alpha-aminopyridine has been researched along with pyrilamine in 108 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 98 (90.74) | 18.7374 |
1990's | 9 (8.33) | 18.2507 |
2000's | 1 (0.93) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Hill, SJ; Marrian, DH; Sanders, JK; Young, JM | 1 |
Duchemin, AM; Quach, TT; Rose, C; Schwartz, JC | 2 |
Chang, RS; Snyder, SH; Tran, VT | 2 |
Al-Haboubi, HA; Zeitlin, IJ | 2 |
Gerner, T; Haffner, JF; Norstein, J | 1 |
Ayres, JW; Block, JH; Levine, HL | 1 |
Hill, SJ; Young, JM | 2 |
Kuhar, MJ; Palacios, JM; Young, WS | 1 |
Cho, CH; Ogle, CW | 1 |
Emson, PC; Hill, SJ; Young, JM | 1 |
Go, K; Namimatsu, A; Okuda, M; Tanimoto, H | 1 |
Bach, JF; Chatenoud, LM; Villemain, FM | 1 |
Ahluwalia, M; Bazan, E; Garver, D; Gruenstein, E; Johnson, CG; Johnson, CL | 1 |
Bloom, J; Freeman, JP; Getek, TA; Holder, CL; Korfmacher, WA | 1 |
Chand, N; Diamantis, W; Hess, FG; McGee, J; Nolan, K; Sofia, RD | 1 |
Khateb, A; Mühlethaler, M; Serafin, M | 1 |
Ido, T; Ishiwata, K; Itoh, M; Matsuzawa, T; Watanabe, T; Yagi, N; Yanai, K | 1 |
Bast, A; Leurs, R; Timmerman, H | 2 |
Donnelly, A; Gellhaus, M; Weiler, JM; Weiler, K | 1 |
Anuka, JA; Thomas, PJ; Walker, J | 1 |
Friedberg, KD; Sekardi, L | 1 |
Fukui, H; Inagaki, N; Taguchi, Y; Wada, H; Wang, NP; Yamatodani, A | 1 |
Mitsuhashi, M; Payan, DG | 1 |
Ruat, M; Schwartz, JC | 1 |
Fukui, H; Sawai, S; Tanaka, F; Wada, H; Wang, NP | 1 |
Dannals, RF; Ravert, HT; Scheffel, U; Tanada, S; Wagner, HN; Wilson, AA; Yanai, K | 2 |
Guo, ZG; Qiu, R | 1 |
Donoso, AO; Seltzer, AM | 1 |
Inoue, T; Kannan, MS | 1 |
Hsu, FL; Munavalli, S; Yeh, SY | 1 |
White, JM | 1 |
Kovatch, RM; Lijinsky, W | 1 |
Ahn, HS; Barnett, A | 1 |
Baker, CH; Davis, DL; Lindsey, BG; Sutton, ET | 1 |
Maslinski, C; Nowak, JZ | 1 |
Alvarez, EO; Banzán, AM | 1 |
Feit, F; Freedberg, RS; Friedman, GR; Palu, RN | 1 |
Bevan, J; Heptinstall, S | 2 |
Bouthenet, ML; Garbarg, M; Ruat, M; Sales, N; Schwartz, JC | 1 |
Treherne, JM; Young, JM | 1 |
Awadhiya, RP; Pillai, AG; Vegad, JL | 1 |
Rosenthal, MD; Williams, PB | 1 |
Ganellin, CR; Garbarg, M; Gros, C; Körner, M; Ruat, M; Schwartz, JC; Tertiuk, W | 1 |
Fukui, H; Wada, H; Wang, NP; Watanabe, T | 1 |
Betowski, LD; Holder, CL; Korfmacher, WA; Mitchum, RK | 1 |
Bach, JF; Cazenave, PA; Chatenoud, L; Ganellin, CR; Garbarg, M; Gros, C; Hoebeke, J; Korner, M; Ruat, M; Villemain, F | 1 |
Chen, J; Johnson, L; Spada, C; Woodward, DF | 1 |
Charap, A; Duzman, E; Leon, J; Shen, CD | 1 |
Ahmed, Ael H; el-Gizawy, SM | 1 |
Driver, AG; Mustafa, SJ | 1 |
Clive, D; Hozier, JC; Sawyer, JR; Turner, NT; Woolley, JL | 1 |
Bielkiewicz-Vollrath, B; Cook, DA | 1 |
Butkow, N; Gelgor, L; Mitchell, D; Phillips, S | 1 |
Marshall, K; Senior, J | 1 |
Bielkiewicz, B; Cook, DA | 2 |
Bouthenet, ML; Ganellin, CR; Garbarg, M; Gros, C; Ife, RJ; Korner, M; Sales, N; Schwartz, JC | 1 |
Eisenbrand, G; Habs, M; Shubik, P | 1 |
Arbonés, L; Claro, E; García, A; Picatoste, F | 1 |
Kanaide, H; Miwa, N; Nakamura, M; Nishimura, J | 1 |
Katayama, S; Tasaka, K | 1 |
Fujisawa, S; Nakai, K; Ohmiya, Y | 1 |
Daum, P; Hill, SJ; Young, JM | 1 |
Brossard, M | 1 |
Wallace, RM; Young, JM | 1 |
Hoffman, LH; Hoos, PC | 1 |
Coutts, II; Gibbs, CJ; Jackson, SM; White, RJ | 1 |
Hösli, E; Hösli, L; Schneider, U; Wiget, W | 1 |
Azuma, Y | 1 |
Andersen, V; Geisler, A; Klysner, R; Manthorpe, R; Nielsen, H; Norn, S; Permin, H; Petersen, J; Skov, PS; Wiik, A | 1 |
Bank, L; Bortz, D; Lipschitz, E; Marks, IN | 1 |
Del Soldato, P | 1 |
Chiou, GC; Miyano, K | 1 |
Haley, TJ | 1 |
Donoghue, ER; Kurland, ML; Lin, RL; Schaffer, MI; Stein, RJ; Wu Chen, NB | 1 |
Alvarez, EO | 1 |
Amerini, S; Bennardini, F; Franconi, F; Ledda, F; Mantelli, L; Matucci, R; Mugelli, A; Sorbi, C | 1 |
Lijinsky, W | 1 |
Hadfield, AJ; Hill, SJ; Robinson, NR | 1 |
Boertje, SB; Domer, FR; Sweeney, SA | 1 |
Godfraind, T; Miller, RC | 1 |
Elias, MS; Evans, PD; Lummis, SC | 1 |
Hui, HW; Robinson, JR; Zeleznick, L | 1 |
Tayal, G; Tripathi, KD | 2 |
Carter, DC; Lewi, HJ | 1 |
Dupont, A; Merand, Y; Savard, P | 1 |
