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adenosine diphosphate and suramin

adenosine diphosphate has been researched along with suramin in 100 studies

Research

Studies (100)

TimeframeStudies, this research(%)All Research%
pre-19902 (2.00)18.7374
1990's42 (42.00)18.2507
2000's42 (42.00)29.6817
2010's13 (13.00)24.3611
2020's1 (1.00)2.80

Authors

AuthorsStudies
Harden, TK; Schachter, JB1
Jacobson, KA; Jarvis, MF; Williams, M1
Boyer, JL; Corbitt, J; Harden, TK; Jacobson, KA; Ji, XD; Kim, HS; Lacy, J; Ravi, G; Waldo, GL1
Boeynaems, JM; Communi, D; Gonzalez, NS; Labouret, C; Le Poul, E; Marteau, F; Savi, P1
Späth, L; Starke, K; von Kügelgen, I1
Hall, DA; Hourani, SM; Nieman, CJ1
Amerini, S; Ledda, F; Mantelli, L; Rubino, A1
Jones, CE; Reid, DM; Shulman, NR; Vostal, JG1
Blakeley, AG; Dunn, PM1
Bäumert, HG; Breddin, HK; Lambrecht, G; Mutschler, E; Radziwon, P; Windscheif, U1
Akaike, N; Ebihara, S; Uneyama, C; Uneyama, H1
Giachetti, A; Maggi, CA; Santicioli, P; Zagorodnyuk, V1
Fu, WM; Liou, JC1
Hashimoto, M; Kokubun, S1
Starke, K; Stoffel, D; von Kügelgen, I1
Balcar, VJ; Bennett, MR; Killinger, S; Li, Y1
Abe, Y; Akaike, N; Furukawa, K; Itoyama, Y; Sorimachi, M1
Chen, ZP; Levy, A; Lightman, SL1
Caparrotta, L; Chinellato, A; Fassina, G; Froldi, G; Pandolfo, L; Ragazzi, E1
Hall, DA; Hourani, SM1
Arnold, HH; Salminen, A1
Bidet, M; Cejka, JC; Poujeol, P; Tauc, M1
Culic, O; Lemmens, R; Teuchy, H; Vanduffel, L1
Barnard, EA; Burnstock, G; King, BF; Simon, J; Webb, TE1
Burnstock, G; Ralevic, V1
Nakamura, S; Ohshita, T; Sawamoto, N; Yamashita, H; Zhang, YX1
Li, CG; Najbar, AT; Rand, MJ1
Bültmann, R; Kurz, G; Nickel, P; Pause, B; Starke, K; Wittenburg, H1
Cazenave, JP; Gachet, C; Hechler, B; Léon, C; Leray, C; Vial, C1
Boeynaems, JM; Communi, D; Robaye, B2
Furukawa, M; Ikeda, K; Suzuki, H; Takasaka, T1
Maggi, CA; Zagorodnyuk, V1
Korngreen, A; Ma, W; Priel, Z; Silberberg, SD1
Dunne, MJ; James, RF; London, NJ; Squires, PE1
Connolly, GP; Demaine, C; Duley, JA1
Bernard, C; Butlen, D; Ferrary, E1
Ito, S; Nakazato, Y; Ohta, T; Otsuguro, K1
Cha, SH; Endou, H; Sekine, T1
Chen, SA; Jan, CR; Li, HF; Wu, SN1
Grantyn, R; Jüttner, R; Taschenberger, H1
Habuchi, Y; Morikawa, J; Nishio, M; Tanaka, H; Yamamoto, T1
Henning, L; Jankowski, J; Junker, R; Schlüter, H; Tente, IM; Tepel, M; van der Giet, M; Zidek, W1
Hourani, SM; Park, HS1
Katsuragi, T; Sato, C; Tsujioka, Y1
Barthó, L; Heinemann, A; Holzer, P; Shahbazian, A1
Figarella, C; Kammouni, W; Merten, MD; Picher, M; Saleh, A1
Dixon, CJ; Green, AK; Webb, TE; Woods, NM1
Nikbakht, MR; Stone, TW1
Carolan, BM; Harden, TK; Keef, KD; Mutafova-Yambolieva, VN1
Boeynaems, JM; Castro, E; Communi, D; Delicado, EG; Jiménez, AI; Miras-Portugal, MT1
Saino, T; Shinohe, Y1
Bültmann, R; Starke, K1
Banes, AJ; Elfervig, MK; Graff, RD; Kelley, SS; Lee, GM; Sood, A1
Bernardes, CF; Castilho, RF; Fagian, MM; Meyer-Fernandes, JR; Vercesi, AE1
Chiba, T; Lee, JH; Marcus, DC1
Imamura, H; Kido, M; Lu, K; Ninomiya, H; Otani, H; Uchiyama, T1
Bell, PD; Johansson, A; Kovacs, G; Liu, R; Persson, AE; Peti-Peterdi, J1
