am 580 and agn 193836

am 580 has been researched along with agn 193836 in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's1 (33.33)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beard, RL; Chandraratna, RA; Duong, TT; Klein, ES; Standevan, AM; Teng, M1
Chandraratna, RA; Duong, TT; Klein, ES; Pino, ME; Teng, M1
Adams, DR; Barlow, S; Borthwick, AD; Brown, JT; Clarke, E; Corcoran, JPT; Goncalves, MB; Jarvis, CI; Kalindjian, SB; Miller, I; Ravier, E; Shiers, JJ; Smith, V; Taddei, DMA1

Other Studies

3 other study(ies) available for am 580 and agn 193836

ArticleYear
Synthesis and biological activity of retinoic acid receptor-alpha specific amides.
    Bioorganic & medicinal chemistry letters, 2002, Nov-04, Volume: 12, Issue:21

    Topics: Amides; Antineoplastic Agents; Breast Neoplasms; Female; Humans; Hydrogen Bonding; Receptors, Retinoic Acid; Retinoic Acid Receptor alpha; Retinoids; Structure-Activity Relationship

2002
Identification of a retinoic acid receptor alpha subtype specific agonist.
    Journal of medicinal chemistry, 1996, Aug-02, Volume: 39, Issue:16

    Topics: Aminobenzoates; Animals; Benzoates; Cell Line; Dose-Response Relationship, Drug; Genes, Reporter; Molecular Structure; Protein Binding; Receptors, Retinoic Acid; Recombinant Fusion Proteins; Retinoic Acid Receptor alpha; Retinoid X Receptors; Retinoids; Tetrahydronaphthalenes; Transcription Factors; Transcriptional Activation; Transfection

1996
Design and synthesis of a potent, highly selective, orally bioavailable, retinoic acid receptor alpha agonist.
    Bioorganic & medicinal chemistry, 2018, 02-15, Volume: 26, Issue:4

    Topics: Administration, Oral; Aminobenzoates; Animals; Benzoates; Cell Survival; Chlorocebus aethiops; COS Cells; Drug Design; Half-Life; Hep G2 Cells; Humans; Mice; Microsomes, Liver; Rats; Receptors, Retinoic Acid; Retinoic Acid Receptor alpha; Retinoic Acid Receptor gamma; Structure-Activity Relationship; Tetrahydronaphthalenes

2018