Page last updated: 2024-09-04

als 8123 and isoproterenol

als 8123 has been researched along with isoproterenol in 1 studies

*Isoproterenol: Isopropyl analog of EPINEPHRINE; beta-sympathomimetic that acts on the heart, bronchi, skeletal muscle, alimentary tract, etc. It is used mainly as bronchodilator and heart stimulant. [MeSH]

*Isoproterenol: Isopropyl analog of EPINEPHRINE; beta-sympathomimetic that acts on the heart, bronchi, skeletal muscle, alimentary tract, etc. It is used mainly as bronchodilator and heart stimulant. [MeSH]

Compound Research Comparison

Studies
(als 8123)
Trials
(als 8123)
Recent Studies (post-2010)
(als 8123)
Studies
(isoproterenol)
Trials
(isoproterenol)
Recent Studies (post-2010) (isoproterenol)
50130,7808032,640

Protein Interaction Comparison

ProteinTaxonomyals 8123 (IC50)isoproterenol (IC50)
Beta-2 adrenergic receptorHomo sapiens (human)0.246
Beta-1 adrenergic receptorHomo sapiens (human)0.333
Beta-2 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)1.77
Beta-1 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-3 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-2 adrenergic receptorCanis lupus familiaris (dog)0.6667

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19901 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gorczynski, RJ; Quon, CY; Shaffer, JE1

Other Studies

1 other study(ies) available for als 8123 and isoproterenol

ArticleYear
Beta-adrenoreceptor antagonist potency and pharmacodynamics of ASL-8123, the primary acid metabolite of esmolol.
    Journal of cardiovascular pharmacology, 1988, Volume: 11, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Dogs; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Infusions, Intravenous; Isoproterenol; Male; Propanolamines

1988