodium; Sodium Channels; Theophylline | 1989 |
Biochemical identification of two types of phenamil binding sites associated with amiloride-sensitive Na+ channels.
Topics: Amiloride; Animals; Cell Membrane; Kidney; Kinetics; Mathematics; Receptors, Drug; Sodium Channels; Swine | 1989 |
Identification and properties of a novel type of Na+-permeable amiloride-sensitive channel in thyroid cells.
Topics: Amiloride; Animals; Cell Membrane; Cells, Cultured; Kinetics; Membrane Potentials; Sodium; Sodium Channels; Swine; Thyroid Gland | 1989 |
Electrogenic sodium absorption in rabbit cecum in vitro.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Amiloride; Animals; Bicarbonates; Biological Transport; Cecum; Chlorides; Cyclic GMP; Dose-Response Relationship, Drug; Electric Conductivity; Electrophysiology; Epinephrine; Furosemide; Intestinal Absorption; Male; Potassium; Rabbits; Sodium; Sulfhydryl Reagents; Water-Electrolyte Balance | 1988 |
Conductive sodium pathway with low affinity to amiloride in LLC-PK1 cells and other epithelia.
Topics: Amiloride; Animals; Cell Line; Cell Membrane; Epithelium; Erythrocyte Membrane; Female; Humans; Kidney Cortex; Kinetics; Male; Membrane Potentials; Microvilli; Rabbits; Rana ridibunda; Rats; Rats, Inbred Strains; Sodium; Sodium Channels; Valinomycin | 1988 |
The structure of the amiloride sensitive apical Na+ channel from pig kidney.
Topics: Amiloride; Animals; Kidney; Sodium Channels; Swine | 1988 |
Inhibition of colonic Na+ transport by amiloride analogues.
Topics: Amiloride; Animals; Biological Transport; Colon; Dexamethasone; Electric Conductivity; Electrophysiology; Epithelium; Female; Kinetics; Rats; Rats, Inbred Strains; Sodium | 1989 |
Evidence for a Na+/H+ exchanger at the basolateral membranes of the isolated frog skin epithelium: effect of amiloride analogues.
Topics: Amiloride; Animals; Biological Transport; Carrier Proteins; Epithelium; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Ouabain; Protons; Rana esculenta; Skin; Sodium; Sodium-Hydrogen Exchangers | 1987 |
Phenamil, an amiloride analogue, inhibits differentiation of Friend murine erythroleukemic cells.
Topics: Amiloride; Animals; Cell Differentiation; Cell Division; Cell Line; Dimethyl Sulfoxide; Friend murine leukemia virus; Leukemia, Erythroblastic, Acute; Mice; Osmolar Concentration; Ouabain; Rubidium; Sodium | 1988 |
Apical nonspecific cation conductances in rabbit cecum.
Topics: Amiloride; Animals; Barium; Calcium; Cations, Divalent; Cecum; Cell Membrane; Colon; Dose-Response Relationship, Drug; Electric Conductivity; Ion Channels; Magnesium; Microelectrodes; Rabbits; Sodium; Sodium Channels; Solutions | 1994 |
Alternatively spliced forms of the alpha subunit of the epithelial sodium channel: distinct sites for amiloride binding and channel pore.
Topics: Alternative Splicing; Amiloride; Amino Acid Sequence; Animals; Base Sequence; Blotting, Southern; Cell Line; Cloning, Molecular; DNA, Complementary; Epithelium; Molecular Sequence Data; Oocytes; Polymerase Chain Reaction; Protein Binding; Rats; Ribonucleases; Sodium Channels; Xenopus | 1995 |
Effects of phenamil on potassium and calcium channels of guinea pig ventricular myocytes.
Topics: Action Potentials; Amiloride; Animals; Calcium Channels; Guinea Pigs; Heart; Potassium Channels; Sodium Channel Blockers | 1995 |
3,4 dichlorobenzamil-sensitive, monovalent cation channel induced by palytoxin in cultured aortic myocytes.
