Page last updated: 2024-08-21

alpha-aminopyridine and pyrilamine

alpha-aminopyridine has been researched along with pyrilamine in 108 studies

Research

Studies (108)

TimeframeStudies, this research(%)All Research%
pre-199098 (90.74)18.7374
1990's9 (8.33)18.2507
2000's1 (0.93)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hill, SJ; Marrian, DH; Sanders, JK; Young, JM1
Duchemin, AM; Quach, TT; Rose, C; Schwartz, JC2
Chang, RS; Snyder, SH; Tran, VT2
Al-Haboubi, HA; Zeitlin, IJ2
Gerner, T; Haffner, JF; Norstein, J1
Ayres, JW; Block, JH; Levine, HL1
Hill, SJ; Young, JM2
Kuhar, MJ; Palacios, JM; Young, WS1
Cho, CH; Ogle, CW1
Emson, PC; Hill, SJ; Young, JM1
Go, K; Namimatsu, A; Okuda, M; Tanimoto, H1
Bach, JF; Chatenoud, LM; Villemain, FM1
Ahluwalia, M; Bazan, E; Garver, D; Gruenstein, E; Johnson, CG; Johnson, CL1
Bloom, J; Freeman, JP; Getek, TA; Holder, CL; Korfmacher, WA1
Chand, N; Diamantis, W; Hess, FG; McGee, J; Nolan, K; Sofia, RD1
Khateb, A; Mühlethaler, M; Serafin, M1
Ido, T; Ishiwata, K; Itoh, M; Matsuzawa, T; Watanabe, T; Yagi, N; Yanai, K1
Bast, A; Leurs, R; Timmerman, H2
Donnelly, A; Gellhaus, M; Weiler, JM; Weiler, K1
Anuka, JA; Thomas, PJ; Walker, J1
Friedberg, KD; Sekardi, L1
Fukui, H; Inagaki, N; Taguchi, Y; Wada, H; Wang, NP; Yamatodani, A1
Mitsuhashi, M; Payan, DG1
Ruat, M; Schwartz, JC1
Fukui, H; Sawai, S; Tanaka, F; Wada, H; Wang, NP1
Dannals, RF; Ravert, HT; Scheffel, U; Tanada, S; Wagner, HN; Wilson, AA; Yanai, K2
Guo, ZG; Qiu, R1
Donoso, AO; Seltzer, AM1
Inoue, T; Kannan, MS1
Hsu, FL; Munavalli, S; Yeh, SY1
White, JM1
Kovatch, RM; Lijinsky, W1
Ahn, HS; Barnett, A1
Baker, CH; Davis, DL; Lindsey, BG; Sutton, ET1
Maslinski, C; Nowak, JZ1
Alvarez, EO; Banzán, AM1
Feit, F; Freedberg, RS; Friedman, GR; Palu, RN1
Bevan, J; Heptinstall, S2
Bouthenet, ML; Garbarg, M; Ruat, M; Sales, N; Schwartz, JC1
Treherne, JM; Young, JM1
Awadhiya, RP; Pillai, AG; Vegad, JL1
Rosenthal, MD; Williams, PB1
Ganellin, CR; Garbarg, M; Gros, C; Körner, M; Ruat, M; Schwartz, JC; Tertiuk, W1
Fukui, H; Wada, H; Wang, NP; Watanabe, T1
Betowski, LD; Holder, CL; Korfmacher, WA; Mitchum, RK1
Bach, JF; Cazenave, PA; Chatenoud, L; Ganellin, CR; Garbarg, M; Gros, C; Hoebeke, J; Korner, M; Ruat, M; Villemain, F1
Chen, J; Johnson, L; Spada, C; Woodward, DF1
Charap, A; Duzman, E; Leon, J; Shen, CD1
Ahmed, Ael H; el-Gizawy, SM1
Driver, AG; Mustafa, SJ1
Clive, D; Hozier, JC; Sawyer, JR; Turner, NT; Woolley, JL1
Bielkiewicz-Vollrath, B; Cook, DA1
Butkow, N; Gelgor, L; Mitchell, D; Phillips, S1
Marshall, K; Senior, J1
Bielkiewicz, B; Cook, DA2
Bouthenet, ML; Ganellin, CR; Garbarg, M; Gros, C; Ife, RJ; Korner, M; Sales, N; Schwartz, JC1
Eisenbrand, G; Habs, M; Shubik, P1
Arbonés, L; Claro, E; García, A; Picatoste, F1
Kanaide, H; Miwa, N; Nakamura, M; Nishimura, J1
Katayama, S; Tasaka, K1
Fujisawa, S; Nakai, K; Ohmiya, Y1
Daum, P; Hill, SJ; Young, JM1
Brossard, M1
Wallace, RM; Young, JM1
Hoffman, LH; Hoos, PC1
Coutts, II; Gibbs, CJ; Jackson, SM; White, RJ1
Hösli, E; Hösli, L; Schneider, U; Wiget, W1
Azuma, Y1
Andersen, V; Geisler, A; Klysner, R; Manthorpe, R; Nielsen, H; Norn, S; Permin, H; Petersen, J; Skov, PS; Wiik, A1
Bank, L; Bortz, D; Lipschitz, E; Marks, IN1
Del Soldato, P1
Chiou, GC; Miyano, K1
Haley, TJ1
Donoghue, ER; Kurland, ML; Lin, RL; Schaffer, MI; Stein, RJ; Wu Chen, NB1
Alvarez, EO1
Amerini, S; Bennardini, F; Franconi, F; Ledda, F; Mantelli, L; Matucci, R; Mugelli, A; Sorbi, C1
Lijinsky, W1
Hadfield, AJ; Hill, SJ; Robinson, NR1
Boertje, SB; Domer, FR; Sweeney, SA1
Godfraind, T; Miller, RC1
Elias, MS; Evans, PD; Lummis, SC1
Hui, HW; Robinson, JR; Zeleznick, L1
Tayal, G; Tripathi, KD2
Carter, DC; Lewi, HJ1
Dupont, A; Merand, Y; Savard, P1
Gross, PM; Harper, AM; Teasdale, GH1
Maśliński, S; Pruszyński, JP; Stajniak, A1
Carswell, H; Nahorski, SR1
Hunt, WA; Kaliner, M; Wescott, SL1
Lombroso, M; Nicosia, S1
Hiley, CR; Hill, SJ; Young, JM1
Heidemann, DR1
De Fabrizio, F2
Johnson, GR1
Chang, RS; Synder, SH1
Krabbe, AA; Olesen, J1
Clifton, PG; Hartfield, AW; Moore, NA1