Gross, PM; Harper, AM; Teasdale, GH | 1 |
Maśliński, S; Pruszyński, JP; Stajniak, A | 1 |
Carswell, H; Nahorski, SR | 1 |
Hunt, WA; Kaliner, M; Wescott, SL | 1 |
Lombroso, M; Nicosia, S | 1 |
Hiley, CR; Hill, SJ; Young, JM | 1 |
Heidemann, DR | 1 |
De Fabrizio, F | 2 |
Johnson, GR | 1 |
Chang, RS; Synder, SH | 1 |
Krabbe, AA; Olesen, J | 1 |
Clifton, PG; Hartfield, AW; Moore, NA | 1 |
1 review(s) available for alpha-aminopyridine and pyrilamine
Article | Year |
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Physical and biological properties of pyrilamine.
Topics: Aminopyridines; Animals; Carcinogens; Chemical Phenomena; Chemistry; Chemistry, Physical; Humans; Immunity; Kinetics; Mutagens; Nervous System Diseases; Pyrilamine; Structure-Activity Relationship; Teratogens; Time Factors | 1983 |
5 trial(s) available for alpha-aminopyridine and pyrilamine
Article | Year |
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Randomized, double-blind, parallel groups, placebo-controlled study of efficacy and safety of Rynatan in the treatment of allergic rhinitis using an acute model.
Topics: Adolescent; Adult; Aged; Aminopyridines; Chlorpheniramine; Double-Blind Method; Drug Combinations; Humans; Middle Aged; Phenylephrine; Placebos; Pyrilamine; Rhinitis, Allergic, Seasonal | 1990 |
Efficacy of cimetidine/pyrilamine eyedrops. A dose response study with histamine challenge.
Topics: Adult; Aminopyridines; Cimetidine; Clinical Trials as Topic; Dose-Response Relationship, Drug; Drug Combinations; Eye; Eye Diseases; Female; Histamine; Humans; Hyperemia; Hypersensitivity; Male; Ophthalmic Solutions; Pyrilamine | 1986 |
Skin test wheal size and erythema not reduced by topical antihistamine.
Topics: Administration, Topical; Aminopyridines; Clinical Trials as Topic; Double-Blind Method; Erythema; Histamine H1 Antagonists; Humans; Hypersensitivity, Immediate; Pruritus; Pyrilamine; Skin Tests | 1983 |
Effect of mepyramine on the untoward side-effects of impromidine.
Topics: Aminopyridines; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Drug Interactions; Female; Flushing; Gastric Acid; Humans; Imidazoles; Impromidine; Male; Middle Aged; Pulse; Pyrilamine; Random Allocation; Receptors, Histamine; Receptors, Histamine H2 | 1984 |
Headache provocation by continuous intravenous infusion of histamine. Clinical results and receptor mechanisms.
Topics: Aminopyridines; Cimetidine; Headache; Histamine; Humans; Migraine Disorders; Pyrilamine | 1980 |
102 other study(ies) available for alpha-aminopyridine and pyrilamine
Article | Year |
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A convenient synthesis of [3H]mepyramine and certain related [3H]antihistamines.
Topics: Aminopyridines; Chemical Phenomena; Chemistry; Histamine H1 Antagonists; Isotope Labeling; Methapyrilene; Methods; Pyrilamine; Tripelennamine; Tritium | 1978 |
In vivo occupation of cerebral histamine H1-receptors evaluated with 3H-mepyramine may predict sedative properties of psychotropic drugs.
Topics: Aminopyridines; Animals; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Cerebral Cortex; Hypnotics and Sedatives; Mice; Psychotropic Drugs; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1 | 1979 |
Characteristics of histamine H1-receptors in peripheral tissues labeled with [3H]mepyramine.
Topics: Adrenal Glands; Aminopyridines; Animals; Aorta; Guinea Pigs; Haplorhini; Ileum; In Vitro Techniques; Lung; Macaca fascicularis; Male; Mice; Muscle, Smooth; Myocardium; Organ Specificity; Pyrilamine; Rabbits; Rats; Receptors, Histamine; Receptors, Histamine H1; Species Specificity | 1979 |
The actions of cimetidine, mepyramine, indomethacin and aprotinin (Trasylol) on the inflammatory response in adjuvant rats [proceedings].
Topics: Aminopyridines; Animals; Aprotinin; Arthritis; Arthritis, Experimental; Cimetidine; Guanidines; Indomethacin; Male; Pyrilamine; Rats | 1979 |
The effects of mepyramine and cimetidine on the motor responses to histamine, cholecystokinin, and gastrin in the fundus and antrum of isolated guinea-pig stomachs.
