alprenolol has been researched along with 1-(2-allylphenoxy)-3-((8-bromoacetylamino-4-menthane-1-yl)amino)-1-propanol in 38 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 21 (55.26) | 18.7374 |
| 1990's | 15 (39.47) | 18.2507 |
| 2000's | 1 (2.63) | 29.6817 |
| 2010's | 1 (2.63) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Lü, ZL; Xia, ZQ; Yi, NY | 1 |
| Eglen, RM; Montgomery, WW; Whiting, RL | 1 |
| Insel, PA; Jasper, JR; Michel, MC | 1 |
| Adham, N; Blue, DR; Bond, RA; Clarke, DE; Delmendo, R; Eglen, RM; Michel, AD; Whiting, RL | 1 |
| Doggrell, SA | 3 |
| Lichtenstein, LM; Peachell, PT; Undem, BJ | 1 |
| Malta, E; Ng, NL | 1 |
| Box, RJ | 1 |
| Black, JW; Gerskowitch, VP; Leff, P; Shankley, NP | 1 |
| Kusiak, JW; Liptak, A; Pitha, J | 1 |
| Insel, PA; Mahan, LC | 2 |
| Abel, PW; May, JM; Minneman, KP | 1 |
| Baker, SP; Muther, TF; Nelson, CA; Pitha, J | 1 |
| Baker, SP; Pitha, J; Raizada, MK; Sumners, C | 1 |
| Baker, SP; Kalberg, CJ; Pitha, J; Standifer, KM; Sumners, C | 1 |
| Dickinson, KE; Inkpen, PM; Rudd, RM; Sever, PS; Winter, RJ | 1 |
| Insel, PA; Jasper, JR; Motulsky, HJ | 1 |
| Ballard, PL; Gonzales, LW; McDonald, JV; Pitha, J; Roberts, JM | 1 |
| Box, RJ; Staehelin, M | 1 |
| Caron, MG; Lefkowitz, RJ; Nasrin, N; Pitha, J; Zjawiony, J | 1 |
| Baker, SP; Dax, EM; Hughes, BA; Kusiak, JW; Pitha, J | 1 |
| Augustine, PC; Kuenzel, WJ; Kusiak, JW; Pitha, J | 1 |
| Zoler, ML | 1 |
| Baum, BJ; Hand, AR; Kousvelari, EE; Kusiak, JW; Pitha, J | 1 |
| Kim, GD; MacEwan, DJ; Milligan, G | 1 |
| Doggrell, SA; Surman, AJ | 2 |
| Kim, GD; Milligan, G | 1 |
| Kurose, H; Nagao, T; Sato, Y | 1 |
| Doggrell, SA; Henderson, CJ; Mistry, DN | 1 |
| Barnett, CW; Doggrell, SA; Petcu, EB | 1 |
| Chong, LK; Drury, DE; Ghahramani, P; Peachell, PT | 1 |
| Lee, JR; Tenner, TE; Zhang, X | 1 |
| Chen, YY; Doggrell, SA | 1 |
| Huang, Z; Li, J; Liao, YH; Qiang, YG; Zhang, XP | 1 |
38 other study(ies) available for alprenolol and 1-(2-allylphenoxy)-3-((8-bromoacetylamino-4-menthane-1-yl)amino)-1-propanol
| Article | Year |
|---|---|
[Synthesis and identification of bromoacetylalprenololmenthane (BAlpM)].
Topics: Adrenergic beta-Antagonists; Alprenolol | 1991 |
Desensitization and functional antagonism by beta-adrenoceptor and muscarinic receptor agonists, respectively: a comparison with receptor alkylation for calculation of apparent agonist affinity.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Alkylation; Alprenolol; Animals; Dose-Response Relationship, Drug; Heart Atria; Male; Prenalterol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Muscarinic | 1991 |
Partial agonistic activity of two irreversible beta-adrenergic receptor ligands, bromoacetylated derivatives of alprenolol and pindolol.
