ag-1296 and quinoxalines

ag-1296 has been researched along with quinoxalines in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (66.67)18.2507
2000's0 (0.00)29.6817
2010's2 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Böhmer, FD; Gazit, A; Heldin, CH; Kovalenko, M; Levitzki, A; Loubtchenkov, M; Rönnstrand, L1
Carlson, P; Krystal, GW; Litz, J1
Chen, H; Gazit, A; Hirth, P; Huber, LJ; Levitzki, A; Lipson, KE; McMahon, G; Pang, L; Tsai, JM1
Banai, S; Fishbein, I; Gazit, A; Gertz, SD; Golomb, G; Huber, R; Lazarovichi, G; Levitzki, A; Pearle, A; Perez, L; Rabinovich, L; Schneider, A; Waltenberger, J; Wolf, Y1
Aihara, M; Ishiuchi, S; Ohtani, T; Watanabe, T1
Baell, JB; Botteon, A; Chang, BCH; Danne, J; Ellis, S; Garcia-Bustos, JF; Gasser, RB; Hofmann, A; Jabbar, A; Jiao, Y; Koehler, AV; Le, T; McNamara, N; Nguyen, N; Preston, S; Skinner, C; Ventura, S; Wang, T1

Other Studies

6 other study(ies) available for ag-1296 and quinoxalines

ArticleYear
Phosphorylation site-specific inhibition of platelet-derived growth factor beta-receptor autophosphorylation by the receptor blocking tyrphostin AG1296.
    Biochemistry, 1997, May-27, Volume: 36, Issue:21

    Topics: Adenosine Triphosphate; Amino Acid Sequence; Animals; Binding, Competitive; Cell Line; Dimerization; Dogs; Enzyme Inhibitors; Humans; Kinetics; Molecular Sequence Data; Nitriles; Phosphatidylinositol 3-Kinases; Phosphorylation; Phosphotransferases (Alcohol Group Acceptor); Protein Binding; Quinoxalines; Receptor Protein-Tyrosine Kinases; Receptors, Platelet-Derived Growth Factor; Swine; Tyrphostins

1997
Induction of apoptosis and inhibition of small cell lung cancer growth by the quinoxaline tyrphostins.
    Cancer research, 1997, Jun-01, Volume: 57, Issue:11

    Topics: Apoptosis; Carcinoma, Small Cell; Cell Division; DNA Fragmentation; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Lung Neoplasms; Nitriles; Phosphorylation; Precipitin Tests; Protein-Tyrosine Kinases; Quinoxalines; Stem Cell Factor; Tumor Cells, Cultured; Tyrphostins

1997
Inhibition of platelet-derived growth factor and epidermal growth factor receptor signaling events after treatment of cells with specific synthetic inhibitors of tyrosine kinase phosphorylation.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 285, Issue:2

    Topics: 3T3 Cells; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cell Cycle Proteins; Cyclin-Dependent Kinase Inhibitor p27; ErbB Receptors; Mice; Microtubule-Associated Proteins; Nitriles; Phosphorylation; Quinoxalines; Receptor Protein-Tyrosine Kinases; Receptors, Platelet-Derived Growth Factor; Signal Transduction; Tumor Suppressor Proteins; Tyrosine; Tyrphostins

1998
PDGF-receptor tyrosine kinase blocker AG1295 selectively attenuates smooth muscle cell growth in vitro and reduces neointimal formation after balloon angioplasty in swine.
    Circulation, 1998, May-19, Volume: 97, Issue:19

    Topics: Angioplasty, Balloon; Animals; Aorta, Abdominal; Carotid Arteries; Cell Division; Cells, Cultured; Endarterectomy, Carotid; Enzyme Inhibitors; Femoral Artery; Humans; Mammary Arteries; Muscle, Smooth, Vascular; Nitriles; Organ Culture Techniques; Phosphorylation; Platelet-Derived Growth Factor; Quinoxalines; Receptor Protein-Tyrosine Kinases; Receptors, Platelet-Derived Growth Factor; Swine; Tunica Intima; Tyrphostins

1998
Enhanced antitumor effect of YM872 and AG1296 combination treatment on human glioblastoma xenograft models.
    Journal of neurosurgery, 2013, Volume: 118, Issue:4

    Topics: Animals; Antineoplastic Agents; Brain Neoplasms; Cell Line, Tumor; Cell Proliferation; Disease Models, Animal; Drug Therapy, Combination; Glioblastoma; Humans; Imidazoles; In Vitro Techniques; Mice; Mice, Nude; Phosphorylation; Proto-Oncogene Proteins c-akt; Proto-Oncogene Proteins c-kit; Quinoxalines; Receptors, AMPA; Receptors, Platelet-Derived Growth Factor; Transplantation, Heterologous; Treatment Outcome; Tyrphostins

2013
Tetrahydroquinoxalines induce a lethal evisceration phenotype in Haemonchus contortus in vitro.
    International journal for parasitology. Drugs and drug resistance, 2019, Volume: 9

    Topics: Animals; Antinematodal Agents; Biological Assay; Drug Discovery; Haemonchus; Inhibitory Concentration 50; Larva; Molting; Phenotype; Quinoxalines; Tyrphostins

2019