Page last updated: 2024-08-16

ag 1879 and staurosporine

ag 1879 has been researched along with staurosporine in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (50.00)29.6817
2010's6 (42.86)24.3611
2020's1 (7.14)2.80

Authors

AuthorsStudies
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Kumar, A; Kumar, D; Mandal, D; Parang, K; Reddy, VB; Tiwari, R1
Ahmad, I; Chhikara, BS; Kumar, A; Mandal, D; Parang, K; Tiwari, R1
Chhikara, BS; Kumar, A; Parang, K; Rao, VK; Shirazi, AN; Tiwari, R1
Mandal, D; Olsen, CE; Parang, K; Parmar, VS; Prasad, AK; Sharma, RK; Singh, S; Tiwari, R1
Brown, A; Mandal, D; Nasrolahi Shirazi, A; Parang, K; Sun, G; Tiwari, RK1
Chand, K; Kumar, S; Parang, K; Prasad, S; Sharma, SK; Shirazi, AN; Tiwari, RK1
Chang, JW; Jo, J; Kim, J; Lee, S; Sim, J; Yun, H1
Boyd, JG; Buckley, RH; Candotti, F; Changelian, PS; Chen, M; Cusack, NA; Gadina, M; Geahlen, RL; Kimmel, LH; Lengi, A; Lin, W; Magnuson, KS; O'Shea, JJ; Roberts, JL; Zhou, YJ1
Dumont, FJ; Gould, S; Koprak, S; Matheravidathu, S; Springer, M1
Cance, WG; Golubovskaya, VM; Gross, S; Kaur, AS; Wilson, RI; Xu, LH; Yang, XH1
Shimoda, LA; Sylvester, JT; Weigand, L1
Abe, K; Ikebukuro, K; Sode, K; Yagi, YI1
Han, A; Hosokawa, K; Maeda, M1

Reviews

1 review(s) available for ag 1879 and staurosporine

ArticleYear
Recent advances in development of hetero-bivalent kinase inhibitors.
    European journal of medicinal chemistry, 2021, Apr-15, Volume: 216

    Topics: Cyclic AMP-Dependent Protein Kinases; Extracellular Signal-Regulated MAP Kinases; Humans; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Receptor, EphA1; Small Molecule Libraries; src-Family Kinases; TOR Serine-Threonine Kinases

2021

Other Studies

13 other study(ies) available for ag 1879 and staurosporine

ArticleYear
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
Click chemistry inspired one-pot synthesis of 1,4-disubstituted 1,2,3-triazoles and their Src kinase inhibitory activity.
    Bioorganic & medicinal chemistry letters, 2011, Jan-01, Volume: 21, Issue:1

    Topics: Alkynes; Aspartic Acid; Binding Sites; Click Chemistry; Computer Simulation; Morpholines; Protein Kinase Inhibitors; Sodium Azide; src-Family Kinases; Structure-Activity Relationship; Triazoles

2011
Synthesis of 3-phenylpyrazolopyrimidine-1,2,3-triazole conjugates and evaluation of their Src kinase inhibitory and anticancer activities.
    Bioorganic & medicinal chemistry letters, 2011, Mar-01, Volume: 21, Issue:5

    Topics: Antineoplastic Agents; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Colonic Neoplasms; Female; Humans; Inhibitory Concentration 50; Models, Molecular; Molecular Structure; Ovarian Neoplasms; Pyrans; Pyrimidines; src-Family Kinases; Triazoles

2011
One-pot regioselective synthesis of tetrahydroindazolones and evaluation of their antiproliferative and Src kinase inhibitory activities.
    Bioorganic & medicinal chemistry letters, 2012, Jan-01, Volume: 22, Issue:1

    Topics: Catalysis; Cell Proliferation; Chemistry, Pharmaceutical; Drug Design; HT29 Cells; Humans; Indazoles; Inhibitory Concentration 50; Ions; Magnetic Resonance Spectroscopy; Models, Chemical; Models, Molecular; Molecular Conformation; src-Family Kinases; Structure-Activity Relationship

2012
O-Aryl α,β-d-ribofuranosides: synthesis & highly efficient biocatalytic separation of anomers and evaluation of their Src kinase inhibitory activity.
    Bioorganic & medicinal chemistry, 2012, Dec-01, Volume: 20, Issue:23

