Page last updated: 2024-09-02

afdx 116 and aq-ra 741

afdx 116 has been researched along with aq-ra 741 in 6 studies

Compound Research Comparison

Studies
(afdx 116)
Trials
(afdx 116)
Recent Studies (post-2010)
(afdx 116)
Studies
(aq-ra 741)
Trials
(aq-ra 741)
Recent Studies (post-2010) (aq-ra 741)
3671242503

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baumgold, J; Cohen, VI; De La Cruz, R; Jin, B; Reba, RC; Rzeszotarski, WJ1
Hendriks, MG; Pfaffendorf, M; Van Zwieten, PA2
Doods, H; Entzeroth, M; Mayer, N1
Hamstra, JJ; Roffel, AF; Santing, RE; ten Berge, RE; Zaagsma, J1
Bechtel, WD; Doods, HN; Engel, W; Ensinger, HA; Entzeroth, M; Ladinsky, H; Mihm, G; Quirion, R; Rudolf, K; Schiavi, GB1

Reviews

1 review(s) available for afdx 116 and aq-ra 741

ArticleYear
Therapeutic potential of CNS-active M2 antagonists: novel structures and pharmacology.
    Life sciences, 1993, Volume: 52, Issue:5-6

    Topics: Animals; Benzodiazepinones; Brain; CHO Cells; Cognition Disorders; Cricetinae; Dibenzazepines; Drug Design; Motor Activity; Parasympatholytics; Piperidines; Pirenzepine; Pyridines; Rats; Receptors, Muscarinic; Structure-Activity Relationship

1993

Other Studies

5 other study(ies) available for afdx 116 and aq-ra 741

ArticleYear
Synthesis and structure-activity relationship of some 5-[[[(dialkylamino)alkyl]-1-piperidinyl]acetyl]-10,11-dihydro-5H- benzo[b,e][1,4]diazepin-11-ones as M2-selective antimuscarinics.
    Journal of medicinal chemistry, 1993, Jan-08, Volume: 36, Issue:1

    Topics: Animals; Benzodiazepinones; Brain; Mice; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Structure-Activity Relationship

1993
Characterization of the muscarinic receptor subtype mediating vasodilation in the rat perfused mesenteric vascular bed preparation.
    Journal of autonomic pharmacology, 1992, Volume: 12, Issue:6

    Topics: Animals; Atropine; Benzodiazepinones; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Arteries; Mesenteric Veins; Methacholine Chloride; Parasympatholytics; Perfusion; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Vasodilation

1992
Cardioselectivity of AQ-RA 741, a novel tricyclic antimuscarinic drug.
    European journal of pharmacology, 1991, Jan-03, Volume: 192, Issue:1

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Cats; Female; Guinea Pigs; Heart; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1991
Dysfunction of muscarinic M2 receptors after the early allergic reaction: possible contribution to bronchial hyperresponsiveness in allergic guinea-pigs.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Administration, Inhalation; Allergens; Animals; Asthma; Benzodiazepinones; Bronchial Hyperreactivity; Diamines; Disease Models, Animal; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Heart; Histamine; Hypersensitivity; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle, Smooth; Neuromuscular Junction; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea

1995
Characterization of the muscarinic receptors in the mesenteric vascular bed of spontaneously hypertensive rats.
    Journal of hypertension, 1993, Volume: 11, Issue:12

    Topics: Animals; Atropine; Benzodiazepinones; Endothelium, Vascular; Hypertension; Male; Mesenteric Artery, Superior; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Muscarinic; Vasodilation

1993