ag 1879 has been researched along with staurosporine in 14 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 7 (50.00) | 29.6817 |
2010's | 6 (42.86) | 24.3611 |
2020's | 1 (7.14) | 2.80 |
Authors | Studies |
---|---|
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M | 1 |
Kumar, A; Kumar, D; Mandal, D; Parang, K; Reddy, VB; Tiwari, R | 1 |
Ahmad, I; Chhikara, BS; Kumar, A; Mandal, D; Parang, K; Tiwari, R | 1 |
Chhikara, BS; Kumar, A; Parang, K; Rao, VK; Shirazi, AN; Tiwari, R | 1 |
Mandal, D; Olsen, CE; Parang, K; Parmar, VS; Prasad, AK; Sharma, RK; Singh, S; Tiwari, R | 1 |
Brown, A; Mandal, D; Nasrolahi Shirazi, A; Parang, K; Sun, G; Tiwari, RK | 1 |
Chand, K; Kumar, S; Parang, K; Prasad, S; Sharma, SK; Shirazi, AN; Tiwari, RK | 1 |
Chang, JW; Jo, J; Kim, J; Lee, S; Sim, J; Yun, H | 1 |
Boyd, JG; Buckley, RH; Candotti, F; Changelian, PS; Chen, M; Cusack, NA; Gadina, M; Geahlen, RL; Kimmel, LH; Lengi, A; Lin, W; Magnuson, KS; O'Shea, JJ; Roberts, JL; Zhou, YJ | 1 |
Dumont, FJ; Gould, S; Koprak, S; Matheravidathu, S; Springer, M | 1 |
Cance, WG; Golubovskaya, VM; Gross, S; Kaur, AS; Wilson, RI; Xu, LH; Yang, XH | 1 |
Shimoda, LA; Sylvester, JT; Weigand, L | 1 |
Abe, K; Ikebukuro, K; Sode, K; Yagi, YI | 1 |
Han, A; Hosokawa, K; Maeda, M | 1 |
1 review(s) available for ag 1879 and staurosporine
Article | Year |
---|---|
Recent advances in development of hetero-bivalent kinase inhibitors.
Topics: Cyclic AMP-Dependent Protein Kinases; Extracellular Signal-Regulated MAP Kinases; Humans; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Receptor, EphA1; Small Molecule Libraries; src-Family Kinases; TOR Serine-Threonine Kinases | 2021 |
13 other study(ies) available for ag 1879 and staurosporine
Article | Year |
---|---|
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases | 2007 |
Click chemistry inspired one-pot synthesis of 1,4-disubstituted 1,2,3-triazoles and their Src kinase inhibitory activity.
Topics: Alkynes; Aspartic Acid; Binding Sites; Click Chemistry; Computer Simulation; Morpholines; Protein Kinase Inhibitors; Sodium Azide; src-Family Kinases; Structure-Activity Relationship; Triazoles | 2011 |
Synthesis of 3-phenylpyrazolopyrimidine-1,2,3-triazole conjugates and evaluation of their Src kinase inhibitory and anticancer activities.
Topics: Antineoplastic Agents; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Colonic Neoplasms; Female; Humans; Inhibitory Concentration 50; Models, Molecular; Molecular Structure; Ovarian Neoplasms; Pyrans; Pyrimidines; src-Family Kinases; Triazoles | 2011 |
One-pot regioselective synthesis of tetrahydroindazolones and evaluation of their antiproliferative and Src kinase inhibitory activities.
Topics: Catalysis; Cell Proliferation; Chemistry, Pharmaceutical; Drug Design; HT29 Cells; Humans; Indazoles; Inhibitory Concentration 50; Ions; Magnetic Resonance Spectroscopy; Models, Chemical; Models, Molecular; Molecular Conformation; src-Family Kinases; Structure-Activity Relationship | 2012 |
O-Aryl α,β-d-ribofuranosides: synthesis & highly efficient biocatalytic separation of anomers and evaluation of their Src kinase inhibitory activity.
