ah 6809 has been researched along with xanthenes in 58 studies
Studies (ah 6809) | Trials (ah 6809) | Recent Studies (post-2010) (ah 6809) | Studies (xanthenes) | Trials (xanthenes) | Recent Studies (post-2010) (xanthenes) |
---|---|---|---|---|---|
163 | 1 | 49 | 5,020 | 92 | 1,325 |
Protein | Taxonomy | ah 6809 (IC50) | xanthenes (IC50) |
---|---|---|---|
Amine oxidase [flavin-containing] B | Homo sapiens (human) | 7.42 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (5.17) | 18.7374 |
1990's | 37 (63.79) | 18.2507 |
2000's | 18 (31.03) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Baxter, GS; Clayton, JK; Marshall, K; Sangha, R; Senior, J | 1 |
Jones, RL; Lawrence, RA | 1 |
Malinowska, B; Molderings, G; Schlicker, E | 1 |
Coleman, RA; Humphrey, PP; Strong, P | 1 |
Hori, T; Matsuda, T; Nakashima, T | 1 |
Diener, M; Nobles, M; Rummel, W; Schmitt, C | 1 |
Matsumura, H | 1 |
Jones, RL; Lawrence, RA; Wilson, NH | 1 |
Biddulph, DM; Capehart, AA | 1 |
McCann, JD; Smith, JJ; Welsh, MJ | 1 |
Jumblatt, MM; Paterson, CA | 1 |
Beasley, TC; Biddulph, DM; Capehart, AA | 1 |
Hayaishi, O; Ito, S; Negishi, M; Okuda, E; Sugama, K | 1 |
Hayaishi, O; Horiguchi, S; Hyodo, M; Ito, S; Uda, R | 1 |
Keery, RJ; Lumley, P | 1 |
Choi, WS; Hayaishi, O; Honda, K; Inoué, S; Matsumura, H; Sakai, T | 1 |
Coleman, RA; Kennedy, I; Sheldrick, RL | 1 |
Burkey, TH; Pepperl, DJ; Regan, JW; Woodward, DF | 1 |
Akarsu, ES; Ayhan, IH | 1 |
Crankshaw, DJ; Gaspar, V | 1 |
Hayaishi, O; Hyodo, M; Ito, S; Minami, T; Nishihara, I; Sakamoto, K | 1 |
Coca-Prados, M; Jumblatt, MM; Neltner, AA; Paterson, CA | 1 |
al-Zadjali, KH; Imler, MP; Ohia, SE | 1 |
Diener, M; Gabato, D | 1 |
Koda, H; Kumazawa, T; Mizumura, K | 1 |
Vardey, CJ; Wheeldon, A | 1 |
Jones, RL; Matthews, JS | 1 |
Barnes, PJ; Belvisi, MG; Kawikova, I; Tadjkarimi, S; Takahashi, T; Yacoub, MH | 1 |
Fukusako, H; Koda, H; Kumazawa, T; Mizumura, K | 1 |
Mazar-Feldman, J; Rimon, G | 1 |
Coleman, R; Hammond, TG; Horton, AA; Hutchinson, SM | 1 |
Berrino, L; Bräutigam, M; Griepenkerl, I; Jäger, R; Möhlig, A; Racké, K; Reimann, A | 1 |
Crider, JY; Griffin, BW; Sharif, NA; Williams, GW | 1 |
Barnes, PJ; Giembycz, MA; Meja, KK | 1 |
Leff, AR; Mitchell, RW; Ndukwu, IM; White, SR | 1 |
Akarsu, ES; Comert, A; Mamuk, S | 1 |
Artibani, W; Corsi, M; Palea, S; Pietra, C; Romano, O; Toson, G; Trist, DG | 1 |
Beadle, RE; Holmes, EP; Seahorn, TL; Venugopalan, CS | 1 |
Crider, JY; Griffin, BW; Sharif, NA | 1 |
Crankshaw, DJ; Hillock, CJ | 1 |
Aussel, C; Ekindjian, OG; Hernvann, A; Le Maire, V; Le Marechal, H; Russo-Marie, F; Solito, E | 1 |
Bessard, G; Chavanon, O; Cracowski, JL; Devillier, P; Hunt, M; Souvignet, C; Stanke-Labesque, F | 1 |
Kinsella, BT; Walsh, MT | 1 |
Grundy, D; Haupt, W; Jiang, W; Kreis, ME | 1 |
Henry, PJ; Knight, DA; Lan, RS; Stewart, GA | 1 |
Breuiller-Fouché, M; Cabrol, D; Dallot, E; Ferré, F; Leroy, MJ; Schmitz, T | 1 |