Topics: Acetylcholine; Aminopyridines; Animals; Cholecystokinin; Cimetidine; Female; Gastrins; Gastrointestinal Motility; Guanidines; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Pressure; Pyloric Antrum; Pyrilamine | 1979 |
Paired-ion reversed-phase high-pressure liquid chromatographic assay of pentobarbital-pyrilamine suppositories.
Topics: Aminopyridines; Chromatography, Gas; Chromatography, High Pressure Liquid; Drug Combinations; Methods; Pentobarbital; Pyrilamine; Suppositories | 1979 |
Heterogeneity of histamine H1-receptors: species variations in [3H]mepyramine binding of brain membranes.
Topics: Aminopyridines; Animals; Binding, Competitive; Brain; Cell Membrane; Cerebral Cortex; Guinea Pigs; Hippocampus; Humans; Kinetics; Male; Mice; Pyrilamine; Rabbits; Rats; Receptors, Histamine H1; Species Specificity | 1979 |
The binding properties of [3H]-mepyramine in the brain of the guinea-pig and the rat [proceedings].
Topics: Aminopyridines; Animals; Brain; Guinea Pigs; Pyrilamine; Rats; Species Specificity | 1979 |
Autoradiographic localization of H1-histamine receptors in brain using 3H-mepyramine: preliminary studies.
Topics: Aminopyridines; Animals; Autoradiography; Brain; Cerebellum; Guinea Pigs; Kinetics; Male; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Time Factors | 1979 |
Histamine H1- and H2-receptor-mediated gastric microcirculatory effects in the aetiology of stress ulceration in the rat stomach.
Topics: Aminopyridines; Animals; Dose-Response Relationship, Drug; Gastric Mucosa; Humans; Male; Mast Cells; Metiamide; Microcirculation; Pyrilamine; Rats; Receptors, Histamine; Stomach Ulcer; Stress, Psychological; Thiourea | 1978 |
The binding of [3H]mepyramine to histamine H1 receptors in guinea-pig brain.
Topics: Aminopyridines; Animals; Brain; Cerebellum; Guinea Pigs; Promethazine; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1 | 1978 |
Mechanism of nasal secretion mediated via nerve reflex in guinea pigs and evaluation of antiallergic drugs.
Topics: Allergens; Aminopyridines; Animals; Atropine Derivatives; Bronchodilator Agents; Capsaicin; Ganglionic Blockers; Guinea Pigs; Hexamethonium; Hexamethonium Compounds; Histamine; Hypersensitivity; Lidocaine; Methacholine Chloride; Nasal Mucosa; ortho-Aminobenzoates; Parasympatholytics; Phthalazines; Pyrilamine; Reflex | 1992 |
Characterization of histamine H1 binding sites on human T lymphocytes by means of 125I-iodobolpyramine. Preferential expression of H1 receptors on CD8 T lymphocytes.
Topics: Aminopyridines; Animals; Antigens, Differentiation, T-Lymphocyte; CD4-Positive T-Lymphocytes; CD8 Antigens; Cell Membrane; Cerebellum; Guinea Pigs; Humans; Kinetics; Pyrilamine; Receptors, Histamine H1; Succinimides; T-Lymphocytes; T-Lymphocytes, Helper-Inducer; T-Lymphocytes, Regulatory | 1990 |
Histamine receptors in human fibroblasts: inositol phosphates, Ca2+, and cell growth.
Topics: Aminopyridines; Calcium; Cell Division; Cell Line; DNA Replication; Fibroblasts; Fluorescent Dyes; Histamine; Humans; Inositol Phosphates; Kinetics; Phorbol 12,13-Dibutyrate; Pyrilamine; Receptors, Histamine; Skin; Tetradecanoylphorbol Acetate; Thymidine | 1990 |
Analysis of rat urine for metabolites of pyrilamine via high-performance liquid chromatography/thermospray mass spectrometry and tandem mass spectrometry.
Topics: Aminopyridines; Animals; Biotransformation; Chromatography, High Pressure Liquid; Female; Male; Mass Spectrometry; Molecular Weight; Pyrilamine; Rats; Rats, Inbred F344; Reference Standards; Spectrophotometry, Ultraviolet | 1990 |
Aeroallergen-induced immediate asthmatic responses and late-phase associated pulmonary eosinophilia in the guinea pig: effect of methylprednisolone and mepyramine.
Topics: Administration, Oral; Aerosols; Aminopyridines; Animals; Asthma; Drug Administration Schedule; Guinea Pigs; Methylprednisolone; Ovalbumin; Premedication; Pulmonary Eosinophilia; Pyrilamine | 1990 |
Histamine excites pedunculopontine neurones in guinea pig brainstem slices.
Topics: Action Potentials; Aminopyridines; Animals; Guinea Pigs; Histamine; In Vitro Techniques; Pons; Pyrilamine; Receptors, Histamine; Tetrodotoxin | 1990 |
Specific binding of [3H]pyrilamine to histamine H1 receptors in guinea pig brain in vivo: determination of binding parameters by a kinetic four-compartment model.
Topics: Aminopyridines; Animals; Binding, Competitive; Brain; Cerebellum; Cerebral Cortex; Chlorpheniramine; Corpus Striatum; Guinea Pigs; Hippocampus; Kinetics; Male; Mathematics; Models, Biological; Pyrilamine; Receptors, Histamine H1; Stereoisomerism; Thalamus; Tissue Distribution; Tritium | 1990 |
Labelling of non-H1-receptor binding sites by [3H]-mepyramine on the rat liver plasma membrane.
