alprazolam and midazolam

alprazolam has been researched along with midazolam in 47 studies

Research

Studies (47)

TimeframeStudies, this research(%)All Research%
pre-19902 (4.26)18.7374
1990's4 (8.51)18.2507
2000's18 (38.30)29.6817
2010's17 (36.17)24.3611
2020's6 (12.77)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Abraham, MH; Acree, WE; Ibrahim, A1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Alelyunas, YW; Bui, K; Empfield, JR; McCarthy, D; Pelosi-Kilby, L; Shen, C; Spreen, RC1
Ahlin, G; Bergström, F; Bredberg, U; Fridén, M; Hammarlund-Udenaes, M; Rehngren, M; Wan, H1
Bracher, F; Fedorov, O; Filippakopoulos, P; Keller, M; Knapp, S; Morgenstern, O; Picaud, S; Wrobel, M1
Artursson, P; Mateus, A; Matsson, P1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Loeffler, PM1
Anderson, BJ; Brown, TC; Exarchos, H; Lee, K1
Jones, CE; Martinez, LA; Merritt, GJ; Wians, FH1
DiMicco, JA1
Adnet, P; Boittiaux, P; Forget, AP; Loeb, P; Mille, FX1
Balian, JD; Flockhart, DA; Yuan, R1
Greenblatt, DJ; Harmatz, JS; Poku, JW; Shader, RI; von Moltke, LL; Warrington, JS1
Cantrell, VE; Eckstein, J; Hall, SD; Hamman, MA; Jones, DR; Ring, BJ; Ruterbories, K; Williams, JA; Wrighton, SA1
Alegret, C; Cammu, G; De Witte, JL; Sessler, DI1
Kanbori, M; Kato, M; Kumaki, Y; Nakahara, Y; Toyo'oka, T1
Kozierowski, T; Małysz, A; Ruciński, M; Rzymski, S; Wołowicka, L1
Masica, AL; Mayo, G; Wilkinson, GR1
Benet, LZ1
Dickson, SJ; Irving, RC1
Galetin, A; Hallifax, D; Houston, JB1
Mandrioli, R; Mercolini, L; Raggi, MA1
Hanioka, N; Kuze, J; Morisaki, K; Mutoh, T; Nakura, H; Narimatsu, S; Takenaka, T1
Gunn, J; Kriger, S; Terrell, AR1
Castell, JV; Donato, MT; Gomez-Lechón, MJ; Hallifax, D; Houston, JB; Lahoz, A; Picazo, L1
Barter, ZE; Cubitt, HE; Howgate, EM; Rostami-Hodjegan, A; Yeo, KR1
Christianson, CD; Johnson, CJ; Laine, DF; Needham, SR; Sheaff, CN; Zimmer, JS1
Houjo, T; Ishigai, M; Kato, M; Ogawa, K1
Ishigai, M; Kato, M; Mitsui, T; Miyake, T; Nagao, S; Nemoto, T; Ogawa, K; Yamada, H1
Boulenc, X; Donazzolo, Y; Hermabessière, S; Martin, V; Nicolas, O; Ollier, C; Zobouyan, I1
Inoue, T; Ishii, S; Nakanishi, K; Sasaki, E; Uehara, S; Uno, Y; Yamazaki, H1
Dang, H; Kaufman, DL; Middleton, B; Tian, J1
Adiwidjaja, J; Boddy, AV; McLachlan, AJ1
Hasegawa, M; Tahara, H; Watanabe, M1
Chan, TS; Raymond, K; Scaringella, YS; Taub, ME1
Madsen, BK; Møller, AM; Rosenberg, J; Zetner, D1
Araújo, JO; Bergamaschi, CC; de Andrade, NK; Guimarães, CC; Lopes, LC; Motta, RHL; Ramacciato, JC1
Cook, JM; Duke, AN; Knutson, DE; Platt, DM; Rowlett, JK; Sharmin, D; Tiruveedhula, VVNPB1
Gui, L; Hu, Y; Jia, W; Lan, K; Liu, C; Miao, J; Wang, C; Wei, W; Wu, Q; Zeng, W1
Morikuni, S; Murayama, N; Noda, Y; Uno, Y; Yamazaki, H1

Reviews

6 review(s) available for alprazolam and midazolam

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Oral benzodiazepines and conscious sedation: a review.
    Journal of oral and maxillofacial surgery : official journal of the American Association of Oral and Maxillofacial Surgeons, 1992, Volume: 50, Issue:9