Reviews

1 review(s) available for alpha-aminopyridine and pyrilamine

ArticleYear
Physical and biological properties of pyrilamine.
    Journal of pharmaceutical sciences, 1983, Volume: 72, Issue:1

    Topics: Aminopyridines; Animals; Carcinogens; Chemical Phenomena; Chemistry; Chemistry, Physical; Humans; Immunity; Kinetics; Mutagens; Nervous System Diseases; Pyrilamine; Structure-Activity Relationship; Teratogens; Time Factors

1983

Trials

5 trial(s) available for alpha-aminopyridine and pyrilamine

ArticleYear
Randomized, double-blind, parallel groups, placebo-controlled study of efficacy and safety of Rynatan in the treatment of allergic rhinitis using an acute model.
    Annals of allergy, 1990, Volume: 64, Issue:1

    Topics: Adolescent; Adult; Aged; Aminopyridines; Chlorpheniramine; Double-Blind Method; Drug Combinations; Humans; Middle Aged; Phenylephrine; Placebos; Pyrilamine; Rhinitis, Allergic, Seasonal

1990
Efficacy of cimetidine/pyrilamine eyedrops. A dose response study with histamine challenge.
    Ophthalmology, 1986, Volume: 93, Issue:1

    Topics: Adult; Aminopyridines; Cimetidine; Clinical Trials as Topic; Dose-Response Relationship, Drug; Drug Combinations; Eye; Eye Diseases; Female; Histamine; Humans; Hyperemia; Hypersensitivity; Male; Ophthalmic Solutions; Pyrilamine

1986
Skin test wheal size and erythema not reduced by topical antihistamine.
    British medical journal (Clinical research ed.), 1983, Nov-12, Volume: 287, Issue:6403

    Topics: Administration, Topical; Aminopyridines; Clinical Trials as Topic; Double-Blind Method; Erythema; Histamine H1 Antagonists; Humans; Hypersensitivity, Immediate; Pruritus; Pyrilamine; Skin Tests

1983
Effect of mepyramine on the untoward side-effects of impromidine.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1984, Aug-18, Volume: 66, Issue:7

    Topics: Aminopyridines; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Drug Interactions; Female; Flushing; Gastric Acid; Humans; Imidazoles; Impromidine; Male; Middle Aged; Pulse; Pyrilamine; Random Allocation; Receptors, Histamine; Receptors, Histamine H2

1984
Headache provocation by continuous intravenous infusion of histamine. Clinical results and receptor mechanisms.
    Pain, 1980, Volume: 8, Issue:2

    Topics: Aminopyridines; Cimetidine; Headache; Histamine; Humans; Migraine Disorders; Pyrilamine

1980

Other Studies

102 other study(ies) available for alpha-aminopyridine and pyrilamine

ArticleYear
A convenient synthesis of [3H]mepyramine and certain related [3H]antihistamines.
    The Journal of pharmacy and pharmacology, 1978, Volume: 30, Issue:10

    Topics: Aminopyridines; Chemical Phenomena; Chemistry; Histamine H1 Antagonists; Isotope Labeling; Methapyrilene; Methods; Pyrilamine; Tripelennamine; Tritium

1978
In vivo occupation of cerebral histamine H1-receptors evaluated with 3H-mepyramine may predict sedative properties of psychotropic drugs.
    European journal of pharmacology, 1979, Dec-20, Volume: 60, Issue:4

    Topics: Aminopyridines; Animals; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Cerebral Cortex; Hypnotics and Sedatives; Mice; Psychotropic Drugs; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1

1979
Characteristics of histamine H1-receptors in peripheral tissues labeled with [3H]mepyramine.
    The Journal of pharmacology and experimental therapeutics, 1979, Volume: 209, Issue:3

    Topics: Adrenal Glands; Aminopyridines; Animals; Aorta; Guinea Pigs; Haplorhini; Ileum; In Vitro Techniques; Lung; Macaca fascicularis; Male; Mice; Muscle, Smooth; Myocardium; Organ Specificity; Pyrilamine; Rabbits; Rats; Receptors, Histamine; Receptors, Histamine H1; Species Specificity

1979
The actions of cimetidine, mepyramine, indomethacin and aprotinin (Trasylol) on the inflammatory response in adjuvant rats [proceedings].
    British journal of pharmacology, 1979, Volume: 67, Issue:3

    Topics: Aminopyridines; Animals; Aprotinin; Arthritis; Arthritis, Experimental; Cimetidine; Guanidines; Indomethacin; Male; Pyrilamine; Rats

1979
The effects of mepyramine and cimetidine on the motor responses to histamine, cholecystokinin, and gastrin in the fundus and antrum of isolated guinea-pig stomachs.
    Scandinavian journal of gastroenterology, 1979, Volume: 14, Issue:1

    Topics: Acetylcholine; Aminopyridines; Animals; Cholecystokinin; Cimetidine; Female; Gastrins; Gastrointestinal Motility; Guanidines; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Pressure; Pyloric Antrum; Pyrilamine

1979
Paired-ion reversed-phase high-pressure liquid chromatographic assay of pentobarbital-pyrilamine suppositories.
    Journal of pharmaceutical sciences, 1979, Volume: 68, Issue:5

    Topics: Aminopyridines; Chromatography, Gas; Chromatography, High Pressure Liquid; Drug Combinations; Methods; Pentobarbital; Pyrilamine; Suppositories

1979
Heterogeneity of histamine H1-receptors: species variations in [3H]mepyramine binding of brain membranes.
    Journal of neurochemistry, 1979, Volume: 32, Issue:6

    Topics: Aminopyridines; Animals; Binding, Competitive; Brain; Cell Membrane; Cerebral Cortex; Guinea Pigs; Hippocampus; Humans; Kinetics; Male; Mice; Pyrilamine; Rabbits; Rats; Receptors, Histamine H1; Species Specificity

1979
The binding properties of [3H]-mepyramine in the brain of the guinea-pig and the rat [proceedings].
    British journal of pharmacology, 1979, Volume: 66, Issue:1

    Topics: Aminopyridines; Animals; Brain; Guinea Pigs; Pyrilamine; Rats; Species Specificity

1979
Autoradiographic localization of H1-histamine receptors in brain using 3H-mepyramine: preliminary studies.
    European journal of pharmacology, 1979, Oct-01, Volume: 58, Issue:3