Topics: Adrenergic beta-Agonists; Alprenolol; Cell Line; Colforsin; Cyclic AMP; Cyclohexane Monoterpenes; Dose-Response Relationship, Drug; Humans; Pindolol | 1991 |
Antagonist characterization of atypical beta adrenoceptors in guinea pig ileum: blockade by alprenolol and dihydroalprenolol.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Dihydroalprenolol; Drug Interactions; Guinea Pigs; Ileum; In Vitro Techniques; Isoproterenol; Male; Muscle, Smooth; Propranolol; Receptors, Adrenergic, beta | 1990 |
The effects of (+/-)-, (+)- and (-)-celiprolol and bromoacetylalprenololmentane at the beta-adrenoceptors of rat isolated cardiovascular preparations.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Celiprolol; Electric Stimulation; Ethanolamines; Heart; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Myocardial Contraction; Procaterol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sotalol | 1990 |
Effects of bromoacetylalprenololmenthane (BAAM), an irreversible beta-adrenoceptor antagonist, on the rat isolated left atria and portal vein.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Electric Stimulation; Heart; In Vitro Techniques; Isoproterenol; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Portal Vein; Rats; Rats, Inbred Strains | 1990 |
Isoproterenol-induced inhibition of immunoglobulin E-mediated release of histamine and arachidonic acid metabolites from the human lung mast cell.
Topics: Alprenolol; Arachidonic Acid; Arachidonic Acids; Calcimycin; Cyclic AMP; Histamine Release; Humans; Immunoglobulin E; Isoproterenol; Lung; Mast Cells; Prostaglandin D2; SRS-A | 1988 |
Organ-bath studies using the irreversible beta-adrenoreceptor antagonist bromoacetylalprenololmenthane (BAAM).
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Female; Guinea Pigs; Heart; Heart Rate; Ileum; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Rats; Refractory Period, Electrophysiological; Uterine Contraction | 1989 |
The effects of beta-adrenoreceptor antagonists on the force responses of the electrically driven rat right ventricle strip to isoprenaline.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Electric Stimulation; Heart; In Vitro Techniques; Isoproterenol; Male; Metoprolol; Myocardial Contraction; Pindolol; Propanolamines; Rats; Rats, Inbred Strains | 1989 |
Quantitative comparison of bromoacetylated derivatives of alprenolol and pindolol on beta-adrenergic receptor binding and mobility in S49 cells.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Cell Membrane; Cyclohexane Monoterpenes; Lipoproteins, LDL; Mice; Pindolol; Receptors, Adrenergic, beta; Transferrin; Tumor Cells, Cultured | 1989 |
Pharmacological analysis of beta-adrenoceptor-mediated agonism in the guinea-pig, isolated, right atrium.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Cholera Toxin; Guinea Pigs; Heart; Heart Atria; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Models, Biological; Receptors, Adrenergic, beta | 1985 |
Alkylating beta-blockers: activity of isomeric bromoacetyl alprenolol menthanes.
Topics: Adrenergic beta-Antagonists; Affinity Labels; Alprenolol; Animals; Cell Membrane; Dihydroalprenolol; Isomerism; Lung; Magnetic Resonance Spectroscopy; Molecular Conformation; Myocardium; Rats; Receptors, Adrenergic, beta; Structure-Activity Relationship | 1985 |
Expression of beta-adrenergic receptors in synchronous and asynchronous S49 lymphoma cells. I. Receptor metabolism after irreversible blockade of receptors and in cells traversing the cell division cycle.
Topics: Adrenergic beta-Antagonists; Alprenolol; Cell Cycle; Cell Division; Cell Line; Centrifugation; Humans; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Lymphoma; Pindolol; Receptors, Adrenergic, beta | 1986 |
Binding of agonists and antagonists to beta-adrenoceptors in rat vas deferens: relationship to functional response.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Animals; Isoproterenol; Male; Pindolol; Rats; Receptors, Adrenergic, beta; Vas Deferens | 1985 |
Differential recovery of beta adrenoreceptor antagonist and agonist high affinity binding sites in the guinea-pig lung after irreversible blockade.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Binding Sites; Dihydroalprenolol; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Lung; Receptors, Adrenergic, beta; Tritium | 1986 |
Characteristics of the beta-adrenoreceptor from neuronal and glial cells in primary cultures of rat brain.