Topics: Aminopyridines; Animals; Cell Membrane; In Vitro Techniques; Kinetics; Liver; Male; Proteins; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Stereoisomerism | 1990 |
Some effects of oestrogens on [3H]-mepyramine binding in rat brain.
Topics: 1-Methyl-3-isobutylxanthine; Aminopyridines; Animals; Brain; Estrogens; Female; Male; Ovariectomy; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1 | 1986 |
Inhibition of immunological histamine release from guinea pig lungs and other organs by mepyramine, ketotifen, and picumast in vivo.
Topics: Aminopyridines; Anaphylaxis; Animals; Coumarins; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine Release; Ketotifen; Lung; Male; Pyrilamine | 1989 |
High affinity, saturable [3H]mepyramine binding sites on rat liver plasma membrane do not represent histamine H1-receptors. A warning.
Topics: Aminopyridines; Animals; Binding, Competitive; Cell Membrane; Histamine H1 Antagonists; Kinetics; Liver; Male; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Structure-Activity Relationship | 1989 |
Characterization of histamine H1-receptors on astrocytes in primary culture: [3H]mepyramine binding studies.
Topics: Aminopyridines; Animals; Animals, Newborn; Astrocytes; Binding, Competitive; Brain; Cells, Cultured; Histamine H1 Antagonists; In Vitro Techniques; Kinetics; Male; Pyrilamine; Rats; Receptors, Histamine H1 | 1989 |
Solubilization and characterization of the pyrilamine-binding protein from cultured smooth muscle cells.
Topics: Aminopyridines; Animals; Cell Line; Chromatography, Gel; Chromatography, High Pressure Liquid; Kinetics; Molecular Weight; Muscle, Smooth; Polyethylene Glycols; Pyrilamine; Receptors, Histamine H1; Solubility; Substrate Specificity | 1989 |
Photoaffinity labeling and electrophoretic identification of the H1-receptor: comparison of several brain regions and animal species.
Topics: Affinity Labels; Aminopyridines; Animals; Brain; Electrophoresis, Polyacrylamide Gel; Guinea Pigs; Male; Membranes; Mice; Mice, Inbred Strains; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Tissue Distribution | 1989 |
Divalent cations increase the binding capacity of the [3H]mepyramine binding site, a possible histamine H1 receptor, in rat liver membranes.
Topics: Aminopyridines; Animals; Brain; Calcium; Cations; Liver; Male; Membranes; Proteins; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1 | 1989 |
Biodistribution and radiation absorbed dose of (N-methyl[11C])pyrilamine: a histamine H-1 receptor radiotracer.
Topics: Aminopyridines; Animals; Brain; Carbon Radioisotopes; Male; Mice; Pyrilamine; Radiation Dosage; Radionuclide Imaging; Receptors, Histamine H2; Tissue Distribution | 1989 |
Protective effects of histamine H1 and H2 antagonists, adenosine and hydrocortisone on cardiac anaphylaxis.
Topics: Adenosine; Aminopyridines; Anaphylaxis; Animals; Arrhythmias, Cardiac; Cardiac Output; Cimetidine; Guinea Pigs; Heart Rate; Hydrocortisone; In Vitro Techniques; Pyrilamine; Receptors, Histamine | 1989 |
Effects of ovariectomy and ovarian steroids on binding of 3H-mepyramine, an H1-histamine antagonist, in rat hypothalamus.
Topics: Aminopyridines; Animals; Estradiol; Female; Hypothalamus; Luteinizing Hormone; Ovariectomy; Progesterone; Pyrilamine; Radioimmunoassay; Radioligand Assay; Rats; Receptors, Histamine H1 | 1989 |
Nonadrenergic and noncholinergic excitatory neurotransmission in rat intrapulmonary artery.
Topics: Aminopyridines; Animals; Atropine; Electric Stimulation; Guanethidine; In Vitro Techniques; Male; Membrane Potentials; Muscle, Smooth, Vascular; Neuromuscular Junction; Norepinephrine; Phentolamine; Propranolol; Pulmonary Artery; Pyrilamine; Rats; Rats, Inbred Strains; Synaptic Transmission; Tetrodotoxin | 1988 |
O-demethylation of pyrilamine.
Topics: Acids; Aminopyridines; Chemical Phenomena; Chemistry; Dealkylation; Hydrobromic Acid; Pyrilamine | 1988 |
The discriminative stimulus properties of mepyramine.
Topics: Aminopyridines; Animals; Chlorpheniramine; Discrimination, Psychological; Histamine H1 Antagonists; Imipramine; Male; Procaine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Scopolamine | 1985 |
Carcinogenicity studies of some analogs of the carcinogen methapyrilene in F344 rats.
Topics: Aminopyridines; Animals; Female; Histamine H1 Antagonists; Liver Neoplasms; Male; Methapyrilene; Pyridines; Pyrilamine; Rats; Rats, Inbred F344; Rats, Inbred Strains; Structure-Activity Relationship | 1986 |
Selective displacement of [3H]mepyramine from peripheral vs. central nervous system receptors by loratadine, a non-sedating antihistamine.
Topics: Aminopyridines; Animals; Binding, Competitive; Cerebral Cortex; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Kinetics; Loratadine; Lung; Male; Piperidines; Pyrilamine; Receptors, Cell Surface | 1986 |
Adrenergic and histaminergic neural interactions in dog paws.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Aminopyridines; Animals; Blood Pressure; Blood Volume; Capillaries; Dogs; Electric Stimulation; Hindlimb; Metiamide; Pyrilamine; Reference Values; Regional Blood Flow; Sciatic Nerve; Thiourea; Vascular Resistance | 1988 |
3H-mepyramine binding and histamine-stimulated cAMP accumulation in mammalian retina.
