Page last updated: 2024-08-16

ag 1879 and sb 203580

ag 1879 has been researched along with sb 203580 in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's11 (61.11)29.6817
2010's7 (38.89)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dai, JR; Deretey, E; Foster, JE; Ng, W; Pasternak, A; Redden, PR; Reid, N; Slon-Usakiewicz, JJ; Toledo-Sherman, L1
Dai, JR; Deretey, E; Foster, JE; Liao, LC; Ng, W; Pasternak, A; Redden, PR; Reid, N; Slon-Usakiewicz, JJ; Toledo-Sherman, L; Uger, MD1
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Hajduk, PJ; Johnson, EF; Kifle, L; Merta, PJ; Metz, JT; Soni, NB1
Dart, ML; Hartnett, JR; Jost, E; Killoran, MP; Kirkland, TA; Machleidt, T; Robers, MB; Schwinn, MK; Shi, C; Wilkinson, JM; Wood, KV; Zimmerman, K1
Dransfield, I; McMeekin, SR; Ruchaud-Sparagano, MH; Walker, TR1
Iso, T; Kanai, H; Kurabayashi, M; Nagai, R; Ohyama, Y; Sakamoto, H; Sato, H; Sato, M; Tamura, J; Uchiyama, T1
Bae, YM; Kim, B; Lee, CK; Lee, HM; Lee, KY; Lee, SH; Lee, YL; Lim, J; Park, PJ; Park, TK; Roh, HY; Won, KJ1
Fujita-Yoshigaki, J; Matsuki-Fukushima, M; Sugiya, H1
Clark, JE; Cotten, M; Eickhoff, J; Flavell, RA; Jacquet, S; Kobayashi, KS; Kumphune, S; Marber, MS; Nishino, Y; Sicard, P1
Daoud, G; Lafond, J; Le bellego, F1
Di Rosa, M; Li Volti, G; Malaguarnera, L; Marsullo, AR; Zambito, AM1
Chen, DB; Feng, L; Liao, WX; Zheng, J1
Harris, T; Mackay, GA; Stewart, AG; Xia, YC1
Chang, HH; Chang, JZ; Deng, YT; Kuo, MY; Liu, CM; Yang, WH1
Jeong, YJ; Kim, CH; Kim, DJ; Kim, JC; Lee, KB; Oh, SM; Park, JH1
Batel, T; Behnen, M; Klinger, M; Laskay, T; Leschczyk, C; Möller, S; Solbach, W1

Other Studies

18 other study(ies) available for ag 1879 and sb 203580

ArticleYear
Frontal affinity chromatography with MS detection of EphB2 tyrosine kinase receptor. 1. Comparison with conventional ELISA.
    Journal of medicinal chemistry, 2004, Oct-07, Volume: 47, Issue:21

    Topics: Chromatography, Affinity; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Ligands; Mass Spectrometry; Models, Molecular; Receptor, EphB2

2004
Frontal affinity chromatography with MS detection of EphB2 tyrosine kinase receptor. 2. Identification of small-molecule inhibitors via coupling with virtual screening.
    Journal of medicinal chemistry, 2005, May-05, Volume: 48, Issue:9

    Topics: Antineoplastic Agents; Binding Sites; Cell Line, Tumor; Chromatography, Affinity; Databases, Factual; Enzyme-Linked Immunosorbent Assay; Heterocyclic Compounds; Humans; Mass Spectrometry; Models, Molecular; Molecular Weight; Naphthoquinones; Phosphorylation; Protein Structure, Tertiary; Quantitative Structure-Activity Relationship; Receptor, EphB2; Sulfides

2005
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
Navigating the kinome.
    Nature chemical biology, 2011, Volume: 7, Issue:4

    Topics: Drug Design; Pharmacogenetics; Protein Kinases; Proteome; Systems Biology

2011
Homogeneous Assay for Target Engagement Utilizing Bioluminescent Thermal Shift.
    ACS medicinal chemistry letters, 2018, Jun-14, Volume: 9, Issue:6

    Topics:

2018
A critical 'threshold' of beta 2-integrin engagement regulates augmentation of cytokine-mediated superoxide anion release.
    British journal of pharmacology, 2004, Volume: 141, Issue:7

