Page last updated: 2024-09-03

afdx 384 and 4-diphenylacetoxy-1,1-dimethylpiperidinium

afdx 384 has been researched along with 4-diphenylacetoxy-1,1-dimethylpiperidinium in 8 studies

Compound Research Comparison

Studies
(afdx 384)
Trials
(afdx 384)
Recent Studies (post-2010)
(afdx 384)
Studies
(4-diphenylacetoxy-1,1-dimethylpiperidinium)
Trials
(4-diphenylacetoxy-1,1-dimethylpiperidinium)
Recent Studies (post-2010) (4-diphenylacetoxy-1,1-dimethylpiperidinium)
7806446152
500446152

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (50.00)18.2507
2000's3 (37.50)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bungardt, E; Feifel, R; Lambrecht, G; Moser, U; Mutschler, E; Surprenant, A; Tacke, R; Vockert, E1
Entzeroth, M; Mayer, N1
Bégos, A; Bizot, JC; Breton, P; Brochet, D; Tambuté, A; Trovero, F1
Elhusseiny, A; Hamel, E1
Iannazzo, L; Majewski, H1
Addison, S; Evangelista, S; Greer, S; Hernon, J; Johns, N; Johnson, I; Lewis, M; Lindqvist, S; Mackay, J; Rhodes, M; Sharp, P; Speakman, C; Stebbings, W; Tighe, R; Watson, M; Williams, M1
Chen, WJ; Dean, B; Lai, CY; Scarr, E; Thomas, N1
Brann, MR; Dörje, F; Lambrecht, G; Mutschler, E; Tacke, R; Wess, J1

Other Studies

8 other study(ies) available for afdx 384 and 4-diphenylacetoxy-1,1-dimethylpiperidinium

ArticleYear
Characterization of muscarinic receptors mediating vasodilation in guinea-pig ileum submucosal arterioles by the use of computer-assisted videomicroscopy.
    European journal of pharmacology, 1992, Mar-17, Volume: 213, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Arterioles; Benzodiazepinones; Carbachol; Guinea Pigs; Ileum; Methacholine Chloride; Muscarine; Muscarinic Antagonists; Oxotremorine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Prostaglandin Endoperoxides, Synthetic; Receptors, Muscarinic; Vasodilation

1992
Labeling of rat heart muscarinic receptors using the new M2 selective antagonist [3H]AF-DX 384.
    Biochemical pharmacology, 1990, Oct-01, Volume: 40, Issue:7

    Topics: Affinity Labels; Animals; Atropine; Binding, Competitive; Male; Muscarinic Antagonists; Myocardium; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1990
Pharmacological profile of CEB-1957 and atropine toward brain muscarinic receptors and comparative study of their efficacy against sarin poisoning.
    Toxicology and applied pharmacology, 1998, Volume: 150, Issue:2

    Topics: Animals; Atropine; Autoradiography; Binding, Competitive; Brain; Cholinesterase Inhibitors; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Poisoning; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Sarin; Thiophenes

1998
Muscarinic--but not nicotinic--acetylcholine receptors mediate a nitric oxide-dependent dilation in brain cortical arterioles: a possible role for the M5 receptor subtype.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2000, Volume: 20, Issue:2

    Topics: Acetylcholine; Animals; Arterioles; Cattle; Cerebral Cortex; Cerebrovascular Circulation; Dose-Response Relationship, Drug; Humans; Microcirculation; Muscarinic Antagonists; Nitric Oxide; Organ Culture Techniques; Parasympatholytics; Piperidines; Pirenzepine; Receptor, Muscarinic M5; Receptors, Muscarinic; Receptors, Nicotinic; Vasodilation; Vasodilator Agents

2000
M(2)/M(4)-muscarinic receptors mediate automodulation of acetylcholine outflow from mouse cortex.
    Neuroscience letters, 2000, Jun-23, Volume: 287, Issue:2

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Autoreceptors; Binding, Competitive; Cerebral Cortex; Furans; Male; Mice; Muscarinic Antagonists; Naphthalenes; Neostigmine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic

2000
The colon-selective spasmolytic otilonium bromide inhibits muscarinic M(3) receptor-coupled calcium signals in isolated human colonic crypts.
    British journal of pharmacology, 2002, Volume: 137, Issue:7

    Topics: Acetylcholine; Animals; Atropine; Calcium; Calcium Signaling; CHO Cells; Colon; Cricetinae; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Quaternary Ammonium Compounds; Receptor, Muscarinic M3; Receptors, Muscarinic; Time Factors; Vasodilator Agents

2002
Changes in cholinergic and glutamatergic markers in the striatum from a sub-set of subjects with schizophrenia.
    Schizophrenia research, 2015, Volume: 169, Issue:1-3

    Topics: Autoradiography; Blotting, Western; Corpus Striatum; Disks Large Homolog 4 Protein; Female; Glial Fibrillary Acidic Protein; Humans; Intracellular Signaling Peptides and Proteins; Male; Membrane Proteins; Middle Aged; Muscarinic Antagonists; Neuroglia; Neurons; Piperidines; Pirenzepine; Radioligand Assay; Radiopharmaceuticals; Receptors, Muscarinic; Schizophrenia; Synaptosomal-Associated Protein 25; Tritium

2015
Antagonist binding profiles of five cloned human muscarinic receptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:2

    Topics: Animals; Cells, Cultured; Cricetinae; Humans; N-Methylscopolamine; Parasympatholytics; Receptors, Muscarinic; Scopolamine Derivatives; Transfection

1991