Page last updated: 2024-09-04

alpha-ergocryptine and metergoline

alpha-ergocryptine has been researched along with metergoline in 1 studies

Compound Research Comparison

Studies
(alpha-ergocryptine)
Trials
(alpha-ergocryptine)
Recent Studies (post-2010)
(alpha-ergocryptine)
Studies
(metergoline)
Trials
(metergoline)
Recent Studies (post-2010) (metergoline)
74186563744

Protein Interaction Comparison

ProteinTaxonomyalpha-ergocryptine (IC50)metergoline (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.0007
Bile salt export pumpHomo sapiens (human)10
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)0.366
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.0041
Alpha-2A adrenergic receptorHomo sapiens (human)0.058
Cytochrome P450 2D6Homo sapiens (human)0.2
D(2) dopamine receptorHomo sapiens (human)0.063
Alpha-2B adrenergic receptorHomo sapiens (human)0.016
Alpha-2C adrenergic receptorHomo sapiens (human)0.189
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0062
Substance-K receptorHomo sapiens (human)4.071
D(1A) dopamine receptorHomo sapiens (human)0.074
AcetylcholinesteraseHomo sapiens (human)1.344
Sodium-dependent noradrenaline transporter Homo sapiens (human)0.366
Histamine H2 receptorHomo sapiens (human)0.975
Alpha-1D adrenergic receptorHomo sapiens (human)0.136
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0004
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0007
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.0062
Sodium-dependent serotonin transporterHomo sapiens (human)0.59
Histamine H1 receptorHomo sapiens (human)4.133
D(3) dopamine receptorHomo sapiens (human)0.0077
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0004
5-hydroxytryptamine receptor 6Homo sapiens (human)0.028
Sodium-dependent dopamine transporter Homo sapiens (human)0.063

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Boess, FG; Monsma, FJ; Sleight, AJ1

Other Studies

1 other study(ies) available for alpha-ergocryptine and metergoline

ArticleYear
Identification of residues in transmembrane regions III and VI that contribute to the ligand binding site of the serotonin 5-HT6 receptor.
    Journal of neurochemistry, 1998, Volume: 71, Issue:5

    Topics: Adenylyl Cyclases; Amino Acid Substitution; Binding Sites; Binding, Competitive; Cell Line; Cyclic AMP; Humans; Ligands; Lysergic Acid Diethylamide; Mutagenesis, Site-Directed; Mutation; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists

1998