Page last updated: 2024-09-02

afdx 116 and darifenacin

afdx 116 has been researched along with darifenacin in 2 studies

Compound Research Comparison

Studies
(afdx 116)
Trials
(afdx 116)
Recent Studies (post-2010)
(afdx 116)
Studies
(darifenacin)
Trials
(darifenacin)
Recent Studies (post-2010) (darifenacin)
3671241652854

Protein Interaction Comparison

ProteinTaxonomyafdx 116 (IC50)darifenacin (IC50)
Beta-1 adrenergic receptorHomo sapiens (human)0.3162
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.8322
Sodium channel protein type 5 subunit alphaHomo sapiens (human)1.5849

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fujino, T; Kageyama, A; Nozawa, Y; Yamada, S; Yoshida, A1
Arrighi, N; Bodei, S; Cosciani Cunico, S; Michel, MC; Sigala, S; Simeone, C; Spano, P; Zani, D1

Other Studies

2 other study(ies) available for afdx 116 and darifenacin

ArticleYear
Loss of muscarinic and purinergic receptors in urinary bladder of rats with hydrochloric acid-induced cystitis.
    Urology, 2010, Volume: 76, Issue:4

    Topics: Adenosine Triphosphate; Animals; Benzhydryl Compounds; Benzofurans; Cresols; Cystitis; Disease Models, Animal; Down-Regulation; Female; Hydrochloric Acid; Mandelic Acids; N-Methylscopolamine; Organophosphonates; Phenols; Phenylpropanolamine; Pirenzepine; Polycyclic Compounds; Pyridoxal Phosphate; Pyrrolidines; Quinuclidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Receptors, Purinergic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urination; Urodynamics

2010
Different muscarinic receptor subtypes modulate proliferation of primary human detrusor smooth muscle cells via Akt/PI3K and map kinases.
    Pharmacological research, 2013, Volume: 74

    Topics: Aged; Atropine; Benzofurans; Carbachol; Cell Proliferation; Cells, Cultured; Cholinergic Agonists; Gene Expression; Humans; Male; Mitogen-Activated Protein Kinases; Muscarinic Antagonists; Myocytes, Smooth Muscle; Phosphatidylinositol 3-Kinases; Piperidines; Pirenzepine; Proto-Oncogene Proteins c-akt; Pyrrolidines; Receptors, Muscarinic; RNA, Messenger; Urinary Bladder

2013