Topics: Acrylamides; Amiloride; Animals; Aorta, Thoracic; Calcium; Cells, Cultured; Cnidarian Venoms; Electrophysiology; In Vitro Techniques; Ion Channels; Muscle, Smooth, Vascular; Ouabain; Potassium; Rats; Rats, Wistar; Sodium; Sodium Channels; Sodium Radioisotopes | 1993 |
Mechanisms of Na+ transport in human distal colonic apical membrane vesicles.
Topics: Amiloride; Biological Transport; Colon; Dose-Response Relationship, Drug; Humans; Intestinal Mucosa; Kinetics; Osmolar Concentration; Sodium; Sodium Channels; Sodium Radioisotopes; Sodium-Hydrogen Exchangers | 1994 |
Diamine oxidase is the amiloride-binding protein and is inhibited by amiloride analogues.
Topics: Amiloride; Amine Oxidase (Copper-Containing); Amino Acid Sequence; Animals; Antibodies, Monoclonal; Carrier Proteins; Colon; DNA, Complementary; Female; Humans; Kidney; Kinetics; Molecular Sequence Data; Molecular Weight; Placenta; Pregnancy; Sequence Homology, Amino Acid; Swine; Transfection | 1994 |
Characterization of an apical sodium conductance in rabbit cecum.
Topics: Amiloride; Animals; Cecum; Cell Membrane; Chlorides; Colon; Electric Conductivity; Hydrogen-Ion Concentration; Potassium; Rabbits; Sodium; Sodium Channels | 1993 |
An epithelial high-affinity amiloride-binding site, different from the Na+ channel.
Topics: Aldosterone; Amiloride; Animals; Binding Sites; Binding, Competitive; Bufo marinus; Cell Membrane; Chickens; Colon; Epithelium; Intestine, Large; Kinetics; Sodium; Sodium Channels; Sodium, Dietary; Urinary Bladder | 1993 |
Activation of sodium transport mediates regulation of thyroid follicle volume in response to hypotonic media.
Topics: Amiloride; Animals; Cells, Cultured; Culture Media; Epithelium; Hypotonic Solutions; Kinetics; Membrane Potentials; Sodium; Sodium Channels; Swine; Thyroid Gland; Thyrotropin; Time Factors | 1993 |
Mechanisms of sodium transport at the blood-brain barrier studied with in situ perfusion of rat brain.
Topics: Amiloride; Animals; Biological Transport; Blood-Brain Barrier; Brain; Bumetanide; Carrier Proteins; Cerebrovascular Circulation; Frontal Lobe; Hydrochlorothiazide; Kinetics; Perfusion; Plasma Volume; Rats; Rats, Inbred Strains; Sodium; Sodium Channels; Sodium-Hydrogen Exchangers; Sodium-Potassium-Chloride Symporters | 1996 |
Mechanism of cardiac inotropy by phenamil, and epithelial sodium channel blocker.
Topics: Amiloride; Animals; Carrier Proteins; Dogs; Female; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Myocardial Contraction; Rats; Sarcoplasmic Reticulum; Sodium Channel Blockers; Sodium-Calcium Exchanger; Sodium-Potassium-Exchanging ATPase | 1996 |
Rotational fluctuation of the sodium-driven flagellar motor of Vibrio alginolyticus induced by binding of inhibitors.
Topics: Amiloride; Cell Division; Computer Simulation; Flagella; Microscopy; Models, Biological; Molecular Structure; Movement; Protein Binding; Sodium; Sodium Channel Blockers; Sodium Channels; Vibrio | 1996 |
The sodium-driven polar flagellar motor of marine Vibrio as the mechanosensor that regulates lateral flagellar expression.
Topics: Amiloride; Bacterial Proteins; Dose-Response Relationship, Drug; Flagella; Flagellin; Gene Expression Regulation, Bacterial; Membrane Proteins; Sodium Channels; Vibrio parahaemolyticus; Viscosity | 1996 |
Vibrio alginolyticus mutants resistant to phenamil, a specific inhibitor of the sodium-driven flagellar motor.
