Page last updated: 2024-09-02

afdx 116 and oxotremorine

afdx 116 has been researched along with oxotremorine in 43 studies

Compound Research Comparison

Studies
(afdx 116)
Trials
(afdx 116)
Recent Studies (post-2010)
(afdx 116)
Studies
(oxotremorine)
Trials
(oxotremorine)
Recent Studies (post-2010) (oxotremorine)
3671241,930699

Protein Interaction Comparison

ProteinTaxonomyafdx 116 (IC50)oxotremorine (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.4
Muscarinic acetylcholine receptor M4Homo sapiens (human)5
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)2.321
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M5Homo sapiens (human)8
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.5012

Research

Studies (43)

TimeframeStudies, this research(%)All Research%
pre-19908 (18.60)18.7374
1990's28 (65.12)18.2507
2000's7 (16.28)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kovacs, I; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1
Casida, JE; Honda, H; Tomizawa, M1
Crino, PB; Jensen, EL; Vogt, BA1
Bhattacharya, SK; Das Gupta, G; Sen, AP; Seth, K; Seth, PK1
Gies, JP; Haddad, EB; Landry, Y1
Daniel, EE; Janssen, LJ1
Inoue, M; Kuriyama, H1
Boddeke, HW1
Richards, MH1
Bird, ED; Crino, PB; Plager, MD; Vogt, BA1
Borkowski, JA; Buck, MA; Mallon, RG; McQuade, RD; Pai, JK; Pepitoni, S1
Danilo, P; Rosen, MR; Steinberg, SF1
Costi, A; Marchi, M; Raiteri, M; Volpe, G1
Delen, FM; Ehlert, FJ; Liem, HA; Yun, SH1
Bagetta, G; Constanti, A1
De Boer, P; Horn, AS; Rollema, H; Westerink, BH; Zaagsma, J1
Arrang, JM; Gulat-Marnay, C; Lafitte, A; Schwartz, JC1
Marchi, M; Raiteri, M1
Kato, T; Mizobe, F; Xu, M; Yamamoto, T1
Araujo, DM; Collier, B; Lapchak, PA; Quirion, R1
Delen, FM; Ehlert, FJ; Friedman, DJ; Self, DW; Yun, SH1
Anderson, W; Dickinson, KE; Hirschowitz, BI; Matsumoto, H; Pruitt, RE; Uemura, N1
Camus, J; Christophe, J; De Neef, P; Fourmy, D; Pradayrol, L; Robberecht, P; Scemama, JL; Tastenoy, M; Vaysse, N; Waelbroeck, M1
Bai, D; Sattelle, DB1
Gabelt, BT; Kaufman, PL; Poyer, JF1
Haass, M; Haunstetter, A; Krüger, C; Kübler, W; Yi, X1
Cynader, MS; Drance, SM; Gupta, N; McAllister, R; Rootman, J1
Aslan, AN; Oktay, S; Onat, F; Ozkutlu, U1
Consolo, S; Garcia Ruiz, AJ; La Porta, C; Ladinsky, H; Zambelli, M1
Ehlert, FJ; Thomas, EA1
Matthews, MR; Zaidi, ZF1
Ehlert, FJ; Sawyer, GW2
Islam, MA; Kimura, I; Nojima, H1
Ehlert, FJ; Ostrom, RS1
DeLapp, NW; Falcone, J; Felder, CC; McClure, D; McKinzie, JH; Sawyer, BD; Vandergriff, A1
Höhle, KD; Möhlig, T; Reinheimer, T; Wessler, I; Zimmermann, S1
Hosoi, T; Nomura, J; Nomura, Y; Okuma, Y1
Bukharaeva, EA; Magazanik, LG; Nikolsky, EE; Samigullin, D; Vyskocil, F1
Ehlert, FJ; Figueroa, KW; Griffin, MT; Liller, S1
Mohler, EG; Palencia, CA; Prior, M; Ragozzino, ME; Rozman, S1
Blackstone, K; Pratt, WE1

Reviews

2 review(s) available for afdx 116 and oxotremorine

ArticleYear
Pharmacology and second messenger interactions of cloned muscarinic receptors.
    Biochemical pharmacology, 1991, Oct-09, Volume: 42, Issue:9

    Topics: Animals; Atropine; Carbachol; Cell Line; Humans; Oxotremorine; Piperidines; Pirenzepine; Receptors, Muscarinic; Recombinant Proteins; Second Messenger Systems; Transfection