    Topics: Administration, Oral; Alprazolam; Ambulatory Surgical Procedures; Anti-Anxiety Agents; Conscious Sedation; Diazepam; Flurazepam; Humans; Lorazepam; Midazolam; Oxazepam; Premedication; Receptors, GABA-A; Temazepam; Triazolam

1992
Pharmacokinetic and pharmacodynamic consequences of metabolism-based drug interactions with alprazolam, midazolam, and triazolam.
    Journal of clinical pharmacology, 1999, Volume: 39, Issue:11

    Topics: Alprazolam; Anti-Anxiety Agents; Data Collection; Drug Interactions; Enzyme Induction; Enzyme Inhibitors; Humans; Itraconazole; Ketoconazole; Midazolam; Triazolam

1999
Benzodiazepine metabolism: an analytical perspective.
    Current drug metabolism, 2008, Volume: 9, Issue:8

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Azepines; Benzodiazepines; Bromazepam; Chromatography, High Pressure Liquid; Diazepam; Humans; Lorazepam; Mass Spectrometry; Midazolam; Triazolam

2008
Melatonin for preoperative and postoperative anxiety in adults.
    The Cochrane database of systematic reviews, 2020, 12-08, Volume: 12

    Topics: Adult; Aged; Aged, 80 and over; Alprazolam; Anti-Anxiety Agents; Anxiety; Bias; Clonidine; Drug Administration Schedule; Humans; Melatonin; Midazolam; Middle Aged; Oxazepam; Postoperative Care; Postoperative Complications; Preoperative Care; Publication Bias; Randomized Controlled Trials as Topic; Surgical Procedures, Operative

2020
Effectiveness and safety of oral sedation in adult patients undergoing dental procedures: a systematic review.
    BMJ open, 2021, 01-25, Volume: 11, Issue:1

    Topics: Adult; Alprazolam; Anesthesia; Benzodiazepines; Diazepam; Humans; Midazolam

2021

Trials

5 trial(s) available for alprazolam and midazolam

ArticleYear
Oral premedication in children: a comparison of chloral hydrate, diazepam, alprazolam, midazolam and placebo for day surgery.
    Anaesthesia and intensive care, 1990, Volume: 18, Issue:2

    Topics: Administration, Oral; Alprazolam; Ambulatory Surgical Procedures; Anesthesia Recovery Period; Attitude; Child Behavior; Child, Preschool; Chloral Hydrate; Diazepam; Double-Blind Method; Female; Humans; Infant; Male; Midazolam; Placebos; Preanesthetic Medication; Random Allocation; Time Factors

1990
Preoperative alprazolam reduces anxiety in ambulatory surgery patients: a comparison with oral midazolam.
    Anesthesia and analgesia, 2002, Volume: 95, Issue:6

    Topics: Administration, Oral; Adult; Alprazolam; Ambulatory Surgical Procedures; Anti-Anxiety Agents; Anxiety; Double-Blind Method; Humans; Midazolam; Premedication; Psychomotor Performance

2002
[Perioperative sedation and analgesia for complications from arthroscopy and arthrotomy of the knee joint].
    Folia medica Cracoviensia, 2001, Volume: 42, Issue:4

    Topics: Administration, Oral; Alprazolam; Analgesia; Arthroscopy; Bupivacaine; Conscious Sedation; Epinephrine; Female; Fentanyl; Humans; Knee Joint; Lidocaine; Male; Midazolam; Pain Measurement; Pain, Postoperative; Patient Satisfaction; Preanesthetic Medication; Premedication

2001
In vivo comparisons of constitutive cytochrome P450 3A activity assessed by alprazolam, triazolam, and midazolam.
    Clinical pharmacology and therapeutics, 2004, Volume: 76, Issue:4

    Topics: Administration, Oral; Adult; Alprazolam; Anti-Anxiety Agents; Aryl Hydrocarbon Hydroxylases; Benzodiazepines; Biological Availability; Cytochrome P-450 CYP3A; Female; Humans; Male; Midazolam; Oxidoreductases, N-Demethylating; Triazolam

2004
CYP3A4-based drug-drug interaction: CYP3A4 substrates' pharmacokinetic properties and ketoconazole dose regimen effect.
    European journal of drug metabolism and pharmacokinetics, 2016, Volume: 41, Issue:1

    Topics: Adolescent; Adult; Alprazolam; Cross-Over Studies; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Humans; Ketoconazole; Male; Midazolam; Substrate Specificity; Young Adult

