Page last updated: 2024-08-26

alphaxalone and etomidate

alphaxalone has been researched along with etomidate in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19903 (14.29)18.7374
1990's3 (14.29)18.2507
2000's6 (28.57)29.6817
2010's9 (42.86)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Asproni, B; Biggio, G; Busonero, F; Cerri, R; Mascia, MP; Pau, A; Sanna, E; Sanna, S; Talani, G1
Atucha, E; Berger, ML; Hammerschmidt, F; Sieghart, W; Zolle, I1
Biziere, K; Keane, PE1
Erhardt, W; Ittner, J; Kramer, A1
Elliott, RC1
Benoit, E1
Biggio, G; Casula, A; Murgia, A; Sanna, E1
Finn, SE; Harrison, NL; Rick, CE; Ye, Q1
Carlson, BX; Engblom, AC; Kristiansen, U; Olsen, RW; Schousboe, A1
Chang, CS; Olcese, R; Olsen, RW1
Krähenbühl, K; Lambert, S; Rudolph, U; Siegwart, R1
Asproni, B; Biggio, G; Busonero, F; Cerri, R; Maciocco, E; Mascia, MP; Pau, A; Sanna, E; Talani, G1
Domínguez Pérez, JM; Fernández Sarmiento, JA; Gómez-Villamandos, RJ; Granados Machuca, MM; Muñoz-Rascón, P; Navarrete-Calvo, R; Quirós Carmona, S; Rodríguez, JM1
Akk, G; Eaton, MM; Li, P; Steinbach, JH1
Andaluz, A; Domínguez, E; Espada, Y; Fresno, L; García, F; Novellas, R; Rivera Del Álamo, MM; Santos, L1
Chandra, D; Homanics, GE; Iyer, SV1
Akk, G; Li, P1
Forman, SA; Stern, AT1
Forman, SA; Hotta, M; Nourmahnad, A; Stern, AT; Stewart, DS; Szabo, A; Ziemba, AM1
Bruzik, KS; Kent, DE; Miller, KW; Savechenkov, PY1

Reviews

1 review(s) available for alphaxalone and etomidate

ArticleYear
The effects of general anaesthetics on GABAergic synaptic transmission.
    Life sciences, 1987, Sep-21, Volume: 41, Issue:12

    Topics: Anesthesia, General; Anesthetics; Animals; Anti-Anxiety Agents; Barbiturates; Benzodiazepines; Ethanol; Etomidate; Humans; Pregnanediones; Receptors, GABA-A; Synaptic Transmission

1987

Other Studies

20 other study(ies) available for alphaxalone and etomidate

ArticleYear
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Synthesis, structure-activity relationships at the GABA(A) receptor in rat brain, and differential electrophysiological profile at the recombinant human GABA(A) receptor of a series of substituted 1,2-diphenylimidazoles.
    Journal of medicinal chemistry, 2005, Apr-07, Volume: 48, Issue:7

    Topics: Amino Acid Sequence; Animals; Behavior, Animal; Brain; Female; GABA-A Receptor Agonists; Humans; Imidazoles; In Vitro Techniques; Male; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Patch-Clamp Techniques; Protein Subunits; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Recombinant Proteins; Reflex; Stereoisomerism; Structure-Activity Relationship; Xenopus laevis

2005
Structure-activity relationship of etomidate derivatives at the GABA(A) receptor: Comparison with binding to 11beta-hydroxylase.
    Bioorganic & medicinal chemistry letters, 2009, Aug-01, Volume: 19, Issue:15

    Topics: Anesthetics, Intravenous; Animals; Binding Sites; Chemistry, Pharmaceutical; Drug Design; Etomidate; Inhibitory Concentration 50; Male; Models, Chemical; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stereoisomerism; Steroid 11-beta-Hydroxylase; Structure-Activity Relationship

2009
[Comparative studies of short-term anesthesia with alfentanil/etomidate and alphaxalone/alphadolone in cats].
    Tierarztliche Praxis. Supplement, 1985, Volume: 1

    Topics: Adjuvants, Anesthesia; Alfentanil; Anesthesia, Intravenous; Anesthetics; Animals; Cats; Etomidate; Fentanyl; Heart Rate; Imidazoles; Pregnanediones; Reflex; Respiration