1991
Cardioselective muscarinic antagonists.
    Federation proceedings, 1987, Volume: 46, Issue:8

    Topics: Animals; Carbachol; Cardiotonic Agents; Carrier Proteins; Cyclic AMP; Cyclic AMP Receptor Protein; Dose-Response Relationship, Drug; Heart; N-Methylscopolamine; Oxotremorine; Phorbol Esters; Pirenzepine; Receptors, Adrenergic; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine Derivatives

1987

Other Studies

41 other study(ies) available for afdx 116 and oxotremorine

ArticleYear
Pharmacological comparison of the cloned human and rat M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: Amino Acid Sequence; Animals; Carbachol; Cloning, Molecular; Cyclic AMP; Humans; Mice; Molecular Sequence Data; Muscarinic Agonists; Muscarinic Antagonists; Phosphatidylinositols; Radioligand Assay; Rats; Receptors, Muscarinic; Sequence Alignment; Sequence Homology, Amino Acid; Signal Transduction; Species Specificity

1998
Insect muscarinic acetylcholine receptor: pharmacological and toxicological profiles of antagonists and agonists.
    Journal of agricultural and food chemistry, 2007, Mar-21, Volume: 55, Issue:6

    Topics: Animals; Brain; Drosophila; Houseflies; Insecta; Muscarinic Agonists; Muscarinic Antagonists; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Tritium

2007
Multiple heteroreceptors on limbic thalamic axons: M2 acetylcholine, serotonin1B, beta 2-adrenoceptors, mu-opioid, and neurotensin.
    Synapse (New York, N.Y.), 1992, Volume: 10, Issue:1

    Topics: Atenolol; Autoradiography; Axons; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethanolamines; Limbic System; Neurotensin; Oxotremorine; Pindolol; Pirenzepine; Receptors, Adrenergic, beta; Receptors, Muscarinic; Receptors, Neurotensin; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, mu; Receptors, Serotonin; Thalamus; Tritium

1992
Central muscarinic receptor subtypes and carrageenin-induced paw oedema in rats.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1991, Volume: 191, Issue:1

    Topics: Animals; Arecoline; Carbachol; Carrageenan; Cerebellum; Corpus Striatum; Edema; Female; Foot; Gallamine Triethiodide; Inflammation; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine

1991
Sialic acid residues as catalysts for M2-muscarinic agonist-receptor interactions.
    Molecular pharmacology, 1990, Volume: 37, Issue:5

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Carbachol; Cell Membrane; Kinetics; Male; Myocardium; Neuraminidase; Oxotremorine; Parasympatholytics; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine; Sialic Acids

1990
Pre- and postjunctional muscarinic receptors in canine bronchi.
    The American journal of physiology, 1990, Volume: 259, Issue:4 Pt 1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Bethanechol Compounds; Bronchi; Carbachol; Dogs; Electric Stimulation; In Vitro Techniques; Membrane Potentials; Microelectrodes; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Receptors, Muscarinic

1990
Muscarinic receptor is coupled with a cation channel through a GTP-binding protein in guinea-pig chromaffin cells.
    The Journal of physiology, 1991, Volume: 436

    Topics: Adrenal Medulla; Animals; Barium; Calcium; Dose-Response Relationship, Drug; Female; GTP-Binding Proteins; Guinea Pigs; Ion Channels; Male; Membrane Potentials; Muscarine; Oxotremorine; Pirenzepine; Receptors, Muscarinic; Tetraethylammonium; Tetraethylammonium Compounds

1991
Different effects of muscarinic agonists in rat superior cervical ganglion and hippocampal slices.
    European journal of pharmacology, 1991, Aug-29, Volume: 201, Issue:2-3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Arecoline; Ganglia, Sympathetic; Hippocampus; In Vitro Techniques; Male; Oxotremorine; Parasympathomimetics; Pilocarpine; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains

1991
Laminar distributions of muscarinic acetylcholine, serotonin, GABA and opioid receptors in human posterior cingulate cortex.
    Neuroscience, 1990, Volume: 36, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aged; Autoradiography; Cerebral Cortex; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Humans; Iodocyanopindolol; Ketanserin; Male; Middle Aged; Oxotremorine; Paroxetine; Pindolol; Piperidines; Pirenzepine; Receptors, Cell Surface; Receptors, Cholinergic; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Opioid; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes

1990
Phospholipase D activity and phosphatidylethanol formation in stimulated HeLa cells expressing the human m1 muscarinic acetylcholine receptor gene.
    Biochemical and biophysical research communications, 1991, Apr-15, Volume: 176, Issue:1

