Page last updated: 2024-08-21

alpha-aminopyridine and bay-68-4986

alpha-aminopyridine has been researched along with bay-68-4986 in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (16.67)29.6817
2010's4 (66.67)24.3611
2020's1 (16.67)2.80

Authors

AuthorsStudies
Elzein, E; Zablocki, J1
Agrawal, R; Bednarkiewicz, Z; Czarnecka, D; Gaszewska-Żurek, E; Jankowska, E; Kawecka-Jaszcz, K; Krzemińska-Pakuła, M; Ochan Kilama, M; Parma, Z; Ponikowski, P; Sosnowski, M; Tendera, M1
Albrecht-Küpper, BE; Diedrichs, N; Gupta, RC; Kohli, S; Rastogi, S; Sabbah, HN; Wang, M; Zhang, K; Zimmermann, K1
Guo, D; Heitman, LH; IJzerman, AP; Lenselink, EB; Louvel, J; Mocking, TA; Mulder-Krieger, T; Soethoudt, M1
Albrecht-Küpper, B; Dinh, W; Gheorghiade, M; Sabbah, HN; van der Laan, M; Voors, AA1
Cooper, SL; Hill, SJ; Jörg, M; March, J; Sabbatini, AR; Scammells, PJ; Woolard, J1

Reviews

2 review(s) available for alpha-aminopyridine and bay-68-4986

ArticleYear
A1 adenosine receptor agonists and their potential therapeutic applications.
    Expert opinion on investigational drugs, 2008, Volume: 17, Issue:12

    Topics: Adenosine A1 Receptor Agonists; Aminopyridines; Angina Pectoris; Animals; Anti-Arrhythmia Agents; Humans; Insulin; Pain; Receptor, Adenosine A1; Thiazoles

2008
Partial Adenosine A1 Agonist in Heart Failure.
    Handbook of experimental pharmacology, 2017, Volume: 243

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Aminopyridines; Angina Pectoris; Animals; Anti-Arrhythmia Agents; Coronary Artery Disease; Diabetes Mellitus; Dipeptides; Drug Partial Agonism; Furans; Heart; Heart Failure; Humans; Insulin Resistance; Ischemic Preconditioning, Myocardial; Lipolysis; Mitochondria, Heart; Myocardium; Oxygen Consumption; Pyridines; Renal Insufficiency; Tachycardia, Supraventricular; Thiazoles

2017

Trials

1 trial(s) available for alpha-aminopyridine and bay-68-4986

ArticleYear
The new oral adenosine A1 receptor agonist capadenoson in male patients with stable angina.
    Clinical research in cardiology : official journal of the German Cardiac Society, 2012, Volume: 101, Issue:7

    Topics: Adenosine A1 Receptor Agonists; Administration, Oral; Adult; Aged; Aminopyridines; Analysis of Variance; Angina, Stable; Dose-Response Relationship, Drug; Double-Blind Method; Exercise Test; Exercise Tolerance; Heart Rate; Humans; Male; Middle Aged; Poland; Receptor, Adenosine A1; Sex Factors; Thiazoles; Time Factors; Treatment Outcome

2012

Other Studies

3 other study(ies) available for alpha-aminopyridine and bay-68-4986

ArticleYear
Chronic therapy with a partial adenosine A1-receptor agonist improves left ventricular function and remodeling in dogs with advanced heart failure.
    Circulation. Heart failure, 2013, Volume: 6, Issue:3

    Topics: Adenosine A1 Receptor Agonists; Aminopyridines; Animals; Dogs; Echocardiography, Doppler; Heart Failure; Hemodynamics; Stroke Volume; Thiazoles; Ventricular Function, Left; Ventricular Pressure; Ventricular Remodeling

2013
Structure-kinetics relationships of Capadenoson derivatives as adenosine A1 receptor agonists.
    European journal of medicinal chemistry, 2015, Aug-28, Volume: 101

    Topics: Adenosine A1 Receptor Agonists; Aminopyridines; Dose-Response Relationship, Drug; Humans; Kinetics; Models, Molecular; Molecular Structure; Receptor, Adenosine A1; Structure-Activity Relationship; Thiazoles

2015
The effect of two selective A
    British journal of pharmacology, 2020, Volume: 177, Issue:2

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Agonists; Aminopyridines; Animals; Cardiovascular System; Consciousness; Drug Partial Agonism; Heart Rate; Hemodynamics; Ligands; Male; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Regional Blood Flow; Thiazoles; Thiophenes

2020