ag 3-5 has been researched along with n-(4-tert-butylphenyl)-4-(3-chloropyridin-2-yl)tetrahydropyrazine-1(2h)-carboxamide in 4 studies
Studies (ag 3-5) | Trials (ag 3-5) | Recent Studies (post-2010) (ag 3-5) | Studies (n-(4-tert-butylphenyl)-4-(3-chloropyridin-2-yl)tetrahydropyrazine-1(2h)-carboxamide) | Trials (n-(4-tert-butylphenyl)-4-(3-chloropyridin-2-yl)tetrahydropyrazine-1(2h)-carboxamide) | Recent Studies (post-2010) (n-(4-tert-butylphenyl)-4-(3-chloropyridin-2-yl)tetrahydropyrazine-1(2h)-carboxamide) |
---|---|---|---|---|---|
126 | 0 | 66 | 83 | 1 | 48 |
Protein | Taxonomy | ag 3-5 (IC50) | n-(4-tert-butylphenyl)-4-(3-chloropyridin-2-yl)tetrahydropyrazine-1(2h)-carboxamide (IC50) |
---|---|---|---|
Transient receptor potential cation channel subfamily V member 1 | Rattus norvegicus (Norway rat) | 0.0051 | |
Amine oxidase [flavin-containing] B | Rattus norvegicus (Norway rat) | 0.0004 | |
Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | 1 | |
Transient receptor potential cation channel subfamily M member 8 | Homo sapiens (human) | 0.6375 | |
Transient receptor potential cation channel subfamily V member 1 | Homo sapiens (human) | 0.0119 | |
Transient receptor potential cation channel subfamily M member 8 | Rattus norvegicus (Norway rat) | 0.475 | |
Transient receptor potential cation channel subfamily M member 8 | Mus musculus (house mouse) | 0.4 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (25.00) | 29.6817 |
2010's | 3 (75.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Colburn, RW; Flores, CM; Liu, Y; Lubin, ML; Qin, N; Reitz, TL; Wang, Y | 1 |
Belmonte, C; Morenilla-Palao, C; Valero, M; Viana, F | 1 |
Beltrán, C; Darszon, A; De Blas, G; de la Vega-Beltrán, JL; Gibbs, GM; Martínez-López, P; Monroy, E; O'Bryan, MK; Orta, G; Treviño, CL | 1 |
Dhandapani, P; Grötzinger, C; Huimann, P; Khajavi, N; Köhrle, J; Ljubojevic, N; Lucius, A; Mergler, S; Reinach, PS | 1 |
4 other study(ies) available for ag 3-5 and n-(4-tert-butylphenyl)-4-(3-chloropyridin-2-yl)tetrahydropyrazine-1(2h)-carboxamide
Article | Year |
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Molecular identification and functional characterization of a temperature-sensitive transient receptor potential channel (TRPM8) from canine.
Topics: Action Potentials; Amino Acid Sequence; Animals; Calcium; Cell Line; Cloning, Molecular; Cold Temperature; DNA, Complementary; Dogs; Dose-Response Relationship, Drug; Fluorometry; Ganglia, Spinal; Gene Library; Humans; Menthol; Mice; Molecular Sequence Data; Mustard Plant; Oocytes; Patch-Clamp Techniques; Plant Oils; Pyrazines; Pyridines; Pyrimidinones; Rats; Reverse Transcriptase Polymerase Chain Reaction; Sequence Alignment; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Transfection; TRPM Cation Channels; Xenopus laevis | 2006 |
Pharmacological and functional properties of TRPM8 channels in prostate tumor cells.
Topics: Arginine; Calcium; Cell Line; Cell Line, Tumor; Cell Membrane; Clotrimazole; Cold Temperature; Endoplasmic Reticulum; Glycine; Humans; Male; Menthol; Prostate; Prostatic Neoplasms; Pyrazines; Pyridines; Pyrimidinones; TRPM Cation Channels | 2011 |
TRPM8 in mouse sperm detects temperature changes and may influence the acrosome reaction.
Topics: Acrosome Reaction; Animals; Capsaicin; Humans; Ion Channel Gating; Male; Menthol; Mice; Mice, Knockout; Pyrazines; Pyridines; Pyrimidinones; Spermatozoa; Temperature; Testis; TRPM Cation Channels | 2011 |
3-Iodothyronamine increases transient receptor potential melastatin channel 8 (TRPM8) activity in immortalized human corneal epithelial cells.
Topics: Calcium; Capsaicin; Cell Line; Epithelial Cells; Humans; Interleukin-6; Membrane Potentials; Patch-Clamp Techniques; Pyrazines; Pyridines; Pyrimidinones; Thyronines; TRPM Cation Channels; TRPV Cation Channels | 2016 |