    Topics: Cloning, Molecular; Enzyme Activation; Genetic Vectors; Glycerophospholipids; HeLa Cells; Humans; Kinetics; Myristic Acid; Myristic Acids; Oxotremorine; Parasympatholytics; Phosphatidic Acids; Phospholipase D; Pirenzepine; Plasmids; Quinuclidinyl Benzilate; Receptors, Muscarinic; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection

1991
Developmental changes in the muscarinic stimulation of canine Purkinje fibers.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:1

    Topics: Acetylcholine; Age Factors; Animals; Dogs; Female; GTP-Binding Proteins; Heart Conduction System; In Vitro Techniques; Male; Membrane Potentials; Oxotremorine; Pertussis Toxin; Pirenzepine; Purkinje Fibers; Receptors, Muscarinic; Virulence Factors, Bordetella

1990
Endogenous aspartate release in the rat hippocampus is inhibited by M2 'cardiac' muscarinic receptors.
    European journal of pharmacology, 1990, Feb-27, Volume: 177, Issue:3

    Topics: Acetylcholine; Animals; Aspartic Acid; Calcium; Carbachol; Chromatography, High Pressure Liquid; Heart; Hippocampus; In Vitro Techniques; Male; Myocardium; Neuromuscular Depolarizing Agents; Oxotremorine; Pirenzepine; Potassium; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Synaptosomes

1990
The interaction of amitriptyline, doxepin, imipramine and their N-methyl quaternary ammonium derivatives with subtypes of muscarinic receptors in brain and heart.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Amitriptyline; Animals; Brain; Doxepin; Heart; Imipramine; In Vitro Techniques; Male; N-Methylscopolamine; Oxotremorine; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives

1990
Muscarinic suppression of the evoked N-wave by oxotremorine-M recorded in the guinea-pig olfactory cortex slice.
    European journal of pharmacology, 1990, Mar-13, Volume: 178, Issue:1

    Topics: Action Potentials; Animals; Carbachol; Cerebral Cortex; Diamines; Electric Stimulation; Electroencephalography; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Olfactory Bulb; Oxotremorine; Parasympatholytics; Parasympathomimetics; Pirenzepine; Receptors, Muscarinic

1990
An M3-like muscarinic autoreceptor regulates the in vivo release of acetylcholine in rat striatum.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Acetylcholine; Animals; Atropine; Chromatography, High Pressure Liquid; Corpus Striatum; Dialysis; Dose-Response Relationship, Drug; Male; Neostigmine; Oxotremorine; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Time Factors

1990
Regulation of histamine release and synthesis in the brain by muscarinic receptors.
    Journal of neurochemistry, 1989, Volume: 52, Issue:1

    Topics: Animals; Brain; Carbachol; Histamine Release; Male; Oxotremorine; Pirenzepine; Potassium; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine

1989
Interaction acetylcholine-glutamate in rat hippocampus: involvement of two subtypes of M-2 muscarinic receptors.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3

    Topics: Acetylcholine; Animals; Carbachol; Glutamates; Glutamic Acid; Hippocampus; In Vitro Techniques; Male; Oxotremorine; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Synaptosomes

1989
Differential effects of M1- and M2-muscarinic drugs on striatal dopamine release and metabolism in freely moving rats.
    Brain research, 1989, Aug-28, Volume: 495, Issue:2

    Topics: Animals; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Thiophenes

1989
Binding sites for [3H]AF-DX 116 and effect of AF-DX 116 on endogenous acetylcholine release from rat brain slices.
    Brain research, 1989, Sep-04, Volume: 496, Issue:1-2

    Topics: Acetylcholine; Animals; Brain; In Vitro Techniques; Male; Oxotremorine; Parasympathomimetics; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1989
Coupling of subtypes of the muscarinic receptor to adenylate cyclase in the corpus striatum and heart.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Binding, Competitive; Corpus Striatum; Gallamine Triethiodide; Male; Myocardium; N-Methylscopolamine; Oxotremorine; Pirenzepine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; RNA, Messenger; Scopolamine Derivatives

1989
Muscarinic cholinergic receptor subtype on frog esophageal peptic cells: binding and secretion studies.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Bethanechol; Bethanechol Compounds; Carbachol; Esophagus; Imipramine; Kinetics; N-Methylscopolamine; Oxotremorine; Pepsinogens; Pirenzepine; Propranolol; Radioligand Assay; Rana catesbeiana; Receptors, Muscarinic; Scopolamine Derivatives

1988
Characterization of muscarinic receptors in human pancreatic membranes.
    Pancreas, 1988, Volume: 3, Issue:6

    Topics: Carbachol; Cell Membrane; Humans; Oxotremorine; Pancreas; Pilocarpine; Pirenzepine; Receptors, Muscarinic