Topics: Aminopyridines; Animals; Brain; Cattle; Cyclic AMP; Dopamine; Guinea Pigs; Histamine; In Vitro Techniques; Pyrilamine; Rabbits; Receptors, Histamine; Retina; Tritium | 1986 |
Histamine in dorsal and ventral hippocampus. II. Effects of H1 and H2 histamine antagonists on exploratory behavior in male rats.
Topics: Aminopyridines; Animals; Brain Mapping; Exploratory Behavior; Hippocampus; Histamine; Histidine Decarboxylase; Male; Methylhistidines; Motor Activity; Neural Inhibition; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Synaptic Transmission | 1986 |
Cardiogenic shock due to antihistamine overdose. Reversal with intra-aortic balloon counterpulsation.
Topics: Aminopyridines; Combined Modality Therapy; Epilepsy, Tonic-Clonic; Female; Humans; Intra-Aortic Balloon Pumping; Middle Aged; Pyrilamine; Shock, Cardiogenic; Suicide, Attempted; Sympathomimetics | 1987 |
Serotonin-induced platelet aggregation in whole blood and the effects of ketanserin and mepyramine.
Topics: Aminopyridines; Dose-Response Relationship, Drug; Humans; Ketanserin; Piperidines; Platelet Aggregation; Pyrilamine; Serotonin; Time Factors | 1985 |
A detailed mapping of histamine H1-receptors in guinea-pig central nervous system established by autoradiography with [125I]iodobolpyramine.
Topics: Aminopyridines; Animals; Autoradiography; Brain; Brain Mapping; Guinea Pigs; Pyrilamine; Receptors, Histamine; Spinal Cord; Succinimides | 1988 |
Temperature-dependence of the kinetics of the binding of [3H]-(+)-N-methyl-4-methyldiphenhydramine to the histamine H1-receptor: comparison with the kinetics of [3H]-mepyramine.
Topics: Aminopyridines; Animals; Cerebellum; Guinea Pigs; Histamine Antagonists; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle, Smooth; Pyrilamine; Receptors, Histamine H1; Temperature | 1988 |
Suppression by mepyramine maleate of the increased vascular permeability in passive cutaneous anaphylaxis in the chicken.
Topics: Aminopyridines; Animals; Capillary Permeability; Chickens; Female; Male; Passive Cutaneous Anaphylaxis; Pyrilamine | 1988 |
Ascorbate increases apparent "specific" binding of [3H]pyrilamine to glass fiber filters.
Topics: Aminopyridines; Ascorbic Acid; Binding Sites; Buffers; Filtration; Glass; Ligands; Pyrilamine | 1988 |
(N-methyl-[11C])pyrilamine, a radiotracer for histamine H-1 receptors: radiochemical synthesis and biodistribution study in mice.
Topics: Aminopyridines; Animals; Brain; Brain Chemistry; Carbon Radioisotopes; Isotope Labeling; Male; Mice; Pyrilamine; Radionuclide Imaging; Receptors, Histamine H1; Tissue Distribution | 1988 |
Characterization of histamine H1-receptor binding peptides in guinea pig brain using [125I]iodoazidophenpyramine, an irreversible specific photoaffinity probe.
Topics: Affinity Labels; Aminopyridines; Animals; Cell Membrane; Cerebellum; Electrophoresis, Polyacrylamide Gel; Guinea Pigs; In Vitro Techniques; Mercaptoethanol; Photochemistry; Protease Inhibitors; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1 | 1988 |
Solubilization, characterization and partial purification of [3H]mepyramine-binding protein, a possible histamine H1 receptor, from rat liver membrane.
Topics: Aminopyridines; Animals; Centrifugation, Density Gradient; Chromatography, Gel; Chromatography, High Pressure Liquid; Gamma Rays; In Vitro Techniques; Liver; Male; Molecular Weight; Protein Binding; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Sucrose | 1988 |
Characterization of doxylamine and pyrilamine metabolites via thermospray/mass spectrometry and tandem mass spectrometry.
Topics: Aminopyridines; Animals; Biotransformation; Doxylamine; Female; Macaca mulatta; Male; Mass Spectrometry; Pyridines; Pyrilamine; Rats; Rats, Inbred F344 | 1988 |
Polyclonal and monoclonal antibodies directed against SK & F 94461, a specific H1 histamine receptor ligand.
Topics: Aminopyridines; Animals; Antibodies, Monoclonal; Antibody Affinity; Antibody Specificity; Binding, Competitive; Immunoglobulin Idiotypes; Mice; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Spectrometry, Fluorescence; Spectrophotometry, Ultraviolet; Time Factors | 1988 |
Effect of cimetidine and pyrilamine on histamine-induced ocular surface hyperemia.
Topics: Aminopyridines; Animals; Cimetidine; Drug Therapy, Combination; Eye Diseases; Female; Histamine; Hyperemia; Pyrilamine; Rabbits | 1986 |
High-performance liquid chromatographic determination of mepyramine maleate, pheniramine maleate and phenylpropanolamine hydrochloride in tablets and drops.
Topics: Aminopyridines; Chromatography, High Pressure Liquid; Histamine Antagonists; Pheniramine; Phenylpropanolamine; Pyrilamine; Solutions; Tablets | 1987 |
Correlation of histamine H1 receptor function and [3H]mepyramine binding in porcine tracheal tissue.