Topics: Adrenergic beta-Agonists; Alprenolol; Animals; Animals, Newborn; Binding, Competitive; Brain; Cell Membrane; Cells, Cultured; Cyclic AMP; Cycloheximide; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Kinetics; Neuroglia; Neurons; Pindolol; Rats; Receptors, Adrenergic, beta | 1986 |
Irreversible binding and recovery of the norepinephrine uptake system using an alkylating derivative of norepinephrine.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Brain; Cells, Cultured; Cerebral Cortex; Corpus Striatum; Cycloheximide; Dopamine; Leucine; Male; Neurons; Norepinephrine; Rats; Rats, Inbred Strains; Synaptosomes | 1988 |
De novo cardiac beta adrenoceptor synthesis in adult rats under normoxic and hypoxic conditions.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Hypoxia; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1988 |
Characterization of a bromoacetylated derivative of pindolol as a high affinity, irreversible beta adrenergic antagonist in cultured cells.
Topics: Adrenergic beta-Antagonists; Alprenolol; Alprostadil; Animals; Cyclic AMP; Cyclohexane Monoterpenes; Dose-Response Relationship, Drug; Iodocyanopindolol; Membrane Proteins; Mice; Pindolol; Receptors, Adrenergic, beta; Tumor Cells, Cultured | 1988 |
Expression of beta-adrenergic receptors in synchronous and asynchronous S49 lymphoma cells. II. Relationship between receptor number and response.
Topics: Adenylyl Cyclases; Alprenolol; Cell Cycle; Cell Line; Colforsin; Cyclic AMP; GTP-Binding Proteins; Guanosine Triphosphate; Isoproterenol; Lymphoma; Receptors, Adrenergic, beta | 1986 |
Lung beta-adrenoreceptor blockade affects perinatal surfactant release but not lung water.
Topics: Alprenolol; Animals; Animals, Newborn; Body Water; Catecholamines; Cyclic AMP; Embryonic and Fetal Development; Female; Fetus; Lung; Phospholipids; Pregnancy; Pulmonary Surfactants; Rabbits; Receptors, Adrenergic, beta | 1986 |
Bromoacetylalprenololmenthane binding to beta-receptors modulates the rate of hormone-induced internalization but not desensitization in S49 cells.
Topics: Alprenolol; Cell Line; Cell Membrane; Cyclic AMP; Isoproterenol; Kinetics; Lymphoma; Propanolamines; Receptors, Adrenergic, beta | 1987 |
Potent beta-adrenergic antagonist possessing chemically reactive group.
Topics: Adrenergic beta-Agonists; Alprenolol; Animals; Binding, Competitive; Cyclohexane Monoterpenes; Dihydroalprenolol; Erythrocyte Membrane; Kinetics; Ranidae; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Regeneration of beta-adrenergic receptors in senescent rats: a study using an irreversible binding antagonist.
Topics: Adrenergic beta-Antagonists; Aging; Alprenolol; Animals; Brain; Cyclohexane Monoterpenes; Dihydroalprenolol; Kinetics; Lung; Myocardium; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Effect of a beta-adrenergic antagonist on blood pressure, heart rate and beta-adrenoceptors in turkey poults.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Blood Pressure; Brain Chemistry; Cyclohexane Monoterpenes; Heart Rate; Myocardium; Receptors, Adrenergic, beta; Turkeys | 1983 |
BAAM: a better beta-blocker--and more?
Topics: Adrenergic beta-Antagonists; Aging; Alprenolol; Animals; Cyclohexane Monoterpenes; Drug Evaluation; Humans; Hypertension; Rats | 1984 |
Bromoacetylalprenololmenthane: a potent irreversible antagonist of beta adrenergic elicited protein exocytosis in rat parotid cells.