Katayama, T; Kawaguchi, N; Minami, M; Nakagawa, T; Nakamura, J; Ohtani, Y; Satoh, M; Yamakuni, H1
Mihaylova-Todorova, ST; Todorov, LD; Westfall, DP1
Chambers, JK; Emson, PC; Moore, DJ; Murdock, PR1
Hoyle, CH; Martín, S; Peláez, T; Peral, A; Pintor, J1
Alessandro, M; Mulè, F; Serio, R; Tamburello, MP; Zizzo, MG1
Laubinger, W; Reiser, G; Wang, H; Welte, T1
Allen, DG; Barden, JA; Huang, W; Jiang, L; Ju, YK1
Delbro, DS; Nordgren, S; Nylund, G1
Buljubasich, R; Ventura, S1
Fachinetto, R; Nogueira, CW; Rocha, JB; Savegnago, L1
Almeida, T; Cunha, RA; Oliveira, CR; Richardson, PJ; Rodrigues, RJ1
Hildebrandt, C; Horner, S; Kassack, MU; Lambrecht, G; Mahaut-Smith, MP; Menke, K; Nickel, P; Ullmann, H1
Burnstock, G; Cowen, T; Knight, GE; Wallace, A1
Barreto-Chaves, ML; Fürstenau, CR; Sarkis, JJ; Trentin, Dda S1
Bielarczyk, H; Jankowska-Kulawy, A; Klimaszewska, J; Michno, A; Pawełczyk, T; Szutowicz, A1
Housley, GD; Soeller, C; Thorne, PR; Vlajkovic, SM; Wang, CJ; Zimmermann, H1
Singleton, SF; Wigle, TJ1
Bowser, DN; Khakh, BS1
Kauffenstein, G; Kukulski, F; Lavoie, EG; Lecka, J; Legendre, C; Lévesque, SA; Munkonda, MN; Pelletier, J; Sévigny, J1
Almeida, ME; Libermann, TA; Rücker, B; Sarkis, JJ; Wink, MR; Zerbini, LF1
Avelino-Cruz, JE; Berra-Romani, R; Moccia, F; Oldani, A; Raqeeb, A; Speroni, F; Taglietti, V; Tanzi, F1
Günthner, T; Jalkanen, S; Jankowski, J; Jankowski, V; Yegutkin, GG; Zidek, W1
Cofan, M; Crumm, S; Hoek, JB; Juskeviciute, E1
Chow, JY; Dong, H; Dong, X; Insel, PA; Kim, HD; Ko, KH; Lee, J; Smoll, EJ1
Barrabin, H; Esteves, FF; Meyer-Fernandes, JR; Moreira, OC; Rios, PF1
Acheson, A; Eames, T; Mundey, M; Nisar, P; Rayment, S; Scholefield, J; Wilson, VG1
Grace, AA; Gurung, IS; Huang, CL; Kalin, A1
Baqi, Y; Glänzel, M; Hoffmann, K; Morena, MS; Müller, CE; von Kügelgen, I1
Andersson, M; Aronsson, P; Ericsson, T; Giglio, D1
Hempel, D; Kurup, IV; Masuda, I; Rosenthal, AK; Ryan, LM1
Kanjanamekanant, K; Luckprom, P; Pavasant, P1
Auld, DS; Blackburn, EA; Boxer, MB; Fothergill-Gilmore, LA; McNae, IW; Michels, PA; Morgan, HP; Nowicki, MW; Shen, M; Veith, H; Walkinshaw, MD; Walsh, MJ; Wear, MA1
Caruso-Neves, C; Costa-Alves, MS; Meyer-Fernandes, JR; Pinheiro, AA; Ribeiro, MC; Wengert, M; Zancan, P1
Bravo, CE; Capettini, LS; Carmo, AO; Chávez-Olórtegui, C; Gomes, MT; Horta, CC; Kalapothakis, E; Lemos, VS; Oliveira-Mendes, BB; Rezende, BA; Silva, JF1
Arakawa, T; Ito, M; Mizoguchi, I; Okayama, M; Shitara, A; Takuma, T1
Bao, Y; Chen, Y; Inoue, Y; Junger, WG; Li, X; Sumi, Y; Tanaka, H; Woehrle, T; Yao, Y1
Drumm, BT; Durnin, L; Hwang, SJ; Kurahashi, M; Mutafova-Yambolieva, VN; Sanders, KM; Sasse, KC; Ward, SM1
Gan, X; Hu, WP; Qiu, CY; Ren, C; Wu, J1
Adefegha, SA; Cabral, FL; Doleski, PH; Leal, DB1
Guo, B; Hu, F; Jiang, P; Lee, I; Li, Z; Pan, L; Wei, W; Xing, F; Xu, J; Yang, J; Zhang, X1
Caringal, H; Gongwer, M; Heer, C; Jacoby, J; Kaufman, R; Kreitzer, MA; Malchow, RP; Shepherd, L; Swygart, D; Tchernookova, BK; Young, M1
Hamaguchi, S; Kariya, M; Namekata, I; Ozaki, AF; Tanaka, H1

