alpidem has been researched along with pk 11195 in 9 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (11.11) | 18.7374 |
1990's | 3 (33.33) | 18.2507 |
2000's | 3 (33.33) | 29.6817 |
2010's | 1 (11.11) | 24.3611 |
2020's | 1 (11.11) | 2.80 |
Authors | Studies |
---|---|
Anzini, M; Basile, AS; Bruni, G; Cappelli, A; Giorgi, G; Langer, T; Romeo, MR; Vomero, S | 1 |
Abignente, E; Chelli, B; Costa, B; Da Settimo, F; Greco, G; Martini, C; Novellino, E; Patrizi, MP; Primofiore, G; Simorini, F; Taliani, S | 1 |
Abignente, E; Chelli, B; Cosimelli, B; Da Settimo, F; Greco, G; Gremigni, V; La Motta, C; Martini, C; Novellino, E; Rossi, L; Sergianni, V; Simorini, F; Spinetti, F; Taliani, S | 1 |
Bellandi, M; Cosimelli, B; Costa, B; Da Pozzo, E; Da Settimo, F; Greco, G; La Motta, C; Marini, AM; Martini, C; Morelli, M; Novellino, E; Salerno, S; Simola, N; Simorini, F; Taliani, S | 1 |
Bendinelli, S; Castellano, S; Cosconati, S; Costa, B; Da Pozzo, E; Da Settimo, F; Greco, G; Martini, C; Milite, C; Novellino, E; Pugliesi, I; Rizzetto, E; Sbardella, G; Stefancich, G; Taliani, S | 1 |
Baglini, E; Barresi, E; Costa, B; Da Pozzo, E; Da Settimo, F; Martini, C; Robello, M; Salerno, S; Taliani, S | 1 |
De Luca, C; De Medici, D; Massotti, M | 1 |
Arbilla, S; Langer, SZ | 1 |
Auta, J; Costa, E; Guidotti, A; Kozikowski, A; Ma, D; Romeo, E | 1 |
1 review(s) available for alpidem and pk 11195
Article | Year |
---|---|
An update into the medicinal chemistry of translocator protein (TSPO) ligands.
Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Anticonvulsants; Apoptosis; Benzimidazoles; Benzodiazepines; Cell Proliferation; Diazepam; Humans; Imidazoles; Membrane Potential, Mitochondrial; Mitochondria; Mitochondrial ADP, ATP Translocases; Mitochondrial Membranes; Mitochondrial Permeability Transition Pore; Oxidative Stress; Protein Binding; Pyridines; Quinolines; Receptors, GABA; Structure-Activity Relationship; Voltage-Dependent Anion Channels | 2021 |
8 other study(ies) available for alpidem and pk 11195
Article | Year |
---|---|
Molecular basis of peripheral vs central benzodiazepine receptor selectivity in a new class of peripheral benzodiazepine receptor ligands related to alpidem.
Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Cerebral Cortex; Drug Design; Flunitrazepam; Imidazoles; Isoquinolines; Models, Molecular; Protein Conformation; Pyridines; Rats; Receptors, GABA-A; Structure-Activity Relationship | 1996 |
N,N-dialkyl-2-phenylindol-3-ylglyoxylamides. A new class of potent and selective ligands at the peripheral benzodiazepine receptor.
Topics: Animals; Binding, Competitive; Brain; Cell Line, Tumor; Glyoxylates; In Vitro Techniques; Indoles; Ligands; Radioligand Assay; Rats; Receptors, GABA-A; Structure-Activity Relationship | 2004 |
New fluorescent 2-phenylindolglyoxylamide derivatives as probes targeting the peripheral-type benzodiazepine receptor: design, synthesis, and biological evaluation.
Topics: Animals; Brain; Cell Line, Tumor; Drug Design; Fluorescent Dyes; In Vitro Techniques; Indoles; Ligands; Radioligand Assay; Rats; Receptors, GABA-A; Spectrophotometry, Ultraviolet | 2007 |
Anxiolytic-like effects of N,N-dialkyl-2-phenylindol-3-ylglyoxylamides by modulation of translocator protein promoting neurosteroid biosynthesis.
Topics: Amides; Animals; Anti-Anxiety Agents; Cell Line, Tumor; Cell Membrane; Cerebral Cortex; Enzyme-Linked Immunosorbent Assay; Isoquinolines; Kidney; Maze Learning; Pregnenolone; Radioligand Assay; Rats | 2008 |
Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein.
Topics: Animals; Binding, Competitive; Carrier Proteins; Cell Line, Tumor; Cell Survival; Inhibitory Concentration 50; Molecular Structure; Quinazolines; Rats; Receptors, GABA-A; Structure-Activity Relationship | 2012 |
Relative efficacies of benzodiazepine receptor agonists in affecting red nucleus electrical activity in rabbits.
Topics: Animals; Bicuculline; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Imidazoles; Isoquinolines; Male; Pentylenetetrazole; Pyridazines; Pyridines; Rabbits; Receptors, GABA-A; Red Nucleus; Zolpidem | 1990 |
Imidazopyridines as a tool for the characterization of benzodiazepine receptors: a proposal for a pharmacological classification as omega receptor subtypes.
Topics: Animals; Brain Chemistry; Flunitrazepam; GABA-A Receptor Antagonists; Imidazoles; In Vitro Techniques; Isoquinolines; Kidney; Ligands; Pyridazines; Pyridines; Rats; Receptors, GABA-A; Spinal Cord; Terminology as Topic; Zolpidem | 1988 |
Participation of mitochondrial diazepam binding inhibitor receptors in the anticonflict, antineophobic and anticonvulsant action of 2-aryl-3-indoleacetamide and imidazopyridine derivatives.
Topics: Aggression; Allosteric Regulation; Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Clonazepam; Desoxycorticosterone; Flumazenil; Imidazoles; Indoleacetic Acids; Isoniazid; Isoquinolines; Mitochondria; Phobic Disorders; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, GABA-A; Seizures; Zolpidem | 1993 |