ah 6809 has been researched along with butaprost in 20 studies
Studies (ah 6809) | Trials (ah 6809) | Recent Studies (post-2010) (ah 6809) | Studies (butaprost) | Trials (butaprost) | Recent Studies (post-2010) (butaprost) |
---|---|---|---|---|---|
163 | 1 | 49 | 6 | 0 | 3 |
163 | 1 | 49 | 161 | 0 | 46 |
Protein | Taxonomy | ah 6809 (IC50) | butaprost (IC50) |
---|---|---|---|
Prostacyclin receptor | Homo sapiens (human) | 0.037 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (10.00) | 18.2507 |
2000's | 10 (50.00) | 29.6817 |
2010's | 6 (30.00) | 24.3611 |
2020's | 2 (10.00) | 2.80 |
Authors | Studies |
---|---|
Ganesh, T | 1 |
Koda, H; Kumazawa, T; Mizumura, K | 1 |
Fukusako, H; Koda, H; Kumazawa, T; Mizumura, K | 1 |
Breuiller-Fouché, M; Cabrol, D; Dallot, E; Ferré, F; Leroy, MJ; Schmitz, T | 1 |
Andelfinger, G; Bouayad, A; Chemtob, S; Clyman, RI; Fouron, JC; Gobeil, F; Kajino, H; Skoll, A; Varma, DR; Vazquez, A; Waleh, N | 1 |
Abayasekara, DR; Bernal, AL; Harris, TE; Michael, AE; Squires, PE | 1 |
Heinemann, A; Holzer, P; Peskar, BA; Shahbazian, A | 1 |
Belvisi, MG; Catley, MC; Clarke, DL; Giembycz, MA; Newton, R; Yacoub, MH | 1 |
Akaike, A; Banno, Y; Fushimi, K; Nakashima, S; Shimizu, K; Takigawa, M | 1 |
Berliner, JA; Cruz, D; Dun, M; Gharavi, N; Koroniak, L; Li, R; Montoya, D; Mouillesseaux, KP | 1 |
Abayasekara, DR; Bernal, AL; Chandras, C; Harris, TE; Michael, AE | 1 |
Bradding, P; Brightling, CE; Cockerill, SL; Cruse, G; Duffy, SM | 1 |
Juvet, SC; Lee, BP; Zhang, L | 1 |
Baun, M; Gupta, S; Jansen-Olesen, I; Myren, M; Olesen, J; Ploug, KB | 1 |
Brant, KA; Fabisiak, JP | 1 |
Chae, IG; Chun, KS; Kwon, TK; Min, KJ; Woo, SM | 1 |
Chadee, K; Lejeune, M; Moreau, F | 1 |
Cao, J; Deng, Y; Fu, C; Gao, L; Gao, R; Liu, B; Mao, W; Shen, Y; Wu, J; Wu, X; Zhang, N; Zhang, S; Zhang, Y | 1 |
Qu, J; Reinach, PS; Srinivasalu, N; Su, Y; Xu, R; Zhang, S; Zhou, X; Zhu, Y | 1 |
Cao, J; Feng, S; Fu, C; Li, Q; Liu, B; Mao, W; Zhang, S; Zhao, J | 1 |
1 review(s) available for ah 6809 and butaprost
Article | Year |
---|---|
Prostanoid receptor EP2 as a therapeutic target.
Topics: Animals; Anti-Inflammatory Agents; Eye Diseases; Gene Knockout Techniques; Humans; Molecular Targeted Therapy; Neurodegenerative Diseases; Prostaglandin-Endoperoxide Synthases; Receptors, Prostaglandin E, EP2 Subtype; Signal Transduction; Stroke | 2014 |
19 other study(ies) available for ah 6809 and butaprost
Article | Year |
---|---|
Involvement of EP3 subtype of prostaglandin E receptors in PGE2-induced enhancement of the bradykinin response of nociceptors.
Topics: Alprostadil; Animals; Bradykinin; Dinoprostone; Dogs; Dose-Response Relationship, Drug; Drug Synergism; Epididymis; Hot Temperature; In Vitro Techniques; Male; Nociceptors; Physical Stimulation; Prostaglandin Antagonists; Receptors, Prostaglandin E; Testis; Xanthenes; Xanthones | 1993 |
EP receptor subtypes implicated in the PGE2-induced sensitization of polymodal receptors in response to bradykinin and heat.
Topics: Alprostadil; Animals; Bradykinin; Cyclic AMP; Dinoprostone; Dogs; Hot Temperature; Nociceptors; Prostaglandin Antagonists; Prostaglandins E, Synthetic; Receptors, Prostaglandin E; Xanthenes; Xanthones | 1996 |
EP(4) receptors mediate prostaglandin E(2)-stimulated glycosaminoglycan synthesis in human cervical fibroblasts in culture.