Reviews

1 review(s) available for adenosine diphosphate and suramin

ArticleYear
Purine and pyrimidine (P2) receptors as drug targets.
    Journal of medicinal chemistry, 2002, Sep-12, Volume: 45, Issue:19

    Topics: Adenosine Triphosphate; Animals; Drug Design; Humans; Ligands; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Pyrimidines; Receptors, Purinergic P2; Uridine Triphosphate

2002

Other Studies

99 other study(ies) available for adenosine diphosphate and suramin

ArticleYear
An examination of deoxyadenosine 5'(alpha-thio)triphosphate as a ligand to define P2Y receptors and its selectivity as a low potency partial agonist of the P2Y1 receptor.
    British journal of pharmacology, 1997, Volume: 121, Issue:2

    Topics: Adenosine Triphosphate; Dose-Response Relationship, Drug; Humans; Radioligand Assay; Receptors, Purinergic P2; Receptors, Purinergic P2Y1

1997
Quantitation of the P2Y(1) receptor with a high affinity radiolabeled antagonist.
    Molecular pharmacology, 2002, Volume: 62, Issue:5

    Topics: Adenosine Diphosphate; Animals; Cells, Cultured; Female; Humans; Insecta; Purinergic P2 Receptor Antagonists; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Tritium

2002
Pharmacological characterization of the human P2Y13 receptor.
    Molecular pharmacology, 2003, Volume: 64, Issue:1

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Cell Membrane; CHO Cells; Cricetinae; Cyclic AMP; Female; GTP-Binding Protein alpha Subunits, Gi-Go; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Inositol Phosphates; Kinetics; Receptors, Purinergic P2; Thionucleotides

2003
Stable adenine nucleotides inhibit [3H]-noradrenaline release in rabbit brain cortex slices by direct action at presynaptic adenosine A1-receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:2

    Topics: Adenine Nucleotides; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Cerebral Cortex; Drug Interactions; Drug Stability; Electric Stimulation; Female; Male; Nerve Endings; Norepinephrine; Purinergic Antagonists; Rabbits; Receptors, Purinergic; Suramin; Synapses; Theophylline; Tritium; Xanthines

1992
Effects of the P2-purinoceptor antagonist, suramin, on human platelet aggregation induced by adenosine 5'-diphosphate.
    British journal of pharmacology, 1992, Volume: 105, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adenosine Diphosphate; Blood Platelets; Humans; In Vitro Techniques; Platelet Aggregation; Platelet Aggregation Inhibitors; Prostaglandin Endoperoxides, Synthetic; Receptors, Purinergic; Serotonin; Suramin

1992
ATP modulates the efferent function of capsaicin-sensitive neurones in guinea-pig isolated atria.
    British journal of pharmacology, 1992, Volume: 105, Issue:3

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Electric Stimulation; Guinea Pigs; Heart Atria; In Vitro Techniques; Male; Neurons, Efferent; Receptors, Purinergic; Suramin; Theophylline

