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alphaxalone and sr 95531

alphaxalone has been researched along with sr 95531 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19902 (20.00)18.7374
1990's7 (70.00)18.2507
2000's1 (10.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andre, JM; Boulanger, T; Durant, F; Hoffmann, R; Rognan, D; Vercauteren, DP; Wermuth, CG1
Korpi, ER; Lüddens, H; Seeburg, PH1
Maksay, G1
McCabe, RT; Olsen, RW; Wamsley, JK; Yezuita, JP1
Acosta-Burruel, M; Goodnough, DB; Hawkinson, JE; Kimbrough, CL; Wood, PL1
Kakemoto, E; Nagata, K; Okuyama, E; Ozoe, Y1
Amato, F; Biggio, G; Deserra, T; Motzo, C; Murgia, A; Sanna, E1
Bracamontes, J; Steinbach, JH; Ueno, S; Weiss, DS; Zorumski, C1
Biggio, G; Casula, A; Murgia, A; Sanna, E1
Goodchild, CS; Nadeson, R1

Other Studies

10 other study(ies) available for alphaxalone and sr 95531

ArticleYear
Structure and molecular modeling of GABAA receptor antagonists.
    Journal of medicinal chemistry, 1992, May-29, Volume: 35, Issue:11

    Topics: Alkaloids; Androstanes; Azasteroids; Azepines; Bicuculline; Crystallization; Dibenzazepines; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Heterocyclic Compounds, 4 or More Rings; Heterocyclic Compounds, Bridged-Ring; Isoxazoles; Lactones; Models, Molecular; Molecular Conformation; Molecular Structure; Piperidines; Pyridazines; Receptors, GABA-A; Structure-Activity Relationship; Tubocurarine; X-Ray Diffraction

1992
GABAA antagonists reveal binding sites for [35S]TBPS in cerebellar granular cell layer.
    European journal of pharmacology, 1992, Feb-18, Volume: 211, Issue:3

    Topics: Androstanes; Animals; Autoradiography; Azasteroids; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellar Cortex; Convulsants; GABA Antagonists; GABA-A Receptor Antagonists; Male; Pyridazines; Rats; Rats, Inbred Strains; Sulfur Radioisotopes

1992
GABAA receptor populations bind agonists and antagonists differentially and with opposite affinities.
    Journal of neurochemistry, 1988, Volume: 50, Issue:6

    Topics: Affinity Labels; Androstanes; Animals; Azasteroids; Brain; Diazepam; Diazonium Compounds; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscimol; Photochemistry; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfanilic Acids; Synaptic Membranes

1988
A novel GABAA antagonist [3H]SR 95531: microscopic analysis of binding in the rat brain and allosteric modulation by several benzodiazepine and barbiturate receptor ligands.
    Synapse (New York, N.Y.), 1988, Volume: 2, Issue:2

    Topics: Allosteric Regulation; Androstanes; Animals; Azasteroids; Binding, Competitive; Brain; Brain Chemistry; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Neurotransmitter

1988
Steroid inhibition of [3H]SR 95531 binding to the GABAA recognition site.
    European journal of pharmacology, 1996, May-23, Volume: 304, Issue:1-3

    Topics: Allosteric Regulation; Androstanes; Animals; Azasteroids; Cell Membrane; Cerebral Cortex; Desoxycorticosterone; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Pregnanolone; Pregnenolone; Protein Binding; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA; Steroids

1996
Interaction of anisatin with rat brain gamma-aminobutyric acidA receptors: allosteric modulation by competitive antagonists.
    Biochemical pharmacology, 1999, Aug-15, Volume: 58, Issue:4

    Topics: Affinity Labels; Allosteric Regulation; Androstanes; Animals; Azasteroids; Binding Sites; Binding, Competitive; Brain; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; GABA Antagonists; In Vitro Techniques; Lactones; Pyridazines; Rats; Receptors, GABA-A; Sesquiterpenes; Spiro Compounds; Tritium

1999
Expression of native GABAA receptors in Xenopus oocytes injected with rat brain synaptosomes.
    Journal of neurochemistry, 1996, Volume: 67, Issue:5

    Topics: Anesthetics; Animals; Brain; Cell Membrane; Chloride Channels; Chlorides; Diazepam; Female; GABA Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Oocytes; Picrotoxin; Pregnanediones; Pyridazines; Rats; Receptors, GABA-A; Synaptosomes; Xenopus laevis; Zinc Compounds

1996
Bicuculline and gabazine are allosteric inhibitors of channel opening of the GABAA receptor.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Jan-15, Volume: 17, Issue:2

    Topics: Allosteric Regulation; Allosteric Site; Amino Acid Sequence; Animals; Bicuculline; Binding Sites; Binding, Competitive; Cell Line; Coturnix; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ion Channel Gating; Ion Transport; Models, Chemical; Molecular Sequence Data; Mutagenesis, Site-Directed; Patch-Clamp Techniques; Pentobarbital; Point Mutation; Pregnanediones; Pregnanolone; Protein Binding; Pyridazines; Receptors, GABA-A; Structure-Activity Relationship

1997
Differential subunit dependence of the actions of the general anesthetics alphaxalone and etomidate at gamma-aminobutyric acid type A receptors expressed in Xenopus laevis oocytes.
    Molecular pharmacology, 1997, Volume: 51, Issue:3

    Topics: Anesthetics; Animals; Binding Sites; Chlorides; Etomidate; Oocytes; Picrotoxin; Pregnanediones; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Xenopus laevis

1997
Antinociceptive properties of neurosteroids II. Experiments with Saffan and its components alphaxalone and alphadolone to reveal separation of anaesthetic and antinociceptive effects and the involvement of spinal cord GABA(A) receptors.
    Pain, 2000, Volume: 88, Issue:1

    Topics: Alfaxalone Alfadolone Mixture; Anesthetics; Animals; Bicuculline; GABA Antagonists; GABA-A Receptor Antagonists; Male; Nociceptors; Pain Measurement; Pregnanediones; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Reference Values; Spinal Cord; Steroids; Time Factors

2000