Andelfinger, G; Bouayad, A; Chemtob, S; Clyman, RI; Fouron, JC; Gobeil, F; Kajino, H; Skoll, A; Varma, DR; Vazquez, A; Waleh, N | 1 |
Abayasekara, DR; Bernal, AL; Harris, TE; Michael, AE; Squires, PE | 1 |
Halm, DR; Halm, ST | 1 |
Brink, C; de Montpreville, V; Norel, X; Walch, L | 1 |
Moreno, JJ; Sanchez, T | 1 |
Casibang, M; Moody, TW | 1 |
Fang, Q; Kim, HJ; Kobayashi, T; Kohyama, T; Liu, X; Rennard, SI; Wen, FQ; Wyatt, TA | 1 |
Manning, BP; Mawe, GM; Sharkey, KA | 1 |
Heinemann, A; Holzer, P; Peskar, BA; Shahbazian, A | 1 |
DeMasi, GM; Hardwick, JC; Jelson, GS; Sager, KL | 1 |
Chakrabarti, S; Chakraborty, C; Lala, PK; Timoshenko, AV; Xu, G | 1 |
Azemovic, D; Massoumi, R; Nielsen, CK; Sjölander, A | 1 |
1 review(s) available for ah 6809 and xanthenes
Article | Year |
---|---|
[Role of prostaglandins D2 and E2 in the regulation of sleep].
Topics: Animals; Arousal; Cyclooxygenase Inhibitors; Dinoprostone; Humans; Norepinephrine; Prostaglandin Antagonists; Prostaglandin D2; Sleep; Xanthenes; Xanthones | 1992 |
57 other study(ies) available for ah 6809 and xanthenes
Article | Year |
---|---|
In vitro characterization of prostanoid EP-receptors in the non-pregnant human myometrium.
Topics: Dinoprostone; Dose-Response Relationship, Drug; Female; Humans; Iloprost; In Vitro Techniques; Misoprostol; Myometrium; Receptors, Prostaglandin E; Rioprostil; Xanthenes; Xanthones | 1991 |
Investigation of the prostaglandin E (EP-) receptor subtype mediating relaxation of the rabbit jugular vein.
Topics: Animals; Chickens; Dinoprostone; Ileum; In Vitro Techniques; Jugular Veins; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Prostaglandins; Rabbits; Receptors, Prostaglandin; Receptors, Prostaglandin E; Xanthenes; Xanthones | 1992 |
Inhibition of noradrenaline release in the rat vena cava via prostanoid receptors of the EP3-subtype.
Topics: Alprostadil; Animals; Dinoprost; Dinoprostone; Electric Stimulation; Indomethacin; Misoprostol; Norepinephrine; Prostaglandin Antagonists; Prostaglandin D2; Prostaglandins; Rats; Receptors, Prostaglandin; Receptors, Prostaglandin E; Vena Cava, Inferior; Xanthenes; Xanthones; Yohimbine | 1992 |
Prostanoid-induced inhibition of lipolysis in rat isolated adipocytes: probable involvement of EP3 receptors.
Topics: Adipose Tissue; Animals; Dinoprostone; Enprostil; In Vitro Techniques; Lipolysis; Prostaglandin Antagonists; Prostaglandins E, Synthetic; Rats; Rats, Inbred Strains; Receptors, Prostaglandin; Xanthenes; Xanthones | 1992 |
Thermal and PGE2 sensitivity of the organum vasculosum lamina terminalis region and preoptic area in rat brain slices.
Topics: Animals; Body Temperature; Cold Temperature; Dinoprostone; Hot Temperature; Hypothalamus; In Vitro Techniques; Male; Neurons; Preoptic Area; Prostaglandin Antagonists; Rats; Rats, Wistar; Xanthenes; Xanthones | 1992 |
Characterization of the antisecretory action of prostaglandin D2 in the rat colon.