1992
Anion channel blockers cause apparent inhibition of exocytosis by reacting with agonist or secretory product, not with cell.
    Proceedings of the National Academy of Sciences of the United States of America, 1989, Volume: 86, Issue:15

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adenosine Diphosphate; Anions; Blood Platelets; Calcimycin; Cell Membrane; Collagen; Erythrocytes; Exocytosis; Humans; Ion Channels; Kinetics; Malondialdehyde; Serotonin; Stilbenes; Suramin; Thrombin

1989
Suramin: a reversible P2-purinoceptor antagonist in the mouse vas deferens.
    British journal of pharmacology, 1988, Volume: 93, Issue:2

    Topics: Adenosine Diphosphate; Animals; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Muscle Contraction; Muscle, Smooth; Receptors, Purinergic; Suramin

1988
Two different inhibitory effects of pyridoxalphosphate-6-azophenyl-2',4'-disulfonic acid on adenosine diphosphate-induced human platelet aggregation.
    Arzneimittel-Forschung, 1995, Volume: 45, Issue:9

    Topics: Adenosine Diphosphate; Humans; In Vitro Techniques; Platelet Aggregation; Platelet Aggregation Inhibitors; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Suramin

1995
Suramin and reactive blue 2 are antagonists for a newly identified purinoceptor on rat megakaryocyte.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Dose-Response Relationship, Drug; Electrophysiology; Female; Inositol 1,4,5-Trisphosphate; Ion Channels; Male; Megakaryocytes; Potassium; Protein Synthesis Inhibitors; Purinergic Antagonists; Rats; Rats, Wistar; Suramin; Thrombin; Triazines

1994
Evidence that tachykinin NK1 and NK2 receptors mediate non-adrenergic non-cholinergic excitation and contraction in the circular muscle of guinea-pig duodenum.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Action Potentials; Adenosine Diphosphate; Animals; Apamin; Arginine; Atropine; Dose-Response Relationship, Drug; Duodenum; Electric Stimulation; Guanethidine; Guinea Pigs; Indomethacin; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Nifedipine; Nitroarginine; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Physalaemin; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Suramin; Thionucleotides

1995
Additive effect of ADP and CGRP in modulation of the acetylcholine receptor channel in Xenopus embryonic myocytes.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Calcitonin Gene-Related Peptide; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Dibutyryl Cyclic GMP; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Activation; Heart; Myocardium; Patch-Clamp Techniques; Protein Kinase C; Receptors, Cholinergic; Receptors, Purinergic; Suramin; Tetradecanoylphorbol Acetate; Xenopus laevis

1995
Contribution of P2-purinoceptors to neurogenic contraction of rat urinary bladder smooth muscle.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Acetylcholine; Adenosine Diphosphate; Adenosine Triphosphate; Analysis of Variance; Animals; Atropine; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Isotonic Contraction; Male; Muscle, Smooth; Parasympatholytics; Protein Synthesis Inhibitors; Rats; Rats, Wistar; Receptors, Purinergic P2; Suramin; Thionucleotides; Triazines; Urinary Bladder

1995
P2-purinoceptor-mediated inhibition of noradrenaline release in rat atria.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Antihypertensive Agents; Atropine; Desipramine; Dose-Response Relationship, Drug; Electric Stimulation; Heart Atria; Indomethacin; Male; Norepinephrine; Phenethylamines; Protein Synthesis Inhibitors; Purinergic P1 Receptor Antagonists; Purinergic P2 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Receptors, Purinergic P2; Suramin; Triazines; Xanthines; Yohimbine

1995
Autoradiography of P2x ATP receptors in the rat brain.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Autoradiography; Binding, Competitive; Brain; Brain Stem; Cerebellum; Cerebral Cortex; Dilazep; Female; Hippocampus; Ligands; Male; Ouabain; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P2; Structure-Activity Relationship; Suramin; Thalamus; Thionucleotides

1995
ATP responses in the embryo chick ciliary ganglion cells.
    Neuroscience, 1995, Volume: 64, Issue:2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Calcium; Chick Embryo; Dose-Response Relationship, Drug; Electrophysiology; Ganglia, Parasympathetic; Patch-Clamp Techniques; Suramin

