ag 1879 has been researched along with bisindolylmaleimide i in 10 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 6 (60.00) | 29.6817 |
2010's | 3 (30.00) | 24.3611 |
2020's | 1 (10.00) | 2.80 |
Authors | Studies |
---|---|
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M | 1 |
Cox, KJ; Gaj, A; Ghosh, I; Jester, BW; Shomin, CD | 1 |
Jadhav, A; Kerns, E; Nguyen, K; Shah, P; Sun, H; Xu, X; Yan, Z; Yu, KR | 1 |
Kabir, M; Kerns, E; Nguyen, K; Shah, P; Sun, H; Wang, Y; Xu, X; Yu, KR | 1 |
Kabir, M; Kerns, E; Neyra, J; Nguyen, K; Nguyễn, ÐT; Shah, P; Siramshetty, VB; Southall, N; Williams, J; Xu, X; Yu, KR | 1 |
Dransfield, I; McMeekin, SR; Ruchaud-Sparagano, MH; Walker, TR | 1 |
Fu, WM; Tang, CH; Yang, RS | 1 |
Shimoda, LA; Sylvester, JT; Weigand, L | 1 |
Clerk, A; Markou, T; Sugden, PH; Yong, CS | 1 |
Fujino, H; Hirabayashi, T; Murayama, T; Nakamura, H; Shimizu, M; Taniguchi, T | 1 |
10 other study(ies) available for ag 1879 and bisindolylmaleimide i
Article | Year |
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A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases | 2007 |
Testing the promiscuity of commercial kinase inhibitors against the AGC kinase group using a split-luciferase screen.
Topics: Animals; Binding, Competitive; Catalytic Domain; Cell-Free System; Cyclic AMP-Dependent Protein Kinase Catalytic Subunits; Cyclic GMP-Dependent Protein Kinase Type I; Cyclic GMP-Dependent Protein Kinases; Databases, Factual; Genes, Reporter; Luciferases; Protein Kinase C; Protein Kinase Inhibitors; Rabbits; Recombinant Fusion Proteins; Structure-Activity Relationship | 2012 |
Highly predictive and interpretable models for PAMPA permeability.
Topics: Artificial Intelligence; Caco-2 Cells; Cell Membrane Permeability; Humans; Models, Biological; Organic Chemicals; Regression Analysis; Support Vector Machine | 2017 |
Predictive models of aqueous solubility of organic compounds built on A large dataset of high integrity.
Topics: Drug Discovery; Organic Chemicals; Pharmaceutical Preparations; Solubility | 2019 |
Retrospective assessment of rat liver microsomal stability at NCATS: data and QSAR models.
Topics: Animals; Computer Simulation; Databases, Factual; Drug Discovery; High-Throughput Screening Assays; Liver; Machine Learning; Male; Microsomes, Liver; National Center for Advancing Translational Sciences (U.S.); Pharmaceutical Preparations; Quantitative Structure-Activity Relationship; Rats; Rats, Sprague-Dawley; Retrospective Studies; United States | 2020 |
A critical 'threshold' of beta 2-integrin engagement regulates augmentation of cytokine-mediated superoxide anion release.
Topics: Binding Sites; CD18 Antigens; Cell Adhesion; Cytochalasin D; Cytokines; Cytoskeleton; Genistein; Humans; Imidazoles; Indoles; Integrin beta Chains; Magnesium; Maleimides; Microspheres; Mitogen-Activated Protein Kinases; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Nocodazole; Particle Size; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Pyridines; Pyrimidines; Serum Albumin; src-Family Kinases; Superoxides; Technology, Pharmaceutical; Tissue Adhesions; Tumor Necrosis Factor-alpha | 2004 |
Prostaglandin E2 stimulates fibronectin expression through EP1 receptor, phospholipase C, protein kinase Calpha, and c-Src pathway in primary cultured rat osteoblasts.
Topics: Animals; Blotting, Western; Bone and Bones; Bone Density; Calcium; Cell Membrane; Cells, Cultured; Chelating Agents; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; Egtazic Acid; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Estrenes; Fibronectins; Genes, Dominant; Genes, Reporter; Immunoblotting; Immunohistochemistry; Immunoprecipitation; Indoles; Integrin alpha5; Integrin beta1; Integrins; Maleimides; Microscopy, Fluorescence; Mutation; Oligonucleotides; Oligonucleotides, Antisense; Osteoblasts; Promoter Regions, Genetic; Protein Isoforms; Protein Kinase C; Pyrimidines; Pyrrolidinones; Rats; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; src-Family Kinases; Transfection; Type C Phospholipases; Up-Regulation | 2005 |
Mechanisms of endothelin-1-induced contraction in pulmonary arteries from chronically hypoxic rats.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amides; Animals; Azepines; Endothelin-1; Enzyme Inhibitors; Genistein; Hypoxia; Indoles; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Male; Maleimides; Myosin-Light-Chain Kinase; Potassium Chloride; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pulmonary Artery; Pyridines; Pyrimidines; Rats; Rats, Wistar; rho-Associated Kinases; src-Family Kinases; Staurosporine; Vasoconstriction | 2006 |
Regulation of protein kinase C delta by phorbol ester, endothelin-1, and platelet-derived growth factor in cardiac myocytes.
Topics: Animals; Animals, Newborn; Cell Culture Techniques; Cell Extracts; Cells, Cultured; Chromatography, Gel; Chromones; Endothelin-1; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Immunoblotting; Indoles; Maleimides; Morpholines; Myocytes, Cardiac; Phosphorylation; Platelet-Derived Growth Factor; Precipitin Tests; Protein Kinase C-delta; Pyrimidines; Rats; Rats, Sprague-Dawley; Solubility; Tetradecanoylphorbol Acetate; Time Factors | 2006 |
Hydrogen peroxide-induced arachidonic acid release in L929 cells; roles of Src, protein kinase C and cytosolic phospholipase A2alpha.
Topics: Animals; Arachidonic Acid; Calcimycin; Calcium; Cell Line, Tumor; Cytosol; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fibroblasts; Group IV Phospholipases A2; Humans; Hydrogen Peroxide; Indoles; Ionophores; Maleimides; Mice; Phospholipases A; Protein Kinase C; Protein Kinase C-alpha; Protein Transport; Pyrimidines; Pyrrolidines; Signal Transduction; src-Family Kinases; Tetradecanoylphorbol Acetate; Transfection | 2006 |