am 251 and am 404

am 251 has been researched along with am 404 in 40 studies

Research

Studies (40)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's23 (57.50)29.6817
2010's15 (37.50)24.3611
2020's2 (5.00)2.80

Authors

AuthorsStudies
Chiou, LC; Gean, PW; Huang, YC; Wang, SJ1
Dougalis, A; Lees, G1
Caraballo, I; El Banoua, F; Fernandez-Espejo, E; Ferrer, B; Flores, JA; Galan-Rodriguez, B; Rodriguez de Fonseca, F1
Mendiguren, A; Pineda, J1
Dinh, T; Freund, TF; Hájos, N; Kathuria, S; Piomelli, D1
Bátkai, S; Bukoski, RD; Harvey-White, J; Kunos, G; Liu, J; Mackie, K; Offertáler, L; Osei-Hyiaman, D; Pacher, P; Radaeva, S; Rudd, MA1
Bianchi, R; Borsani, E; Buffoli, B; Rezzani, R; Ricci, F; Rodella, LF1
Gorzalka, BB; Hill, MN; Sun, JC1
Gorzalka, BB; Hill, MN1
Baik, SK; Gaskari, SA; Lee, SS; Li, Y; Liu, H; Moezi, L1
Bazan, NG; Boudaba, C; Di, S; Harris, C; Marcheselli, VL; Popescu, IR; Tasker, JG; Weng, FJ1
Cheer, JF; Wassum, KM; Wightman, RM1
Ballini, C; Blandina, P; Cenni, G; Della Corte, L; Formigli, L; Giannoni, P; Mackie, K; Mannaioni, PF; Nosi, D; Passani, MB1
Galea, LA; Gorzalka, BB; Hill, MN; Kambo, JS; Sun, JC1
Aguiar, DC; Guimarães, FS; Moreira, FA1
Bianchi, R; Borsani, E; Labanca, M; Rodella, LF1
Beaulieu, P; Dani, M; Guindon, J; Lambert, C1
Gorzalka, BB; Hill, MN; Morrish, AC1
Greenwood, R; Jayamanne, A; Mitchell, VA; Vaughan, CW1
Alizadeh, AM; Haghparast, A; Khani, A; Motamedi, F; Naderi, N; Rezaii, N; Saber-Tehrani, A1
Finn, DP; Kelly, JP; O'Driscoll, M; Roche, M1
Aguiar, DC; Corrêa, FM; Guimarães, FS; Lisboa, SF; Resstel, LB1
Hasanein, P1
Alger, BE; Kim, J1
Bingham, B; Gorzalka, BB; Gray, JM; Hill, MN; Hillard, CJ; Lee, TT; McLaughlin, RJ; Shrestha, L; Viau, V1
Lu, L; Shimizu, T; Yokotani, K1
Corrêa, FM; da Silva, AL; Guimarães, FS; Lisboa, SF; Reis, DG; Resstel, LB1
Casarotto, PC; Gomes, FV; Guimarães, FS; Resstel, LB1
Calapai, G; Caputi, AP; Mannucci, C; Navarra, M; Pieratti, A; Russo, GA1
Bechard, M; Bishop, SF; Chi, N; Lauzon, NM; Laviolette, SR; Tan, H1
Jain, NS; Manna, SS; Umathe, SN1
Ayoub, SS; Baker, D; Bolton, C; Flower, RJ; Pryce, G; Seed, MP1
Alves, FH; Corrêa, FM; Fedoce, AG; Ferreira-Junior, NC; Resstel, LB1
Cho, HS; Choi, SJ; Jeun, SH; Kim, KJ; Li, QZ; Sung, KW1
Garcia-Bereguiain, MA; Gonzalez-Islas, C; Wenner, P1
Benkő, R; Benyó, Z; Di Marzo, V; Horváth, B; Iring, A; Járai, Z; Lacza, Z; Leszl-Ishiguro, M; Pacher, P; Ruisanchez, É; Sándor, P1
Aliev, R; Kitchigina, V; Shubina, L1
Higashi, Y; Nakamura, K; Saito, M; Shimizu, S; Shimizu, T; Tanaka, K; Taniuchi, K; Ueba, T; Yawata, T; Yuri, K1
Gianessi, CA; Groman, SM; Jiang, M; Taylor, JR; Thompson, SL; van der Stelt, M1
Hara, K; Haranishi, Y; Terada, T1