    Topics: Aminopyridines; Animals; Autoradiography; Brain; Cerebellum; Guinea Pigs; Kinetics; Male; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Time Factors

1979
Histamine H1- and H2-receptor-mediated gastric microcirculatory effects in the aetiology of stress ulceration in the rat stomach.
    Experientia, 1978, Oct-15, Volume: 34, Issue:10

    Topics: Aminopyridines; Animals; Dose-Response Relationship, Drug; Gastric Mucosa; Humans; Male; Mast Cells; Metiamide; Microcirculation; Pyrilamine; Rats; Receptors, Histamine; Stomach Ulcer; Stress, Psychological; Thiourea

1978
The binding of [3H]mepyramine to histamine H1 receptors in guinea-pig brain.
    Journal of neurochemistry, 1978, Volume: 31, Issue:4

    Topics: Aminopyridines; Animals; Brain; Cerebellum; Guinea Pigs; Promethazine; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1

1978
Mechanism of nasal secretion mediated via nerve reflex in guinea pigs and evaluation of antiallergic drugs.
    International archives of allergy and immunology, 1992, Volume: 97, Issue:2

    Topics: Allergens; Aminopyridines; Animals; Atropine Derivatives; Bronchodilator Agents; Capsaicin; Ganglionic Blockers; Guinea Pigs; Hexamethonium; Hexamethonium Compounds; Histamine; Hypersensitivity; Lidocaine; Methacholine Chloride; Nasal Mucosa; ortho-Aminobenzoates; Parasympatholytics; Phthalazines; Pyrilamine; Reflex

1992
Characterization of histamine H1 binding sites on human T lymphocytes by means of 125I-iodobolpyramine. Preferential expression of H1 receptors on CD8 T lymphocytes.
    Journal of immunology (Baltimore, Md. : 1950), 1990, Feb-15, Volume: 144, Issue:4

    Topics: Aminopyridines; Animals; Antigens, Differentiation, T-Lymphocyte; CD4-Positive T-Lymphocytes; CD8 Antigens; Cell Membrane; Cerebellum; Guinea Pigs; Humans; Kinetics; Pyrilamine; Receptors, Histamine H1; Succinimides; T-Lymphocytes; T-Lymphocytes, Helper-Inducer; T-Lymphocytes, Regulatory

1990
Histamine receptors in human fibroblasts: inositol phosphates, Ca2+, and cell growth.
    The American journal of physiology, 1990, Volume: 258, Issue:3 Pt 1

    Topics: Aminopyridines; Calcium; Cell Division; Cell Line; DNA Replication; Fibroblasts; Fluorescent Dyes; Histamine; Humans; Inositol Phosphates; Kinetics; Phorbol 12,13-Dibutyrate; Pyrilamine; Receptors, Histamine; Skin; Tetradecanoylphorbol Acetate; Thymidine

1990
Analysis of rat urine for metabolites of pyrilamine via high-performance liquid chromatography/thermospray mass spectrometry and tandem mass spectrometry.
    Biomedical & environmental mass spectrometry, 1990, Volume: 19, Issue:3

    Topics: Aminopyridines; Animals; Biotransformation; Chromatography, High Pressure Liquid; Female; Male; Mass Spectrometry; Molecular Weight; Pyrilamine; Rats; Rats, Inbred F344; Reference Standards; Spectrophotometry, Ultraviolet

1990
Aeroallergen-induced immediate asthmatic responses and late-phase associated pulmonary eosinophilia in the guinea pig: effect of methylprednisolone and mepyramine.
    International archives of allergy and applied immunology, 1990, Volume: 91, Issue:3

    Topics: Administration, Oral; Aerosols; Aminopyridines; Animals; Asthma; Drug Administration Schedule; Guinea Pigs; Methylprednisolone; Ovalbumin; Premedication; Pulmonary Eosinophilia; Pyrilamine

1990
Histamine excites pedunculopontine neurones in guinea pig brainstem slices.
    Neuroscience letters, 1990, May-04, Volume: 112, Issue:2-3

    Topics: Action Potentials; Aminopyridines; Animals; Guinea Pigs; Histamine; In Vitro Techniques; Pons; Pyrilamine; Receptors, Histamine; Tetrodotoxin

1990
Specific binding of [3H]pyrilamine to histamine H1 receptors in guinea pig brain in vivo: determination of binding parameters by a kinetic four-compartment model.
    Journal of neurochemistry, 1990, Volume: 55, Issue:2

    Topics: Aminopyridines; Animals; Binding, Competitive; Brain; Cerebellum; Cerebral Cortex; Chlorpheniramine; Corpus Striatum; Guinea Pigs; Hippocampus; Kinetics; Male; Mathematics; Models, Biological; Pyrilamine; Receptors, Histamine H1; Stereoisomerism; Thalamus; Tissue Distribution; Tritium

1990
Labelling of non-H1-receptor binding sites by [3H]-mepyramine on the rat liver plasma membrane.
    Agents and actions, 1990, Volume: 30, Issue:1-2

    Topics: Aminopyridines; Animals; Cell Membrane; In Vitro Techniques; Kinetics; Liver; Male; Proteins; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Stereoisomerism

1990
Some effects of oestrogens on [3H]-mepyramine binding in rat brain.
    Methods and findings in experimental and clinical pharmacology, 1986, Volume: 8, Issue:11

    Topics: 1-Methyl-3-isobutylxanthine; Aminopyridines; Animals; Brain; Estrogens; Female; Male; Ovariectomy; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1

1986
Inhibition of immunological histamine release from guinea pig lungs and other organs by mepyramine, ketotifen, and picumast in vivo.
    Arzneimittel-Forschung, 1989, Volume: 39, Issue:10A

    Topics: Aminopyridines; Anaphylaxis; Animals; Coumarins; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine Release; Ketotifen; Lung; Male; Pyrilamine

1989
High affinity, saturable [3H]mepyramine binding sites on rat liver plasma membrane do not represent histamine H1-receptors. A warning.
    Biochemical pharmacology, 1989, Jul-01, Volume: 38, Issue:13

    Topics: Aminopyridines; Animals; Binding, Competitive; Cell Membrane; Histamine H1 Antagonists; Kinetics; Liver; Male; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Structure-Activity Relationship

1989
Characterization of histamine H1-receptors on astrocytes in primary culture: [3H]mepyramine binding studies.
    European journal of pharmacology, 1989, Nov-28, Volume: 173, Issue:1