Topics: Amiloride; Drug Resistance, Microbial; Flagella; Mutation; Sodium; Vibrio | 1997 |
Cystic fibrosis and non-cystic-fibrosis human nasal epithelium show analogous Na+ absorption and reversible block by phenamil.
Topics: Amiloride; Cells, Cultured; Cystic Fibrosis; Dose-Response Relationship, Drug; Epithelium; Humans; Nasal Mucosa; Sodium | 1997 |
Effects of topically delivered benzamil and amiloride on nasal potential difference in cystic fibrosis.
Topics: Administration, Intranasal; Adolescent; Adult; Aerosols; Amiloride; Cells, Cultured; Cystic Fibrosis; Epithelium; Female; Humans; In Vitro Techniques; Male; Membrane Potentials; Nasal Mucosa; Sodium Channel Blockers; Sodium Channels | 1998 |
Na+-driven flagellar motor resistant to phenamil, an amiloride analog, caused by mutations in putative channel components.
Topics: Amiloride; Amino Acid Sequence; Bacterial Proteins; Base Sequence; Binding Sites; DNA Primers; Drug Resistance, Microbial; Flagella; Genes, Bacterial; Models, Molecular; Molecular Motor Proteins; Molecular Sequence Data; Mutagenesis, Site-Directed; Mutation; Protein Conformation; Sodium; Sodium Channels; Vibrio | 1999 |
Mechanisms of basolateral Na+ transport in rabbit esophageal epithelial cells.
Topics: Amiloride; Ammonia; Animals; Bicarbonates; Biological Transport; Bumetanide; Chlorides; Epithelial Cells; Esophagus; Homeostasis; Hydrogen-Ion Concentration; In Vitro Techniques; Intracellular Membranes; Isotonic Solutions; Rabbits; Sodium | 1999 |
Mutations conferring resistance to phenamil and amiloride, inhibitors of sodium-driven motility of Vibrio parahaemolyticus.
Topics: Amiloride; Amino Acid Sequence; Bacterial Outer Membrane Proteins; Bacterial Proteins; Cell Movement; Conserved Sequence; Membrane Proteins; Molecular Sequence Data; Mutation; Phenotype; Sodium; Vibrio parahaemolyticus | 1999 |
Ca-sensitive Na transport in sheep omasum.
Topics: Aldosterone; Amiloride; Animals; Biological Transport; Calcium; Electric Conductivity; Feedback; Female; Magnesium; Male; Mannitol; Microelectrodes; Omasum; Serous Membrane; Sheep; Sodium; Theophylline | 1999 |
Mechanism of branchial apical silver uptake by rainbow trout is via the proton-coupled Na(+) channel.
Topics: Amiloride; Animals; Anti-Bacterial Agents; Binding, Competitive; Biological Transport; Cations; Cell Membrane; Enzyme Inhibitors; Gills; Kinetics; Macrolides; Oncorhynchus mykiss; Protons; Silver Nitrate; Sodium Channel Blockers; Sodium Channels; Time Factors | 1999 |
Modulation of the Ca(2+) release channel of sarcoplasmic reticulum by amiloride analogs.
Topics: Amiloride; Animals; Caffeine; Calcium; Calcium Channels; Cetomacrogol; Diuretics; Electrophysiology; In Vitro Techniques; Isometric Contraction; Magnesium; Membranes; Muscle Fibers, Skeletal; Phosphodiesterase Inhibitors; Rabbits; Ruthenium Red; Ryanodine Receptor Calcium Release Channel; Sarcoplasmic Reticulum; Sodium Channels; Solutions | 2000 |
Multimeric structure of PomA, a component of the Na+-driven polar flagellar motor of vibrio alginolyticus.
Topics: Amiloride; Bacterial Proteins; Cell Membrane; Cell Movement; Dimerization; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Flagella; Mutation; Protein Structure, Tertiary; Recombinant Fusion Proteins; Sodium; Sodium Channels; Sodium Chloride; Vibrio | 2000 |
Evidence for a Na+-H+ exchange across human colonic basolateral plasma membranes purified from organ donor colons.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acetazolamide; Amiloride; Biological Transport; Bumetanide; Carbonic Anhydrase Inhibitors; Cell Membrane; Colon; Humans; Hydrogen; In Vitro Techniques; Ion Exchange; Sodium; Sodium-Potassium-Exchanging ATPase; Tissue Donors | 2000 |
Copper uptake across rainbow trout gills: mechanisms of apical entry.