1995
Activation of specific ATP receptors induces a rapid increase in intracellular calcium ions in rat hypothalamic neurons.
    Brain research, 1994, Apr-04, Volume: 641, Issue:2

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Calcium; Cells, Cultured; Cytosol; Fetus; Guanosine Triphosphate; Hypothalamus; Kinetics; Neurons; Rats; Rats, Sprague-Dawley; Receptors, Neurotransmitter; Receptors, Purinergic P2; Structure-Activity Relationship; Suramin

1994
Purine- and nucleotide-mediated relaxation of rabbit thoracic aorta: common and different sites of action.
    The Journal of pharmacy and pharmacology, 1994, Volume: 46, Issue:5

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; In Vitro Techniques; Inosine; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nucleotides; Purines; Rabbits; Suramin; Uridine Triphosphate; Vasodilator Agents

1994
Effects of suramin on increases in cytosolic calcium and on inhibition of adenylate cyclase induced by adenosine 5'-diphosphate in human platelets.
    Biochemical pharmacology, 1994, Mar-15, Volume: 47, Issue:6

    Topics: Adenosine Diphosphate; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Alprostadil; Blood Platelets; Calcium; Cyclic AMP; Cytosol; Epinephrine; Humans; In Vitro Techniques; Suramin

1994
Differentiation of BA-HAN-1C rhabdomyosarcoma cells is controlled by a pertussis toxin sensitive signaling pathway.
    Cellular & molecular biology research, 1993, Volume: 39, Issue:3

    Topics: Adenosine Diphosphate; Animals; Cell Differentiation; Cell Transformation, Neoplastic; Cyclic AMP; Fibroblast Growth Factor 2; Gene Expression Regulation; GTP Phosphohydrolases; GTP-Binding Proteins; Muscles; Myogenin; Pertussis Toxin; Phenotype; Rats; Rhabdomyosarcoma; Ribose; Signal Transduction; Suramin; Tumor Cells, Cultured; Virulence Factors, Bordetella

1993
Nucleotides mobilize intracellular calcium stores of renal proximal cells in primary culture: existence of a suramin-sensitive mechanism.
    Biochimica et biophysica acta, 1993, Mar-10, Volume: 1176, Issue:1-2

    Topics: Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Bordetella pertussis; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Fura-2; Kidney Tubules, Proximal; Male; Nucleotides; Rabbits; Suramin

1993
Regulation of proliferation of LLC-MK2 cells by nucleosides and nucleotides: the role of ecto-enzymes.
    The Biochemical journal, 1996, Jun-01, Volume: 316 ( Pt 2)

    Topics: 5'-Nucleotidase; Acid Anhydride Hydrolases; Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Alkaline Phosphatase; Animals; Cell Division; Cell Line; Cell Line, Transformed; Dinucleoside Phosphates; Dipyridamole; Enzyme Inhibitors; HeLa Cells; Humans; Levamisole; Nucleoside-Triphosphatase; Nucleosides; Nucleotides; Suramin; Thymidine; Triazines

1996
Characterisation of a recombinant P2Y purinoceptor.
    European journal of pharmacology, 1995, Nov-30, Volume: 291, Issue:3

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Affinity Labels; Animals; Brain; Cell Line; Electrophysiology; Inositol Phosphates; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Recombinant Proteins; Suramin; Thionucleotides; Triazines; Uridine Triphosphate; Xenopus

1995
Relative contribution of P2U- and P2Y-purinoceptors to endothelium-dependent vasodilatation in the golden hamster isolated mesenteric arterial bed.
    British journal of pharmacology, 1996, Volume: 117, Issue:8

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Cricetinae; Endothelium, Vascular; Male; Mesenteric Arteries; Methoxamine; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Rats; Receptors, Purinergic P2; Suramin; Uridine Triphosphate; Vasoconstrictor Agents; Vasodilation

1996
ATP induces release of newly synthesized dopamine in the rat striatum.
    Neurochemistry international, 1996, Volume: 28, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenosine; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; alpha-Methyltyrosine; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Corpus Striatum; Dopamine; Homovanillic Acid; Kinetics; Male; Methyltyrosines; Microdialysis; Neurons; omega-Conotoxin GVIA; Peptides; Purinergic P2 Receptor Antagonists; Rats; Rats, Wistar; Reserpine; Suramin; Tetrodotoxin; Xanthines

