Page last updated: 2024-09-02

afdx 116 and 4-fluorohexahydrosiladifenidol

afdx 116 has been researched along with 4-fluorohexahydrosiladifenidol in 10 studies

Compound Research Comparison

Studies
(afdx 116)
Trials
(afdx 116)
Recent Studies (post-2010)
(afdx 116)
Studies
(4-fluorohexahydrosiladifenidol)
Trials
(4-fluorohexahydrosiladifenidol)
Recent Studies (post-2010) (4-fluorohexahydrosiladifenidol)
36712482010

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (90.00)18.2507
2000's1 (10.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kashihara, K; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1
Ehlert, FJ; Esqueda, EE; Gerstin, EH; Griffin, MT1
Hendriks, MG; Pfaffendorf, M; Van Zwieten, PA2
Anderson, DJ; Connolly, T; McKinney, M; Miller, JH; Vella-Rountree, L1
Jaiswal, N; Lambrecht, G; Malik, KU; Mutschler, E; Tacke, R1
Boddeke, HW1
Baron, E; Boer, R; Eltze, M; Kromer, W1
Garland, CJ; Hillier, K; Kerr, PM; Wallis, RM1
Höhle, KD; Möhlig, T; Reinheimer, T; Wessler, I; Zimmermann, S1

Other Studies

10 other study(ies) available for afdx 116 and 4-fluorohexahydrosiladifenidol

ArticleYear
Cloning of the rat M3, M4 and M5 muscarinic acetylcholine receptor genes by the polymerase chain reaction (PCR) and the pharmacological characterization of the expressed genes.
    Life sciences, 1992, Volume: 51, Issue:12

    Topics: Acetylcholine; Amino Acid Sequence; Animals; Base Sequence; Carbachol; Cell Line; Cloning, Molecular; Cyclic AMP; Fibroblasts; Gene Expression; Inositol Phosphates; Molecular Sequence Data; Parasympatholytics; Polymerase Chain Reaction; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Receptors, Muscarinic; Transfection

1992
Stimulation of cyclic AMP accumulation and phosphoinositide hydrolysis by M3 muscarinic receptors in the rat peripheral lung.
    Biochemical pharmacology, 1996, Aug-23, Volume: 52, Issue:4

    Topics: Animals; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Hydrolysis; Lung; Male; Oxotremorine; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic

1996
Characterization of the muscarinic receptor subtype mediating vasodilation in the rat perfused mesenteric vascular bed preparation.
    Journal of autonomic pharmacology, 1992, Volume: 12, Issue:6

    Topics: Animals; Atropine; Benzodiazepinones; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Arteries; Mesenteric Veins; Methacholine Chloride; Parasympatholytics; Perfusion; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Vasodilation

1992
Pharmacological profiles for rat cortical M1 and M2 muscarinic receptors using selective antagonists: comparison with N1E-115 muscarinic receptors.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:3

    Topics: Animals; Cerebral Cortex; Cyclic AMP; Diamines; In Vitro Techniques; Muscarinic Antagonists; Parasympatholytics; Phenethylamines; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Tumor Cells, Cultured

1991
Pharmacological characterization of the vascular muscarinic receptors mediating relaxation and contraction in rabbit aorta.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Antihypertensive Agents; Aorta, Abdominal; Arecoline; Atropine; Diamines; Endothelium, Vascular; Hexamethonium; Hexamethonium Compounds; Indomethacin; Male; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Norepinephrine; Parasympatholytics; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic

1991
Different effects of muscarinic agonists in rat superior cervical ganglion and hippocampal slices.
    European journal of pharmacology, 1991, Aug-29, Volume: 201, Issue:2-3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Arecoline; Ganglia, Sympathetic; Hippocampus; In Vitro Techniques; Male; Oxotremorine; Parasympathomimetics; Pilocarpine; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains

1991
Telenzepine inhibits electrically-stimulated, acetylcholine plus histamine-mediated acid secretion in the mouse isolated stomach by blockade of M1 muscarine receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:1

    Topics: Acetylcholine; Alkaloids; Animals; Anti-Ulcer Agents; Electric Stimulation; Furans; Gastric Acid; Gastric Mucosa; Histamine; Mice; Muscarinic Antagonists; Naphthalenes; p-Methoxy-N-methylphenethylamine; Parasympatholytics; Piperidines; Pirenzepine; Stomach; Thiazepines; Vagus Nerve

1991
Characterization of the muscarinic receptors in the mesenteric vascular bed of spontaneously hypertensive rats.
    Journal of hypertension, 1993, Volume: 11, Issue:12

    Topics: Animals; Atropine; Benzodiazepinones; Endothelium, Vascular; Hypertension; Male; Mesenteric Artery, Superior; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Muscarinic; Vasodilation

1993
Characterization of muscarinic receptors mediating contractions of circular and longitudinal muscle of human isolated colon.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: Alkaloids; Atropine; Carbachol; Carcinoma; Colon; Colonic Neoplasms; Dose-Response Relationship, Drug; Furans; Humans; In Vitro Techniques; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Naphthalenes; Piperidines; Pirenzepine

1995
Muscarinic control of histamine release from airways. Inhibitory M1-receptors in human bronchi but absence in rat trachea.
    American journal of respiratory and critical care medicine, 2000, Volume: 162, Issue:2 Pt 1

    Topics: Acetylcholine; Animals; Bronchi; Calcimycin; Clozapine; Female; Histamine Release; Humans; Ionophores; Male; Mast Cells; Muscarinic Antagonists; Organ Culture Techniques; Oxotremorine; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Species Specificity; Trachea

2000