Topics: Aminopyridines; Animals; In Vitro Techniques; Models, Biological; Muscle Contraction; Muscle, Smooth; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Swine; Time Factors; Trachea | 1987 |
Methapyrilene is a genotoxic carcinogen: studies on methapyrilene and pyrilamine in the L5178Y/TK +/- mouse lymphoma assay.
Topics: Aminopyridines; Animals; Biotransformation; Carcinogens; Chromosome Aberrations; Leukemia L5178; Methapyrilene; Mice; Microsomes, Liver; Mutagenicity Tests; Neoplasm Proteins; Preservation, Biological; Pyrilamine; Rats; Thymidine Kinase; Tumor Cells, Cultured; Tumor Stem Cell Assay | 1987 |
Binding of 3H-mepyramine to dog portal vein and cerebral cortex.
Topics: Aminopyridines; Animals; Cerebral Cortex; Dogs; In Vitro Techniques; Muscle, Smooth, Vascular; Portal Vein; Pyrilamine; Receptors, Histamine H1 | 1986 |
Injectable aspirin and mepyramine abolish post-ischaemic hyperalgesia in rats.
Topics: Aminopyridines; Animals; Aspirin; Histamine; Hyperalgesia; Hyperesthesia; Ischemia; Male; Prostaglandins; Pyrilamine; Rats; Rats, Inbred Strains | 1986 |
The effect of mepyramine and ranitidine on the oestrogen and anti-oestrogen stimulated rat uterus.
Topics: Aminopyridines; Animals; Estrogen Antagonists; Estrogens; Female; Organ Size; Pyrilamine; Ranitidine; Rats; Receptors, Histamine; Regional Blood Flow; Tamoxifen; Uterine Contraction; Uterus | 1986 |
The binding of [3H]mepyramine to histamine H1 receptors in monkey brain.
Topics: Aminopyridines; Animals; Brain; Haplorhini; In Vitro Techniques; Kinetics; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1 | 1985 |
[125I]Iodobolpyramine, a highly sensitive probe for histamine H1-receptors in guinea-pig brain.
Topics: Aminopyridines; Animals; Autoradiography; Brain; Cerebellum; Guinea Pigs; In Vitro Techniques; Indicators and Reagents; Iodine Radioisotopes; Kinetics; Male; Membranes; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Succinimides | 1986 |
Carcinogenicity of methapyrilene hydrochloride, mepyramine hydrochloride, thenyldiamine hydrochloride, and pyribenzamine hydrochloride in Sprague-Dawley rats.
Topics: Adenoma; Adrenal Gland Neoplasms; Aminopyridines; Animals; Dose-Response Relationship, Drug; Female; Liver Neoplasms; Liver Neoplasms, Experimental; Male; Methapyrilene; Neoplasms, Experimental; Pyridines; Pyrilamine; Rats; Structure-Activity Relationship; Tripelennamine | 1986 |
[3H]mepyramine binding to histamine H1 receptors in bovine retina.
Topics: Aminopyridines; Animals; Binding, Competitive; Cattle; Kinetics; Pyrilamine; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H1; Retina | 1986 |
Specific binding of [3H] mepyramine to histamine H1-receptors in the sarcolemma from porcine aorta and coronary artery.
Topics: Aminopyridines; Animals; Aorta; Centrifugation, Density Gradient; Coronary Vessels; Kinetics; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Sarcolemma; Subcellular Fractions; Swine | 1985 |
Effects of H1-receptor blocking drugs on the frog sartorius neuromuscular junction.
Topics: Action Potentials; Aminopyridines; Animals; Diphenhydramine; Dose-Response Relationship, Drug; Electric Conductivity; Electrophysiology; Membrane Potentials; Neuromuscular Junction; Perfusion; Promethazine; Pyrilamine; Ranidae; Receptors, Histamine; Receptors, Histamine H1; Time Factors | 1985 |
Comparison of pulmonary accumulation of pyrilamine and pyrilamine N-oxide.
Topics: Aminopyridines; Animals; Cyclic N-Oxides; In Vitro Techniques; Kinetics; Lung; Male; Mice; Mice, Inbred ICR; Pyrilamine | 1985 |
Characterization of [3H]mepyramine binding to the longitudinal muscle of guinea pig small intestine.
Topics: Aminopyridines; Animals; Binding Sites; Calcium; Guinea Pigs; Histamine; Histamine H1 Antagonists; Hydrogen-Ion Concentration; In Vitro Techniques; Intestine, Small; Magnesium; Male; Muscle, Smooth; Pyrilamine; Receptors, Histamine H1 | 1981 |
Affinities of histamine H1-antagonists in guinea pig brain: similarity of values determined from [3H]mepyramine binding and from inhibition of a functional response.
Topics: Aminopyridines; Animals; Binding, Competitive; Brain; Female; Guinea Pigs; Histamine H1 Antagonists; Kinetics; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Structure-Activity Relationship | 1981 |
Rabbits infested with adult Ixodes ricinus L.: effects of mepyramine on acquired resistance.
Topics: Aminopyridines; Animals; Female; Histamine H1 Antagonists; Immunity, Innate; Male; Oviposition; Pyrilamine; Rabbits; Tick Infestations; Ticks | 1982 |
Labeling of histamine H1-receptors in the brain of the living mouse.
Topics: Aminopyridines; Animals; Binding Sites; Binding, Competitive; Brain; Histamine H1 Antagonists; Male; Mice; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1 | 1980 |
Temperature dependence of the binding of [3H]mepyramine and related compounds to the histamine H1 receptor.