Other Studies

40 other study(ies) available for am 251 and am 404

ArticleYear
Mediation of amphetamine-induced long-term depression of synaptic transmission by CB1 cannabinoid receptors in the rat amygdala.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Nov-12, Volume: 23, Issue:32

    Topics: Amphetamine; Amygdala; Animals; Arachidonic Acids; Benzoxazines; Calcium; Calcium Channels; Central Nervous System Stimulants; Dopamine Antagonists; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; In Vitro Techniques; Ligands; Long-Term Synaptic Depression; Male; Morpholines; Naphthalenes; Patch-Clamp Techniques; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Synaptic Transmission

2003
Differential effects of the sleep-inducing lipid oleamide and cannabinoids on the induction of long-term potentiation in the CA1 neurons of the rat hippocampus in vitro.
    Brain research, 2004, Jan-30, Volume: 997, Issue:1

    Topics: Amidohydrolases; Analysis of Variance; Animals; Animals, Newborn; Arachidonic Acids; Benzoxazines; Cannabinoids; Capsaicin; Drug Interactions; Electric Stimulation; Electrophysiology; Endocannabinoids; Excitatory Postsynaptic Potentials; Hippocampus; Hypnotics and Sedatives; In Vitro Techniques; Long-Term Potentiation; Male; Morpholines; Naphthalenes; Neurons; Oleic Acids; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rimonabant; Sleep

2004
Experimental parkinsonism alters anandamide precursor synthesis, and functional deficits are improved by AM404: a modulator of endocannabinoid function.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2004, Volume: 29, Issue:6

    Topics: Acyltransferases; Amidohydrolases; Amphetamine; Analysis of Variance; Animals; Antiparkinson Agents; Arachidonic Acids; Behavior, Animal; Brain Chemistry; Cell Count; Central Nervous System Stimulants; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Endocannabinoids; Functional Laterality; Male; Motor Activity; Oxidopamine; Parkinsonian Disorders; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Rotation; Serotonin Antagonists; Serotonin Receptor Agonists; Substantia Nigra; Tyrosine 3-Monooxygenase

2004
Cannabinoids enhance N-methyl-D-aspartate-induced excitation of locus coeruleus neurons by CB1 receptors in rat brain slices.
    Neuroscience letters, 2004, Jun-03, Volume: 363, Issue:1

    Topics: Action Potentials; Analgesics; Animals; Arachidonic Acids; Benzoxazines; Calcium Channel Blockers; Cannabinoids; Cyclohexanols; Drug Interactions; Electrophysiology; Endocannabinoids; Excitatory Amino Acid Agonists; In Vitro Techniques; Locus Coeruleus; Male; Morpholines; N-Methylaspartate; Naphthalenes; Neurons; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant

2004
Endocannabinoid transport tightly controls 2-arachidonoyl glycerol actions in the hippocampus: effects of low temperature and the transport inhibitor AM404.
    The European journal of neuroscience, 2004, Volume: 19, Issue:11

    Topics: Animals; Animals, Newborn; Arachidonic Acids; Biological Transport; Cannabinoid Receptor Modulators; Dose-Response Relationship, Drug; Drug Interactions; Endocannabinoids; Excitatory Postsynaptic Potentials; Glycerides; Hippocampus; In Vitro Techniques; Male; Neural Inhibition; Neurons; Patch-Clamp Techniques; Piperidines; Pyrazoles; Rats; Rats, Wistar; Temperature; Tritium

2004
Endocannabinoids acting at cannabinoid-1 receptors regulate cardiovascular function in hypertension.
    Circulation, 2004, Oct-05, Volume: 110, Issue:14

    Topics: Amidohydrolases; Angiotensin II; Animals; Arachidonic Acids; Benzamides; Benzyl Compounds; Blood Pressure; Camphanes; Carbamates; Dronabinol; Endocannabinoids; Endothelium, Vascular; Hypertension; Male; Models, Cardiovascular; Myocardial Contraction; Myocardium; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Inbred Dahl; Rats, Inbred SHR; Rats, Inbred WKY; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Up-Regulation; Vascular Resistance; Vasodilation; Ventricular Function, Left

