Page last updated: 2024-08-21

amiloride and chloroquine

amiloride has been researched along with chloroquine in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19901 (5.56)18.7374
1990's8 (44.44)18.2507
2000's4 (22.22)29.6817
2010's5 (27.78)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Bansal, DD; MacGregor, RR1
Augustine, EC; Kensinger, RS1
Broxterman, HJ; Kuiper, CM; Lankelma, J; Pinedo, HM; Schuurhuis, GJ1
Lanzer, M; Sanchez, CP; Wünsch, S1
Gekle, M; Grosse-Wortmann, L; Lanzer, M; Sanchez, CP; Wiesner, J; Wünsch, S1
Kulda, J; Schrével, J; Suchan, P; Tachezy, J1
Bray, PG; Ginsburg, H; Janneh, O; Mungthin, M; Raynes, KJ; Ward, SA1
Bray, PG; Ginsburg, H; Ward, SA1
Cerami, A; Dzekunov, S; Ferrer, AS; Martiney, JA; Roepe, P1
Norbury, CC1
Ma, DX; Qi, XR1
Ashraf, S; Gil, PR; Nazarenus, M; Parak, WJ1
Alper, SL; Alves, J; Hsu, A; Hubner, CA; Rivera, A; Rust, MB; Shmukler, BE; Trudel, M1

Reviews

3 review(s) available for amiloride and chloroquine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Na+/H+ antiporter, chloroquine uptake and drug resistance: inconsistencies in a newly proposed model.
    Parasitology today (Personal ed.), 1999, Volume: 15, Issue:9

    Topics: Amiloride; Animals; Antimalarials; Chloroquine; Drug Resistance; Humans; Malaria, Falciparum; Plasmodium falciparum; Sodium-Hydrogen Exchangers; Vacuoles

1999
Chloroquine uptake, altered partitioning and the basis of drug resistance: evidence for chloride-dependent ionic regulation.
    Novartis Foundation symposium, 1999, Volume: 226

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Animals; Antimalarials; Chlorides; Chloroquine; Diuretics; Drug Resistance; Plasmodium falciparum; Sodium-Hydrogen Exchangers

1999

Other Studies

15 other study(ies) available for amiloride and chloroquine

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Secretion of plasminogen activator from bovine parathyroid cells.
    Endocrinology, 1990, Volume: 126, Issue:5

    Topics: Adenine; Amiloride; Animals; Calcitriol; Calcium; Cattle; Cells, Cultured; Chloroquine; Fibrin; Hydrocortisone; Microsomes; Molecular Weight; Oligopeptides; Organelles; Parathyroid Glands; Parathyroid Hormone; Plasminogen Activators; Plasminogen Inactivators; Urokinase-Type Plasminogen Activator

1990
Endocytosis and degradation of ovine prolactin by Nb2 lymphoma cells: characterization and effects of agents known to alter prolactin-induced mitogenesis.
    Endocrinology, 1990, Volume: 127, Issue:1

    Topics: Amiloride; Animals; Calcimycin; Cell Division; Cell Membrane; Chloroquine; Endocytosis; Kinetics; Leupeptins; Lymphoma; Methylamines; Mitosis; Monensin; Prolactin; Rats; Receptors, Prolactin; Sheep; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured

1990
Glycolysis in P-glycoprotein-overexpressing human tumor cell lines. Effects of resistance-modifying agents.
    FEBS letters, 1989, Apr-24, Volume: 247, Issue:2

    Topics: Adenosine Triphosphate; Amiloride; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood Proteins; Chloroquine; Cytochalasin B; Drug Resistance; Energy Metabolism; Glutathione Transferase; Glycolysis; Humans; Hydrogen-Ion Concentration; Lactates; Lactic Acid; Membrane Glycoproteins; Monensin; Nigericin; Oxygen Consumption; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Verapamil

1989
Identification of a chloroquine importer in Plasmodium falciparum. Differences in import kinetics are genetically linked with the chloroquine-resistant phenotype.
    The Journal of biological chemistry, 1997, Jan-31, Volume: 272, Issue:5