    Topics: Aminopyridines; Animals; Animals, Newborn; Astrocytes; Binding, Competitive; Brain; Cells, Cultured; Histamine H1 Antagonists; In Vitro Techniques; Kinetics; Male; Pyrilamine; Rats; Receptors, Histamine H1

1989
Solubilization and characterization of the pyrilamine-binding protein from cultured smooth muscle cells.
    Molecular pharmacology, 1989, Volume: 35, Issue:6

    Topics: Aminopyridines; Animals; Cell Line; Chromatography, Gel; Chromatography, High Pressure Liquid; Kinetics; Molecular Weight; Muscle, Smooth; Polyethylene Glycols; Pyrilamine; Receptors, Histamine H1; Solubility; Substrate Specificity

1989
Photoaffinity labeling and electrophoretic identification of the H1-receptor: comparison of several brain regions and animal species.
    Journal of neurochemistry, 1989, Volume: 53, Issue:2

    Topics: Affinity Labels; Aminopyridines; Animals; Brain; Electrophoresis, Polyacrylamide Gel; Guinea Pigs; Male; Membranes; Mice; Mice, Inbred Strains; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Tissue Distribution

1989
Divalent cations increase the binding capacity of the [3H]mepyramine binding site, a possible histamine H1 receptor, in rat liver membranes.
    Japanese journal of pharmacology, 1989, Volume: 49, Issue:3

    Topics: Aminopyridines; Animals; Brain; Calcium; Cations; Liver; Male; Membranes; Proteins; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1

1989
Biodistribution and radiation absorbed dose of (N-methyl[11C])pyrilamine: a histamine H-1 receptor radiotracer.
    International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology, 1989, Volume: 16, Issue:4

    Topics: Aminopyridines; Animals; Brain; Carbon Radioisotopes; Male; Mice; Pyrilamine; Radiation Dosage; Radionuclide Imaging; Receptors, Histamine H2; Tissue Distribution

1989
Protective effects of histamine H1 and H2 antagonists, adenosine and hydrocortisone on cardiac anaphylaxis.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1989, Volume: 10, Issue:1

    Topics: Adenosine; Aminopyridines; Anaphylaxis; Animals; Arrhythmias, Cardiac; Cardiac Output; Cimetidine; Guinea Pigs; Heart Rate; Hydrocortisone; In Vitro Techniques; Pyrilamine; Receptors, Histamine

1989
Effects of ovariectomy and ovarian steroids on binding of 3H-mepyramine, an H1-histamine antagonist, in rat hypothalamus.
    Brain research bulletin, 1989, Volume: 23, Issue:3

    Topics: Aminopyridines; Animals; Estradiol; Female; Hypothalamus; Luteinizing Hormone; Ovariectomy; Progesterone; Pyrilamine; Radioimmunoassay; Radioligand Assay; Rats; Receptors, Histamine H1

1989
Nonadrenergic and noncholinergic excitatory neurotransmission in rat intrapulmonary artery.
    The American journal of physiology, 1988, Volume: 254, Issue:6 Pt 2

    Topics: Aminopyridines; Animals; Atropine; Electric Stimulation; Guanethidine; In Vitro Techniques; Male; Membrane Potentials; Muscle, Smooth, Vascular; Neuromuscular Junction; Norepinephrine; Phentolamine; Propranolol; Pulmonary Artery; Pyrilamine; Rats; Rats, Inbred Strains; Synaptic Transmission; Tetrodotoxin

1988
O-demethylation of pyrilamine.
    Journal of pharmaceutical sciences, 1988, Volume: 77, Issue:8

    Topics: Acids; Aminopyridines; Chemical Phenomena; Chemistry; Dealkylation; Hydrobromic Acid; Pyrilamine

1988
The discriminative stimulus properties of mepyramine.
    Life sciences, 1985, Sep-23, Volume: 37, Issue:12

    Topics: Aminopyridines; Animals; Chlorpheniramine; Discrimination, Psychological; Histamine H1 Antagonists; Imipramine; Male; Procaine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Scopolamine

1985
Carcinogenicity studies of some analogs of the carcinogen methapyrilene in F344 rats.
    Journal of cancer research and clinical oncology, 1986, Volume: 112, Issue:1

    Topics: Aminopyridines; Animals; Female; Histamine H1 Antagonists; Liver Neoplasms; Male; Methapyrilene; Pyridines; Pyrilamine; Rats; Rats, Inbred F344; Rats, Inbred Strains; Structure-Activity Relationship

1986
Selective displacement of [3H]mepyramine from peripheral vs. central nervous system receptors by loratadine, a non-sedating antihistamine.
    European journal of pharmacology, 1986, Aug-07, Volume: 127, Issue:1-2

    Topics: Aminopyridines; Animals; Binding, Competitive; Cerebral Cortex; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Kinetics; Loratadine; Lung; Male; Piperidines; Pyrilamine; Receptors, Cell Surface

1986
Adrenergic and histaminergic neural interactions in dog paws.
    The American journal of physiology, 1988, Volume: 255, Issue:3 Pt 2

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Aminopyridines; Animals; Blood Pressure; Blood Volume; Capillaries; Dogs; Electric Stimulation; Hindlimb; Metiamide; Pyrilamine; Reference Values; Regional Blood Flow; Sciatic Nerve; Thiourea; Vascular Resistance

1988
3H-mepyramine binding and histamine-stimulated cAMP accumulation in mammalian retina.
    Agents and actions, 1986, Volume: 18, Issue:1-2

    Topics: Aminopyridines; Animals; Brain; Cattle; Cyclic AMP; Dopamine; Guinea Pigs; Histamine; In Vitro Techniques; Pyrilamine; Rabbits; Receptors, Histamine; Retina; Tritium

1986
Histamine in dorsal and ventral hippocampus. II. Effects of H1 and H2 histamine antagonists on exploratory behavior in male rats.
    Physiology & behavior, 1986, Volume: 37, Issue:1

    Topics: Aminopyridines; Animals; Brain Mapping; Exploratory Behavior; Hippocampus; Histamine; Histidine Decarboxylase; Male; Methylhistidines; Motor Activity; Neural Inhibition; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Synaptic Transmission

1986
Cardiogenic shock due to antihistamine overdose. Reversal with intra-aortic balloon counterpulsation.
    JAMA, 1987, Feb-06, Volume: 257, Issue:5