    Topics: Binding Sites; CD18 Antigens; Cell Adhesion; Cytochalasin D; Cytokines; Cytoskeleton; Genistein; Humans; Imidazoles; Indoles; Integrin beta Chains; Magnesium; Maleimides; Microspheres; Mitogen-Activated Protein Kinases; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Nocodazole; Particle Size; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Pyridines; Pyrimidines; Serum Albumin; src-Family Kinases; Superoxides; Technology, Pharmaceutical; Tissue Adhesions; Tumor Necrosis Factor-alpha

2004
Mitochondrial reactive oxygen species and c-Src play a critical role in hypoxic response in vascular smooth muscle cells.
    Cardiovascular research, 2005, Sep-01, Volume: 67, Issue:4

    Topics: Androstadienes; Animals; Blotting, Northern; Catalase; Cell Hypoxia; Cell Line; Flavonoids; Hydrogen Peroxide; Hypoxia-Inducible Factor 1, alpha Subunit; Imidazoles; Immunoblotting; Microscopy, Fluorescence; Mitochondria; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Naphthalenes; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Plasminogen Activator Inhibitor 1; Protein Kinase Inhibitors; Proto-Oncogene Proteins pp60(c-src); Pyrazoles; Pyridines; Pyrimidines; Rabbits; RNA, Messenger; Rotenone; Wortmannin

2005
p38 mitogen-activated protein kinase contributes to angiotensin II-stimulated migration of rat aortic smooth muscle cells.
    Journal of pharmacological sciences, 2007, Volume: 105, Issue:1

    Topics: Actins; Angiotensin II; Animals; Aorta; Calcium-Calmodulin-Dependent Protein Kinases; Cell Movement; Cell Proliferation; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Imidazoles; Intracellular Signaling Peptides and Proteins; Male; Mitogen-Activated Protein Kinase 1; Muscle, Smooth, Vascular; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; Rats; Rats, Sprague-Dawley; Signal Transduction; Stilbenes; Syk Kinase; Vasoconstrictor Agents

2007
Inhibition of Src and p38 MAP kinases suppresses the change of claudin expression induced on dedifferentiation of primary cultured parotid acinar cells.
    American journal of physiology. Cell physiology, 2008, Volume: 294, Issue:3

    Topics: Amylases; Animals; Anthracenes; Aquaporin 5; Butadienes; Cell Adhesion; Cell Culture Techniques; Cell Differentiation; Cell Proliferation; Cell Shape; Cells, Cultured; Claudin-4; Claudins; Enzyme Activation; Extracellular Matrix; Imidazoles; Keratin-14; Male; Membrane Proteins; Nitriles; p38 Mitogen-Activated Protein Kinases; Parotid Gland; Protein Kinase Inhibitors; Pyrazoles; Pyridines; Pyrimidines; Rats; Rats, Sprague-Dawley; Signal Transduction; src-Family Kinases; Tight Junctions; Time Factors; Vimentin

2008
The role of RIP2 in p38 MAPK activation in the stressed heart.
    The Journal of biological chemistry, 2008, May-02, Volume: 283, Issue:18

    Topics: Acetylmuramyl-Alanyl-Isoglutamine; Animals; Cells, Cultured; Enzyme Activation; Imidazoles; In Vitro Techniques; Male; Mice; Myocardial Contraction; Myocardial Infarction; Myocardium; Myocytes, Cardiac; p38 Mitogen-Activated Protein Kinases; Protein Structure, Tertiary; Pyridines; Pyrimidines; Rats; Receptor-Interacting Protein Serine-Threonine Kinase 2

2008
PP2 regulates human trophoblast cells differentiation by activating p38 and ERK1/2 and inhibiting FAK activation.
    Placenta, 2008, Volume: 29, Issue:10

    Topics: Benzoquinones; Cell Differentiation; Cells, Cultured; CSK Tyrosine-Protein Kinase; Enzyme Activation; Female; Flavonoids; Focal Adhesion Protein-Tyrosine Kinases; Humans; Imidazoles; Lactams, Macrocyclic; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; p38 Mitogen-Activated Protein Kinases; Pregnancy; Protein-Tyrosine Kinases; Proto-Oncogene Proteins pp60(c-src); Pyridines; Pyrimidines; Rifabutin; Signal Transduction; src-Family Kinases; Trophoblasts

2008
Prolactin induces chitotriosidase expression in human macrophages through PTK, PI3-K, and MAPK pathways.
    Journal of cellular biochemistry, 2009, Aug-01, Volume: 107, Issue:5