Topics: Acetylcholine; Animals; Chlorides; Colon; Epoprostenol; Female; In Vitro Techniques; Intestinal Mucosa; Neurons; Prostaglandin D2; Rats; Rats, Inbred Strains; Receptors, Prostaglandin; Tetrodotoxin; Xanthenes; Xanthones | 1992 |
Characterization of receptors involved in the direct and indirect actions of prostaglandins E and I on the guinea-pig ileum.
Topics: Animals; Epoprostenol; Guinea Pigs; Histamine Antagonists; Ileum; In Vitro Techniques; Male; Morphine; Muscle Relaxation; Prostaglandin Antagonists; Prostaglandins E; Prostaglandins E, Synthetic; Receptors, Prostaglandin; Trachea; Vas Deferens; Xanthenes; Xanthones | 1992 |
Effects of a putative prostaglandin E2 antagonist, AH6809, on chondrogenesis in serum-free cultures of chick limb mesenchyme.
Topics: Adenylyl Cyclases; Animals; Cartilage; Cells, Cultured; Chick Embryo; Cyclic AMP; Dinoprost; Extremities; Mesoderm; Prostaglandin Antagonists; Radioimmunoassay; Receptors, Prostaglandin; Receptors, Prostaglandin E; Xanthenes; Xanthones | 1991 |
Bradykinin stimulates airway epithelial Cl- secretion via two second messenger pathways.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Bradykinin; Calcimycin; Cells, Cultured; Charybdotoxin; Chlorides; Cyclic AMP; Dogs; Epithelium; Indomethacin; Inositol 1,4,5-Trisphosphate; Isoproterenol; Kinetics; Mucous Membrane; Muscle, Smooth; Prostaglandin Antagonists; Quinacrine; Scorpion Venoms; Second Messenger Systems; Thionucleotides; Trachea; Xanthenes; Xanthones | 1990 |
Prostaglandin E2 effects on corneal endothelial cyclic adenosine monophosphate synthesis and cell shape are mediated by a receptor of the EP2 subtype.
Topics: Animals; Cells, Cultured; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Endothelium, Corneal; Prostaglandins E, Synthetic; Rabbits; Receptors, Prostaglandin; Receptors, Prostaglandin E; Xanthenes; Xanthones | 1991 |
Comparative effects of cytosine arabinoside and a prostaglandin E2 antagonist, AH6809, on chondrogenesis in serum-free cultures of chick limb mesenchyme.
Topics: Animals; Cartilage; Cell Differentiation; Cell Division; Cells, Cultured; Chick Embryo; Cytarabine; Dinoprostone; DNA; Embryonic and Fetal Development; Extremities; Mesoderm; Prostaglandin Antagonists; Receptors, Prostaglandin; Xanthenes; Xanthones | 1991 |
Evaluation of ZK110841 and AH6809, an agonist and an antagonist of prostaglandin DP-receptors on human platelets, with a PGD2-responsive cell line from bovine embryonic trachea.
Topics: Animals; Blood Platelets; Cattle; Cell Line; Cyclic AMP; Dinoprost; Prostaglandin D2; Receptors, Prostaglandin; Trachea; Xanthenes; Xanthones | 1990 |
Nociceptive effects induced by intrathecal administration of prostaglandin D2, E2, or F2 alpha to conscious mice.
Topics: Animals; Dose-Response Relationship, Drug; Hyperalgesia; Hyperesthesia; Injections, Spinal; Male; Mice; Nociceptors; Prostaglandins; Spinal Cord; Xanthenes; Xanthones | 1990 |
AH6809, a prostaglandin DP-receptor blocking drug on human platelets.
Topics: 1-Methyl-3-isobutylxanthine; 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adenosine; Adenosine Diphosphate; Adenosine-5'-(N-ethylcarboxamide); Dinoprost; Epoprostenol; Humans; Hydantoins; In Vitro Techniques; Male; Platelet Activating Factor; Platelet Aggregation; Prostaglandin D2; Prostaglandin Endoperoxides, Synthetic; Receptors, Immunologic; Receptors, Prostaglandin; Xanthenes; Xanthones | 1988 |
Evidence that brain prostaglandin E2 is involved in physiological sleep-wake regulation in rats.
Topics: Animals; Body Temperature; Brain; Circadian Rhythm; Dinoprostone; Male; Prostaglandin Antagonists; Rats; Rats, Inbred Strains; Reference Values; Sleep; Sleep, REM; Wakefulness; Xanthenes; Xanthones | 1989 |
New evidence with selective agonists and antagonists for the subclassification of PGE2-sensitive (EP) receptors.