    Topics: Aminopyridines; Combined Modality Therapy; Epilepsy, Tonic-Clonic; Female; Humans; Intra-Aortic Balloon Pumping; Middle Aged; Pyrilamine; Shock, Cardiogenic; Suicide, Attempted; Sympathomimetics

1987
Serotonin-induced platelet aggregation in whole blood and the effects of ketanserin and mepyramine.
    Thrombosis research, 1985, Apr-15, Volume: 38, Issue:2

    Topics: Aminopyridines; Dose-Response Relationship, Drug; Humans; Ketanserin; Piperidines; Platelet Aggregation; Pyrilamine; Serotonin; Time Factors

1985
A detailed mapping of histamine H1-receptors in guinea-pig central nervous system established by autoradiography with [125I]iodobolpyramine.
    Neuroscience, 1988, Volume: 26, Issue:2

    Topics: Aminopyridines; Animals; Autoradiography; Brain; Brain Mapping; Guinea Pigs; Pyrilamine; Receptors, Histamine; Spinal Cord; Succinimides

1988
Temperature-dependence of the kinetics of the binding of [3H]-(+)-N-methyl-4-methyldiphenhydramine to the histamine H1-receptor: comparison with the kinetics of [3H]-mepyramine.
    British journal of pharmacology, 1988, Volume: 94, Issue:3

    Topics: Aminopyridines; Animals; Cerebellum; Guinea Pigs; Histamine Antagonists; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle, Smooth; Pyrilamine; Receptors, Histamine H1; Temperature

1988
Suppression by mepyramine maleate of the increased vascular permeability in passive cutaneous anaphylaxis in the chicken.
    Veterinary research communications, 1988, Volume: 12, Issue:2-3

    Topics: Aminopyridines; Animals; Capillary Permeability; Chickens; Female; Male; Passive Cutaneous Anaphylaxis; Pyrilamine

1988
Ascorbate increases apparent "specific" binding of [3H]pyrilamine to glass fiber filters.
    Journal of pharmacological methods, 1988, Volume: 20, Issue:4

    Topics: Aminopyridines; Ascorbic Acid; Binding Sites; Buffers; Filtration; Glass; Ligands; Pyrilamine

1988
(N-methyl-[11C])pyrilamine, a radiotracer for histamine H-1 receptors: radiochemical synthesis and biodistribution study in mice.
    International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology, 1988, Volume: 15, Issue:6

    Topics: Aminopyridines; Animals; Brain; Brain Chemistry; Carbon Radioisotopes; Isotope Labeling; Male; Mice; Pyrilamine; Radionuclide Imaging; Receptors, Histamine H1; Tissue Distribution

1988
Characterization of histamine H1-receptor binding peptides in guinea pig brain using [125I]iodoazidophenpyramine, an irreversible specific photoaffinity probe.
    Proceedings of the National Academy of Sciences of the United States of America, 1988, Volume: 85, Issue:8

    Topics: Affinity Labels; Aminopyridines; Animals; Cell Membrane; Cerebellum; Electrophoresis, Polyacrylamide Gel; Guinea Pigs; In Vitro Techniques; Mercaptoethanol; Photochemistry; Protease Inhibitors; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1

1988
Solubilization, characterization and partial purification of [3H]mepyramine-binding protein, a possible histamine H1 receptor, from rat liver membrane.
    Japanese journal of pharmacology, 1988, Volume: 46, Issue:2

    Topics: Aminopyridines; Animals; Centrifugation, Density Gradient; Chromatography, Gel; Chromatography, High Pressure Liquid; Gamma Rays; In Vitro Techniques; Liver; Male; Molecular Weight; Protein Binding; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Sucrose

1988
Characterization of doxylamine and pyrilamine metabolites via thermospray/mass spectrometry and tandem mass spectrometry.
    Biomedical & environmental mass spectrometry, 1988, May-01, Volume: 15, Issue:9

    Topics: Aminopyridines; Animals; Biotransformation; Doxylamine; Female; Macaca mulatta; Male; Mass Spectrometry; Pyridines; Pyrilamine; Rats; Rats, Inbred F344

1988
Polyclonal and monoclonal antibodies directed against SK & F 94461, a specific H1 histamine receptor ligand.
    Molecular pharmacology, 1988, Volume: 34, Issue:2

    Topics: Aminopyridines; Animals; Antibodies, Monoclonal; Antibody Affinity; Antibody Specificity; Binding, Competitive; Immunoglobulin Idiotypes; Mice; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Spectrometry, Fluorescence; Spectrophotometry, Ultraviolet; Time Factors

1988
Effect of cimetidine and pyrilamine on histamine-induced ocular surface hyperemia.
    Journal of ocular pharmacology, 1986,Summer, Volume: 2, Issue:3

    Topics: Aminopyridines; Animals; Cimetidine; Drug Therapy, Combination; Eye Diseases; Female; Histamine; Hyperemia; Pyrilamine; Rabbits

1986
High-performance liquid chromatographic determination of mepyramine maleate, pheniramine maleate and phenylpropanolamine hydrochloride in tablets and drops.
    The Analyst, 1987, Volume: 112, Issue:6

    Topics: Aminopyridines; Chromatography, High Pressure Liquid; Histamine Antagonists; Pheniramine; Phenylpropanolamine; Pyrilamine; Solutions; Tablets

1987
Correlation of histamine H1 receptor function and [3H]mepyramine binding in porcine tracheal tissue.
    European journal of pharmacology, 1987, Jul-23, Volume: 139, Issue:3

    Topics: Aminopyridines; Animals; In Vitro Techniques; Models, Biological; Muscle Contraction; Muscle, Smooth; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Swine; Time Factors; Trachea

1987
Methapyrilene is a genotoxic carcinogen: studies on methapyrilene and pyrilamine in the L5178Y/TK +/- mouse lymphoma assay.
    Mutation research, 1987, Volume: 189, Issue:3

    Topics: Aminopyridines; Animals; Biotransformation; Carcinogens; Chromosome Aberrations; Leukemia L5178; Methapyrilene; Mice; Microsomes, Liver; Mutagenicity Tests; Neoplasm Proteins; Preservation, Biological; Pyrilamine; Rats; Thymidine Kinase; Tumor Cells, Cultured; Tumor Stem Cell Assay

1987
Binding of 3H-mepyramine to dog portal vein and cerebral cortex.
    Proceedings of the Western Pharmacology Society, 1986, Volume: 29

    Topics: Aminopyridines; Animals; Cerebral Cortex; Dogs; In Vitro Techniques; Muscle, Smooth, Vascular; Portal Vein; Pyrilamine; Receptors, Histamine H1