    Topics: Acetylation; Ascomycota; Candida; Enzymes, Immobilized; Humans; Inhibitory Concentration 50; Lipase; Models, Molecular; Protein Kinase Inhibitors; Ribose; src-Family Kinases; Stereoisomerism

2012
Cyclic peptides containing tryptophan and arginine as Src kinase inhibitors.
    Bioorganic & medicinal chemistry letters, 2013, Jun-01, Volume: 23, Issue:11

    Topics: Arginine; Cell Line, Tumor; Cell Membrane Permeability; Humans; Kinetics; Peptides, Cyclic; Protein Binding; Protein Kinase Inhibitors; src-Family Kinases; Tryptophan

2013
Synthesis and evaluation of c-Src kinase inhibitory activity of pyridin-2(1H)-one derivatives.
    Bioorganic chemistry, 2014, Volume: 53

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Survival; CSK Tyrosine-Protein Kinase; Enzyme Activation; ErbB Receptors; Humans; MCF-7 Cells; Mitogen-Activated Protein Kinase Kinases; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyridones; Pyruvate Dehydrogenase Acetyl-Transferring Kinase; src-Family Kinases

2014
Unexpected effects of FERM domain mutations on catalytic activity of Jak3: structural implication for Janus kinases.
    Molecular cell, 2001, Volume: 8, Issue:5

    Topics: Adenosine Triphosphate; Amino Acid Sequence; Animals; Catalysis; COS Cells; Enzyme Inhibitors; Humans; Interleukin Receptor Common gamma Subunit; Janus Kinase 3; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Mutation; Protein Structure, Tertiary; Protein-Tyrosine Kinases; Pyrimidines; Receptors, Interleukin-7; Recombinant Fusion Proteins; Sequence Alignment; src-Family Kinases; Staurosporine

2001
Down-regulation of cell surface CXCR6 expression during T cell activation is predominantly mediated by calcineurin.
    Cellular immunology, 2003, Volume: 223, Issue:1

    Topics: Antigens, CD; Antigens, Differentiation, T-Lymphocyte; Butadienes; Calcineurin; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cytokines; Down-Regulation; Flow Cytometry; Humans; Immunosuppressive Agents; Interleukin-2; Lectins, C-Type; Lymphocyte Activation; Nitriles; Pyrimidines; Receptors, CCR7; Receptors, Chemokine; Receptors, CXCR6; Receptors, Cytokine; Receptors, G-Protein-Coupled; Receptors, Virus; Signal Transduction; Staurosporine; Tacrolimus

2003
Simultaneous inhibition of focal adhesion kinase and SRC enhances detachment and apoptosis in colon cancer cell lines.
    Molecular cancer research : MCR, 2003, Volume: 1, Issue:10

    Topics: Adenoviridae; Apoptosis; Blotting, Western; Caspase 3; Caspases; Cell Adhesion; Cell Line, Tumor; Down-Regulation; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; HT29 Cells; Humans; Immunoblotting; Microscopy, Fluorescence; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyrimidines; Signal Transduction; src-Family Kinases; Staurosporine

2003
Mechanisms of endothelin-1-induced contraction in pulmonary arteries from chronically hypoxic rats.
    American journal of physiology. Lung cellular and molecular physiology, 2006, Volume: 290, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amides; Animals; Azepines; Endothelin-1; Enzyme Inhibitors; Genistein; Hypoxia; Indoles; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Male; Maleimides; Myosin-Light-Chain Kinase; Potassium Chloride; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pulmonary Artery; Pyridines; Pyrimidines; Rats; Rats, Wistar; rho-Associated Kinases; src-Family Kinases; Staurosporine; Vasoconstriction

2006
Kinetic mechanism and inhibitor characterization of WNK1 kinase.
    Biochemistry, 2009, Nov-03, Volume: 48, Issue:43

    Topics: Electrophoretic Mobility Shift Assay; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Intracellular Signaling Peptides and Proteins; Kinetics; Minor Histocompatibility Antigens; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Staurosporine; Tyrphostins; WNK Lysine-Deficient Protein Kinase 1

2009
Phosphate-affinity electrophoresis on a microchip for determination of protein kinase activity.
    Electrophoresis, 2009, Volume: 30, Issue:20

    Topics: Acrylamides; Electrophoresis, Microchip; Indoles; Limit of Detection; Phosphopeptides; Protein Kinases; Pyridines; Pyrimidines; src-Family Kinases; Staurosporine; Sulfonamides

2009