Topics: Alprostadil; Animals; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Dinoprostone; In Vitro Techniques; Muscle Contraction; Prostaglandins E; Prostaglandins E, Synthetic; Receptors, Prostaglandin; Receptors, Prostaglandin E; Xanthenes; Xanthones | 1987 |
6-Isopropoxy-9-oxoxanthene-2-carboxylic acid (AH 6809), a human EP2 receptor antagonist.
Topics: Animals; Binding, Competitive; Cells, Cultured; Cyclic AMP; Dinoprostone; Humans; Kinetics; Prostaglandin Antagonists; Receptors, Prostaglandin E; Tritium; Xanthenes; Xanthones | 1995 |
Iloprost, a stable analogue of PGI2, potentiates the hyperthermic effect of PGE2 in rats.
Topics: Animals; Body Temperature; Dinoprostone; Dose-Response Relationship, Drug; Drug Synergism; Iloprost; Indomethacin; Injections; Injections, Intraventricular; Male; Preoptic Area; Prostaglandin Antagonists; Rats; Rats, Wistar; Receptors, Prostaglandin E; Xanthenes; Xanthones | 1993 |
Pharmacological characterization in vitro of prostanoid receptors in the myometrium of nonpregnant ewes.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Carbazoles; Cloprostenol; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; Female; Iloprost; In Vitro Techniques; Isoproterenol; Myometrium; Prostaglandin Antagonists; Prostaglandin D2; Prostaglandin Endoperoxides, Synthetic; Prostaglandins; Prostaglandins E, Synthetic; Prostaglandins, Synthetic; Receptors, Prostaglandin; Sheep; Thromboxane A2; Thromboxanes; Uterine Contraction; Vasoconstrictor Agents; Xanthenes; Xanthones | 1995 |
Blockade by ONO-NT-012, a unique prostanoid analogue, of prostaglandin E2-induced allodynia in conscious mice.
Topics: Analysis of Variance; Animals; Bridged Bicyclo Compounds; Dinoprostone; Hyperalgesia; Injections, Spinal; Male; Mice; Pain; Skin; Styrenes; Xanthenes; Xanthones | 1995 |
EP2-receptor stimulated cyclic AMP synthesis in cultured human non-pigmented ciliary epithelium.
Topics: Cell Line, Transformed; Ciliary Body; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Epithelium; Humans; Prostaglandin Antagonists; Receptors, Prostaglandin E; Xanthenes; Xanthones | 1994 |
Inhibitory effect of prostaglandins on dopamine release from the retina.
Topics: Animals; Apomorphine; Cyclooxygenase Inhibitors; Dinoprostone; Dopamine; Electric Stimulation; Flurbiprofen; In Vitro Techniques; Male; Melatonin; Prostaglandin Antagonists; Prostaglandins; Rabbits; Receptors, Cell Surface; Receptors, Dopamine D2; Receptors, Melatonin; Receptors, Prostaglandin; Retina; Xanthenes; Xanthones | 1994 |
Thromboxane-like actions of prostaglandin D2 on the contractility of the rat colon in vitro.
Topics: Animals; Carbachol; Colon; Eicosanoids; Female; In Vitro Techniques; Isometric Contraction; Muscle Contraction; Muscle, Smooth; Parasympathetic Nervous System; Prostaglandin Antagonists; Prostaglandin D2; Rats; Rats, Inbred Strains; SRS-A; Sulfonamides; Tetrodotoxin; Thromboxane A2; Thromboxanes; Xanthenes; Xanthones | 1994 |
Involvement of EP3 subtype of prostaglandin E receptors in PGE2-induced enhancement of the bradykinin response of nociceptors.
Topics: Alprostadil; Animals; Bradykinin; Dinoprostone; Dogs; Dose-Response Relationship, Drug; Drug Synergism; Epididymis; Hot Temperature; In Vitro Techniques; Male; Nociceptors; Physical Stimulation; Prostaglandin Antagonists; Receptors, Prostaglandin E; Testis; Xanthenes; Xanthones | 1993 |
Characterization of the inhibitory prostanoid receptors on human neutrophils.