1986
Injectable aspirin and mepyramine abolish post-ischaemic hyperalgesia in rats.
    Pain, 1986, Volume: 26, Issue:3

    Topics: Aminopyridines; Animals; Aspirin; Histamine; Hyperalgesia; Hyperesthesia; Ischemia; Male; Prostaglandins; Pyrilamine; Rats; Rats, Inbred Strains

1986
The effect of mepyramine and ranitidine on the oestrogen and anti-oestrogen stimulated rat uterus.
    British journal of pharmacology, 1986, Volume: 89, Issue:1

    Topics: Aminopyridines; Animals; Estrogen Antagonists; Estrogens; Female; Organ Size; Pyrilamine; Ranitidine; Rats; Receptors, Histamine; Regional Blood Flow; Tamoxifen; Uterine Contraction; Uterus

1986
The binding of [3H]mepyramine to histamine H1 receptors in monkey brain.
    Canadian journal of physiology and pharmacology, 1985, Volume: 63, Issue:6

    Topics: Aminopyridines; Animals; Brain; Haplorhini; In Vitro Techniques; Kinetics; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1

1985
[125I]Iodobolpyramine, a highly sensitive probe for histamine H1-receptors in guinea-pig brain.
    European journal of pharmacology, 1986, Jan-21, Volume: 120, Issue:2

    Topics: Aminopyridines; Animals; Autoradiography; Brain; Cerebellum; Guinea Pigs; In Vitro Techniques; Indicators and Reagents; Iodine Radioisotopes; Kinetics; Male; Membranes; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Succinimides

1986
Carcinogenicity of methapyrilene hydrochloride, mepyramine hydrochloride, thenyldiamine hydrochloride, and pyribenzamine hydrochloride in Sprague-Dawley rats.
    Journal of cancer research and clinical oncology, 1986, Volume: 111, Issue:1

    Topics: Adenoma; Adrenal Gland Neoplasms; Aminopyridines; Animals; Dose-Response Relationship, Drug; Female; Liver Neoplasms; Liver Neoplasms, Experimental; Male; Methapyrilene; Neoplasms, Experimental; Pyridines; Pyrilamine; Rats; Structure-Activity Relationship; Tripelennamine

1986
[3H]mepyramine binding to histamine H1 receptors in bovine retina.
    Biochemical and biophysical research communications, 1986, Mar-13, Volume: 135, Issue:2

    Topics: Aminopyridines; Animals; Binding, Competitive; Cattle; Kinetics; Pyrilamine; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H1; Retina

1986
Specific binding of [3H] mepyramine to histamine H1-receptors in the sarcolemma from porcine aorta and coronary artery.
    Biochemical and biophysical research communications, 1985, Jan-16, Volume: 126, Issue:1

    Topics: Aminopyridines; Animals; Aorta; Centrifugation, Density Gradient; Coronary Vessels; Kinetics; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Sarcolemma; Subcellular Fractions; Swine

1985
Effects of H1-receptor blocking drugs on the frog sartorius neuromuscular junction.
    British journal of pharmacology, 1985, Volume: 85, Issue:4

    Topics: Action Potentials; Aminopyridines; Animals; Diphenhydramine; Dose-Response Relationship, Drug; Electric Conductivity; Electrophysiology; Membrane Potentials; Neuromuscular Junction; Perfusion; Promethazine; Pyrilamine; Ranidae; Receptors, Histamine; Receptors, Histamine H1; Time Factors

1985
Comparison of pulmonary accumulation of pyrilamine and pyrilamine N-oxide.
    Japanese journal of pharmacology, 1985, Volume: 38, Issue:4

    Topics: Aminopyridines; Animals; Cyclic N-Oxides; In Vitro Techniques; Kinetics; Lung; Male; Mice; Mice, Inbred ICR; Pyrilamine

1985
Characterization of [3H]mepyramine binding to the longitudinal muscle of guinea pig small intestine.
    Molecular pharmacology, 1981, Volume: 19, Issue:3

    Topics: Aminopyridines; Animals; Binding Sites; Calcium; Guinea Pigs; Histamine; Histamine H1 Antagonists; Hydrogen-Ion Concentration; In Vitro Techniques; Intestine, Small; Magnesium; Male; Muscle, Smooth; Pyrilamine; Receptors, Histamine H1

1981
Affinities of histamine H1-antagonists in guinea pig brain: similarity of values determined from [3H]mepyramine binding and from inhibition of a functional response.
    Journal of neurochemistry, 1981, Volume: 37, Issue:5

    Topics: Aminopyridines; Animals; Binding, Competitive; Brain; Female; Guinea Pigs; Histamine H1 Antagonists; Kinetics; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Structure-Activity Relationship

1981
Rabbits infested with adult Ixodes ricinus L.: effects of mepyramine on acquired resistance.
    Experientia, 1982, Jun-15, Volume: 38, Issue:6

    Topics: Aminopyridines; Animals; Female; Histamine H1 Antagonists; Immunity, Innate; Male; Oviposition; Pyrilamine; Rabbits; Tick Infestations; Ticks

1982
Labeling of histamine H1-receptors in the brain of the living mouse.
    Neuroscience letters, 1980, Volume: 17, Issue:1-2

    Topics: Aminopyridines; Animals; Binding Sites; Binding, Competitive; Brain; Histamine H1 Antagonists; Male; Mice; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1

1980
Temperature dependence of the binding of [3H]mepyramine and related compounds to the histamine H1 receptor.
    Molecular pharmacology, 1983, Volume: 23, Issue:1

    Topics: Aminopyridines; Animals; Cerebellum; Chlorpromazine; Guinea Pigs; Histamine H1 Antagonists; Kinetics; Male; Phenothiazines; Promethazine; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Temperature; Tripelennamine

1983
Effect of histamine receptor antagonists and indomethacin on implantation in the rabbit.
    Biology of reproduction, 1983, Volume: 29, Issue:4

    Topics: Aminopyridines; Animals; Capillary Permeability; Cimetidine; Drug Combinations; Drug Interactions; Embryo Implantation; Female; Histamine H1 Antagonists; Indomethacin; Pregnancy; Pyrilamine; Rabbits; Uterus

1983
Evidence for the existence of histamine H1- and H2-receptors on astrocytes of cultured rat central nervous system.
    Neuroscience letters, 1984, Aug-10, Volume: 48, Issue:3