1985
The action of intravenous anaesthetic and central depressant drugs on the contractures elicited by tetraethylammonium in the chick biventer cervicis muscle.
    General pharmacology, 1985, Volume: 16, Issue:6

    Topics: Alfaxalone Alfadolone Mixture; Anesthetics; Animals; Central Nervous System Depressants; Chickens; Chloralose; Diazepam; Drug Synergism; Ethanol; Etomidate; In Vitro Techniques; Methohexital; Muscle Contraction; Neck Muscles; Paraldehyde; Pregnanediones; Propanidid; Tetraethylammonium; Tetraethylammonium Compounds; Thiopental; Urethane

1985
Effects of intravenous anaesthetics on nerve axons.
    European journal of anaesthesiology, 1995, Volume: 12, Issue:1

    Topics: Action Potentials; Anesthetics, Intravenous; Animals; Axons; Dose-Response Relationship, Drug; Etomidate; Ion Channel Gating; Ketamine; Membrane Potentials; Nerve Fibers, Myelinated; Potassium; Potassium Channels; Pregnanediones; Rana esculenta; Sodium; Sodium Channels; Time Factors

1995
Differential subunit dependence of the actions of the general anesthetics alphaxalone and etomidate at gamma-aminobutyric acid type A receptors expressed in Xenopus laevis oocytes.
    Molecular pharmacology, 1997, Volume: 51, Issue:3

    Topics: Anesthetics; Animals; Binding Sites; Chlorides; Etomidate; Oocytes; Picrotoxin; Pregnanediones; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Xenopus laevis

1997
Neurosteroids act on the GABA(A) receptor at sites on the N-terminal side of the middle of TM2.
    Neuroreport, 1998, Feb-16, Volume: 9, Issue:3

    Topics: Anesthetics; Cell Line; Ethanol; Etomidate; GABA-A Receptor Agonists; Humans; Patch-Clamp Techniques; Pregnanediones; Receptors, Glycine; Steroids

1998
A single glycine residue at the entrance to the first membrane-spanning domain of the gamma-aminobutyric acid type A receptor beta(2) subunit affects allosteric sensitivity to GABA and anesthetics.
    Molecular pharmacology, 2000, Volume: 57, Issue:3

    Topics: Allosteric Regulation; Amino Acid Sequence; Anesthetics; Animals; Cells, Cultured; Chloride Channels; Electrophysiology; Etomidate; GABA Modulators; gamma-Aminobutyric Acid; Glycine; Ligands; Molecular Sequence Data; Mutagenesis, Site-Directed; Pentobarbital; Pregnanediones; Propofol; Protein Conformation; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Sequence Homology, Amino Acid; Spodoptera

2000
A single M1 residue in the beta2 subunit alters channel gating of GABAA receptor in anesthetic modulation and direct activation.
    The Journal of biological chemistry, 2003, Oct-31, Volume: 278, Issue:44

    Topics: Adjuvants, Anesthesia; Allosteric Site; Amino Acid Sequence; Anesthetics; Anesthetics, Intravenous; Animals; Cloning, Molecular; DNA Mutational Analysis; Dose-Response Relationship, Drug; Etomidate; Kinetics; Ligands; Models, Biological; Molecular Sequence Data; Mutagenesis; Mutation; Oocytes; Patch-Clamp Techniques; Pentobarbital; Point Mutation; Pregnanediones; Propofol; Protein Structure, Tertiary; Rats; Receptors, GABA-A; Recombinant Proteins; RNA, Messenger; Xenopus

2003
Mutational analysis of molecular requirements for the actions of general anaesthetics at the gamma-aminobutyric acidA receptor subtype, alpha1beta2gamma2.
    BMC pharmacology, 2003, Nov-12, Volume: 3

    Topics: Anesthetics, General; Animals; Cells, Cultured; Enflurane; Etomidate; gamma-Aminobutyric Acid; Humans; Point Mutation; Pregnanediones; Propofol; Protein Subunits; Rats; Receptors, GABA-A; Recombinant Proteins

2003
Ethyl 2-(4-bromophenyl)-1-(2,4-dichlorophenyl)-1H-4-imidazolecarboxylate is a novel positive modulator of GABAA receptors.
    European journal of pharmacology, 2005, Jun-15, Volume: 516, Issue:3

