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alpha-aminopyridine and almorexant

alpha-aminopyridine has been researched along with almorexant in 2 studies

Research

Studies (2)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	0 (0.00)	18.2507
2000's	0 (0.00)	29.6817
2010's	2 (100.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Bissantz, C; Kratzeisen, C; Malherbe, P; Marcuz, A; Roche, O; Wettstein, JG	1
Brown, J; Langmead, CJ; Marshall, FH; Mould, R	1

Other Studies

2 other study(ies) available for alpha-aminopyridine and almorexant

Article	Year
Mapping the binding pocket of dual antagonist almorexant to human orexin 1 and orexin 2 receptors: comparison with the selective OX1 antagonist SB-674042 and the selective OX2 antagonist N-ethyl-2-[(6-methoxy-pyridin-3-yl)-(toluene-2-sulfonyl)-amino]-N-py Molecular pharmacology, 2010, Volume: 78, Issue:1 Topics: Acetamides; Amino Acid Sequence; Aminopyridines; Binding Sites; Cell Line; Humans; Isoquinolines; Molecular Sequence Data; Mutagenesis, Site-Directed; Orexin Receptors; Pyrrolidines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sequence Homology, Amino Acid; Sulfonamides; Thiazoles	2010
Binding kinetics differentiates functional antagonism of orexin-2 receptor ligands. British journal of pharmacology, 2014, Volume: 171, Issue:2 Topics: Acetamides; Algorithms; Aminopyridines; Animals; Binding, Competitive; CHO Cells; Cricetulus; HEK293 Cells; Humans; Inositol Phosphates; Isoquinolines; Kinetics; Ligands; MAP Kinase Signaling System; Orexin Receptor Antagonists; Orexin Receptors; Phosphorylation; Protein Binding; Radioligand Assay; Sleep; Sulfonamides	2014

Article

Year

Mapping the binding pocket of dual antagonist almorexant to human orexin 1 and orexin 2 receptors: comparison with the selective OX1 antagonist SB-674042 and the selective OX2 antagonist N-ethyl-2-[(6-methoxy-pyridin-3-yl)-(toluene-2-sulfonyl)-amino]-N-py

Molecular pharmacology, 2010, Volume: 78, Issue:1

Topics: Acetamides; Amino Acid Sequence; Aminopyridines; Binding Sites; Cell Line; Humans; Isoquinolines; Molecular Sequence Data; Mutagenesis, Site-Directed; Orexin Receptors; Pyrrolidines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sequence Homology, Amino Acid; Sulfonamides; Thiazoles

2010

Binding kinetics differentiates functional antagonism of orexin-2 receptor ligands.

British journal of pharmacology, 2014, Volume: 171, Issue:2

Topics: Acetamides; Algorithms; Aminopyridines; Animals; Binding, Competitive; CHO Cells; Cricetulus; HEK293 Cells; Humans; Inositol Phosphates; Isoquinolines; Kinetics; Ligands; MAP Kinase Signaling System; Orexin Receptor Antagonists; Orexin Receptors; Phosphorylation; Protein Binding; Radioligand Assay; Sleep; Sulfonamides

2014