2016

Other Studies

36 other study(ies) available for alprazolam and midazolam

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Air to lung partition coefficients for volatile organic compounds and blood to lung partition coefficients for volatile organic compounds and drugs.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:3

    Topics: Air; Animals; Humans; Lung; Organic Chemicals; Probability; Rats; Tissue Distribution; Volatilization

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Central Nervous System Agents; Drug Evaluation, Preclinical; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Solubility

2010
Measurement of unbound drug exposure in brain: modeling of pH partitioning explains diverging results between the brain slice and brain homogenate methods.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:3

    Topics: Animals; Biological Transport; Brain; Chemical Phenomena; Dialysis; Hydrogen-Ion Concentration; In Vitro Techniques; Lysosomes; Male; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Tissue Distribution

2011
Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family.
    Bioorganic & medicinal chemistry, 2012, Mar-15, Volume: 20, Issue:6

    Topics: Alprazolam; Benzazepines; Benzodiazepines; Cell Cycle Proteins; GABA Modulators; Humans; Midazolam; Models, Molecular; Nuclear Proteins; Protein Interaction Maps; Protein Structure, Tertiary; Transcription Factors

2012
A high-throughput cell-based method to predict the unbound drug fraction in the brain.
    Journal of medicinal chemistry, 2014, Apr-10, Volume: 57, Issue:7

    Topics: Animals; Brain; Dialysis; HEK293 Cells; High-Throughput Screening Assays; Humans; Pharmaceutical Preparations; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization

2014
Benzodiazepines identified by capillary gas chromatography-mass spectrometry, with specific ion screening used to detect benzophenone derivatives.
    Clinical chemistry, 1989, Volume: 35, Issue:7

    Topics: Alprazolam; Benzodiazepines; Benzophenones; Forensic Medicine; Gas Chromatography-Mass Spectrometry; Humans; Hydrolysis; Immunoenzyme Techniques; Midazolam; Triazolam

1989
Evidence for control of cardiac vagal tone by benzodiazepine receptors.
    Neuropharmacology, 1987, Volume: 26, Issue:6

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Atropine; Chlordiazepoxide; Flumazenil; Heart; Heart Rate; Male; Midazolam; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vagus Nerve

1987
[Benzodiazepine withdrawal presenting as pseudo-surgical abdominal pain].
    Annales francaises d'anesthesie et de reanimation, 1997, Volume: 16, Issue:5

    Topics: Abdomen, Acute; Adult; Alprazolam; Anti-Anxiety Agents; Bromazepam; Diagnosis, Differential; Headache; Humans; Hydroxyzine; Male; Midazolam; Self Administration; Substance Withdrawal Syndrome; Substance-Related Disorders; Truth Disclosure; Vomiting

1997
Effects of age on in vitro midazolam biotransformation in male CD-1 mouse liver microsomes.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 292, Issue:3

    Topics: Age Factors; Alprazolam; Animals; Anti-Anxiety Agents; Aryl Hydrocarbon Hydroxylases; Biotransformation; Blotting, Western; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; In Vitro Techniques; Ketoconazole; Male; Mice; Microsomes, Liver; Midazolam; Oxidoreductases, N-Demethylating

2000
Comparative metabolic capabilities of CYP3A4, CYP3A5, and CYP3A7.
    Drug metabolism and disposition: the biological fate of chemicals, 2002, Volume: 30, Issue:8

    Topics: Alprazolam; Aryl Hydrocarbon Hydroxylases; Biotransformation; Clarithromycin; Coumarins; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Cytochromes b5; Diltiazem; Estradiol; Humans; In Vitro Techniques; Kinetics; Microsomes, Liver; Midazolam; Nifedipine; Tamoxifen; Testosterone; Triazolam

2002
Determination of hypnotic benzodiazepines (alprazolam, estazolam, and midazolam) and their metabolites in rat hair and plasma by reversed-phase liquid-chromatography with electrospray ionization mass spectrometry.
    Journal of pharmaceutical and biomedical analysis, 2003, Jan-15, Volume: 30, Issue:6

    Topics: Alprazolam; Animals; Benzodiazepines; Chromatography, High Pressure Liquid; Estazolam; Hair; Male; Midazolam; Rats; Spectrometry, Mass, Electrospray Ionization

2003
There are no useful CYP3A probes that quantitatively predict the in vivo kinetics of other CYP3A substrates and no expectation that one will be found.
    Molecular interventions, 2005, Volume: 5, Issue:2