2004
AM404, an inhibitor of anandamide reuptake decreases Fos-immunoreactivity in the spinal cord of neuropathic rats after non-noxious stimulation.
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Animals; Arachidonic Acids; Capsaicin; Constriction; Dose-Response Relationship, Drug; Endocannabinoids; Immunohistochemistry; Indoles; Male; Physical Stimulation; Piperidines; Polyunsaturated Alkamides; Proto-Oncogene Proteins c-fos; Pyrazoles; Rats; Rats, Sprague-Dawley; Sciatic Nerve; Spinal Cord

2005
Functional role of the endocannabinoid system and AMPA/kainate receptors in 5-HT2A receptor-mediated wet dog shakes.
    European journal of pharmacology, 2005, May-23, Volume: 516, Issue:1

    Topics: Amphetamines; Animals; Arachidonic Acids; Behavior, Animal; Cannabinoid Receptor Modulators; Dose-Response Relationship, Drug; Endocannabinoids; Excitatory Amino Acid Antagonists; Injections, Intraperitoneal; Ketanserin; Male; Piperidines; Pyrazoles; Quinoxalines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT2A; Receptors, AMPA; Receptors, Kainic Acid; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists

2005
Pharmacological enhancement of cannabinoid CB1 receptor activity elicits an antidepressant-like response in the rat forced swim test.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2005, Volume: 15, Issue:6

    Topics: Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Arachidonic Acids; Desipramine; Dose-Response Relationship, Drug; Dronabinol; Male; Motor Activity; Oleic Acids; Piperidines; Pyrazoles; Rats; Rats, Long-Evans; Receptor, Cannabinoid, CB1; Swimming

2005
Role of endocannabinoids in the pathogenesis of cirrhotic cardiomyopathy in bile duct-ligated rats.
    British journal of pharmacology, 2005, Volume: 146, Issue:3

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Bile Ducts; Cardiomyopathies; Endocannabinoids; Gene Expression; Liver Cirrhosis, Experimental; Male; Myocardial Contraction; Papillary Muscles; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrodotoxin; Ventricular Function, Left

2005
Activity-dependent release and actions of endocannabinoids in the rat hypothalamic supraoptic nucleus.
    The Journal of physiology, 2005, Dec-15, Volume: 569, Issue:Pt 3

    Topics: Animals; Arachidonic Acids; Benzoxazines; Benzyl Compounds; Cannabinoid Receptor Modulators; Cannabinoids; Endocannabinoids; Excitatory Postsynaptic Potentials; Glutamic Acid; Glycerides; In Vitro Techniques; Male; Morpholines; Naphthalenes; Neurons; Piperidines; Polyunsaturated Alkamides; Presynaptic Terminals; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Presynaptic; Supraoptic Nucleus; Synaptic Transmission

2005
Cannabinoid modulation of electrically evoked pH and oxygen transients in the nucleus accumbens of awake rats.
    Journal of neurochemistry, 2006, Volume: 97, Issue:4

    Topics: Animals; Arachidonic Acids; Benzoxazines; Calcium Channel Blockers; Cannabinoids; Cerebrovascular Circulation; Electric Stimulation; Energy Metabolism; Hydrogen-Ion Concentration; Male; Medial Forebrain Bundle; Morpholines; Naphthalenes; Nucleus Accumbens; Oxygen Consumption; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant

2006
Differential effect of cannabinoid agonists and endocannabinoids on histamine release from distinct regions of the rat brain.
    The European journal of neuroscience, 2006, Volume: 24, Issue:6

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Bicuculline; Cannabinoid Receptor Modulators; Cannabinoids; Cell Differentiation; Chromatography, High Pressure Liquid; Endocannabinoids; GABA Antagonists; gamma-Aminobutyric Acid; Histamine; Hypothalamus; Immunohistochemistry; Male; Microdialysis; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Time Factors; Wakefulness

2006
Endocannabinoids modulate stress-induced suppression of hippocampal cell proliferation and activation of defensive behaviours.
    The European journal of neuroscience, 2006, Volume: 24, Issue:7

    Topics: Aggression; Animals; Arachidonic Acids; Behavior, Animal; Bromodeoxyuridine; Cannabinoid Receptor Modulators; Cell Count; Cell Proliferation; Endocannabinoids; Enzyme Inhibitors; Hippocampus; Immunohistochemistry; Male; Neural Inhibition; Odorants; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Stress, Psychological; Thiazoles

2006
Anxiolytic-like effect of cannabinoids injected into the rat dorsolateral periaqueductal gray.
    Neuropharmacology, 2007, Volume: 52, Issue:3