Topics: Amiloride; Animals; Anti-Bacterial Agents; Biological Transport; Calcium; Copper; Copper Radioisotopes; Gills; Kinetics; Macrolides; Oncorhynchus mykiss; Potassium; Proton Pump Inhibitors; Sodium; Sodium Channel Blockers | 2002 |
Localization and characterization of phenamil-sensitive Na+ influx in isolated rainbow trout gill epithelial cells.
Topics: Amiloride; Animals; Anti-Bacterial Agents; Biological Transport; Bumetanide; Epithelial Cells; Female; Gills; Guanidines; Hydrogen-Ion Concentration; Macrolides; Male; Mitochondria; Models, Biological; Oncorhynchus mykiss; Ouabain; Peanut Agglutinin; Sodium; Sodium Radioisotopes; Sulfones | 2003 |
Flagellar motors of marine bacteria Halomonas are driven by both protons and sodium ions.
Topics: Adaptation, Biological; Amiloride; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Flagella; Halomonas; Microscopy, Electron; Movement; Proton Pumps; Seawater; Sodium-Potassium-Exchanging ATPase; Uncoupling Agents; Water Microbiology | 2004 |
Evaluation of second generation amiloride analogs as therapy for cystic fibrosis lung disease.
Topics: Absorption; Amiloride; Animals; Bronchi; Cystic Fibrosis; Electrophysiology; Epithelial Cells; Epithelial Sodium Channels; Epithelium; Female; Humans; In Vitro Techniques; Lung Diseases; Mannitol; Microscopy, Confocal; Mucus; Muscle Contraction; Sheep; Sodium; Sodium Channel Blockers; Sodium Channels; Viscosity | 2004 |
Sodium-sensitive and -insensitive copper accumulation by isolated intestinal cells of rainbow trout Oncorhynchus mykiss.
Topics: Amiloride; Analysis of Variance; Animals; Cells, Cultured; Chlorides; Copper; Hydrogen-Ion Concentration; Intestinal Mucosa; Oncorhynchus mykiss; Sodium; Sodium Channel Blockers; Sodium Channels | 2005 |
Influence of water chemistry and natural organic matter on active and passive uptake of inorganic mercury by gills of rainbow trout (Oncorhynchus mykiss).
Topics: Amiloride; Animals; Biological Transport; Biological Transport, Active; Cysteine; Dose-Response Relationship, Drug; Edetic Acid; Ethylenediamines; Fresh Water; Gills; Ions; Lanthanum; Mercury; Models, Biological; Nitrilotriacetic Acid; Oncorhynchus mykiss; Ontario; Spectrophotometry, Atomic; Verapamil | 2005 |
A mathematical model of electrolyte and fluid transport across corneal endothelium.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Biological Transport, Active; Chloride Channels; Computer Simulation; Electrolytes; Endothelium, Corneal; Ion Channels; Kinetics; Models, Biological; Osmosis; Ouabain; Permeability; Proton-Translocating ATPases; Sodium-Potassium-Exchanging ATPase; Symporters | 2005 |
A possible role for membrane depolarization in epithelial wound healing.
Topics: Actins; Amiloride; Animals; Cattle; Cells, Cultured; Choline; Endothelium, Corneal; Epithelial Cells; Membrane Potentials; Sodium; Wound Healing | 2005 |
Mechanisms behind Pb-induced disruption of Na+ and Cl- balance in rainbow trout (Oncorhynchus mykiss).
