Page last updated: 2024-09-05

ahc 52 and nicardipine

ahc 52 has been researched along with nicardipine in 2 studies

Compound Research Comparison

Studies
(ahc 52)
Trials
(ahc 52)
Recent Studies (post-2010)
(ahc 52)
Studies
(nicardipine)
Trials
(nicardipine)
Recent Studies (post-2010) (nicardipine)
7002,646444312

Protein Interaction Comparison

ProteinTaxonomyahc 52 (IC50)nicardipine (IC50)
Bile salt export pumpHomo sapiens (human)8.314
ATP-dependent translocase ABCB1Mus musculus (house mouse)8
ATP-dependent translocase ABCB1Homo sapiens (human)4.2992
Cytochrome P450 3A4Homo sapiens (human)0.42
Cytochrome P450 2C9 Homo sapiens (human)1.69
ATP-dependent translocase ABCB1Mus musculus (house mouse)2.5
Cytochrome P450 2J2Homo sapiens (human)1.69
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)4.925
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)4.8

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kobayashi, Y; Watanabe, N; Yamashiro, T1
Kobayashi, Y; Koga, C; Tsuruo, T; Watanabe, N; Yamashiro, T; Yokoyama, KK1

Other Studies

2 other study(ies) available for ahc 52 and nicardipine

ArticleYear
Reduction of intracellular pH by inhibitors of natural killer cell activity, nicardipine, methyl 2-(N-benzyl-N-methylamino)ethyl-2,6-dimethyl-4-(2-isopropyl-pyrazolo[1, 5-a]pyridine-3-yl)-1,4-dihydro-pyridine-3,5-dicarboxylate (AHC-52), and 4,4'-diisothio
    Biochemical pharmacology, 1997, Jul-01, Volume: 54, Issue:1

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cytotoxicity, Immunologic; Dihydropyridines; Flow Cytometry; Humans; Hydrogen-Ion Concentration; Killer Cells, Natural; Nicardipine; Pyrazoles; Tumor Cells, Cultured

1997
Requirement of expression of P-glycoprotein on human natural killer leukemia cells for cell-mediated cytotoxicity.
    Biochemical pharmacology, 1998, May-01, Volume: 55, Issue:9

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line; Cell Survival; Cytotoxicity, Immunologic; Dihydropyridines; Drug Resistance, Multiple; Humans; Killer Cells, Natural; Nicardipine; Oligonucleotides, Antisense; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Pyrazoles; RNA, Messenger; Thymoma; Thymus Neoplasms; Transcription, Genetic; Tumor Cells, Cultured

1998