Page last updated: 2024-09-02

afdx 116 and quinuclidines

afdx 116 has been researched along with quinuclidines in 8 studies

Compound Research Comparison

Studies
(afdx 116)
Trials
(afdx 116)
Recent Studies (post-2010)
(afdx 116)
Studies
(quinuclidines)
Trials
(quinuclidines)
Recent Studies (post-2010) (quinuclidines)
3671242,567453991

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19901 (12.50)18.7374
1990's5 (62.50)18.2507
2000's1 (12.50)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bartolini, A; Fantetti, L; Ghelardini, C; Giotti, A; Malcangio, M; Malmberg-Aiello, P1
Bhattacharya, SK; Das Gupta, G; Sen, AP; Seth, K; Seth, PK1
Kato, T; Mizobe, F; Xu, M; Yamamoto, T1
Gabelt, BT; Kaufman, PL; Poyer, JF1
Doods, HN; van Zwieten, PA1
Gabelt, BT; Kaufman, PL1
Ehlert, FJ; Figueroa, KW; Griffin, MT; Liller, S1
Fujino, T; Kageyama, A; Nozawa, Y; Yamada, S; Yoshida, A1

Reviews

1 review(s) available for afdx 116 and quinuclidines

ArticleYear
Muscarinic receptors and drugs in cardiovascular medicine.
    Cardiovascular drugs and therapy, 1995, Volume: 9, Issue:1

    Topics: Bradycardia; Cardiovascular Diseases; Cholinergic Agents; Endothelium, Vascular; Humans; Muscarinic Agonists; Muscarinic Antagonists; Muscle, Smooth, Vascular; Nitric Oxide; Parasympatholytics; Pirenzepine; Quinuclidines; Receptors, Muscarinic; Regression Analysis; Structure-Activity Relationship

1995

Other Studies

7 other study(ies) available for afdx 116 and quinuclidines

ArticleYear
Role of muscarinic receptor subtypes in central antinociception.
    British journal of pharmacology, 1992, Volume: 105, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analgesia; Animals; Male; Mice; Pain Measurement; Pirenzepine; Quinuclidines; Receptors, Muscarinic; Thiophenes

1992
Central muscarinic receptor subtypes and carrageenin-induced paw oedema in rats.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1991, Volume: 191, Issue:1

    Topics: Animals; Arecoline; Carbachol; Carrageenan; Cerebellum; Corpus Striatum; Edema; Female; Foot; Gallamine Triethiodide; Inflammation; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine

1991
Differential effects of M1- and M2-muscarinic drugs on striatal dopamine release and metabolism in freely moving rats.
    Brain research, 1989, Aug-28, Volume: 495, Issue:2

    Topics: Animals; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Thiophenes

1989
The effect of muscarinic agonists and selective receptor subtype antagonists on the contractile response of the isolated rhesus monkey ciliary muscle.
    Experimental eye research, 1994, Volume: 59, Issue:6

    Topics: Animals; Carbachol; Ciliary Body; Dose-Response Relationship, Drug; In Vitro Techniques; Macaca mulatta; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Quinuclidines

1994
Inhibition of aceclidine-stimulated outflow facility, accommodation and miosis in rhesus monkeys by muscarinic receptor subtype antagonists.
    Experimental eye research, 1994, Volume: 58, Issue:5

    Topics: Accommodation, Ocular; Animals; Aqueous Humor; Dose-Response Relationship, Drug; Female; Macaca mulatta; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Pupil; Quinuclidines

1994
Estimation of agonist activity at G protein-coupled receptors: analysis of M2 muscarinic receptor signaling through Gi/o,Gs, and G15.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Algorithms; Animals; Carbachol; Cell Line; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Diphenylacetic Acids; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Protein alpha Subunits, Gs; Heterotrimeric GTP-Binding Proteins; Humans; Isoproterenol; Oxotremorine; Pertussis Toxin; Phosphatidylinositols; Piperidines; Pirenzepine; Quinuclidines; Receptor, Muscarinic M2; Signal Transduction; Transfection

2007
Loss of muscarinic and purinergic receptors in urinary bladder of rats with hydrochloric acid-induced cystitis.
    Urology, 2010, Volume: 76, Issue:4

    Topics: Adenosine Triphosphate; Animals; Benzhydryl Compounds; Benzofurans; Cresols; Cystitis; Disease Models, Animal; Down-Regulation; Female; Hydrochloric Acid; Mandelic Acids; N-Methylscopolamine; Organophosphonates; Phenols; Phenylpropanolamine; Pirenzepine; Polycyclic Compounds; Pyridoxal Phosphate; Pyrrolidines; Quinuclidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Receptors, Purinergic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urination; Urodynamics

2010