    Topics: Animals; Anxiety; Arachidonic Acids; Behavior, Animal; Cannabinoids; Disease Models, Animal; Dose-Response Relationship, Drug; Endocannabinoids; Male; Maze Learning; Periaqueductal Gray; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1

2007
AM404 decreases Fos-immunoreactivity in the spinal cord in a model of inflammatory pain.
    Brain research, 2007, Jun-04, Volume: 1152

    Topics: Animals; Arachidonic Acids; Capsaicin; Endocannabinoids; Immunohistochemistry; Indoles; Inflammation; Male; Pain; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Proto-Oncogene Proteins c-fos; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Spinal Cord; TRPV Cation Channels

2007
The local antinociceptive effects of paracetamol in neuropathic pain are mediated by cannabinoid receptors.
    European journal of pharmacology, 2007, Nov-14, Volume: 573, Issue:1-3

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Animals; Arachidonic Acids; Cannabinoid Receptor Antagonists; Disease Models, Animal; Dose-Response Relationship, Drug; Hindlimb; Hot Temperature; Hyperalgesia; Indoles; Male; Neuralgia; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Sciatic Nerve

2007
Endocannabinoid modulation of male rat sexual behavior.
    Psychopharmacology, 2008, Volume: 198, Issue:4

    Topics: Amidohydrolases; Animals; Appetitive Behavior; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Consummatory Behavior; Dose-Response Relationship, Drug; Ejaculation; Endocannabinoids; Enzyme Inhibitors; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Long-Evans; Receptor, Cannabinoid, CB1; Sexual Behavior, Animal

2008
Actions of the endocannabinoid transport inhibitor AM404 in neuropathic and inflammatory pain models.
    Clinical and experimental pharmacology & physiology, 2007, Volume: 34, Issue:11

    Topics: Analgesics; Animals; Arachidonic Acids; Cannabinoid Receptor Modulators; Carrier Proteins; Disease Models, Animal; Endocannabinoids; Freund's Adjuvant; Inflammation; Ligation; Male; Motor Activity; Pain; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Sciatic Nerve; Sciatic Neuropathy; Time Factors

2007
Interaction between cannabinoid compounds and diazepam on anxiety-like behaviour of mice.
    Pharmacology, biochemistry, and behavior, 2008, Volume: 89, Issue:1

    Topics: Amidohydrolases; Animals; Anxiety; Arachidonic Acids; Behavior, Animal; Benzamides; Benzoxazines; Cannabinoids; Carbamates; Data Interpretation, Statistical; Diazepam; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Enzyme Inhibitors; GABA Modulators; Hypnotics and Sedatives; Male; Mice; Morpholines; Naphthalenes; Piperidines; Postural Balance; Pyrazoles; Receptor, Cannabinoid, CB1

2008
Augmentation of endogenous cannabinoid tone modulates lipopolysaccharide-induced alterations in circulating cytokine levels in rats.
    Immunology, 2008, Volume: 125, Issue:2

    Topics: Anilides; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Cinnamates; Cytokines; Drug Synergism; Indoles; Interleukin-1beta; Interleukin-6; Lipopolysaccharides; Male; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Tumor Necrosis Factor-alpha

2008
Activation of CB1 cannabinoid receptors in the dorsolateral periaqueductal gray reduces the expression of contextual fear conditioning in rats.
    Psychopharmacology, 2008, Volume: 198, Issue:3

    Topics: Animals; Arachidonic Acids; Blood Pressure; Conditioning, Operant; Endocannabinoids; Fear; Heart Rate; Male; Microinjections; Neurotransmitter Uptake Inhibitors; Periaqueductal Gray; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1

2008
The endocannabinoid transport inhibitor AM404 modulates nociception in cholestasis.
    Neuroscience letters, 2009, Oct-25, Volume: 462, Issue:3

    Topics: Animals; Arachidonic Acids; Biological Transport; Camphanes; Cannabinoid Receptor Modulators; Cholestasis; Endocannabinoids; Male; Naloxone; Opioid Peptides; Pain; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2

2009
Reduction in endocannabinoid tone is a homeostatic mechanism for specific inhibitory synapses.
    Nature neuroscience, 2010, Volume: 13, Issue:5

