alprenolol and ici 118551

alprenolol has been researched along with ici 118551 in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19907 (41.18)18.7374
1990's2 (11.76)18.2507
2000's7 (41.18)29.6817
2010's1 (5.88)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carrupt, PA; el Tayar, N; Testa, B; Van de Waterbeemd, H1
Baker, JG1
Deupi, X; Farrens, D; Kobilka, B; Parnot, C; Ratnala, VR; Swaminath, G; Yao, X1
Bonin, H; Bouvier, M; Frielle, T; Nantel, F; Nguyen, CT; Suzuki, T; Valiquette, M1
Doggrell, SA1
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW1
Abrahamsson, T1
Hughes, RJ; Insel, PA; Mahan, LC1
Brunswick, DJ; Conway, PG; Tondo, L1
Crankshaw, DJ; Ruzycky, AL1
Allen, LF; Apparsundaram, S; Bond, RA; Hyek, MF; Johnson, TD; Kenakin, TP; Leff, P; McMinn, TR; Milano, CA; Rockman, HA1
Bond, RA; Callaerts-Vegh, Z; Evans, KL; Liu, X1
Bond, RA; Callaerts-Vegh, Z; Cuba, DL; Davies, PJ; Evans, KL; Giles, H; Gurji, HA; Shipley, GL1
Denda, M; Fuziwara, S; Inoue, K1
Devanathan, S; Kobilka, B; Salamon, Z; Tollin, G; Yao, Z1
Brahmadevara, N; MacDonald, A; Shaw, AM1
Bai, Q; Ban, Y; Liu, H; Yao, X; Zhang, Y1

Reviews

1 review(s) available for alprenolol and ici 118551

ArticleYear
Modeling of beta-adrenoceptors based on molecular electrostatic potential studies of agonists and antagonists.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:11

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Models, Molecular; Receptors, Adrenergic, beta; Structure-Activity Relationship

1988

Other Studies

16 other study(ies) available for alprenolol and ici 118551

ArticleYear
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
    British journal of pharmacology, 2005, Volume: 144, Issue:3

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

2005
Coupling ligand structure to specific conformational switches in the beta2-adrenoceptor.
    Nature chemical biology, 2006, Volume: 2, Issue:8

    Topics: Adrenergic beta-2 Receptor Agonists; Albuterol; Alprenolol; Amino Acid Sequence; Binding Sites; Crystallography, X-Ray; Epinephrine; Humans; Isoproterenol; Ligands; Models, Molecular; Molecular Sequence Data; Molecular Structure; Propanolamines; Protein Conformation; Protein Structure, Tertiary; Receptors, Adrenergic, beta-2; Sensitivity and Specificity; Spectrometry, Fluorescence

2006
Distinct regulation of beta 1- and beta 2-adrenergic receptors in Chinese hamster fibroblasts.
    Molecular pharmacology, 1992, Volume: 41, Issue:3

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Alprenolol; Animals; Betaxolol; Binding, Competitive; Cells, Cultured; Cricetinae; Cricetulus; DNA; Down-Regulation; Epinephrine; Fibroblasts; Iodocyanopindolol; Isoproterenol; Norepinephrine; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Transfection

1992
The effects of beta-adrenoreceptor antagonists on the force responses of the electrically driven rat right ventricle strip to isoprenaline.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:4

    Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Electric Stimulation; Heart; In Vitro Techniques; Isoproterenol; Male; Metoprolol; Myocardial Contraction; Pindolol; Propanolamines; Rats; Rats, Inbred Strains

1989
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
    European journal of pharmacology, 1989, Aug-29, Volume: 167, Issue:3

    Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta

1989
The beta 1- and beta 2-adrenoceptor stimulatory effects of alprenolol, oxprenolol and pindolol: a study in the isolated right atrium and uterus of the rat.
    British journal of pharmacology, 1986, Volume: 87, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Female; Heart; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Oxprenolol; Pindolol; Practolol; Propanolamines; Rats; Rats, Inbred Strains; Uterus

