am 251 and am4113
am 251 has been researched along with am4113 in 9 studies
Research
Studies (9)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 4 (44.44) | 29.6817 |
2010's | 5 (55.56) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
---|---|
Brown, C; Fan, P; Makriyannis, A; McLaughlin, PJ; Olszewska, T; Olzewska, T; Pang, Y; Parker, LA; Peng, Y; Salamone, JD; Sink, KS; Thakur, GA; Vemuri, VK; Wood, JA | 1 |
Makriyannis, A; Olszewska, T; Salamone, JD; Sink, KS; Vemuri, VK | 1 |
Bow, JP; Hodge, J; Makriyannis, A; McLaughlin, PJ; Plyler, KS; Salamone, JD; Vemuri, VK; Wisniecki, A | 1 |
Collins, LE; Makriyannis, A; Nunes, EJ; Salamone, JD; Segovia, KN; Sink, KS; Thakur, G; Vemuri, VK | 1 |
Collins, LE; Correa, M; Makriyannis, A; Markus, EJ; Randall, PA; Salamone, JD; Segovia, KN; Sink, J; Sink, KS; Vemuri, VK | 1 |
Bashashati, M; Duncan, M; Hirota, C; Keenan, CM; Lutz, B; Mackie, K; Macnaughton, WK; Makriyannis, A; Sharkey, KA; Storr, MA; Vemuri, VK | 1 |
Collins, LE; Makriyannis, A; Markus, EJ; Salamone, JD; Segovia, KN; Sink, KS; Vemuri, VK | 1 |
Bedard, H; Chambers, AP; Cluny, NL; Limebeer, CL; Lutz, B; Makriyannis, A; Parker, LA; Sharkey, KA; Vemuri, VK; Wood, JT; Zimmer, A | 1 |
Keller, A; Raver, SM | 1 |
Other Studies
9 other study(ies) available for am 251 and am4113
Article | Year |
---|---|
The novel cannabinoid CB1 receptor neutral antagonist AM4113 suppresses food intake and food-reinforced behavior but does not induce signs of nausea in rats.
Topics: Adamantane; Analysis of Variance; Animals; Behavior, Animal; Conditioning, Operant; Cyclic AMP; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Eating; Male; Motor Activity; Nausea; Piperidines; Protein Binding; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reinforcement, Psychology | 2008 |
Cannabinoid CB1 antagonists and dopamine antagonists produce different effects on a task involving response allocation and effort-related choice in food-seeking behavior.
Topics: Animals; Benzazepines; Choice Behavior; Conditioning, Operant; Dopamine Antagonists; Feeding Behavior; Food Preferences; Injections, Intraperitoneal; Male; Motivation; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reinforcement Schedule; Salicylamides | 2008 |
The cannabinoid CB1 receptor inverse agonist AM 251 and antagonist AM 4113 produce similar effects on the behavioral satiety sequence in rats.
Topics: Animals; Appetite; Behavior, Animal; Feeding Behavior; Grooming; Injections, Intraperitoneal; Male; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Satiety Response | 2008 |
Intracerebroventricular administration of cannabinoid CB1 receptor antagonists AM251 and AM4113 fails to alter food-reinforced behavior in rats.
Topics: Analysis of Variance; Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Administration Routes; Drug Interactions; Eating; Food Deprivation; Injections, Intraventricular; Male; Motor Activity; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reinforcement Schedule; Reinforcement, Psychology | 2009 |
Potential anxiogenic effects of cannabinoid CB1 receptor antagonists/inverse agonists in rats: comparisons between AM4113, AM251, and the benzodiazepine inverse agonist FG-7142.
Topics: Animals; Anxiety; Brain; Carbolines; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Inverse Agonism; Exploratory Behavior; GABA Antagonists; Male; Maze Learning; Piperidines; Proto-Oncogene Proteins c-fos; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1 | 2010 |
Differential effects of CB(1) neutral antagonists and inverse agonists on gastrointestinal motility in mice.
Topics: Animals; Colon; Epithelium; Feces; Gastrointestinal Motility; Gastrointestinal Transit; Ileum; Immunohistochemistry; Ions; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle, Smooth; Permeability; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Water | 2010 |
The CB1 inverse agonist AM251, but not the CB1 antagonist AM4113, enhances retention of contextual fear conditioning in rats.
Topics: Acoustic Stimulation; Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Inverse Agonism; Fear; Freezing Reaction, Cataleptic; Male; Motor Activity; Piperidines; Pyrazoles; Random Allocation; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Time Factors | 2010 |
A novel peripherally restricted cannabinoid receptor antagonist, AM6545, reduces food intake and body weight, but does not cause malaise, in rodents.
Topics: Animals; Avoidance Learning; Benzoxazines; Body Weight; Brain; Conditioning, Classical; Cyclic AMP; Dose-Response Relationship, Drug; Eating; Female; Gastrointestinal Motility; HEK293 Cells; Humans; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2 | 2010 |
Permanent suppression of cortical oscillations in mice after adolescent exposure to cannabinoids: receptor mechanisms.
Topics: Animals; Benzoxazines; Cannabinoid Receptor Modulators; Dronabinol; Indoles; Male; Mice; Morpholines; Naphthalenes; Piperidines; Prefrontal Cortex; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Somatosensory Cortex; Tissue Culture Techniques | 2014 |