Page last updated: 2024-09-03

afdx 384 and oxotremorine

afdx 384 has been researched along with oxotremorine in 6 studies

Compound Research Comparison

Studies
(afdx 384)
Trials
(afdx 384)
Recent Studies (post-2010)
(afdx 384)
Studies
(oxotremorine)
Trials
(oxotremorine)
Recent Studies (post-2010) (oxotremorine)
78061,930699
5001,930699

Protein Interaction Comparison

ProteinTaxonomyafdx 384 (IC50)oxotremorine (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.4
Muscarinic acetylcholine receptor M4Homo sapiens (human)5
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)2.321
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M5Homo sapiens (human)8
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.5012

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (50.00)18.2507
2000's2 (33.33)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bungardt, E; Feifel, R; Lambrecht, G; Moser, U; Mutschler, E; Surprenant, A; Tacke, R; Vockert, E1
Wells, JW; Wreggett, KA1
Araujo, DM; Hefti, F; Lapchak, PA1
Auld, DS; Day, JC; Mennicken, F; Quirion, R1
Dean, B; Gibbons, AS; Jeon, WJ; Scarr, E1
Casida, JE; Honda, H; Tomizawa, M1

Other Studies

6 other study(ies) available for afdx 384 and oxotremorine

ArticleYear
Characterization of muscarinic receptors mediating vasodilation in guinea-pig ileum submucosal arterioles by the use of computer-assisted videomicroscopy.
    European journal of pharmacology, 1992, Mar-17, Volume: 213, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Arterioles; Benzodiazepinones; Carbachol; Guinea Pigs; Ileum; Methacholine Chloride; Muscarine; Muscarinic Antagonists; Oxotremorine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Prostaglandin Endoperoxides, Synthetic; Receptors, Muscarinic; Vasodilation

1992
Cooperativity manifest in the binding properties of purified cardiac muscarinic receptors.
    The Journal of biological chemistry, 1995, Sep-22, Volume: 270, Issue:38

    Topics: Allosteric Regulation; Animals; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Molecular Weight; Muscarinic Antagonists; Myocardium; N-Methylscopolamine; Oxotremorine; Parasympatholytics; Pirenzepine; Quinuclidinyl Benzilate; Radioligand Assay; Receptors, Muscarinic; Sarcolemma; Scopolamine Derivatives; Swine

1995
Regulation of hippocampal muscarinic receptor function by chronic nerve growth factor treatment in adult rats with fimbrial transections.
    Neuroscience, 1993, Volume: 53, Issue:2

    Topics: Animals; Autoradiography; Female; Guanosine Monophosphate; Hippocampus; In Vitro Techniques; Injections, Intraventricular; Inosine Triphosphate; Nerve Growth Factors; Oxotremorine; Parasympathetic Nervous System; Parasympatholytics; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptors, Muscarinic; Second Messenger Systems

1993
Pharmacological characterization of endogenous acetylcholine release from primary septal cultures.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 292, Issue:2

    Topics: Acetylcholine; Animals; Cells, Cultured; Choline; Choline O-Acetyltransferase; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Muscarinic Agonists; Neuromuscular Depolarizing Agents; Oxotremorine; Parasympatholytics; Piperidines; Pirenzepine; Potassium; Rats; Septum of Brain; Time Factors; Veratridine

2000
Changes in Muscarinic M2 Receptor Levels in the Cortex of Subjects with Bipolar Disorder and Major Depressive Disorder and in Rats after Treatment with Mood Stabilisers and Antidepressants.
    The international journal of neuropsychopharmacology, 2016, Volume: 19, Issue:4

    Topics: Animals; Antidepressive Agents; Antimanic Agents; Bipolar Disorder; Cerebral Cortex; Depressive Disorder, Major; Disease Models, Animal; Female; Fluoxetine; Humans; Imipramine; Male; Middle Aged; Muscarinic Agonists; Oxotremorine; Pirenzepine; Radiopharmaceuticals; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Tritium

2016
Insect muscarinic acetylcholine receptor: pharmacological and toxicological profiles of antagonists and agonists.
    Journal of agricultural and food chemistry, 2007, Mar-21, Volume: 55, Issue:6

    Topics: Animals; Brain; Drosophila; Houseflies; Insecta; Muscarinic Agonists; Muscarinic Antagonists; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Tritium

2007