    Topics: Amiloride; Animals; Binding, Competitive; Biological Transport; Chloroquine; Crosses, Genetic; Drug Resistance; Erythrocytes; Humans; Kinetics; Phenotype; Plasmodium falciparum; Sodium-Hydrogen Exchangers; Temperature

1997
Differential stimulation of the Na+/H+ exchanger determines chloroquine uptake in Plasmodium falciparum.
    The Journal of cell biology, 1998, Jan-26, Volume: 140, Issue:2

    Topics: Amiloride; Animals; Antimalarials; Chloroquine; Cytoplasm; Drug Resistance; Fluorometry; Humans; Hydrogen-Ion Concentration; Phenotype; Plasmodium falciparum; Sodium-Hydrogen Exchangers

1998
The host-protein-independent iron uptake by Tritrichomonas foetus.
    Experimental parasitology, 1998, Volume: 90, Issue:2

    Topics: Amiloride; Ammonium Chloride; Animals; Antiprotozoal Agents; Ascorbic Acid; Cattle; Chloroquine; Ferric Compounds; Iron; Iron Chelating Agents; Lactoferrin; Nitrilotriacetic Acid; Oxidation-Reduction; Sodium Fluoride; Transferrin; Tritrichomonas foetus

1998
Cellular uptake of chloroquine is dependent on binding to ferriprotoporphyrin IX and is independent of NHE activity in Plasmodium falciparum.
    The Journal of cell biology, 1999, Apr-19, Volume: 145, Issue:2

    Topics: Amiloride; Animals; Antimalarials; Bicarbonates; Biological Transport; Chloroquine; Erythrocyte Membrane; Erythrocytes; Hemin; Hemoglobins; Humans; Hydrogen-Ion Concentration; Kinetics; Leupeptins; Plasmodium falciparum; Sodium-Hydrogen Exchangers; Verapamil

1999
Tracing the route taken by peptides and major histocompatibility complex class I molecules in presentation of exogenous antigens.
    Methods in molecular biology (Clifton, N.J.), 2001, Volume: 156

    Topics: Amiloride; Animals; Antigen Presentation; Antigen-Presenting Cells; Antigens; beta 2-Microglobulin; Chloroquine; Cytochalasins; Endocytosis; Fluorescein-5-isothiocyanate; Histocompatibility Antigens Class I; Killer Cells, Natural; Phagocytosis; Sensitivity and Specificity; Spectrometry, Fluorescence; T-Lymphocytes

2001
[Comparison of mechanisms and cellular uptake of cell-penetrating peptide on different cell lines].
    Yao xue xue bao = Acta pharmaceutica Sinica, 2010, Volume: 45, Issue:9

    Topics: Adsorption; Amiloride; Cell Line, Tumor; Cell Membrane; Cell-Penetrating Peptides; Chloroquine; Chlorpromazine; Dose-Response Relationship, Drug; Exocytosis; Heparin; Humans; Proteoglycans; Temperature; Time Factors

2010
pH-sensitive capsules as intracellular optical reporters for monitoring lysosomal pH changes upon stimulation.
    Small (Weinheim an der Bergstrasse, Germany), 2012, Mar-26, Volume: 8, Issue:6

    Topics: Amiloride; Chloroquine; Fluorescence; Hydrogen-Ion Concentration; Lysosomes; Macrolides; Monensin

2012
N-ethylmaleimide activates a Cl(-)-independent component of K(+) flux in mouse erythrocytes.
    Blood cells, molecules & diseases, 2013, Volume: 51, Issue:1

    Topics: Amiloride; Animals; Chlorides; Chloroquine; Drug Resistance; Erythrocytes; Ethylmaleimide; Hemoglobin, Sickle; Intermediate-Conductance Calcium-Activated Potassium Channels; K Cl- Cotransporters; Mice; Mice, Knockout; Potassium; Symporters; Temperature

2013