    Topics: Alprazolam; Benzodiazepines; Biopharmaceutics; Chemistry, Pharmaceutical; Cytochrome P-450 CYP3A; Drug Design; Humans; Kinetics; Midazolam; Molecular Probes; Protein Binding; Solubility; Triazolam

2005
The detection of sedatives in hair and nail samples using tandem LC-MS-MS.
    Forensic science international, 2007, Feb-14, Volume: 166, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Alprazolam; Azabicyclo Compounds; Benzodiazepines; Chromatography, Liquid; Clobazam; Clonazepam; Diazepam; Female; Forensic Pathology; Hair; Humans; Hypnotics and Sedatives; Male; Mass Spectrometry; Midazolam; Middle Aged; Nails; Oxazepam; Piperazines; Predictive Value of Tests; Rape; Temazepam; Triazolam

2007
Prediction of metabolic clearance using fresh human hepatocytes: comparison with cryopreserved hepatocytes and hepatic microsomes for five benzodiazepines.
    Xenobiotica; the fate of foreign compounds in biological systems, 2008, Volume: 38, Issue:4

    Topics: Alprazolam; Benzodiazepines; Cell Survival; Cells, Cultured; Cryopreservation; Cytochrome P-450 CYP3A; Diazepam; Flunitrazepam; Hepatocytes; Humans; Metabolic Clearance Rate; Microsomes, Liver; Midazolam; Substrate Specificity; Triazolam

2008
Separate evaluation of intestinal and hepatic metabolism of three benzodiazepines in rats with cannulated portal and jugular veins: comparison with the profile in non-cannulated mice.
    Xenobiotica; the fate of foreign compounds in biological systems, 2009, Volume: 39, Issue:11

    Topics: Administration, Oral; Alprazolam; Animals; Benzodiazepines; Biological Availability; Catheterization; Intestinal Mucosa; Jugular Veins; Liver; Male; Mice; Mice, Inbred BALB C; Midazolam; Portal Vein; Rats; Rats, Sprague-Dawley; Triazolam

2009
Simultaneous determination and quantification of 12 benzodiazepines in serum or whole blood using UPLC/MS/MS.
    Methods in molecular biology (Clifton, N.J.), 2010, Volume: 603

    Topics: Alprazolam; Benzodiazepines; Chlordiazepoxide; Chromatography, Liquid; Clonazepam; Flunitrazepam; Humans; Lorazepam; Midazolam; Nordazepam; Oxazepam; Reproducibility of Results; Tandem Mass Spectrometry

2010
Metabolite formation kinetics and intrinsic clearance of phenacetin, tolbutamide, alprazolam, and midazolam in adenoviral cytochrome P450-transfected HepG2 cells and comparison with hepatocytes and in vivo.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:9

    Topics: Adenoviridae; Alprazolam; Base Sequence; Cell Line; Cytochrome P-450 Enzyme System; DNA Primers; Hepatocytes; Humans; Midazolam; Phenacetin; Tolbutamide

2010
Sources of interindividual variability in IVIVE of clearance: an investigation into the prediction of benzodiazepine clearance using a mechanistic population-based pharmacokinetic model.
    Xenobiotica; the fate of foreign compounds in biological systems, 2011, Volume: 41, Issue:8

    Topics: Alprazolam; Benzodiazepines; Cytochrome P-450 CYP3A; Humans; Kinetics; Liver; Metabolic Clearance Rate; Midazolam; Triazolam

2011
Use of conventional bioanalytical devices to automate DBS extractions in liquid-handling dispensing tips.
    Bioanalysis, 2011, Volume: 3, Issue:20

    Topics: Alprazolam; Automation; Chromatography, High Pressure Liquid; Dried Blood Spot Testing; Humans; Midazolam; Tandem Mass Spectrometry

2011
A new approach to predicting human hepatic clearance of CYP3A4 substrates using monkey pharmacokinetic data.
    Xenobiotica; the fate of foreign compounds in biological systems, 2013, Volume: 43, Issue:5

    Topics: Alprazolam; Animals; Cytochrome P-450 CYP3A; Diltiazem; Humans; Liver; Macaca fascicularis; Midazolam; Tacrolimus

2013
A useful model capable of predicting the clearance of cytochrome 3A4 (CYP3A4) substrates in humans: validity of CYP3A4 transgenic mice lacking their own Cyp3a enzymes.
    Drug metabolism and disposition: the biological fate of chemicals, 2014, Volume: 42, Issue:9

    Topics: Alprazolam; Animals; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Felodipine; Humans; Male; Mice; Mice, Transgenic; Microsomes, Liver; Midazolam; Nifedipine; Nitrendipine; Quinidine