Topics: Aminopyridines; Animals; Cerebellum; Chlorpromazine; Guinea Pigs; Histamine H1 Antagonists; Kinetics; Male; Phenothiazines; Promethazine; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Temperature; Tripelennamine | 1983 |
Effect of histamine receptor antagonists and indomethacin on implantation in the rabbit.
Topics: Aminopyridines; Animals; Capillary Permeability; Cimetidine; Drug Combinations; Drug Interactions; Embryo Implantation; Female; Histamine H1 Antagonists; Indomethacin; Pregnancy; Pyrilamine; Rabbits; Uterus | 1983 |
Evidence for the existence of histamine H1- and H2-receptors on astrocytes of cultured rat central nervous system.
Topics: Aminopyridines; Animals; Astrocytes; Brain Stem; Cells, Cultured; Cimetidine; Histamine; Histamine H1 Antagonists; Membrane Potentials; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Spinal Cord; Thiazoles | 1984 |
[Pharmacological studies on rat passive cutaneous anaphylaxis (PCA) (author's transl)].
Topics: Aminopyridines; Aminopyrine; Animals; Benzydamine; Cyclic AMP; Epinephrine; Histamine Release; Isoproterenol; Male; Passive Cutaneous Anaphylaxis; Pyrilamine; Rabbits; Rats; Tissue Distribution | 1980 |
Possible role of histamine in rheumatoid arthritis. Treatment with cimetidine and mepyramine.
Topics: Adolescent; Adult; Aminopyridines; Arthritis, Rheumatoid; Cimetidine; Drug Therapy, Combination; Female; Guanidines; Histamine H1 Antagonists; Histamine Release; Humans; Male; Middle Aged; Pyrilamine | 1981 |
Studies with specific agonists and antagonists of the role of histamine H1- and H2-receptor activation in the pathogenesis of gastric lesions in rats.
Topics: Aminopyridines; Animals; Atropine; Dimaprit; Drug Interactions; Female; Histamine; Pyridines; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach Ulcer; Thiourea | 1984 |
Pharmacological prevention of ocular inflammation induced by lens proteins.
Topics: Aminopyridines; Animals; Catechols; Cimetidine; Crystallins; Disease Models, Animal; Drug Therapy, Combination; Endophthalmitis; Female; Indomethacin; Masoprocol; Pyrilamine; Rabbits | 1984 |
The general toxicology unknown. II. A case report: doxylamine and pyrilamine intoxication.
Topics: Adult; Aminopyridines; Chromatography, Gas; Doxylamine; Gas Chromatography-Mass Spectrometry; Humans; Immunoenzyme Techniques; Male; Mass Spectrometry; Pyridines; Pyrilamine; Spectrophotometry; Suicide; Toxicology | 1983 |
Effects of histamine antagonists injected in the preoptic-anterior hypothalamic area on the prolactin surge induced by estrogen in ovariectomized rats.
Topics: Aminopyridines; Animals; Castration; Circadian Rhythm; Drug Implants; Estrogens; Female; Hypothalamus, Anterior; Metiamide; Preoptic Area; Prolactin; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea | 1984 |
Specific and non-specific displaceable binding of 3H-mepyramine to homogenates of monkey cortex.
Topics: Aminopyridines; Animals; Binding, Competitive; Cerebral Cortex; Haplorhini; In Vitro Techniques; Pyrilamine | 1984 |
On the presence of H1-receptors in various sections of guinea-pig heart: a correlation between binding and functional studies.
Topics: Aminopyridines; Animals; Binding Sites; Guinea Pigs; Heart Atria; Heart Ventricles; In Vitro Techniques; Male; Membranes; Myocardium; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1 | 1984 |
Chronic toxicity tests of pyrilamine maleate and methapyrilene hydrochloride in F344 rats.
Topics: Aminopyridines; Animals; Carcinogens; Diet; Dose-Response Relationship, Drug; Female; Liver Neoplasms; Male; Methapyrilene; Pyrilamine; Rats; Rats, Inbred F344; Structure-Activity Relationship; Time Factors | 1984 |
Effects of ketanserin and mepyramine on platelet aggregation and on the uptake of 5-hydroxytryptamine into platelets.
Topics: Adenosine Diphosphate; Aminopyridines; Blood Platelets; Humans; Ketanserin; Piperidines; Platelet Aggregation; Pyrilamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1983 |
The nature of the binding of [3H]mepyramine to homogenates of guinea-pig cerebral cortex at different [3H]ligand concentrations.
Topics: Aminopyridines; Animals; Cerebral Cortex; Guinea Pigs; In Vitro Techniques; Kinetics; Pyrilamine; Receptors, Histamine H1; Tritium | 1983 |
Blockade of the acetylcholine-and histamine-induced changes in the permeability of the blood-brain barrier of normotensive and spontaneously hypertensive rats by atropine and pyrilamine.
Topics: Acetylcholine; Aminopyridines; Animals; Atropine; Blood Pressure; Blood-Brain Barrier; Female; Histamine; Hypertension; Male; Pyrilamine; Rats; Rats, Inbred Strains | 1983 |
Effects of histamine and the histamine antagonists mepyramine and cimetidine on human coronary arteries in vitro.
Topics: Adolescent; Adult; Aged; Aminopyridines; Child; Cimetidine; Coronary Vessels; Histamine; Humans; In Vitro Techniques; Middle Aged; Muscle Contraction; Muscle Relaxation; Potassium; Pyrilamine | 1983 |
[3H]mepyramine binding sites in the optic lobe of the locust: autoradiographic and pharmacological studies.
Topics: Aminopyridines; Animals; Autoradiography; Binding Sites; Binding, Competitive; Grasshoppers; Kinetics; Optic Lobe, Nonmammalian; Pyrilamine; Tritium | 1984 |
Ocular disposition of topically applied histamine, cimetidine, and pyrilamine in the albino rabbit.