Topics: Amiloride; Animals; Carbonic Anhydrases; Chlorides; Enzyme Inhibitors; Gills; Lead; Macrolides; Oncorhynchus mykiss; Proton-Translocating ATPases; Sodium; Sodium Channel Blockers; Sodium-Potassium-Exchanging ATPase; Time Factors; Water-Electrolyte Balance | 2005 |
Interactions between Na+ channels and Na+-HCO3- cotransporters in the freshwater fish gill MR cell: a model for transepithelial Na+ uptake.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Animals; Bicarbonates; Cell Survival; Epithelial Cells; Fluoresceins; Fluorescent Dyes; Gills; Hydrogen-Ion Concentration; In Vitro Techniques; Ion Channel Gating; Ion Transport; Membrane Potentials; Mitochondria; Models, Animal; Oncorhynchus mykiss; Sodium; Sodium Channels; Sodium-Bicarbonate Symporters | 2007 |
Mechanisms of dietary Cu uptake in freshwater rainbow trout: evidence for Na-assisted Cu transport and a specific metal carrier in the intestine.
Topics: Amiloride; Animals; Carbon Dioxide; Chlorides; Copper; Hydrogen-Ion Concentration; Hypercapnia; Intestinal Absorption; Intestinal Mucosa; Microvilli; Oncorhynchus mykiss; Osmolar Concentration; Osmotic Pressure; Silver; Sodium; Sodium Channel Blockers; Sulfates | 2007 |
The small molecule phenamil induces osteoblast differentiation and mineralization.
Topics: Amiloride; Animals; Base Sequence; Bone Morphogenetic Protein 2; Bone Morphogenetic Protein 7; Bone Remodeling; Cell Cycle Proteins; Cell Differentiation; Cell Line; DNA Primers; Gene Expression; Mesenchymal Stem Cells; Mice; Minerals; Organ Culture Techniques; Osteoblasts; Recombinant Proteins; RNA, Small Interfering; Signal Transduction; Smad Proteins | 2009 |
Ca(2+) regulation of endocochlear potential in marginal cells.
Topics: Amiloride; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Cochlea; Egtazic Acid; Endolymph; Epithelial Sodium Channels; Evoked Potentials, Auditory; Furosemide; Guinea Pigs; Imidazoles; Nifedipine; Sodium Channel Blockers; Sodium Potassium Chloride Symporter Inhibitors; Thapsigargin; TRPC Cation Channels | 2009 |
The small molecule phenamil is a modulator of adipocyte differentiation and PPARgamma expression.
Topics: 3T3 Cells; Adipocytes; Amiloride; Animals; CCAAT-Enhancer-Binding Protein-delta; Cell Differentiation; DNA-Binding Proteins; Gene Expression Regulation; Harmine; Mice; Molecular Structure; Monoamine Oxidase Inhibitors; Oxazoles; PPAR gamma; Proto-Oncogene Proteins c-ets; Signal Transduction; Sodium Channel Blockers; Transcription Factors; Tyrosine | 2010 |
The amiloride derivative phenamil attenuates pulmonary vascular remodeling by activating NFAT and the bone morphogenetic protein signaling pathway.
Topics: Acid Sensing Ion Channels; Amiloride; Animals; Base Sequence; Binding Sites; Bone Morphogenetic Proteins; Cell Proliferation; Humans; Hypertension, Pulmonary; Hypoxia; Lung; Male; Models, Biological; Molecular Sequence Data; Muscle Contraction; Nerve Tissue Proteins; NFATC Transcription Factors; Promoter Regions, Genetic; Protein Kinases; Protein Serine-Threonine Kinases; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Signal Transduction; Sodium Channels; Transcriptional Activation | 2011 |
Cross-reactivity of acid-sensing ion channel and Na⁺-H⁺ exchanger antagonists with nicotinic acetylcholine receptors.
Topics: Acid Sensing Ion Channels; Amiloride; Animals; Brain; Cell Line; Guanidines; In Vitro Techniques; Mice; Mice, Inbred C57BL; Mice, Knockout; Nerve Tissue Proteins; Neurons; Nicotine; Nicotinic Agonists; Oocytes; Pyrazoles; Receptors, Nicotinic; Sodium Channel Blockers; Sodium Channels; Sodium-Hydrogen Exchangers; Synaptic Transmission; Xenopus | 2011 |
Pharmacological characterisation of apical Na+ and Cl- transport mechanisms of the anal papillae in the larval mosquito Aedes aegypti.
