Page last updated: 2024-09-03

afdx 384 and carbachol

afdx 384 has been researched along with carbachol in 2 studies

Compound Research Comparison

Studies
(afdx 384)
Trials
(afdx 384)
Recent Studies (post-2010)
(afdx 384)
Studies
(carbachol)
Trials
(carbachol)
Recent Studies (post-2010) (carbachol)
780613,91881968
50013,91881968

Protein Interaction Comparison

ProteinTaxonomyafdx 384 (IC50)carbachol (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.7849
Muscarinic acetylcholine receptor M4Homo sapiens (human)2.0626
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)3.4134
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.535
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.6638
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.849
Muscarinic acetylcholine receptor M3Homo sapiens (human)4.99

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lau, WM; Szilagyi, M1
Bungardt, E; Feifel, R; Lambrecht, G; Moser, U; Mutschler, E; Surprenant, A; Tacke, R; Vockert, E1

Other Studies

2 other study(ies) available for afdx 384 and carbachol

ArticleYear
A pharmacological profile of glycopyrrolate: interactions at the muscarinic acetylcholine receptor.
    General pharmacology, 1992, Volume: 23, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Binding, Competitive; Carbachol; Diamines; Female; Gallamine Triethiodide; Glycopyrrolate; Guinea Pigs; In Vitro Techniques; Ligands; Muscarinic Antagonists; Myocardial Contraction; Parasympatholytics; Pirenzepine; Quinuclidinyl Benzilate

1992
Characterization of muscarinic receptors mediating vasodilation in guinea-pig ileum submucosal arterioles by the use of computer-assisted videomicroscopy.
    European journal of pharmacology, 1992, Mar-17, Volume: 213, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Arterioles; Benzodiazepinones; Carbachol; Guinea Pigs; Ileum; Methacholine Chloride; Muscarine; Muscarinic Antagonists; Oxotremorine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Prostaglandin Endoperoxides, Synthetic; Receptors, Muscarinic; Vasodilation

1992