am 251 and orlistat

am 251 has been researched along with orlistat in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (16.67)29.6817
2010's5 (83.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adams, Y; Ahenkorah, S; Laitinen, JT; Laitinen, T; Navia-Paldanius, D; Nevalainen, TJ; Parkkari, T; Patel, JZ; Savinainen, JR; Staszewski, M; Vaara, M; Walczyński, K1
Kaczor, AA; Laitinen, JT; Laitinen, T; Navia-Paldanius, D; Nevalainen, TJ; Parkkari, T; Patel, JZ; Savinainen, JR; van Bruchem, J1
Hashimoto, K; Kano, M; Kawata, S; Tanimura, A1
Chiou, LC; Fu, SY; Ho, YC; Lee, HJ; Liao, HT; Liao, YY; Mackie, K; Teng, SF; Tung, LW1
Gyires, K; Hunyady, L; Németh, J; Rónai, AZ; Szekeres, M; Tóth, VE; Zádori, ZS1
Becerril-Meléndez, AL; Marichal-Cancino, BA; Méndez-Díaz, M; Prospéro-Garcia, O; Ruiz-Contreras, AE; Sánchez-Fuentes, A1

Other Studies

6 other study(ies) available for am 251 and orlistat

ArticleYear
Loratadine analogues as MAGL inhibitors.
    Bioorganic & medicinal chemistry letters, 2015, Apr-01, Volume: 25, Issue:7

    Topics: Amidohydrolases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Loratadine; Models, Molecular; Molecular Structure; Monoacylglycerol Lipases; Recombinant Proteins; Structure-Activity Relationship

2015
Revisiting 1,3,4-Oxadiazol-2-ones: Utilization in the Development of ABHD6 Inhibitors.
    Bioorganic & medicinal chemistry, 2015, Oct-01, Volume: 23, Issue:19

    Topics: Animals; Binding Sites; Catalytic Domain; Enzyme Inhibitors; Mice; Molecular Docking Simulation; Monoacylglycerol Lipases; Oxadiazoles; Protein Binding; Receptors, Cannabinoid; Serine Proteases; Structure-Activity Relationship

2015
Not glutamate but endocannabinoids mediate retrograde suppression of cerebellar parallel fiber to Purkinje cell synaptic transmission in young adult rodents.
    Neuropharmacology, 2009, Volume: 57, Issue:2

    Topics: Aging; Animals; Calcium; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Cerebellum; Endocannabinoids; Enzyme Inhibitors; Glutamic Acid; Humans; In Vitro Techniques; Lactones; Mice; Mice, Inbred C57BL; Mice, Knockout; Neural Inhibition; Orlistat; Piperidines; Purkinje Cells; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Cannabinoid; Synaptic Transmission

2009
Activation of orexin 1 receptors in the periaqueductal gray of male rats leads to antinociception via retrograde endocannabinoid (2-arachidonoylglycerol)-induced disinhibition.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Oct-12, Volume: 31, Issue:41

    Topics: Analysis of Variance; Animals; Animals, Newborn; Arachidonic Acids; Benzoxazines; Benzoxazoles; Biphenyl Compounds; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Disease Models, Animal; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Estrenes; gamma-Aminobutyric Acid; Glycerides; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Intracellular Signaling Peptides and Proteins; Lactones; Male; Morpholines; Naphthalenes; Naphthyridines; Neural Inhibition; Neural Pathways; Neuropeptides; Orexin Receptors; Orexins; Orlistat; Pain; Pain Measurement; Patch-Clamp Techniques; Periaqueductal Gray; Piperidines; Pyrazoles; Pyrrolidinones; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea

2011
Angiotensin II-induced activation of central AT1 receptors exerts endocannabinoid-mediated gastroprotective effect in rats.
    Molecular and cellular endocrinology, 2014, Feb-15, Volume: 382, Issue:2

    Topics: Angiotensin II; Animals; Atropine; CHO Cells; Cricetulus; Ethanol; Gastric Mucosa; Gene Expression Regulation; Injections, Intraventricular; Lactones; Lipoprotein Lipase; Male; Mice; Mice, Knockout; Orlistat; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Angiotensin, Type 1; Receptor, Cannabinoid, CB1; Signal Transduction; Stomach; Stomach Ulcer; Vagotomy; Vagus Nerve

2014
mGluR1/5 activation in the lateral hypothalamus increases food intake via the endocannabinoid system.
    Neuroscience letters, 2016, Sep-19, Volume: 631

    Topics: Animals; Eating; Endocannabinoids; Enzyme Inhibitors; Glycine; Hypothalamic Area, Lateral; Lactones; Lipoprotein Lipase; Male; Orlistat; Phenylacetates; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate

2016
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