    Topics: Agatoxins; Animals; Arachidonic Acids; Benzamides; Benzoxazines; Biophysics; Calcium; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Carbamates; Conotoxins; Dose-Response Relationship, Drug; Down-Regulation; Drug Interactions; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glycerides; Hippocampus; Homeostasis; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Morpholines; Naphthalenes; Nerve Net; Neural Inhibition; Neurons; Patch-Clamp Techniques; Piperidines; Polyamines; Polyunsaturated Alkamides; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Rimonabant; Sodium Channel Blockers; Synapses; Tetrodotoxin

2010
Endogenous cannabinoid signaling is essential for stress adaptation.
    Proceedings of the National Academy of Sciences of the United States of America, 2010, May-18, Volume: 107, Issue:20

    Topics: Adaptation, Physiological; Analysis of Variance; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Corticosterone; Endocannabinoids; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Signal Transduction; Stress, Physiological

2010
Possible inhibitory roles of endogenous 2-arachidonoylglycerol during corticotropin-releasing factor-induced activation of central sympatho-adrenomedullary outflow in anesthetized rats.
    European journal of pharmacology, 2010, Sep-01, Volume: 641, Issue:1

    Topics: Adrenal Medulla; Anesthesia; Animals; Arachidonic Acids; Brain; Cannabinoid Receptor Agonists; Cannabinoid Receptor Modulators; Catecholamines; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Endocannabinoids; Glycerides; Male; Monoacylglycerol Lipases; Piperidines; Pyrazoles; Rats; Rats, Wistar; Sympathetic Nervous System

2010
Cannabinoid CB1 receptors in the medial prefrontal cortex modulate the expression of contextual fear conditioning.
    The international journal of neuropsychopharmacology, 2010, Volume: 13, Issue:9

    Topics: Animals; Arachidonic Acids; Behavior, Animal; Blood Pressure; Cannabinoid Receptor Modulators; Carbolines; Conditioning, Classical; Electroshock; Endocannabinoids; Fear; Freezing Reaction, Cataleptic; GABA Antagonists; Heart Rate; Male; Piperidines; Polyunsaturated Alkamides; Prefrontal Cortex; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Synaptic Transmission

2010
Facilitation of CB1 receptor-mediated neurotransmission decreases marble burying behavior in mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 2011, Mar-30, Volume: 35, Issue:2

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Benzoxazines; Calcium Channel Blockers; Cannabinoids; Carbamates; Drug Interactions; Endocannabinoids; Male; Mice; Mice, Inbred C57BL; Morpholines; Motor Activity; Naphthalenes; Obsessive-Compulsive Disorder; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Synaptic Transmission

2011
Interactions between endocannabinoid and serotonergic systems in mood disorders caused by nicotine withdrawal.
    Nicotine & tobacco research : official journal of the Society for Research on Nicotine and Tobacco, 2011, Volume: 13, Issue:4

    Topics: Animals; Arachidonic Acids; Behavior, Animal; Cannabinoid Receptor Modulators; Disease Models, Animal; Drug Interactions; Endocannabinoids; Male; Mice; Mood Disorders; Motor Activity; Nicotine; Piperazines; Piperidines; Pyrazoles; Pyridines; Random Allocation; Receptor, Cannabinoid, CB1; Receptor, Serotonin, 5-HT1A; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Smoking Cessation; Substance Withdrawal Syndrome

2011
Cannabinoid transmission in the basolateral amygdala modulates fear memory formation via functional inputs to the prelimbic cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Apr-06, Volume: 31, Issue:14

    Topics: Action Potentials; Afferent Pathways; Amygdala; Analysis of Variance; Animals; Arachidonic Acids; Benzoxazines; Calcium Channel Blockers; Cannabinoids; Dose-Response Relationship, Drug; Electroshock; Fear; Functional Laterality; Male; Memory; Morpholines; Naphthalenes; Neural Inhibition; Neurons; Piperidines; Prefrontal Cortex; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Smell

2011
Involvement of endocannabinoids in antidepressant and anti-compulsive effect of fluoxetine in mice.
    Behavioural brain research, 2011, Sep-30, Volume: 223, Issue:1

    Topics: Animals; Antidepressive Agents; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Compulsive Behavior; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Endocannabinoids; Fluoxetine; Injections, Intraventricular; Male; Mice; Motor Activity; Piperidines; Polyunsaturated Alkamides; Pyrazoles

2011
Paracetamol-induced hypothermia is independent of cannabinoids and transient receptor potential vanilloid-1 and is not mediated by AM404.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:9