1996
Evidence for two distinct P2-purinoceptors subserving contraction of the rat anococcygeus smooth muscle.
    British journal of pharmacology, 1996, Volume: 118, Issue:3

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Dose-Response Relationship, Drug; Male; Muscle Contraction; Muscle, Smooth; Rats; Rats, Sprague-Dawley; Receptors, Purinergic; Suramin

1996
P2-purinoceptor antagonists: III. Blockade of P2-purinoceptor subtypes and ecto-nucleotidases by compounds related to suramin.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 354, Issue:4

    Topics: Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Colon; Guinea Pigs; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Purinergic P2 Receptor Antagonists; Rats; Structure-Activity Relationship; Suramin; Thionucleotides; Vas Deferens

1996
The P2Y1 receptor is an ADP receptor antagonized by ATP and expressed in platelets and megakaryoblastic cells.
    FEBS letters, 1997, Feb-10, Volume: 403, Issue:1

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Binding, Competitive; Blood Platelets; Calcium; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Humans; Jurkat Cells; Megakaryocytes; Membrane Proteins; Polymerase Chain Reaction; Pyridoxal Phosphate; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Receptors, Purinergic P2Y12; Suramin

1997
Slow desensitization of the human P2Y6 receptor.
    European journal of pharmacology, 1997, Jun-25, Volume: 329, Issue:2-3

    Topics: Adenosine Diphosphate; GTP-Binding Proteins; Humans; Inositol 1,4,5-Trisphosphate; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Receptors, Purinergic P2; Suramin; Triazines; Tumor Cells, Cultured; Uridine Diphosphate

1997
P2 purinoceptor of the globular substance in the otoconial membrane of the guinea pig inner ear.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Calcium; Cells, Cultured; Enzyme Inhibitors; Estrenes; Guinea Pigs; Kinetics; Otolithic Membrane; PC12 Cells; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Pyrrolidinones; Rats; Receptors, Purinergic P2; Saccule and Utricle; Suramin; Triazines; Type C Phospholipases; Uridine Triphosphate

1997
Pharmacological evidence for the existence of multiple P2 receptors in the circular muscle of guinea-pig colon.
    British journal of pharmacology, 1998, Volume: 123, Issue:1

    Topics: Adenosine Diphosphate; Animals; Apamin; Autonomic Nervous System; Colon; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Platelet Aggregation Inhibitors; Purinergic P2 Receptor Agonists; Pyridoxal Phosphate; Receptors, Purinergic P2; Suramin; Thionucleotides; Vasodilator Agents

1998
Extracellular ATP directly gates a cation-selective channel in rabbit airway ciliated epithelial cells.
    The Journal of physiology, 1998, May-01, Volume: 508 ( Pt 3)

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Antineoplastic Agents; Barium Compounds; Cations, Divalent; Cesium; Chlorides; Cilia; Electric Conductivity; Electric Stimulation; Epithelial Cells; Extracellular Space; GTP-Binding Proteins; Ion Channel Gating; Ion Channels; Male; Mucous Membrane; Patch-Clamp Techniques; Rabbits; Receptors, Purinergic P2; Suramin; Tetraethylammonium; Trachea; Uridine Triphosphate

1998
Characterization of purinergic receptor-evoked increases in intracellular Ca2+ transients in isolated human and rodent insulin-secreting cells. Purinergic receptor signalling and [Ca2+]i in human beta-cells.
    Advances in experimental medicine and biology, 1997, Volume: 426

    Topics: Adenine Nucleotides; Adenosine; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Cadaver; Calcium; Cells, Cultured; Humans; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Models, Biological; Receptors, Purinergic; Rodentia; Signal Transduction; Suramin; Tissue Donors; Uridine Triphosphate

1997
Ecto-nucleotidases in isolated intact rat vagi, nodose ganglia, and superior cervical ganglia.
    Advances in experimental medicine and biology, 1998, Volume: 431

    Topics: Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Enzyme Inhibitors; Evoked Potentials; In Vitro Techniques; Male; Nodose Ganglion; Rats; Rats, Wistar; Superior Cervical Ganglion; Suramin; Vagus Nerve

1998
Pharmacological characterization of ATP receptors in ampulla from frog semicircular canal.
    The American journal of physiology, 1998, Volume: 275, Issue:1