Topics: Acetylation; Ascomycota; Candida; Enzymes, Immobilized; Humans; Inhibitory Concentration 50; Lipase; Models, Molecular; Protein Kinase Inhibitors; Ribose; src-Family Kinases; Stereoisomerism | 2012 |
Cyclic peptides containing tryptophan and arginine as Src kinase inhibitors.
Topics: Arginine; Cell Line, Tumor; Cell Membrane Permeability; Humans; Kinetics; Peptides, Cyclic; Protein Binding; Protein Kinase Inhibitors; src-Family Kinases; Tryptophan | 2013 |
Synthesis and evaluation of c-Src kinase inhibitory activity of pyridin-2(1H)-one derivatives.
Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Survival; CSK Tyrosine-Protein Kinase; Enzyme Activation; ErbB Receptors; Humans; MCF-7 Cells; Mitogen-Activated Protein Kinase Kinases; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyridones; Pyruvate Dehydrogenase Acetyl-Transferring Kinase; src-Family Kinases | 2014 |
Unexpected effects of FERM domain mutations on catalytic activity of Jak3: structural implication for Janus kinases.
Topics: Adenosine Triphosphate; Amino Acid Sequence; Animals; Catalysis; COS Cells; Enzyme Inhibitors; Humans; Interleukin Receptor Common gamma Subunit; Janus Kinase 3; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Mutation; Protein Structure, Tertiary; Protein-Tyrosine Kinases; Pyrimidines; Receptors, Interleukin-7; Recombinant Fusion Proteins; Sequence Alignment; src-Family Kinases; Staurosporine | 2001 |
Down-regulation of cell surface CXCR6 expression during T cell activation is predominantly mediated by calcineurin.
Topics: Antigens, CD; Antigens, Differentiation, T-Lymphocyte; Butadienes; Calcineurin; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cytokines; Down-Regulation; Flow Cytometry; Humans; Immunosuppressive Agents; Interleukin-2; Lectins, C-Type; Lymphocyte Activation; Nitriles; Pyrimidines; Receptors, CCR7; Receptors, Chemokine; Receptors, CXCR6; Receptors, Cytokine; Receptors, G-Protein-Coupled; Receptors, Virus; Signal Transduction; Staurosporine; Tacrolimus | 2003 |
Simultaneous inhibition of focal adhesion kinase and SRC enhances detachment and apoptosis in colon cancer cell lines.
Topics: Adenoviridae; Apoptosis; Blotting, Western; Caspase 3; Caspases; Cell Adhesion; Cell Line, Tumor; Down-Regulation; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; HT29 Cells; Humans; Immunoblotting; Microscopy, Fluorescence; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyrimidines; Signal Transduction; src-Family Kinases; Staurosporine | 2003 |
Mechanisms of endothelin-1-induced contraction in pulmonary arteries from chronically hypoxic rats.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amides; Animals; Azepines; Endothelin-1; Enzyme Inhibitors; Genistein; Hypoxia; Indoles; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Male; Maleimides; Myosin-Light-Chain Kinase; Potassium Chloride; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pulmonary Artery; Pyridines; Pyrimidines; Rats; Rats, Wistar; rho-Associated Kinases; src-Family Kinases; Staurosporine; Vasoconstriction | 2006 |
Kinetic mechanism and inhibitor characterization of WNK1 kinase.
Topics: Electrophoretic Mobility Shift Assay; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Intracellular Signaling Peptides and Proteins; Kinetics; Minor Histocompatibility Antigens; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Staurosporine; Tyrphostins; WNK Lysine-Deficient Protein Kinase 1 | 2009 |
Phosphate-affinity electrophoresis on a microchip for determination of protein kinase activity.
Topics: Acrylamides; Electrophoresis, Microchip; Indoles; Limit of Detection; Phosphopeptides; Protein Kinases; Pyridines; Pyrimidines; src-Family Kinases; Staurosporine; Sulfonamides | 2009 |