    Topics: Acetaminophen; Amidohydrolases; Anilides; Animals; Arachidonic Acids; Cannabinoids; Cinnamates; Hypothermia; Hypothermia, Induced; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2011
Medial prefrontal cortex endocannabinoid system modulates baroreflex activity through CB(1) receptors.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2012, Volume: 302, Issue:7

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Baroreflex; Benzamides; Blood Pressure; Cannabinoid Receptor Modulators; Carbamates; Endocannabinoids; Glutamic Acid; Male; Piperidines; Prefrontal Cortex; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1

2012
Involvement of the endocannabinoid system in ethanol-induced corticostriatal synaptic depression.
    Journal of pharmacological sciences, 2012, Volume: 120, Issue:1

    Topics: Animals; Arachidonic Acids; Benzoxazines; Brain; Cannabinoids; Ethanol; Excitatory Postsynaptic Potentials; Morpholines; Naphthalenes; Neurons; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1

2012
Tonic and transient endocannabinoid regulation of AMPAergic miniature postsynaptic currents and homeostatic plasticity in embryonic motor networks.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Sep-26, Volume: 32, Issue:39

    Topics: Age Factors; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analgesics; Animals; Arachidonic Acids; Benzoxazines; Chick Embryo; Electric Stimulation; Endocannabinoids; Excitatory Amino Acid Agonists; Female; gamma-Aminobutyric Acid; Heterocyclic Compounds, 1-Ring; Homeostasis; Male; Morpholines; Motor Neurons; Naphthalenes; Nerve Net; Neuronal Plasticity; Patch-Clamp Techniques; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Signal Transduction; Spinal Cord; Synaptic Potentials; Urea

2012
Role of endocannabinoids and cannabinoid-1 receptors in cerebrocortical blood flow regulation.
    PloS one, 2013, Volume: 8, Issue:1

    Topics: Animals; Arachidonic Acids; Arterial Pressure; Cerebrovascular Circulation; Endocannabinoids; Heart Rate; Hemodynamics; Hypercapnia; Hypertension; Hypoxia; Laser-Doppler Flowmetry; Male; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1

2013
Attenuation of kainic acid-induced status epilepticus by inhibition of endocannabinoid transport and degradation in guinea pigs.
    Epilepsy research, 2015, Volume: 111

    Topics: Amidohydrolases; Animals; Anticonvulsants; Arachidonic Acids; Benzamides; Biological Transport; Brain; Cannabinoid Receptor Antagonists; Carbamates; Endocannabinoids; Guinea Pigs; Kainic Acid; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Seizures; Status Epilepticus

2015
Possible inhibitory role of endogenous 2-arachidonoylglycerol as an endocannabinoid in (±)-epibatidine-induced activation of central adrenomedullary outflow in the rat.
    Neuropharmacology, 2015, Volume: 95

    Topics: Adrenal Medulla; Animals; Arachidonic Acids; Bridged Bicyclo Compounds, Heterocyclic; Catecholamines; Dose-Response Relationship, Drug; Endocannabinoids; Glycerides; Immunohistochemistry; Male; Neurons; Neurotransmitter Agents; Nicotinic Agonists; Paraventricular Hypothalamic Nucleus; Piperidines; Pyrazoles; Pyridines; Rats, Wistar; Receptor, Cannabinoid, CB1

2015
Endocannabinoid contributions to alcohol habits and motivation: Relevance to treatment.
    Addiction biology, 2020, Volume: 25, Issue:3

    Topics: Alcohol Drinking; Animals; Arachidonic Acids; Benzodioxoles; Cannabinoid Receptor Antagonists; Central Nervous System Depressants; Drug-Seeking Behavior; Endocannabinoids; Ethanol; Glycerides; Habits; Lipoprotein Lipase; Lithium Chloride; Mice; Monoacylglycerol Lipases; Motivation; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1

2020
Inhibitory effect of intrathecally administered AM404, an endocannabinoid reuptake inhibitor, on neuropathic pain in a rat chronic constriction injury model.
    Pharmacological reports : PR, 2021, Volume: 73, Issue:3

    Topics: Animals; Arachidonic Acids; Capsaicin; Constriction; Disease Models, Animal; Endocannabinoids; Hyperalgesia; Indoles; Male; Neuralgia; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rotarod Performance Test; Spinal Cord; TRPV Cation Channels

2021
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