Topics: Humans; Hydantoins; In Vitro Techniques; Leukotriene B4; Misoprostol; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Oxygen Consumption; Prostaglandin Antagonists; Prostaglandins; Prostanoic Acids; Receptors, Prostaglandin; Superoxides; Xanthenes; Xanthones; Zymosan | 1993 |
Potentiation of aggregation and inhibition of adenylate cyclase in human platelets by prostaglandin E analogues.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Dinoprostone; Drug Synergism; Humans; Platelet Activating Factor; Platelet Aggregation; Prostaglandin Antagonists; Prostaglandin Endoperoxides, Synthetic; Prostaglandins E, Synthetic; Xanthenes; Xanthones | 1993 |
8-Epi-PGF2 alpha, a novel noncyclooxygenase-derived prostaglandin, constricts airways in vitro.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adolescent; Adult; Animals; Bronchoconstriction; Dinoprost; Dioxanes; Dose-Response Relationship, Drug; F2-Isoprostanes; Female; Guinea Pigs; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Prostaglandin Antagonists; Prostaglandin Endoperoxides, Synthetic; Receptors, Prostaglandin; Thromboxane A2; Trachea; Xanthenes; Xanthones | 1996 |
EP receptor subtypes implicated in the PGE2-induced sensitization of polymodal receptors in response to bradykinin and heat.
Topics: Alprostadil; Animals; Bradykinin; Cyclic AMP; Dinoprostone; Dogs; Hot Temperature; Nociceptors; Prostaglandin Antagonists; Prostaglandins E, Synthetic; Receptors, Prostaglandin E; Xanthenes; Xanthones | 1996 |
A common low-affinity binding site for primary prostanoids on bovine aortic endothelial cells.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Aorta; Binding Sites; Biphenyl Compounds; Carbazoles; Cattle; Cells, Cultured; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Dinoprostone; Endothelium, Vascular; Epoprostenol; Heptanoic Acids; Iloprost; Prostaglandin Endoperoxides, Synthetic; Prostaglandins; Sulfonamides; Thromboxane A2; Thromboxanes; Xanthenes; Xanthones | 1996 |
Effects of eicosanoids on parameters in isolated rat hepatocytes and isolated rat hepatocyte couplets: protective effects of eicosanoid receptor antagonists.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Cell Membrane; Cells, Cultured; Cholic Acids; Dinoprost; Dinoprostone; Dioxanes; Eicosanoids; Fluoresceins; Liver; Prostaglandin Antagonists; Prostaglandin D2; Prostaglandin Endoperoxides, Synthetic; Rats; Receptors, Eicosanoid; Thromboxane A2; Vasoconstrictor Agents; Xanthenes; Xanthones | 1997 |
Modulation of noradrenaline release in rat isolated stomach by prostanoids, but not by histaminergic mechanisms.
Topics: Abortifacient Agents, Nonsteroidal; Animals; Dinoprostone; Electric Stimulation; Female; Gastric Mucosa; Histamine Agonists; Indomethacin; Methylhistamines; Misoprostol; Muscarinic Agonists; Norepinephrine; Oxotremorine; Parasympatholytics; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Histamine; Receptors, Prostaglandin; Scopolamine; Stomach; Tetrodotoxin; Xanthenes; Xanthones; Yohimbine | 1995 |
FP prostaglandin receptors mediating inositol phosphates generation and calcium mobilization in Swiss 3T3 cells: a pharmacological study.
Topics: 3T3 Cells; Animals; Calcium; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Hydantoins; Inositol Phosphates; Mice; Prostaglandin Antagonists; Protein Binding; Receptors, Prostaglandin; Xanthenes; Xanthones | 1997 |
Characterization of the prostanoid receptor(s) on human blood monocytes at which prostaglandin E2 inhibits lipopolysaccharide-induced tumour necrosis factor-alpha generation.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Biphenyl Compounds; Dinoprostone; Drug Interactions; Epoprostenol; Humans; Leukocytes, Mononuclear; Lipopolysaccharides; Prostaglandin Antagonists; Prostaglandin Endoperoxides, Synthetic; Prostanoic Acids; Receptors, Prostaglandin; Thromboxane A2; Tumor Necrosis Factor-alpha; Xanthenes; Xanthones | 1997 |
EP1 receptor blockade attenuates both spontaneous tone and PGE2-elicited contraction in guinea pig trachealis.