    Topics: Acetophenones; Benzopyrans; Butadienes; Chromones; Gene Expression Regulation, Enzymologic; Genistein; Hexosaminidases; Humans; Imidazoles; Macrophages; MAP Kinase Signaling System; Monocytes; Morpholines; Nitriles; Phosphatidylinositol 3-Kinases; Phosphorylation; Prolactin; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-akt; Pyridines; Pyrimidines; RNA, Messenger; Tyrphostins

2009
Deciphering mechanisms controlling placental artery endothelial cell migration stimulated by vascular endothelial growth factor.
    Endocrinology, 2010, Volume: 151, Issue:7

    Topics: Androstadienes; Animals; Anthracenes; Arteries; Butadienes; Caveolin 1; Cell Movement; Cells, Cultured; CSK Tyrosine-Protein Kinase; Electrophoresis, Polyacrylamide Gel; Endothelial Cells; Enzyme Inhibitors; Female; Focal Adhesion Protein-Tyrosine Kinases; Imidazoles; Immunoprecipitation; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Nitric Oxide Synthase Type III; Nitriles; Nitrogen Oxides; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Placenta; Pregnancy; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; Sheep; Signal Transduction; src-Family Kinases; Vascular Endothelial Growth Factor A; Wortmannin

2010
Secreted factors from human mast cells trigger inflammatory cytokine production by human airway smooth muscle cells.
    International archives of allergy and immunology, 2013, Volume: 160, Issue:1

    Topics: Asthma; Cell Line; Culture Media, Conditioned; Exosomes; Humans; Imidazoles; Immunoglobulin E; Inflammation; Interleukin-6; Interleukin-8; Mast Cells; Myocytes, Smooth Muscle; p38 Mitogen-Activated Protein Kinases; Pyridines; Pyrimidines; Receptors, Fc; Respiratory System; RNA, Messenger; src-Family Kinases

2013
Curcumin inhibits TGFβ1-induced CCN2 via Src, JNK, and Smad3 in gingiva.
    Journal of dental research, 2013, Volume: 92, Issue:7

    Topics: Anthracenes; Anti-Inflammatory Agents, Non-Steroidal; Catechin; Cell Culture Techniques; Cell Movement; Cells, Cultured; Connective Tissue Growth Factor; Curcumin; Enzyme Inhibitors; Fibroblasts; Flavonoids; Gingiva; Gingival Overgrowth; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Imidazoles; Lovastatin; MAP Kinase Kinase 4; Phosphorylation; Protein Kinase Inhibitors; Pyridines; Pyrimidines; Signal Transduction; Smad3 Protein; src-Family Kinases; Transforming Growth Factor beta1

2013
RIP2/RICK-dependent cytokine production upon Yersinia enterocolitica infection in macrophages with TLR4 deficiency.
    Scandinavian journal of immunology, 2013, Volume: 78, Issue:5

    Topics: Animals; Enzyme Inhibitors; Gefitinib; Imidazoles; Interleukin-10; Interleukin-6; Macrophages; Mice; Mice, Inbred C57BL; Mice, Knockout; Nod1 Signaling Adaptor Protein; Nod2 Signaling Adaptor Protein; Protein Kinase Inhibitors; Pyridines; Pyrimidines; Quinazolines; Receptor-Interacting Protein Serine-Threonine Kinase 2; Receptor-Interacting Protein Serine-Threonine Kinases; Signal Transduction; Toll-Like Receptor 4; Tumor Necrosis Factor-alpha; Yersinia enterocolitica; Yersinia Infections

2013
Immobilized immune complexes induce neutrophil extracellular trap release by human neutrophil granulocytes via FcγRIIIB and Mac-1.
    Journal of immunology (Baltimore, Md. : 1950), 2014, Aug-15, Volume: 193, Issue:4

    Topics: Aminopyrine; Antigen-Antibody Complex; Antioxidants; Ascorbic Acid; Autoimmune Diseases; Butadienes; CD11a Antigen; CD18 Antigens; Cell Degranulation; Cells, Cultured; Extracellular Signal-Regulated MAP Kinases; GPI-Linked Proteins; Humans; Imidazoles; Inflammation; Intracellular Signaling Peptides and Proteins; Lymphocyte Function-Associated Antigen-1; Macrophage-1 Antigen; Mesalamine; Neutrophil Activation; Neutrophils; Nitriles; Onium Compounds; p38 Mitogen-Activated Protein Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-akt; Pyridines; Pyrimidines; Reactive Oxygen Species; Receptors, IgG; src-Family Kinases; Syk Kinase

2014