2014
Marmoset Cytochrome P450 3A4 Ortholog Expressed in Liver and Small-Intestine Tissues Efficiently Metabolizes Midazolam, Alprazolam, Nifedipine, and Testosterone.
    Drug metabolism and disposition: the biological fate of chemicals, 2017, Volume: 45, Issue:5

    Topics: Adolescent; Adult; Aged; Alprazolam; Animals; Callithrix; Cytochrome P-450 CYP3A; Female; Humans; Intestine, Small; Liver; Macaca fascicularis; Male; Microsomes; Midazolam; Middle Aged; Multigene Family; Nifedipine; Pharmaceutical Preparations; Phylogeny; Sequence Alignment; Sequence Homology, Amino Acid; Species Specificity; Testosterone; Young Adult

2017
Clinically applicable GABA receptor positive allosteric modulators promote ß-cell replication.
    Scientific reports, 2017, 03-23, Volume: 7, Issue:1

    Topics: Allosteric Regulation; Alprazolam; Animals; Benzodiazepines; Carrier Proteins; Cell Division; Cell Proliferation; Clonazepam; GABA Modulators; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Insulin-Secreting Cells; Islets of Langerhans; Mice; Midazolam; Rats; Receptors, GABA-A

2017
Physiologically Based Pharmacokinetic Modelling of Hyperforin to Predict Drug Interactions with St John's Wort.
    Clinical pharmacokinetics, 2019, Volume: 58, Issue:7

    Topics: Adult; Alprazolam; Antineoplastic Agents; Computer Simulation; Cytochrome P-450 CYP2C19; Cytochrome P-450 CYP2C9; Cytochrome P-450 CYP3A; Female; Herb-Drug Interactions; Humans; Hypericum; Imatinib Mesylate; Intestinal Mucosa; Liver; Male; Midazolam; Middle Aged; Models, Biological; Phloroglucinol; Terpenes

2019
A comparative study for detecting CYP3A induction by CYP3A probe drugs and endogenous markers in cynomolgus monkeys.
    Biopharmaceutics & drug disposition, 2019, Volume: 40, Issue:2

    Topics: Alprazolam; Animals; Area Under Curve; Biomarkers; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inducers; Dose-Response Relationship, Drug; Drug Interactions; Hydrocortisone; Hydroxycholesterols; Macaca fascicularis; Male; Midazolam; Rifampin; Triazolam

2019
Evaluation of Erythromycin as a Tool to Assess CYP3A Contribution of Low Clearance Compounds in a Long-Term Hepatocyte Culture.
    Drug metabolism and disposition: the biological fate of chemicals, 2020, Volume: 48, Issue:8

    Topics: Adult; Alprazolam; Cells, Cultured; Coculture Techniques; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inducers; Cytochrome P-450 CYP3A Inhibitors; Drug Evaluation, Preclinical; Erythromycin; Female; Glucuronosyltransferase; Hepatobiliary Elimination; Hepatocytes; Humans; Male; Midazolam; Middle Aged; Primary Cell Culture; Rifampin; Time Factors

2020
Tolerance and dependence following chronic alprazolam treatment in rhesus monkeys: Role of GABA
    Drug and alcohol dependence, 2021, 11-01, Volume: 228

    Topics: Alprazolam; Animals; Benzodiazepines; Drug Tolerance; Female; Macaca mulatta; Midazolam; Receptors, GABA-A; Substance Withdrawal Syndrome; Zolpidem

2021
Reevaluate In Vitro CYP3A Index Reactions of Benzodiazepines and Steroids between Humans and Dogs.
    Drug metabolism and disposition: the biological fate of chemicals, 2022, Volume: 50, Issue:6

    Topics: Alprazolam; Animals; Benzodiazepines; Cytochrome P-450 CYP3A; Deoxycholic Acid; Dogs; Humans; Hydroxylation; Kinetics; Microsomes, Liver; Midazolam; Protein Isoforms; Species Specificity; Steroids; Triazolam

2022
Liver microsomal cytochrome P450 3A-dependent drug oxidation activities in individual dogs.
    Xenobiotica; the fate of foreign compounds in biological systems, 2023, Volume: 53, Issue:3

    Topics: Alprazolam; Animals; Cytochrome P-450 CYP3A; Dogs; Estradiol; Hydroxylation; Liver; Microsomes, Liver; Midazolam; Nifedipine; Rats; RNA, Messenger

2023
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