Page last updated: 2024-09-03

afdx 384 and methoctramine

afdx 384 has been researched along with methoctramine in 6 studies

Compound Research Comparison

Studies
(afdx 384)
Trials
(afdx 384)
Recent Studies (post-2010)
(afdx 384)
Studies
(methoctramine)
Trials
(methoctramine)
Recent Studies (post-2010) (methoctramine)
7806332132
50040015
500332132

Protein Interaction Comparison

ProteinTaxonomyafdx 384 (IC50)methoctramine (IC50)
CholinesteraseHomo sapiens (human)0.9772
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.0407
AcetylcholinesteraseHomo sapiens (human)5.3703
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)0.138
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)0.138
Carboxylic ester hydrolase Rattus norvegicus (Norway rat)0.9772

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (83.33)18.2507
2000's1 (16.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lau, WM; Szilagyi, M2
Pepeu, G; Vannucchi, MG1
Avignone, E; Cattaneo, A; Cherubini, E; Guarnieri, E; Rosati, AM; Traversa, U1
Brann, MR; Dörje, F; Lambrecht, G; Mutschler, E; Tacke, R; Wess, J1
Casida, JE; Honda, H; Tomizawa, M1

Other Studies

6 other study(ies) available for afdx 384 and methoctramine

ArticleYear
A pharmacological profile of glycopyrrolate: interactions at the muscarinic acetylcholine receptor.
    General pharmacology, 1992, Volume: 23, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Binding, Competitive; Carbachol; Diamines; Female; Gallamine Triethiodide; Glycopyrrolate; Guinea Pigs; In Vitro Techniques; Ligands; Muscarinic Antagonists; Myocardial Contraction; Parasympatholytics; Pirenzepine; Quinuclidinyl Benzilate

1992
Muscarinic receptor modulation of acetylcholine release from rat cerebral cortex and hippocampus.
    Neuroscience letters, 1995, Apr-28, Volume: 190, Issue:1

    Topics: Acetylcholine; Animals; Cerebral Cortex; Diamines; Hippocampus; Male; Muscarinic Antagonists; Parasympatholytics; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Scopolamine

1995
Interaction of tacrine at M1 and M2 cholinoceptors in guinea pig brain.
    Pharmacology, 1993, Volume: 47, Issue:4

    Topics: Animals; Binding Sites; Brain; Diamines; Drug Interactions; Female; Guinea Pigs; Parasympatholytics; Pirenzepine; Receptors, Cholinergic; Tacrine

1993
Increased density of M1 receptors in the hippocampus of juvenile rats chronically deprived of NGF.
    Brain research, 1999, Jan-09, Volume: 815, Issue:2

    Topics: Animals; Animals, Newborn; Binding, Competitive; Diamines; Hippocampus; Neoplasm Transplantation; Nerve Growth Factors; Pirenzepine; Protein Binding; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptors, Muscarinic; Tumor Cells, Cultured

1999
Antagonist binding profiles of five cloned human muscarinic receptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:2

    Topics: Animals; Cells, Cultured; Cricetinae; Humans; N-Methylscopolamine; Parasympatholytics; Receptors, Muscarinic; Scopolamine Derivatives; Transfection

1991
Insect muscarinic acetylcholine receptor: pharmacological and toxicological profiles of antagonists and agonists.
    Journal of agricultural and food chemistry, 2007, Mar-21, Volume: 55, Issue:6

    Topics: Animals; Brain; Drosophila; Houseflies; Insecta; Muscarinic Agonists; Muscarinic Antagonists; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Tritium

2007