Topics: Acetylcholine; Animals; Biphenyl Compounds; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Dinoprostone; Electric Stimulation; Epithelium; Guinea Pigs; Iloprost; In Vitro Techniques; Indomethacin; Kinetics; Male; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Prostaglandin Antagonists; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Trachea; Xanthenes; Xanthones | 1997 |
Inhibition of pentylenetetrazol-induced seizures in rats by prostaglandin D2.
Topics: Animals; Anticonvulsants; Cerebral Ventricles; Dinoprost; Epilepsy, Tonic-Clonic; Injections, Intraventricular; Male; Pentylenetetrazole; Prostaglandin Antagonists; Prostaglandin D2; Rats; Rats, Wistar; Seizures; Sodium Selenite; Xanthenes; Xanthones | 1998 |
Pharmacological characterization of thromboxane and prostanoid receptors in human isolated urinary bladder.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Alprostadil; Biphenyl Compounds; Dinoprost; Dinoprostone; Electric Stimulation; Heptanoic Acids; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Prostaglandin Antagonists; Prostaglandin D2; Receptors, Prostaglandin; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Receptors, Prostaglandin E, EP2 Subtype; Receptors, Thromboxane; Thromboxane A2; Urinary Bladder; Xanthenes; Xanthones | 1998 |
Responses of guinea-pig lung parenchymal strips to tracheobronchial lavage fluid from horses affected with summer pasture-associated obstructive pulmonary disease.
Topics: Animal Feed; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bronchoalveolar Lavage Fluid; Dinoprostone; Guinea Pigs; Histamine; Horse Diseases; Horses; In Vitro Techniques; Leukotriene D4; Lung; Lung Diseases, Obstructive; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phospholipid Ethers; Platelet Activating Factor; Platelet Aggregation Inhibitors; Poaceae; Prostaglandin Antagonists; Quinolines; Reference Values; Seasons; Trachea; Xanthenes; Xanthones | 1998 |
Prostaglandin DP receptors positively coupled to adenylyl cyclase in embryonic bovine tracheal (EBTr) cells: pharmacological characterization using agonists and antagonists.
Topics: Adenosine Monophosphate; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cattle; Cells, Cultured; Cyclic AMP; Embryo, Mammalian; Enzyme Inhibitors; Hydantoins; Prostaglandin Antagonists; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; Stimulation, Chemical; Trachea; Xanthenes; Xanthones | 1999 |
Inhibitory prostanoid EP receptors in human non-pregnant myometrium.
Topics: Anti-Arrhythmia Agents; Biphenyl Compounds; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Muscle Relaxation; Myometrium; Prostaglandin Antagonists; Prostaglandins; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP2 Subtype; Xanthenes; Xanthones | 1999 |
System A neutral amino acid transporter regulation by interleukin-1beta in human osteoarthritic synovial cells: evidence for involvement of prostaglandin E(2) as a second messenger.
Topics: Amino Acid Transport Systems; Arachidonic Acids; beta-Alanine; Biological Transport; Carrier Proteins; Cells, Cultured; Cyclooxygenase 2; Cytosol; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Humans; Indans; Interleukin-1; Isoenzymes; Kinetics; Membrane Proteins; Osteoarthritis; Phospholipases A; Prostaglandin-Endoperoxide Synthases; Second Messenger Systems; Synovial Membrane; Xanthenes; Xanthones | 2000 |
Human internal mammary artery contraction by isoprostaglandin f(2alpha) type-III [8-iso-prostaglandin F(2alpha)].
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adult; Aged; Benzoquinones; Biphenyl Compounds; Dinoprost; Dose-Response Relationship, Drug; F2-Isoprostanes; Female; Flavanones; Flavonoids; Heptanoic Acids; Humans; In Vitro Techniques; Leukotrienes; Lipoxygenase Inhibitors; Male; Mammary Arteries; Middle Aged; Prostaglandin Antagonists; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Receptors, Thromboxane; Thromboxane B2; Vasoconstriction; Vasoconstrictor Agents; Xanthenes; Xanthones | 2000 |
Regulation of the human prostanoid TPalpha and TPbeta receptor isoforms mediated through activation of the EP(1) and IP receptors.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Biological Transport; Blood Platelets; Calcium; Cells, Cultured; Dinoprostone; Drug Interactions; Enzyme Inhibitors; Epoprostenol; Humans; Indoles; Isoquinolines; Maleimides; Prostaglandin Antagonists; Prostaglandins; Protein Isoforms; Receptors, Epoprostenol; Receptors, Prostaglandin; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Receptors, Thromboxane; Signal Transduction; Sulfonamides; Vasoconstrictor Agents; Xanthenes; Xanthones | 2000 |
Prostaglandin EP receptor subtypes have distinctive effects on jejunal afferent sensitivity in the rat.