Topics: Aedes; Amiloride; Anal Canal; Animals; Bumetanide; Carbonic Anhydrases; Chlorides; Ion Transport; Ion-Selective Electrodes; Larva; Macrolides; Methazolamide; Microelectrodes; Models, Biological; Ouabain; Sodium; Sodium-Potassium-Chloride Symporters; Sodium-Potassium-Exchanging ATPase; Vacuolar Proton-Translocating ATPases | 2011 |
Comparative characterization of Na+ transport in Cyprinodon variegatus variegatus and Cyprinodon variegatus hubbsi: a model species complex for studying teleost invasion of freshwater.
Topics: Acclimatization; Amiloride; Animals; Cell Size; Chlorides; Epithelium; Fresh Water; Gills; Introduced Species; Ion Transport; Killifishes; Kinetics; Macrolides; Metolazone; Mitochondria; Models, Animal; Sodium; Species Specificity; Time Factors | 2012 |
Evaluating the feasibility of utilizing the small molecule phenamil as a novel biofactor for bone regenerative engineering.
Topics: Alkaline Phosphatase; Amiloride; Animals; Biocompatible Materials; Bone Matrix; Bone Regeneration; Calcification, Physiologic; Cell Adhesion; Cell Line; Cell Proliferation; Feasibility Studies; Lactic Acid; Mice; Microspheres; Osteoblasts; Polyglycolic Acid; Polylactic Acid-Polyglycolic Acid Copolymer; Small Molecule Libraries; Tissue Engineering; Tissue Scaffolds | 2014 |
Short-term administration of small molecule phenamil induced a protracted osteogenic effect on osteoblast-like MC3T3-E1 cells.
Topics: Amiloride; Animals; Antigens, Differentiation; Cell Differentiation; Cell Line; Drug Carriers; Lactic Acid; Mice; Osteoblasts; Osteogenesis; Polyglycolic Acid; Polylactic Acid-Polyglycolic Acid Copolymer | 2016 |
Stimulating effects of quercetin and phenamil on differentiation of human dental pulp cells.
Topics: Alkaline Phosphatase; Amiloride; Antioxidants; Cell Differentiation; Cells, Cultured; Dental Pulp; Dentinogenesis; Extracellular Matrix Proteins; Extracellular Signal-Regulated MAP Kinases; Gene Expression; Humans; MAP Kinase Signaling System; Osteoblasts; Osteocalcin; Phosphoproteins; Quercetin; Real-Time Polymerase Chain Reaction; RNA, Messenger; Sialoglycoproteins | 2013 |
Ammonia transport across the skin of adult rainbow trout (Oncorhynchus mykiss) exposed to high environmental ammonia (HEA).
Topics: Amiloride; Ammonia; Animals; Body Surface Area; Cation Transport Proteins; Environment; Fish Proteins; In Vitro Techniques; Oncorhynchus mykiss; Proton-Translocating ATPases; RNA, Messenger; Skin; Sodium; Sodium Channel Blockers; Sodium-Hydrogen Exchangers | 2014 |
Quorum sensing positively regulates flagellar motility in pathogenic Vibrio harveyi.
Topics: Amiloride; Animals; Aquatic Organisms; Artemia; Bacterial Proteins; Flagella; Quorum Sensing; Repressor Proteins; Sodium Channels; Trans-Activators; Transcription Factors; Vibrio; Virulence Factors | 2015 |
An in vitro investigation of gastrointestinal Na(+) uptake mechanisms in freshwater rainbow trout.
Topics: Amiloride; Animals; Biological Transport; Fresh Water; Furosemide; Gastrointestinal Tract; Hydrochlorothiazide; In Vitro Techniques; Kinetics; Macrolides; Models, Biological; Oncorhynchus mykiss; Osmolar Concentration; Osmoregulation; Regression Analysis; Sodium Radioisotopes | 2014 |
Delivery of Phenamil Enhances BMP-2-Induced Osteogenic Differentiation of Adipose-Derived Stem Cells and Bone Formation in Calvarial Defects.