    Topics: Aminopyridines; Animals; Astrocytes; Brain Stem; Cells, Cultured; Cimetidine; Histamine; Histamine H1 Antagonists; Membrane Potentials; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Spinal Cord; Thiazoles

1984
[Pharmacological studies on rat passive cutaneous anaphylaxis (PCA) (author's transl)].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1980, Volume: 76, Issue:8

    Topics: Aminopyridines; Aminopyrine; Animals; Benzydamine; Cyclic AMP; Epinephrine; Histamine Release; Isoproterenol; Male; Passive Cutaneous Anaphylaxis; Pyrilamine; Rabbits; Rats; Tissue Distribution

1980
Possible role of histamine in rheumatoid arthritis. Treatment with cimetidine and mepyramine.
    Allergy, 1981, Volume: 36, Issue:6

    Topics: Adolescent; Adult; Aminopyridines; Arthritis, Rheumatoid; Cimetidine; Drug Therapy, Combination; Female; Guanidines; Histamine H1 Antagonists; Histamine Release; Humans; Male; Middle Aged; Pyrilamine

1981
Studies with specific agonists and antagonists of the role of histamine H1- and H2-receptor activation in the pathogenesis of gastric lesions in rats.
    Agents and actions, 1984, Volume: 14, Issue:2

    Topics: Aminopyridines; Animals; Atropine; Dimaprit; Drug Interactions; Female; Histamine; Pyridines; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach Ulcer; Thiourea

1984
Pharmacological prevention of ocular inflammation induced by lens proteins.
    Ophthalmic research, 1984, Volume: 16, Issue:5

    Topics: Aminopyridines; Animals; Catechols; Cimetidine; Crystallins; Disease Models, Animal; Drug Therapy, Combination; Endophthalmitis; Female; Indomethacin; Masoprocol; Pyrilamine; Rabbits

1984
The general toxicology unknown. II. A case report: doxylamine and pyrilamine intoxication.
    Journal of forensic sciences, 1983, Volume: 28, Issue:2

    Topics: Adult; Aminopyridines; Chromatography, Gas; Doxylamine; Gas Chromatography-Mass Spectrometry; Humans; Immunoenzyme Techniques; Male; Mass Spectrometry; Pyridines; Pyrilamine; Spectrophotometry; Suicide; Toxicology

1983
Effects of histamine antagonists injected in the preoptic-anterior hypothalamic area on the prolactin surge induced by estrogen in ovariectomized rats.
    Brain research bulletin, 1984, Volume: 12, Issue:1

    Topics: Aminopyridines; Animals; Castration; Circadian Rhythm; Drug Implants; Estrogens; Female; Hypothalamus, Anterior; Metiamide; Preoptic Area; Prolactin; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea

1984
Specific and non-specific displaceable binding of 3H-mepyramine to homogenates of monkey cortex.
    Proceedings of the Western Pharmacology Society, 1984, Volume: 27

    Topics: Aminopyridines; Animals; Binding, Competitive; Cerebral Cortex; Haplorhini; In Vitro Techniques; Pyrilamine

1984
On the presence of H1-receptors in various sections of guinea-pig heart: a correlation between binding and functional studies.
    Agents and actions, 1984, Volume: 15, Issue:3-4

    Topics: Aminopyridines; Animals; Binding Sites; Guinea Pigs; Heart Atria; Heart Ventricles; In Vitro Techniques; Male; Membranes; Myocardium; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1

1984
Chronic toxicity tests of pyrilamine maleate and methapyrilene hydrochloride in F344 rats.
    Food and chemical toxicology : an international journal published for the British Industrial Biological Research Association, 1984, Volume: 22, Issue:1

    Topics: Aminopyridines; Animals; Carcinogens; Diet; Dose-Response Relationship, Drug; Female; Liver Neoplasms; Male; Methapyrilene; Pyrilamine; Rats; Rats, Inbred F344; Structure-Activity Relationship; Time Factors

1984
Effects of ketanserin and mepyramine on platelet aggregation and on the uptake of 5-hydroxytryptamine into platelets.
    Thrombosis research, 1983, Jun-01, Volume: 30, Issue:5

    Topics: Adenosine Diphosphate; Aminopyridines; Blood Platelets; Humans; Ketanserin; Piperidines; Platelet Aggregation; Pyrilamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1983
The nature of the binding of [3H]mepyramine to homogenates of guinea-pig cerebral cortex at different [3H]ligand concentrations.
    Biochemical pharmacology, 1983, Aug-15, Volume: 32, Issue:16

    Topics: Aminopyridines; Animals; Cerebral Cortex; Guinea Pigs; In Vitro Techniques; Kinetics; Pyrilamine; Receptors, Histamine H1; Tritium

1983
Blockade of the acetylcholine-and histamine-induced changes in the permeability of the blood-brain barrier of normotensive and spontaneously hypertensive rats by atropine and pyrilamine.
    Research communications in chemical pathology and pharmacology, 1983, Volume: 42, Issue:1

    Topics: Acetylcholine; Aminopyridines; Animals; Atropine; Blood Pressure; Blood-Brain Barrier; Female; Histamine; Hypertension; Male; Pyrilamine; Rats; Rats, Inbred Strains

1983
Effects of histamine and the histamine antagonists mepyramine and cimetidine on human coronary arteries in vitro.
    British journal of pharmacology, 1983, Volume: 79, Issue:4

    Topics: Adolescent; Adult; Aged; Aminopyridines; Child; Cimetidine; Coronary Vessels; Histamine; Humans; In Vitro Techniques; Middle Aged; Muscle Contraction; Muscle Relaxation; Potassium; Pyrilamine

1983
[3H]mepyramine binding sites in the optic lobe of the locust: autoradiographic and pharmacological studies.
    Brain research, 1984, Mar-05, Volume: 294, Issue:2

    Topics: Aminopyridines; Animals; Autoradiography; Binding Sites; Binding, Competitive; Grasshoppers; Kinetics; Optic Lobe, Nonmammalian; Pyrilamine; Tritium

1984
Ocular disposition of topically applied histamine, cimetidine, and pyrilamine in the albino rabbit.
    Current eye research, 1984, Volume: 3, Issue:2

    Topics: Administration, Topical; Aminopyridines; Animals; Aqueous Humor; Biological Availability; Ciliary Body; Cimetidine; Conjunctiva; Cornea; Eye; Histamine; Iris; Male; Pyrilamine; Rabbits

1984
Histamine antagonists modify systemic digoxin cardiotoxicity by their central action.
    The Indian journal of medical research, 1984, Volume: 79