Topics: Animals; Calcium Channel Blockers; Dinoprostone; Dose-Response Relationship, Drug; Electrophysiology; Gastrointestinal Motility; Jejunum; Male; Neurons, Afferent; Nifedipine; Prostaglandin Antagonists; Prostaglandins; Protein Isoforms; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Prostaglandin E; Xanthenes; Xanthones | 2000 |
Role of PGE(2) in protease-activated receptor-1, -2 and -4 mediated relaxation in the mouse isolated trachea.
Topics: Animals; Caenorhabditis elegans Proteins; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dinoprostone; Enzyme Activation; In Vitro Techniques; Indomethacin; Isoenzymes; Ligands; Male; Membrane Proteins; Mice; Mice, Inbred CBA; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Prostaglandin Antagonists; Prostaglandin-Endoperoxide Synthases; Protein Serine-Threonine Kinases; Receptor, PAR-2; Receptors, Thrombin; Thrombin; Trachea; Trypsin; Xanthenes; Xanthones | 2001 |
EP(4) receptors mediate prostaglandin E(2)-stimulated glycosaminoglycan synthesis in human cervical fibroblasts in culture.
Topics: Alprostadil; Biphenyl Compounds; Cells, Cultured; Cervix Uteri; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; Female; Fibroblasts; Glycosaminoglycans; Humans; Prostaglandin Antagonists; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP4 Subtype; Xanthenes; Xanthones | 2001 |
Characterization of PGE2 receptors in fetal and newborn lamb ductus arteriosus.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine Triphosphate; Alprostadil; Animals; Animals, Newborn; Anti-Arrhythmia Agents; Anti-Ulcer Agents; Binding, Competitive; Biphenyl Compounds; Colforsin; Dinoprost; Ductus Arteriosus; Female; Fetus; Polymerase Chain Reaction; Potassium Channels; Pregnancy; Prostaglandin Antagonists; Prostaglandins E, Synthetic; Radioligand Assay; Receptors, Prostaglandin E; Sheep; Tritium; Vasoconstriction; Xanthenes; Xanthones | 2001 |
Human granulosa-lutein cells express functional EP1 and EP2 prostaglandin receptors.
Topics: 16,16-Dimethylprostaglandin E2; Alprostadil; Calcium; Cells, Cultured; Cyclic AMP; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Dinoprostone; Dose-Response Relationship, Drug; Female; Granulosa Cells; Humans; Intracellular Fluid; Lutein; Progesterone; Prostaglandin Antagonists; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Receptors, Prostaglandin E, EP2 Subtype; RNA, Messenger; Xanthenes; Xanthones | 2001 |
Prostanoids stimulate K secretion and Cl secretion in guinea pig distal colon via distinct pathways.
Topics: Animals; Bumetanide; Chlorides; Colon; Cyclooxygenase Inhibitors; Dinoprostone; Diuretics; Dose-Response Relationship, Drug; Guinea Pigs; Humans; In Vitro Techniques; Indomethacin; Intestinal Mucosa; Male; Potassium; Prostaglandin Antagonists; Receptors, Prostaglandin; Xanthenes; Xanthones | 2001 |
Prostanoid EP(1)- and TP-receptors involved in the contraction of human pulmonary veins.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Biphenyl Compounds; Carbazoles; Culture Techniques; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Dinoprostone; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Heptanoic Acids; Humans; Iloprost; Male; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Prostaglandin Antagonists; Prostaglandins F, Synthetic; Pulmonary Veins; Receptors, Prostaglandin; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Receptors, Prostaglandin E, EP3 Subtype; Receptors, Thromboxane; Sulfonamides; Vasoconstriction; Xanthenes; Xanthones | 2001 |
Role of EP(1) and EP(4) PGE(2) subtype receptors in serum-induced 3T6 fibroblast cycle progression and proliferation.