Topics: Adrenergic beta-Antagonists; Alprenolol; Amylases; Animals; Cyclohexane Monoterpenes; Depression, Chemical; Dihydroalprenolol; Exocytosis; Isoproterenol; Male; Microscopy, Electron; Parotid Gland; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1983 |
Analysis of the role of receptor number in defining the intrinsic activity and potency of partial agonists in neuroblastoma x glioma hybrid NG108-15 cells transfected to express differing levels of the human beta 2-adrenoceptor.
Topics: Adenylyl Cyclases; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Albuterol; Alprenolol; Dobutamine; Ephedrine; Epinephrine; Humans; Hybrid Cells; Isoproterenol; Receptors, Adrenergic, beta-2; Transfection; Tumor Cells, Cultured | 1995 |
Alprenolol and bromoacetylalprenololmenthane are competitive slowly reversible antagonists at the beta 1-adrenoceptors of rat left atria.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Atrial Function; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Rats; Rats, Wistar | 1993 |
Receptor availability defines the extent of agonist-mediated G-protein down-regulation in neuroblastoma x glioma hybrid cells transfected to express the beta 2-adrenoceptor.
Topics: Adenylyl Cyclases; Adrenergic beta-2 Receptor Antagonists; Alprenolol; Down-Regulation; Gene Expression; Glioma; GTP-Binding Proteins; Humans; Hybrid Cells; Isoproterenol; Neuroblastoma; Receptors, Adrenergic, beta-2; Tumor Cells, Cultured | 1994 |
Loss of maximum attenuation and receptor reserve for isoprenaline at the beta 2-adrenoceptors of the portal veins of hypertensive rats.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Hypertension; Hypertrophy; Isoproterenol; Male; Nitroprusside; Portal Vein; Pyrazines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Vasodilator Agents; Verapamil | 1995 |
Relationship between desensitization and downregulation of beta-adrenoceptors in cardiac tissues after prolonged in vivo infusion of T-0509, a beta 1-adrenoceptor agonist.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Analysis of Variance; Animals; Binding, Competitive; Down-Regulation; Drug Interactions; Ethanolamines; GTP-Binding Proteins; Heart; Heart Ventricles; Injections, Subcutaneous; Iodocyanopindolol; Isoproterenol; Male; Myocardium; Pindolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-2 | 1997 |
The effects of bromoacetylalprenololmenthane on the responses to isoprenaline of the left ventricle from normo-, prehyper- and hypertensive rats.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Blood Pressure; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Female; Heart; Heart Ventricles; Hypertension; Isoproterenol; Male; Myocardial Contraction; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Ventricular Function, Left | 1997 |
Affinity constants and beta-adrenoceptor reserves for isoprenaline on cardiac tissue from normotensive and hypertensive rats.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Female; Heart; Heart Atria; Heart Ventricles; Hypertension; Hypertrophy, Left Ventricular; Isoproterenol; Male; Myocardial Contraction; Myocardium; Papillary Muscles; Pyrazines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta | 1998 |
Influence of receptor reserve on beta-adrenoceptor-mediated responses in human lung mast cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Antibodies, Anti-Idiotypic; Histamine Release; Humans; Immunoglobulin E; In Vitro Techniques; Isoproterenol; Lung; Mast Cells; Receptors, Adrenergic, beta | 1998 |
Evidence for spare beta-adrenoceptors in the rabbit heart.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Central Nervous System Stimulants; Ethanol; Heart; Heart Ventricles; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Myocardial Contraction; Rabbits; Radioligand Assay; Receptors, Adrenergic, beta | 1999 |
Responsiveness, affinity constants and beta-adrenoceptor reserves for isoprenaline on aortae from normo-, pre- and hypertensive rats.
Topics: Adrenergic beta-Agonists; Algorithms; Alprenolol; Animals; Aorta, Thoracic; Binding, Competitive; Blood Pressure; Colforsin; Dose-Response Relationship, Drug; Female; Hypertension; In Vitro Techniques; Isoproterenol; Male; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Vasoconstriction | 2002 |
Modulation of β-adrenergic receptor in rat lung after gamma irradiation.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Female; Gamma Rays; Kinetics; Lung; Male; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 2014 |