    Topics: Aminopyridines; Animals; Arrhythmias, Cardiac; Brain; Cats; Cimetidine; Digoxin; Female; Pyrilamine; Time Factors

1984
Bile salt-induced gastric mucosal damage and histamine receptor antagonists.
    Gut, 1983, Volume: 24, Issue:1

    Topics: Aminopyridines; Animals; Biological Transport; Cimetidine; Dogs; Gastric Mucosa; Guanidines; Hydrogen-Ion Concentration; Male; Potassium; Pyrilamine; Sodium; Stomach; Taurocholic Acid

1983
Specific binding of [3H]mepyramine to histamine H1-receptors in vascular smooth muscle membranes.
    Agents and actions, 1983, Volume: 13, Issue:2-3

    Topics: Aminopyridines; Animals; Aorta; Cattle; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Tritium

1983
3H-mepyramine binding in various regions of rat brain following chronic treatment with different classes of antidepressant drugs.
    Progress in neuro-psychopharmacology & biological psychiatry, 1982, Volume: 6, Issue:4-6

    Topics: Aminopyridines; Animals; Antidepressive Agents; Brain; Clomipramine; Desipramine; Female; Iprindole; Nomifensine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1

1982
Regional effect of mepyramine on cerebral glucose utilization in conscious rats.
    European journal of pharmacology, 1982, Feb-05, Volume: 77, Issue:4

    Topics: Aminopyridines; Animals; Binding Sites; Brain; Cerebral Cortex; Glucose; Male; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1

1982
The actions of cimetidine hydrochloride and mepyramine maleate in rat adjuvant arthritis.
    European journal of pharmacology, 1982, Feb-26, Volume: 78, Issue:2

    Topics: Aminopyridines; Animals; Arthritis; Arthritis, Experimental; Cimetidine; Guanidines; Male; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H2

1982
Histamine and gastric acid secretion in rabbits: mechanism of inhibition.
    Agents and actions, 1982, Volume: 12, Issue:1-2

    Topics: Aminopyridines; Animals; Blood Pressure; Catecholamines; Gastric Acid; Gastric Mucosa; Histamine; Pyrilamine; Rabbits; Stomach; Time Factors

1982
Distribution and characteristics of histamine H1-receptors in guinea-pig airways identified by [3H]mepyramine.
    European journal of pharmacology, 1982, Jul-09, Volume: 81, Issue:2

    Topics: Aminopyridines; Animals; Brain; Guinea Pigs; In Vitro Techniques; Lung; Male; Pyrilamine; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H1; Sodium; Trachea; Tritium

1982
Histamine H-1 receptors on rat peritoneal mast cells.
    Life sciences, 1982, Nov-01, Volume: 31, Issue:18

    Topics: Aminopyridines; Animals; Ascitic Fluid; Binding, Competitive; Cimetidine; Diphenhydramine; Histamine; Male; Mast Cells; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1

1982
3H-Mepyramine binding to histamine H1-receptors in guinea pig lung: characteristics and regulation by ions.
    Life sciences, 1981, Feb-09, Volume: 28, Issue:6

    Topics: Aminopyridines; Animals; Cations, Divalent; Cations, Monovalent; Cell Membrane; Guinea Pigs; Kinetics; Lung; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Tritium

1981
Temperature dependent receptor interconversion hypothesis: chronotropic histamine receptors in isolated guineapig atria.
    Indian journal of experimental biology, 1980, Volume: 18, Issue:10

    Topics: Aminopyridines; Animals; Atrial Function; Cimetidine; Female; Guanidines; Guinea Pigs; Heart; Heart Atria; Heart Rate; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Temperature

1980
Extended mepyramine treatment and histamine H1-receptors in guinea-pig brain.
    European journal of pharmacology, 1981, May-22, Volume: 71, Issue:4

    Topics: Aminopyridines; Animals; Binding Sites; Blood Pressure; Brain; Guinea Pigs; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Time Factors

1981
High-pressure liquid chromatographic determination of methscopolamine nitrate, phenylpropanolamine hydrochloride, pyrilamine maleate, and pheniramine maleate in tablets.
    Journal of pharmaceutical sciences, 1981, Volume: 70, Issue:7

    Topics: Aminopyridines; Chromatography, High Pressure Liquid; Drug Combinations; Drug Stability; N-Methylscopolamine; Pheniramine; Phenylpropanolamine; Pyrilamine; Scopolamine Derivatives; Tablets

1981
GLC analysis of menthol, phenol, benzocaine, and pyrilamine maleate in aerosol spray lotion.
    Journal of pharmaceutical sciences, 1981, Volume: 70, Issue:10

    Topics: Aerosols; Aminopyridines; Benzocaine; Chromatography, Gas; Menthol; Phenol; Phenols; Pyrilamine

1981
A fatal case involving pyrilamine.
    Clinical toxicology, 1981, Volume: 18, Issue:8

    Topics: Adult; Aminopyridines; Female; Humans; Pyrilamine; Suicide

1981
Histamine H1-receptor binding sites in guinea pig brain membranes: regulation of agonist interactions by guanine nucleotides and cations.
    Journal of neurochemistry, 1980, Volume: 34, Issue:4

    Topics: Aminopyridines; Animals; Binding, Competitive; Brain; Cations, Divalent; Guanine Nucleotides; Guinea Pigs; Kinetics; Male; Osmolar Concentration; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Ribonucleotides; Structure-Activity Relationship

1980
Simultaneous GLC analysis of salicylamide, phenylpropanolamine hydrochloride, caffeine, chlorpheniramine maleate, phenylephrine hydrochloride, and pyrilamine maleate in capsule preparations.
    Journal of pharmaceutical sciences, 1980, Volume: 69, Issue:7

    Topics: Aminopyridines; Caffeine; Capsules; Chlorpheniramine; Chromatography, Gas; Phenylephrine; Phenylpropanolamine; Pyrilamine; Salicylamides

1980
Serotonergic and histaminergic mechanisms involved in intralipid drinking?
    Pharmacology, biochemistry, and behavior, 2003, Volume: 76, Issue:2

    Topics: Aminopyridines; Animals; Cyproheptadine; Dietary Fats; Dose-Response Relationship, Drug; Drinking Behavior; Eating; Histamine; Histamine H1 Antagonists; Hyperphagia; Indoles; Male; Metergoline; Pyrilamine; Rats; Serotonin; Serotonin Antagonists

2003