Page last updated: 2024-09-02

afdx 116 and dexetimide

afdx 116 has been researched along with dexetimide in 4 studies

Compound Research Comparison

Studies
(afdx 116)
Trials
(afdx 116)
Recent Studies (post-2010)
(afdx 116)
Studies
(dexetimide)
Trials
(dexetimide)
Recent Studies (post-2010) (dexetimide)
36712411744

Protein Interaction Comparison

ProteinTaxonomyafdx 116 (IC50)dexetimide (IC50)
Muscarinic acetylcholine receptor M1Mus musculus (house mouse)0.0033
Muscarinic acetylcholine receptor M4Mus musculus (house mouse)0.0033
Muscarinic acetylcholine receptor M5Mus musculus (house mouse)0.0033
Muscarinic acetylcholine receptor M3Mus musculus (house mouse)0.0033
Muscarinic acetylcholine receptor M2Mus musculus (house mouse)0.0033

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19902 (50.00)18.7374
1990's1 (25.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kovacs, I; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1
Elzinga, CR; Meurs, H; Roffel, AF; Zaagsma, J1
de Zeeuw, RA; in't Hout, WG; Roffel, AF; Zaagsma, J1
Christopoulos, A; Lanzafame, A; Mitchelson, F1

Other Studies

4 other study(ies) available for afdx 116 and dexetimide

ArticleYear
Pharmacological comparison of the cloned human and rat M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: Amino Acid Sequence; Animals; Carbachol; Cloning, Molecular; Cyclic AMP; Humans; Mice; Molecular Sequence Data; Muscarinic Agonists; Muscarinic Antagonists; Phosphatidylinositols; Radioligand Assay; Rats; Receptors, Muscarinic; Sequence Alignment; Sequence Homology, Amino Acid; Signal Transduction; Species Specificity

1998
Allosteric interactions of three muscarine antagonists at bovine tracheal smooth muscle and cardiac M2 receptors.
    European journal of pharmacology, 1989, Mar-07, Volume: 172, Issue:1

    Topics: Animals; Cattle; Dexetimide; Diamines; Gallamine Triethiodide; Heart; In Vitro Techniques; Membrane Proteins; Muscle, Smooth; Parasympatholytics; Pirenzepine; Receptors, Muscarinic; Trachea

1989
The M2 selective antagonist AF-DX 116 shows high affinity for muscarine receptors in bovine tracheal membranes.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:5

    Topics: Animals; Binding, Competitive; Cattle; Dexetimide; In Vitro Techniques; Membrane Proteins; Muscle, Smooth; Myocardium; Pirenzepine; Receptors, Muscarinic; Trachea

1987
The allosteric interaction of otenzepad (AF-DX 116) at muscarinic M2 receptors in guinea pig atria.
    European journal of pharmacology, 2001, Mar-30, Volume: 416, Issue:3

    Topics: Acetylcholine; Allosteric Regulation; Animals; Atropine; Carbachol; Cardiotonic Agents; Dexetimide; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Heart Atria; In Vitro Techniques; Kinetics; Male; Muscarinic Antagonists; N-Methylscopolamine; Nicotinic Antagonists; Parasympatholytics; Phthalimides; Pirenzepine; Quaternary Ammonium Compounds; Radioligand Assay; Receptor, Muscarinic M2; Receptors, Muscarinic

2001