am 251 and leptin

am 251 has been researched along with leptin in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (22.22)29.6817
2010's7 (77.78)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Black, SC; Hildebrandt, AL; Kelly-Sullivan, DM1
Judge, MK; Scarpace, PJ; Zhang, Y1
Cunnane, SC; D'Asti, E; Di Marzo, V; Grajzer, M; Long, H; Tremblay-Mercier, J; Walker, CD1
Dodd, GT; Luckman, SM; Lutz, B; Mancini, G1
Bermúdez-Silva, FJ; Cifuentes, M; de Fonseca, FR; Fernández-Llebrez, P; Grondona, JM; López-Ávalos, MD; Pavón, FJ; Pérez-Martín, M; Rivera, P; Romero-Zerbo, Y; Serrano, A; Suárez, J1
Agar, E; Alici, SK; Arslan, G; Ayyildiz, M1
Aranda, P; Errami, M; Galisteo, M; Llopis, J; López-Chaves, C; López-Jurado, M; Martínez, R; Merroun, I; Porres, JM; Sánchez-González, C; Zarzuelo, A1
Bojanowska, E; Wierucka-Rybak, M; Wolak, M1
Bojanowska, E; Drobnik, J; Juszczak, M; Wierucka-Rybak, M; Wolak, M1

Other Studies

9 other study(ies) available for am 251 and leptin

ArticleYear
Antiobesity effects of chronic cannabinoid CB1 receptor antagonist treatment in diet-induced obese mice.
    European journal of pharmacology, 2003, Feb-21, Volume: 462, Issue:1-3

    Topics: Animals; Blood Glucose; Body Weight; Cholesterol; Dietary Fats; Dose-Response Relationship, Drug; Eating; Insulin; Leptin; Male; Mice; Mice, Inbred C57BL; Obesity; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Triglycerides

2003
Responses to the cannabinoid receptor-1 antagonist, AM251, are more robust with age and with high-fat feeding.
    The Journal of endocrinology, 2009, Volume: 203, Issue:2

    Topics: Age Factors; Animals; Appetite Depressants; Body Composition; Dietary Fats; Energy Intake; Hyperphagia; Ion Channels; Leptin; Male; Mitochondrial Proteins; Obesity; Piperidines; Pyrazoles; Rats; Rats, Inbred F344; Receptor, Cannabinoid, CB1; STAT3 Transcription Factor; Uncoupling Protein 1; Weight Gain

2009
Maternal dietary fat determines metabolic profile and the magnitude of endocannabinoid inhibition of the stress response in neonatal rat offspring.
    Endocrinology, 2010, Volume: 151, Issue:4

    Topics: Adipose Tissue; Adrenocorticotropic Hormone; Analysis of Variance; Animals; Animals, Suckling; Body Weight; Brain; Brain Chemistry; Cannabinoid Receptor Modulators; Corticosterone; Dietary Fats; Endocannabinoids; Fatty Acids; Female; Hypothalamo-Hypophyseal System; Insulin; Lactation; Leptin; Piperidines; Pituitary-Adrenal System; Pregnancy; Prenatal Exposure Delayed Effects; Prenatal Nutritional Physiological Phenomena; Pyrazoles; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Regression Analysis; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stress, Physiological

2010
The peptide hemopressin acts through CB1 cannabinoid receptors to reduce food intake in rats and mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, May-26, Volume: 30, Issue:21

    Topics: Analysis of Variance; Animals; Behavior, Animal; Benzoxazines; Chlorocebus aethiops; Circadian Rhythm; COS Cells; Cyclohexanols; Dose-Response Relationship, Drug; Drinking Behavior; Dronabinol; Drug Administration Routes; Eating; Food Deprivation; Green Fluorescent Proteins; Hemoglobins; Hyperphagia; Leptin; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Morpholines; Naphthalenes; Peptide Fragments; Piperidines; Protein Transport; Psychotropic Drugs; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Time Factors; Transfection

2010
Obesity-dependent cannabinoid modulation of proliferation in adult neurogenic regions.
    The European journal of neuroscience, 2011, Volume: 33, Issue:9

    Topics: Adiponectin; Animals; Blood Glucose; Body Weight; Cannabinoid Receptor Modulators; Cell Proliferation; Cholesterol; Dietary Fats; Energy Intake; Female; Insulin; Leptin; Male; Neurogenesis; Obesity; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Triglycerides

2011
The role of CB1-receptors in the proconvulsant effect of leptin on penicillin-induced epileptiform activity in rats.
    CNS neuroscience & therapeutics, 2013, Volume: 19, Issue:4

    Topics: Animals; Convulsants; Epilepsy; Infusions, Intraventricular; Leptin; Male; Penicillins; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1

2013
Novel effects of the cannabinoid inverse agonist AM 251 on parameters related to metabolic syndrome in obese Zucker rats.
    Metabolism: clinical and experimental, 2013, Volume: 62, Issue:11

    Topics: Animals; Biomarkers; Cannabinoid Receptor Antagonists; Eating; Energy Metabolism; Fatty Liver; Insulin; Insulin Resistance; Leptin; Lipid Metabolism; Liver; Male; Metabolic Syndrome; Obesity; Piperidines; Pyrazoles; Rats; Rats, Zucker; Receptor, Cannabinoid, CB1; Weight Gain

2013
The effects of leptin in combination with a cannabinoid receptor 1 antagonist, AM 251, or cannabidiol on food intake and body weight in rats fed a high-fat or a free-choice high sugar diet.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2014, Volume: 65, Issue:4

    Topics: Animals; Body Weight; Cannabidiol; Cannabinoid Receptor Antagonists; Diet, High-Fat; Dietary Sucrose; Drug Combinations; Eating; Leptin; Male; Piperidines; Pyrazoles; Rats, Wistar; Receptor, Cannabinoid, CB1

2014
The inhibitory effect of combination treatment with leptin and cannabinoid CB1 receptor agonist on food intake and body weight gain is mediated by serotonin 1B and 2C receptors.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2016, Volume: 67, Issue:3

    Topics: Aminopyridines; Animals; Cannabinoid Receptor Agonists; Drug Synergism; Eating; Indoles; Leptin; Male; Oxadiazoles; Piperazines; Piperidines; Pyrazoles; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Weight Gain

2016
chemdatabank.com