Topics: Administration, Topical; Aminopyridines; Animals; Aqueous Humor; Biological Availability; Ciliary Body; Cimetidine; Conjunctiva; Cornea; Eye; Histamine; Iris; Male; Pyrilamine; Rabbits | 1984 |
Histamine antagonists modify systemic digoxin cardiotoxicity by their central action.
Topics: Aminopyridines; Animals; Arrhythmias, Cardiac; Brain; Cats; Cimetidine; Digoxin; Female; Pyrilamine; Time Factors | 1984 |
Bile salt-induced gastric mucosal damage and histamine receptor antagonists.
Topics: Aminopyridines; Animals; Biological Transport; Cimetidine; Dogs; Gastric Mucosa; Guanidines; Hydrogen-Ion Concentration; Male; Potassium; Pyrilamine; Sodium; Stomach; Taurocholic Acid | 1983 |
Specific binding of [3H]mepyramine to histamine H1-receptors in vascular smooth muscle membranes.
Topics: Aminopyridines; Animals; Aorta; Cattle; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Tritium | 1983 |
3H-mepyramine binding in various regions of rat brain following chronic treatment with different classes of antidepressant drugs.
Topics: Aminopyridines; Animals; Antidepressive Agents; Brain; Clomipramine; Desipramine; Female; Iprindole; Nomifensine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1 | 1982 |
Regional effect of mepyramine on cerebral glucose utilization in conscious rats.
Topics: Aminopyridines; Animals; Binding Sites; Brain; Cerebral Cortex; Glucose; Male; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1 | 1982 |
The actions of cimetidine hydrochloride and mepyramine maleate in rat adjuvant arthritis.
Topics: Aminopyridines; Animals; Arthritis; Arthritis, Experimental; Cimetidine; Guanidines; Male; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H2 | 1982 |
Histamine and gastric acid secretion in rabbits: mechanism of inhibition.
Topics: Aminopyridines; Animals; Blood Pressure; Catecholamines; Gastric Acid; Gastric Mucosa; Histamine; Pyrilamine; Rabbits; Stomach; Time Factors | 1982 |
Distribution and characteristics of histamine H1-receptors in guinea-pig airways identified by [3H]mepyramine.
Topics: Aminopyridines; Animals; Brain; Guinea Pigs; In Vitro Techniques; Lung; Male; Pyrilamine; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H1; Sodium; Trachea; Tritium | 1982 |
Histamine H-1 receptors on rat peritoneal mast cells.
Topics: Aminopyridines; Animals; Ascitic Fluid; Binding, Competitive; Cimetidine; Diphenhydramine; Histamine; Male; Mast Cells; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1 | 1982 |
3H-Mepyramine binding to histamine H1-receptors in guinea pig lung: characteristics and regulation by ions.
Topics: Aminopyridines; Animals; Cations, Divalent; Cations, Monovalent; Cell Membrane; Guinea Pigs; Kinetics; Lung; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Tritium | 1981 |
Temperature dependent receptor interconversion hypothesis: chronotropic histamine receptors in isolated guineapig atria.
Topics: Aminopyridines; Animals; Atrial Function; Cimetidine; Female; Guanidines; Guinea Pigs; Heart; Heart Atria; Heart Rate; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Temperature | 1980 |
Extended mepyramine treatment and histamine H1-receptors in guinea-pig brain.
Topics: Aminopyridines; Animals; Binding Sites; Blood Pressure; Brain; Guinea Pigs; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Time Factors | 1981 |
High-pressure liquid chromatographic determination of methscopolamine nitrate, phenylpropanolamine hydrochloride, pyrilamine maleate, and pheniramine maleate in tablets.
Topics: Aminopyridines; Chromatography, High Pressure Liquid; Drug Combinations; Drug Stability; N-Methylscopolamine; Pheniramine; Phenylpropanolamine; Pyrilamine; Scopolamine Derivatives; Tablets | 1981 |
GLC analysis of menthol, phenol, benzocaine, and pyrilamine maleate in aerosol spray lotion.
Topics: Aerosols; Aminopyridines; Benzocaine; Chromatography, Gas; Menthol; Phenol; Phenols; Pyrilamine | 1981 |
A fatal case involving pyrilamine.
Topics: Adult; Aminopyridines; Female; Humans; Pyrilamine; Suicide | 1981 |
Histamine H1-receptor binding sites in guinea pig brain membranes: regulation of agonist interactions by guanine nucleotides and cations.
Topics: Aminopyridines; Animals; Binding, Competitive; Brain; Cations, Divalent; Guanine Nucleotides; Guinea Pigs; Kinetics; Male; Osmolar Concentration; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Ribonucleotides; Structure-Activity Relationship | 1980 |
Simultaneous GLC analysis of salicylamide, phenylpropanolamine hydrochloride, caffeine, chlorpheniramine maleate, phenylephrine hydrochloride, and pyrilamine maleate in capsule preparations.
Topics: Aminopyridines; Caffeine; Capsules; Chlorpheniramine; Chromatography, Gas; Phenylephrine; Phenylpropanolamine; Pyrilamine; Salicylamides | 1980 |
Serotonergic and histaminergic mechanisms involved in intralipid drinking?
Topics: Aminopyridines; Animals; Cyproheptadine; Dietary Fats; Dose-Response Relationship, Drug; Drinking Behavior; Eating; Histamine; Histamine H1 Antagonists; Hyperphagia; Indoles; Male; Metergoline; Pyrilamine; Rats; Serotonin; Serotonin Antagonists | 2003 |