Topics: Alprostadil; Biphenyl Compounds; Cells, Cultured; Cervix Uteri; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; Female; Fibroblasts; Glycosaminoglycans; Humans; Prostaglandin Antagonists; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP4 Subtype; Xanthenes; Xanthones | 2001 |
Characterization of PGE2 receptors in fetal and newborn lamb ductus arteriosus.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine Triphosphate; Alprostadil; Animals; Animals, Newborn; Anti-Arrhythmia Agents; Anti-Ulcer Agents; Binding, Competitive; Biphenyl Compounds; Colforsin; Dinoprost; Ductus Arteriosus; Female; Fetus; Polymerase Chain Reaction; Potassium Channels; Pregnancy; Prostaglandin Antagonists; Prostaglandins E, Synthetic; Radioligand Assay; Receptors, Prostaglandin E; Sheep; Tritium; Vasoconstriction; Xanthenes; Xanthones | 2001 |
Human granulosa-lutein cells express functional EP1 and EP2 prostaglandin receptors.
Topics: 16,16-Dimethylprostaglandin E2; Alprostadil; Calcium; Cells, Cultured; Cyclic AMP; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Dinoprostone; Dose-Response Relationship, Drug; Female; Granulosa Cells; Humans; Intracellular Fluid; Lutein; Progesterone; Prostaglandin Antagonists; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Receptors, Prostaglandin E, EP2 Subtype; RNA, Messenger; Xanthenes; Xanthones | 2001 |
Differential peristaltic motor effects of prostanoid (DP, EP, IP, TP) and leukotriene receptor agonists in the guinea-pig isolated small intestine.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Alprostadil; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dinoprostone; Dose-Response Relationship, Drug; Fatty Acids, Unsaturated; Female; Guinea Pigs; Hydantoins; Hydrazines; Iloprost; In Vitro Techniques; Intestine, Small; Leukotriene Antagonists; Leukotriene D4; Male; Oxazepines; Peristalsis; Prostaglandin D2; Prostaglandins A; Receptors, Leukotriene; Receptors, Prostaglandin; Xanthenes; Xanthones; Yohimbine | 2002 |
Identification in human airways smooth muscle cells of the prostanoid receptor and signalling pathway through which PGE2 inhibits the release of GM-CSF.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 8-Bromo Cyclic Adenosine Monophosphate; Adenoviridae; Adolescent; Adult; Aged; Alprostadil; Cell Survival; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; Enzyme Inhibitors; Female; Gene Expression; Genetic Vectors; Granulocyte Colony-Stimulating Factor; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Indomethacin; Interleukin-1; Isoquinolines; Male; Middle Aged; Misoprostol; Myocytes, Smooth Muscle; Prostaglandins E, Synthetic; Protein Isoforms; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP2 Subtype; Receptors, Prostaglandin E, EP4 Subtype; Signal Transduction; Sulfonamides; Trachea; Xanthones | 2004 |
Implication of prostaglandin E(2) in TNF-alpha-induced release of m-calpain from HCS-2/8 chondrocytes. Inhibition of m-calpain release by NSAIDs.
Topics: Alprostadil; Anti-Inflammatory Agents, Non-Steroidal; Apoptosis; Aspirin; Calpain; Cell Line, Tumor; Chondrocytes; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Diclofenac; Dinoprostone; Humans; Nitrobenzenes; Phenylpropionates; Prostaglandin Antagonists; Sulfonamides; Tumor Necrosis Factor-alpha; Up-Regulation; Xanthones | 2004 |
Identification of prostaglandin E2 receptor subtype 2 as a receptor activated by OxPAPC.
Topics: Alprostadil; Atherosclerosis; Cells, Cultured; Dinoprostone; Foam Cells; Humans; Interleukin-10; Isoprostanes; Macrophages; Monocytes; Oxidation-Reduction; Phosphatidylcholines; Phospholipid Ethers; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP2 Subtype; RNA, Messenger; Tumor Necrosis Factor-alpha; Xanthones | 2006 |
PTGER1 and PTGER2 receptors mediate regulation of progesterone synthesis and type 1 11beta-hydroxysteroid dehydrogenase activity by prostaglandin E2 in human granulosa lutein cells.
Topics: 11-beta-Hydroxysteroid Dehydrogenase Type 1; Alprostadil; Cells, Cultured; Cortisone; Cyclic AMP; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Dinoprostone; Dose-Response Relationship, Drug; Female; Humans; Hydrocortisone; Luteal Cells; Progesterone; Prostaglandin Antagonists; Prostaglandins E, Synthetic; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Receptors, Prostaglandin E, EP2 Subtype; Xanthones | 2007 |
Engagement of the EP2 prostanoid receptor closes the K+ channel KCa3.1 in human lung mast cells and attenuates their migration.