1986
Certain beta-blockers can decrease beta-adrenergic receptor number: II. Down-regulation of receptor number by alprenolol and propranolol in cultured lymphoma and muscle cells.
    Circulation research, 1988, Volume: 63, Issue:2

    Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Cell Line; Cyclic AMP; Humans; Lymphoma; Muscles; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Tumor Cells, Cultured

1988
Labeling in vivo of beta adrenergic receptors in the central nervous system of the rat after administration of [125I] iodopindolol.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:1

    Topics: Alprenolol; Animals; Betaxolol; Binding, Competitive; Brain Stem; Central Nervous System; Cerebellum; Cerebral Cortex; Clenbuterol; Isotope Labeling; Male; Mathematics; Pindolol; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Spinal Cord; Tissue Distribution

1985
Characterization of putative beta-adrenoceptors in the myometrium of the pregnant ewe: correlation between the binding of [3H] dihydroalprenolol and the inhibition of myometrial contractility in vitro.
    Biology of reproduction, 1984, Volume: 30, Issue:3

    Topics: Adrenergic beta-Agonists; Albuterol; Alprenolol; Animals; Atenolol; Dihydroalprenolol; Dose-Response Relationship, Drug; Female; Myometrium; Pregnancy; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Sheep; Uterine Contraction

1984
Physiological effects of inverse agonists in transgenic mice with myocardial overexpression of the beta 2-adrenoceptor.
    Nature, 1995, Mar-16, Volume: 374, Issue:6519

    Topics: Adrenergic beta-Agonists; Alprenolol; Animals; Cyclohexane Monoterpenes; GTP-Binding Proteins; Heart; Mice; Mice, Transgenic; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1995
Chronic infusion of beta-adrenoceptor antagonist and inverse agonists decreases elevated protein kinase A activity in transgenic mice with cardiac-specific overexpression of human beta 2-adrenoceptor.
    Journal of cardiovascular pharmacology, 2002, Volume: 40, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Carbazoles; Carvedilol; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Heart Atria; Heart Ventricles; Humans; Infusion Pumps, Implantable; Mice; Mice, Transgenic; Myocardium; Propanolamines; Receptors, Adrenergic, beta-2

2002
Effects of different beta adrenoceptor ligands in mice with permanent occlusion of the left anterior descending coronary artery.
    British journal of pharmacology, 2003, Volume: 138, Issue:8

    Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Carbazoles; Carvedilol; Coronary Disease; Coronary Vessels; Ligands; Male; Mice; Mice, Inbred C57BL; Propanolamines; Receptors, Adrenergic, beta

2003
Beta2-adrenergic receptor antagonist accelerates skin barrier recovery and reduces epidermal hyperplasia induced by barrier disruption.
    The Journal of investigative dermatology, 2003, Volume: 121, Issue:1

    Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Biological Transport; Calcium; Calcium Channel Blockers; Calcium Channels; Clenbuterol; Epidermis; Humidity; Hyperplasia; Male; Mice; Mice, Hairless; Nifedipine; Procaterol; Propanolamines; Verapamil

2003
Plasmon-waveguide resonance studies of ligand binding to the human beta 2-adrenergic receptor.
    Biochemistry, 2004, Mar-23, Volume: 43, Issue:11

    Topics: Adrenergic Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Anisotropy; Epinephrine; Humans; Isoproterenol; Kinetics; Ligands; Lipid Bilayers; Phosphatidylcholines; Propanolamines; Protein Binding; Proteolipids; Receptors, Adrenergic, beta-2; Spectrum Analysis; Surface Plasmon Resonance

2004
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction

2004
Computational study on the different ligands induced conformation change of β2 adrenergic receptor-Gs protein complex.
    PloS one, 2013, Volume: 8, Issue:7

    Topics: Alprenolol; Benzoxazines; Binding Sites; Computational Biology; GTP-Binding Protein alpha Subunits, Gs; GTP-Binding Protein beta Subunits; Humans; Hydrogen Bonding; Ligands; Models, Molecular; Multiprotein Complexes; Propanolamines; Protein Conformation; Receptors, Adrenergic, beta-2; Thermodynamics

2013