    Topics: Animals; Binding, Competitive; Cell Membrane; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Etomidate; Female; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Glycine; Humans; Hydrocarbons, Halogenated; Imidazoles; Male; Membrane Potentials; Oocytes; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Glycine; Receptors, Serotonin, 5-HT3; Serotonin; Tritium; Xenopus laevis

2005
Comparison of the cardiopulmonary parameters after induction of anaesthesia with alphaxalone or etomidate in dogs.
    Veterinary anaesthesia and analgesia, 2012, Volume: 39, Issue:4

    Topics: Anesthesia, Intravenous; Animals; Blood Gas Monitoring, Transcutaneous; Blood Pressure; Body Temperature; Dogs; Etomidate; Female; Heart; Heart Rate; Lung; Male; Pregnanediones; Respiratory Rate; Stroke Volume; Vascular Resistance

2012
The benzodiazepine diazepam potentiates responses of α1β2γ2L γ-aminobutyric acid type A receptors activated by either γ-aminobutyric acid or allosteric agonists.
    Anesthesiology, 2013, Volume: 118, Issue:6

    Topics: Anesthetics; Animals; Binding Sites; Diazepam; Drug Synergism; Etomidate; GABA Modulators; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Patch-Clamp Techniques; Pentobarbital; Pregnanediones; Rats; Receptors, GABA-A

2013
Doppler evaluation of the effects of propofol, etomidate and alphaxalone on fetoplacental circulation hemodynamics in the pregnant ewe.
    Placenta, 2013, Volume: 34, Issue:9

    Topics: Anesthesia, Obstetrical; Anesthetics, Intravenous; Animals; Animals, Inbred Strains; Blood Flow Velocity; Etomidate; Female; Fetus; Heart Rate, Fetal; Placental Circulation; Pregnancy; Pregnanediones; Propofol; Pulsatile Flow; Random Allocation; Sheep, Domestic; Ultrasonography, Doppler; Ultrasonography, Prenatal; Umbilical Arteries; Vascular Resistance

2013
GABAA-R α4 subunits are required for the low dose locomotor stimulatory effect of alphaxalone, but not for several other behavioral responses to alphaxalone, etomidate or propofol.
    Neurochemical research, 2014, Volume: 39, Issue:6

    Topics: Anesthetics; Animals; Etomidate; Female; Male; Mice; Mice, 129 Strain; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Pregnanediones; Propofol; Protein Subunits; Receptors, GABA-A

2014
Synaptic-type α1β2γ2L GABAA receptors produce large persistent currents in the presence of ambient GABA and anesthetic drugs.
    Molecular pharmacology, 2015, Volume: 87, Issue:5

    Topics: Anesthetics; Animals; Cell Line; Chromosome Pairing; Etomidate; gamma-Aminobutyric Acid; HEK293 Cells; Humans; Pentobarbital; Pregnanediones; Propofol; Rats; Receptors, GABA-A

2015
A Cysteine Substitution Probes β3H267 Interactions with Propofol and Other Potent Anesthetics in α1β3γ2L γ-Aminobutyric Acid Type A Receptors.
    Anesthesiology, 2016, Volume: 124, Issue:1

    Topics: Amino Acid Substitution; Anesthetics; Anesthetics, Intravenous; Animals; Barbiturates; Cysteine; Electrophysiological Phenomena; Etomidate; Female; Pregnanediones; Propofol; Receptors, GABA; Xenopus laevis

2016
Tryptophan and Cysteine Mutations in M1 Helices of α1β3γ2L γ-Aminobutyric Acid Type A Receptors Indicate Distinct Intersubunit Sites for Four Intravenous Anesthetics and One Orphan Site.
    Anesthesiology, 2016, Volume: 125, Issue:6

    Topics: Amino Acid Substitution; Anesthetics, Intravenous; Animals; Barbiturates; Binding Sites; Cysteine; Etomidate; Female; Ion Channel Gating; Mutation; Pregnanediones; Propofol; Receptors, GABA-A; Tryptophan; Xenopus

2016
Binding site location on GABA
    British journal of pharmacology, 2019, Volume: 176, Issue:24

    Topics: Anesthetics, Intravenous; Animals; Behavior, Animal; Binding Sites; Dose-Response Relationship, Drug; Drug Combinations; Drug Synergism; Etomidate; Larva; Mephobarbital; Pregnanediones; Receptors, GABA-A; Xenopus laevis

2019