1988
Muscarinic acetylcholine receptors on an identified motor neurone in the cockroach, Periplaneta americana.
    Neuroscience letters, 1994, Jul-04, Volume: 175, Issue:1-2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Arecoline; Atropine; Dose-Response Relationship, Drug; Evoked Potentials; Ganglia, Invertebrate; In Vitro Techniques; Male; Motor Neurons; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Periplaneta; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine; Vertebrates

1994
The effect of muscarinic agonists and selective receptor subtype antagonists on the contractile response of the isolated rhesus monkey ciliary muscle.
    Experimental eye research, 1994, Volume: 59, Issue:6

    Topics: Animals; Carbachol; Ciliary Body; Dose-Response Relationship, Drug; In Vitro Techniques; Macaca mulatta; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Quinuclidines

1994
Muscarinic inhibition of cardiac norepinephrine and neuropeptide Y release during ischemia and reperfusion.
    The American journal of physiology, 1994, Volume: 267, Issue:6 Pt 2

    Topics: Animals; Atropine; Carbachol; Electric Stimulation; Guinea Pigs; Heart; Male; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; Neuropeptide Y; Norepinephrine; Oxotremorine; Parasympatholytics; Pirenzepine; Receptors, Muscarinic

1994
Muscarinic receptor M1 and M2 subtypes in the human eye: QNB, pirenzipine, oxotremorine, and AFDX-116 in vitro autoradiography.
    The British journal of ophthalmology, 1994, Volume: 78, Issue:7

    Topics: Adult; Aged; Aged, 80 and over; Anterior Eye Segment; Autoradiography; Ciliary Body; Eye; Female; Humans; Iris; Male; Middle Aged; Oxotremorine; Parasympatholytics; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Retina

1994
Central muscarinic M2 cholinoceptors involved in cholinergic hypertension.
    European journal of pharmacology, 1993, Dec-21, Volume: 250, Issue:3

    Topics: Animals; Blood Pressure; Diamines; Dose-Response Relationship, Drug; Female; Heart Rate; Injections, Intravenous; Injections, Intraventricular; Male; Muscarinic Antagonists; Oxotremorine; Physostigmine; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic

1993
Differences between rat dorsal and ventral hippocampus in muscarinic receptor agonist binding and interaction with phospholipase C.
    European journal of pharmacology, 1993, Jan-15, Volume: 244, Issue:2

    Topics: Alkaloids; Animals; Carbachol; Furans; Guanylyl Imidodiphosphate; Hippocampus; Male; Membranes; Mitochondria; N-Methylscopolamine; Naphthalenes; Oxotremorine; Parasympatholytics; Parasympathomimetics; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Synaptosomes; Type C Phospholipases

1993
Involvement of the M2 muscarinic receptor in contractions of the guinea pig trachea, guinea pig esophagus, and rat fundus.
    Biochemical pharmacology, 1996, Mar-22, Volume: 51, Issue:6

    Topics: Adrenergic beta-Agonists; Animals; Colforsin; Cyclic AMP; Esophagus; Gastric Fundus; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pertussis Toxin; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Serotonin; Trachea; Virulence Factors, Bordetella

1996
Exocytotic release from neuronal cell bodies, dendrites and nerve terminals in sympathetic ganglia of the rat, and its differential regulation.
    Neuroscience, 1997, Volume: 80, Issue:3

    Topics: Animals; Atropine; Carbachol; Cell Membrane; Dendrites; Exocytosis; Ganglia, Sympathetic; Male; Membrane Potentials; Nerve Endings; Neurons; Nicotine; Oxotremorine; Parasympatholytics; Pirenzepine; Potassium; Rats; Rats, Wistar; Receptors, Muscarinic; Regression Analysis; Synapses

1997
Contractile roles of the M2 and M3 muscarinic receptors in the guinea pig colon.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:1

    Topics: Animals; Colforsin; Colon; Cyclic AMP; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Oxotremorine; Pertussis Toxin; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Virulence Factors, Bordetella

1998
Muscarinic M1 receptor activation reduces maximum upstroke velocity of action potential in mouse right atria.
    European journal of pharmacology, 1998, Apr-10, Volume: 346, Issue:2-3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Action Potentials; Animals; Heart; Heart Atria; Heart Rate; In Vitro Techniques; Kinetics; Male; Membrane Potentials; Mice; Microelectrodes; Muscarinic Agonists; Oxotremorine; Parasympatholytics; Pirenzepine; Receptors, Muscarinic