Topics: Adipose Tissue; Amiloride; Animals; Bone Morphogenetic Protein 2; Bone Regeneration; Cell Cycle Proteins; Cell Differentiation; Cell Proliferation; Cells, Cultured; Lactic Acid; Mice, Inbred C57BL; Mice, Nude; Microscopy, Electron, Scanning; Osteogenesis; Polyglycolic Acid; Polylactic Acid-Polyglycolic Acid Copolymer; Skull; Smad Proteins; Stem Cells; Tissue Scaffolds; Ubiquitin-Protein Ligases; X-Ray Microtomography | 2015 |
Cloning and characterization of Na(+)/H(+) Exchanger isoforms NHE2 and NHE3 from the gill of Pacific dogfish Squalus suckleyi.
Topics: Amiloride; Animals; Biological Transport, Active; Cell Line; Cloning, Molecular; Cricetinae; Dogfish; Epithelial Sodium Channel Blockers; Fish Proteins; Gills; Inhibitory Concentration 50; Protein Isoforms; Sodium-Hydrogen Exchangers | 2015 |
Enhanced Osteogenesis of Adipose-Derived Stem Cells by Regulating Bone Morphogenetic Protein Signaling Antagonists and Agonists.
Topics: Adipose Tissue; Adult Stem Cells; Amiloride; Animals; Bone Morphogenetic Proteins; Carrier Proteins; Cell Differentiation; Cells, Cultured; Male; Mice; Mice, Inbred C57BL; Mice, Nude; Osteogenesis; Signal Transduction; Smad Proteins | 2016 |
Re-Epithelialization of Pathological Cutaneous Wounds Is Improved by Local Mineralocorticoid Receptor Antagonism.
Topics: Administration, Cutaneous; Amiloride; Animals; Clobetasol; Epidermis; Glucocorticoids; Humans; Keratinocytes; Mice; Mineralocorticoid Receptor Antagonists; Ointments; Re-Epithelialization; Receptors, Mineralocorticoid; Skin; Wound Healing | 2016 |
5-(N, N-Hexamethylene) amiloride is a GABA-A ρ1 receptor positive allosteric modulator.
Topics: Allosteric Regulation; Amiloride; Binding Sites; Electrophysiology; gamma-Aminobutyric Acid; Guanidine; HEK293 Cells; Humans; Mutagenesis, Site-Directed; Receptors, GABA-B | 2016 |
Phenamil enhances the adipogenic differentiation of hen preadipocytes.
Topics: Adipocytes; Adipogenesis; Amiloride; Animals; CCAAT-Enhancer-Binding Protein-alpha; CCAAT-Enhancer-Binding Protein-beta; Cell Differentiation; Cells, Cultured; Chickens; Fatty Acid-Binding Proteins; Female; Oleic Acid; PPAR gamma | 2016 |
Enhanced Mandibular Bone Repair by Combined Treatment of Bone Morphogenetic Protein 2 and Small-Molecule Phenamil.
Topics: Amiloride; Animals; Bone Morphogenetic Protein 2; Drug Implants; Humans; Mandible; Mandibular Injuries; Mesenchymal Stem Cells; Rats, Sprague-Dawley | 2017 |
Effects of Bioactive Compounds on Odontogenic Differentiation and Mineralization.
Topics: Amiloride; Animals; Calcification, Physiologic; Dental Pulp; Dose-Response Relationship, Drug; Genistein; Metformin; Mice; Mice, Nude; Morpholines; Odontogenesis; Purines; Stem Cell Transplantation | 2017 |
Phenamil, an amiloride derivative, restricts long bone growth and alters keeled-sternum bone architecture in growing chickens.
Topics: Amiloride; Animal Feed; Animals; Avian Proteins; Calcification, Physiologic; Chickens; Female; Male; Osteogenesis; Sternum; Tibia | 2017 |
Intracellular co-delivery of Sr ion and phenamil drug through mesoporous bioglass nanocarriers synergizes BMP signaling and tissue mineralization.