Topics: Animals; Biphenyl Compounds; Calcium; Cell Cycle; Cell Division; Cells, Cultured; Cyclic AMP; Cyclins; Dinoprostone; Fibroblasts; Mice; Prostaglandin Antagonists; Protein Isoforms; Xanthenes; Xanthones | 2002 |
AH6809 antagonizes non-small cell lung cancer prostaglandin receptors.
Topics: Binding Sites; Calcium; Carcinoma, Non-Small-Cell Lung; Cell Division; Cell Membrane; Colony-Forming Units Assay; Cyclic AMP; Cytoplasm; Dinoprostone; DNA Primers; Humans; Lung Neoplasms; Prostaglandin Antagonists; Receptors, Prostaglandin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured; Xanthenes; Xanthones | 2002 |
PGD(2) modulates fibroblast-mediated native collagen gel contraction.
Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Carbazoles; Cells, Cultured; Collagen; Cyclic GMP; Enzyme Inhibitors; Estrenes; Fatty Acids, Unsaturated; Fibroblasts; Gels; Humans; Hydrazines; Indoles; Lung; Mesylates; Naphthalenes; Prostaglandin Antagonists; Prostaglandin D2; Protein Kinase C; Pyrroles; Pyrrolidinones; Rats; Receptors, Immunologic; Receptors, Prostaglandin; Thionucleotides; Type C Phospholipases; Wound Healing; Xanthenes; Xanthones | 2002 |
Effects of PGE2 in guinea pig colonic myenteric ganglia.
Topics: Action Potentials; Animals; Colon; Dinoprostone; Dose-Response Relationship, Drug; Electric Impedance; Electrophysiology; Female; Ganglia; Guinea Pigs; Male; Membrane Potentials; Microelectrodes; Myenteric Plexus; Neurokinin-1 Receptor Antagonists; Neurons; Receptors, Neurokinin-3; Receptors, Prostaglandin; Tetrodotoxin; Xanthenes; Xanthones | 2002 |
Differential peristaltic motor effects of prostanoid (DP, EP, IP, TP) and leukotriene receptor agonists in the guinea-pig isolated small intestine.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Alprostadil; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dinoprostone; Dose-Response Relationship, Drug; Fatty Acids, Unsaturated; Female; Guinea Pigs; Hydantoins; Hydrazines; Iloprost; In Vitro Techniques; Intestine, Small; Leukotriene Antagonists; Leukotriene D4; Male; Oxazepines; Peristalsis; Prostaglandin D2; Prostaglandins A; Receptors, Leukotriene; Receptors, Prostaglandin; Xanthenes; Xanthones; Yohimbine | 2002 |
Modulation of guinea pig intrinsic cardiac neurons by prostaglandins.
Topics: Animals; Dinoprostone; Female; Ganglia, Parasympathetic; Guinea Pigs; Heart; Hydantoins; Male; Mast Cells; Membrane Potentials; Phospholipases A; Phospholipases A2; Potassium Channel Blockers; Prostaglandin D2; Receptors, Prostaglandin; Xanthenes; Xanthones | 2003 |
Role of prostaglandin E2 receptors in migration of murine and human breast cancer cells.
Topics: Alprostadil; Animals; Breast Neoplasms; Carcinoma; Cell Movement; Colforsin; Cyclic AMP; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Dinoprostone; Dose-Response Relationship, Drug; Female; Humans; Indoles; Isoenzymes; Mammary Neoplasms, Experimental; Membrane Proteins; Mice; Neoplasm Invasiveness; Prostaglandin-Endoperoxide Synthases; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP2 Subtype; Receptors, Prostaglandin E, EP4 Subtype; Tumor Cells, Cultured; Up-Regulation; Xanthenes; Xanthones | 2003 |
Leukotriene D4-induced adhesion of Caco-2 cells is mediated by prostaglandin E2 and upregulation of alpha2beta1-integrin.
Topics: Caco-2 Cells; Carcinoma; Cell Adhesion; Colitis; Collagen Type I; Colonic Neoplasms; Cyclooxygenase 2; Dinoprostone; Extracellular Matrix; Humans; Integrin alpha2beta1; Isoenzymes; Leukotriene D4; Membrane Proteins; Nitrobenzenes; Prostaglandin-Endoperoxide Synthases; Receptors, Leukotriene; Sulfonamides; Up-Regulation; Xanthenes; Xanthones | 2003 |