1998
Comparison of functional antagonism between isoproterenol and M2 muscarinic receptors in guinea pig ileum and trachea.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 288, Issue:3

    Topics: Animals; Colforsin; Diphenylacetic Acids; Guinea Pigs; Histamine; Ileum; Isoproterenol; Muscle Relaxation; Oxotremorine; Pertussis Toxin; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptors, Muscarinic; Trachea; Virulence Factors, Bordetella

1999
Muscarinic M3 receptor inactivation reveals a pertussis toxin-sensitive contractile response in the guinea pig colon: evidence for M2/M3 receptor interactions.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:1

    Topics: Animals; Colon; Diphenylacetic Acids; Guinea Pigs; Hydrolysis; In Vitro Techniques; Male; Models, Biological; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pertussis Toxin; Phosphatidylinositols; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Virulence Factors, Bordetella

1999
Determination of [35S]guanosine-5'-O-(3-thio)triphosphate binding mediated by cholinergic muscarinic receptors in membranes from Chinese hamster ovary cells and rat striatum using an anti-G protein scintillation proximity assay.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:2

    Topics: Algorithms; Animals; Antibodies; Cell Membrane; CHO Cells; Cricetinae; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Mice; Muscarinic Agonists; Muscarinic Antagonists; Neostriatum; Oxotremorine; Pirenzepine; Precipitin Tests; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic

1999
Muscarinic control of histamine release from airways. Inhibitory M1-receptors in human bronchi but absence in rat trachea.
    American journal of respiratory and critical care medicine, 2000, Volume: 162, Issue:2 Pt 1

    Topics: Acetylcholine; Animals; Bronchi; Calcimycin; Clozapine; Female; Histamine Release; Humans; Ionophores; Male; Mast Cells; Muscarinic Antagonists; Organ Culture Techniques; Oxotremorine; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Species Specificity; Trachea

2000
The presence and functions of muscarinic receptors in human T cells: the involvement in IL-2 and IL-2 receptor system.
    Life sciences, 2003, Mar-28, Volume: 72, Issue:18-19

    Topics: Acetylcholine; Blotting, Northern; DNA; DNA Probes; DNA, Complementary; Enzyme-Linked Immunosorbent Assay; Humans; Interleukin-2; Jurkat Cells; Muscarinic Agonists; Oxotremorine; Parasympatholytics; Pirenzepine; Receptors, Interleukin-2; Receptors, Muscarinic; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; T-Lymphocytes

2003
Cholinergic regulation of the evoked quantal release at frog neuromuscular junction.
    The Journal of physiology, 2004, Oct-01, Volume: 560, Issue:Pt 1

    Topics: Acetylcholine; Action Potentials; Animals; Arecoline; Carbachol; Cholinergic Agonists; Diamines; Motor Neurons; Muscarinic Agonists; Muscarinic Antagonists; Neural Conduction; Neuromuscular Junction; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oxotremorine; Parasympatholytics; Pirenzepine; Rana ridibunda; Receptors, Muscarinic; Synaptic Transmission; Tubocurarine

2004
Estimation of agonist activity at G protein-coupled receptors: analysis of M2 muscarinic receptor signaling through Gi/o,Gs, and G15.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Algorithms; Animals; Carbachol; Cell Line; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Diphenylacetic Acids; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Protein alpha Subunits, Gs; Heterotrimeric GTP-Binding Proteins; Humans; Isoproterenol; Oxotremorine; Pertussis Toxin; Phosphatidylinositols; Piperidines; Pirenzepine; Quinuclidines; Receptor, Muscarinic M2; Signal Transduction; Transfection

2007
Acetylcholine activity in selective striatal regions supports behavioral flexibility.
    Neurobiology of learning and memory, 2009, Volume: 91, Issue:1

    Topics: Acetylcholine; Analysis of Variance; Animals; Cognition; Corpus Striatum; Male; Maze Learning; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Pirenzepine; Random Allocation; Rats; Rats, Long-Evans; Receptor, Muscarinic M2; Reversal Learning

2009
Nucleus accumbens acetylcholine and food intake: decreased muscarinic tone reduces feeding but not food-seeking.
    Behavioural brain research, 2009, Mar-02, Volume: 198, Issue:1

    Topics: Acetylcholine; Animals; Dose-Response Relationship, Drug; Eating; Feeding Behavior; Male; Microinjections; Muscarinic Agonists; Muscarinic Antagonists; N-Methylscopolamine; Nucleus Accumbens; Oxotremorine; Parasympatholytics; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic

2009