Topics: Amiloride; Bone Morphogenetic Proteins; Calcification, Physiologic; Cell Culture Techniques; Cells, Cultured; Drug Carriers; Humans; Mesenchymal Stem Cells; Nanoparticles; Odontogenesis; Osteogenesis; Porosity; Signal Transduction; Strontium | 2017 |
Small molecule-mediated tribbles homolog 3 promotes bone formation induced by bone morphogenetic protein-2.
Topics: Adipogenesis; Amiloride; Animals; Bone Density Conservation Agents; Bone Morphogenetic Protein 2; Bone Regeneration; Cell Differentiation; Drug Synergism; Drug Therapy, Combination; Enzyme Activation; Gene Expression Regulation; Inflammation; Male; Mandible; Mandibular Injuries; Mesenchymal Stem Cells; NF-kappa B; Osteoblasts; Osteogenesis; PPAR gamma; Protein Serine-Threonine Kinases; Rats; Rats, Sprague-Dawley; Signal Transduction; Treatment Outcome | 2017 |
Sodium-powered stators of the bacterial flagellar motor can generate torque in the presence of phenamil with mutations near the peptidoglycan-binding region.
Topics: Amiloride; ATP-Binding Cassette Transporters; Bacterial Proteins; Escherichia coli; Escherichia coli Proteins; Flagella; Molecular Motor Proteins; Peptidoglycan; Phylogeny; Point Mutation; Sodium; Sodium Channel Blockers; Sodium Channels; Torque; Vibrio alginolyticus | 2019 |
Enhanced Cellular Uptake Of Phenamil Through Inclusion Complex With Histidine Functionalized β-Cyclodextrin As Penetrative Osteoinductive Agent.
Topics: 2-Hydroxypropyl-beta-cyclodextrin; Adipose Tissue; Amiloride; Calcification, Physiologic; Cell Survival; Endocytosis; Histidine; Humans; Molecular Docking Simulation; Osseointegration; Osteogenesis; Particle Size; Proton Magnetic Resonance Spectroscopy; Solubility; Spectroscopy, Fourier Transform Infrared; Static Electricity; Stem Cells | 2019 |
Mineralized nanofibrous scaffold promotes phenamil-induced osteoblastic differentiation while mitigating adipogenic differentiation.
Topics: Adipogenesis; Amiloride; Animals; Cell Differentiation; Cell Line; Mice; Nanofibers; Osteoblasts; Tissue Scaffolds | 2020 |
One-pot porogen free method fabricated porous microsphere-aggregated 3D PCL scaffolds for bone tissue engineering.
Topics: Amiloride; Apatites; Biocompatible Materials; Bone Morphogenetic Protein 2; Bone Regeneration; Cell Differentiation; Cell Survival; Drug Liberation; Gene Expression; Humans; Microspheres; Nanostructures; Polyesters; Porosity; Recombinant Proteins; Tissue Engineering; Tissue Scaffolds; Transforming Growth Factor beta | 2020 |
An Elastic Mineralized 3D Electrospun PCL Nanofibrous Scaffold for Drug Release and Bone Tissue Engineering.
Topics: Amiloride; Animals; Bone Regeneration; Cell Differentiation; Cell Line; Durapatite; Elastic Modulus; Extracellular Matrix; Mice; Minerals; Nanofibers; Osteoclasts; Osteogenesis; Polyesters; Porosity; Printing, Three-Dimensional; Serum Albumin, Bovine; Surface Properties; Tissue Engineering | 2021 |
Dual drug delivery system of teicoplanin and phenamil based on pH-sensitive silk fibroin/sodium alginate hydrogel scaffold for treating chronic bone infection.
Topics: Alginates; Amiloride; Animals; Anti-Bacterial Agents; Drug Delivery Systems; Fibroins; Hydrogels; Hydrogen-Ion Concentration; Methicillin-Resistant Staphylococcus aureus; Osteomyelitis; Rats; Teicoplanin | 2022 |