Topics: Alprostadil; Benzimidazoles; Calcium Channel Agonists; Cell Movement; Chemotaxis; Dinoprostone; Histamine Release; Humans; Mast Cells; Potassium Channels; Prostaglandin Antagonists; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP2 Subtype; Xanthones | 2008 |
Prostaglandin E2 signaling through E prostanoid receptor 2 impairs proliferative response of double negative regulatory T cells.
Topics: Alprostadil; Animals; CD4 Antigens; CD8 Antigens; Cell Proliferation; Clone Cells; Cytotoxicity, Immunologic; Dinoprostone; Immunomagnetic Separation; Mice; Mice, Inbred C57BL; Mice, Transgenic; Prostaglandin Antagonists; Receptors, Antigen, T-Cell, alpha-beta; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP2 Subtype; T-Lymphocytes, Regulatory; Xanthones | 2009 |
Functional and molecular characterization of prostaglandin E2 dilatory receptors in the rat craniovascular system in relevance to migraine.
Topics: Adenine; Alprostadil; Animals; Cerebral Arteries; Dinoprostone; Enzyme Inhibitors; Male; Meningeal Arteries; Migraine Disorders; Prostaglandin Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Prostaglandin E, EP2 Subtype; Receptors, Prostaglandin E, EP4 Subtype; RNA, Messenger; Trigeminal Nerve; Vasodilation; Xanthones | 2010 |
Role of hypoxia-inducible factor 1, α subunit and cAMP-response element binding protein 1 in synergistic release of interleukin 8 by prostaglandin E2 and nickel in lung fibroblasts.
Topics: Alprostadil; Biomimetics; Cells, Cultured; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Dinoprostone; Drug Synergism; Fibroblasts; Humans; Hypoxia-Inducible Factor 1, alpha Subunit; Inflammation; Interleukin-8; Lung; Nickel; p38 Mitogen-Activated Protein Kinases; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP2 Subtype; Receptors, Prostaglandin E, EP4 Subtype; Signal Transduction; Xanthones | 2013 |
Silymarin suppresses the PGE2 -induced cell migration through inhibition of EP2 activation; G protein-dependent PKA-CREB and G protein-independent Src-STAT3 signal pathways.
Topics: Alprostadil; Antioxidants; Benzodioxoles; Carcinoma, Renal Cell; Cell Line, Tumor; Cell Movement; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; Down-Regulation; Enzyme Activation; Enzyme Inhibitors; GTP-Binding Proteins; HCT116 Cells; HT29 Cells; Humans; Integrases; Kidney Neoplasms; Phosphorylation; Prostaglandin Antagonists; Quinazolines; Receptors, Prostaglandin E, EP2 Subtype; RNA Interference; RNA, Small Interfering; Signal Transduction; Silymarin; src-Family Kinases; STAT3 Transcription Factor; Wound Healing; Xanthones | 2015 |
Loss of EP2 receptor subtype in colonic cells compromise epithelial barrier integrity by altering claudin-4.
Topics: Alprostadil; Caco-2 Cells; Cell Membrane Permeability; Claudin-4; Cytokines; Down-Regulation; Humans; Interferon-gamma; Receptors, Prostaglandin E, EP2 Subtype; RNA Interference; RNA, Messenger; RNA, Small Interfering; Tight Junctions; Xanthones | 2014 |
PTGER2 activation induces PTGS-2 and growth factor gene expression in endometrial epithelial cells of cattle.
Topics: Alprostadil; Animals; Cattle; Cells, Cultured; Cyclooxygenase 2; Dinoprostone; Endometrium; Epithelial Cells; Female; Gene Expression Regulation; Intercellular Signaling Peptides and Proteins; Interleukin-8; MAP Kinase Signaling System; Prostaglandin Antagonists; Receptors, Prostaglandin E, EP2 Subtype; Transforming Growth Factor beta1; Vascular Endothelial Growth Factor A; Xanthones | 2017 |
Crosstalk between EP2 and PPARα Modulates Hypoxic Signaling and Myopia Development in Guinea Pigs.
Topics: Alprostadil; Animals; Cyclic AMP; Extracellular Matrix; Guinea Pigs; Hypoxia-Inducible Factor 1, alpha Subunit; Myopia, Degenerative; PPAR alpha; Prostaglandin Antagonists; Prostaglandins E, Synthetic; Receptors, Prostaglandin E, EP2 Subtype; Signal Transduction; Xanthones | 2020 |
Proliferation of bovine endometrial epithelial cells is promoted by prostaglandin E
Topics: Alprostadil; Aminopyridines; Animals; Cattle; Cell Cycle; Cell Proliferation; Cells, Cultured; Cyclin-Dependent Kinases; Cyclooxygenase 1; Cyclooxygenase 2; Dinoprostone; Endometrium; Epithelial Cells; Female; Proliferating Cell Nuclear Antigen; Purines; Receptors, Prostaglandin E, EP2 Subtype; Signal Transduction; Up-Regulation; Xanthones | 2021 |