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Binding, Competitive; Female; Kinetics; Male; Radioligand Assay; Rana ridibunda; Receptors, Purinergic P2; Semicircular Canals; Suramin; Thionucleotides

1998
Two types of relaxation-mediating P2 receptors in rat gastric circular muscle.
    Japanese journal of pharmacology, 1998, Volume: 78, Issue:2

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Antineoplastic Agents; Apamin; Dose-Response Relationship, Drug; Gastric Mucosa; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Platelet Aggregation Inhibitors; Pyridoxal Phosphate; Rats; Rats, Wistar; Receptors, Purinergic P2; Stomach; Suramin; Thionucleotides

1998
P2 purinoceptor localization along rat nephron and evidence suggesting existence of subtypes P2Y1 and P2Y2.
    The American journal of physiology, 1998, Volume: 274, Issue:6

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Calcium; Calcium Channel Blockers; Gallic Acid; Kidney Glomerulus; Kidney Tubules, Collecting; Male; Nephrons; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P2; Suramin; Thionucleotides; Uridine Triphosphate

1998
Stimulation of large-conductance Ca2+-activated K+ channels by Evans blue in cultured endothelial cells of human umbilical veins.
    Biochemical and biophysical research communications, 1999, Jan-27, Volume: 254, Issue:3

    Topics: Adenosine Diphosphate; Capillary Permeability; Cells, Cultured; Endothelium, Vascular; Evans Blue; Humans; Kinetics; Large-Conductance Calcium-Activated Potassium Channels; Membrane Potentials; Patch-Clamp Techniques; Potassium Channels; Potassium Channels, Calcium-Activated; Suramin; Umbilical Veins

1999
Ca2+-permeable P2X receptor channels in cultured rat retinal ganglion cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, May-01, Volume: 19, Issue:9

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Calcium; Cells, Cultured; Kinetics; Membrane Potentials; Patch-Clamp Techniques; Rats; Receptors, Purinergic P2; Regression Analysis; Retinal Ganglion Cells; Suramin

1999
P2 purinoceptors contribute to ATP-induced inhibition of L-type Ca2+ current in rabbit atrial myocytes.
    Cardiovascular research, 1999, Volume: 41, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 5'-Nucleotidase; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Adrenergic beta-Agonists; Animals; Calcium-Transporting ATPases; Colforsin; Cyclic AMP; Enzyme Inhibitors; Isoproterenol; Myocardium; Patch-Clamp Techniques; Pertussis Toxin; Potassium Channels; Potassium Channels, Voltage-Gated; Purinergic P1 Receptor Antagonists; Purinergic P2 Receptor Antagonists; Rabbits; Receptors, Purinergic P2; Shal Potassium Channels; Suramin; Virulence Factors, Bordetella; Xanthines

1999
Identification and characterization of P(1), P(7)-Di(adenosine-5')-heptaphosphate from human platelets.
    The Journal of biological chemistry, 1999, Aug-20, Volume: 274, Issue:34

    Topics: Adenosine Diphosphate; Animals; Blood Platelets; Dinucleoside Phosphates; Humans; Platelet Aggregation; Rats; Suramin; Thrombin; Vasoconstriction; Vasoconstrictor Agents

1999
Differential effects of adenine nucleotide analogues on shape change and aggregation induced by adnosine 5-diphosphate (ADP) in human platelets.
    British journal of pharmacology, 1999, Volume: 127, Issue:6

    Topics: Adenine Nucleotides; Adenosine Diphosphate; Adenosine Triphosphate; Blood Platelets; Cell Size; Dose-Response Relationship, Drug; Humans; Platelet Aggregation; Suramin; Thionucleotides; Trypanocidal Agents; Uridine Triphosphate

1999
Cross desensitizations on contractions by P2-agonists of guinea pig ileum.
    Japanese journal of pharmacology, 1999, Volume: 80, Issue:4

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Receptors, Purinergic P2; Suramin; Tetrodotoxin

1999
Different receptors mediating the inhibitory action of exogenous ATP and endogenously released purines on guinea-pig intestinal peristalsis.
    British journal of pharmacology, 1999, Volume: 128, Issue:2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Apamin; Female; Guinea Pigs; Ileum; In Vitro Techniques; Intestines; Male; Peristalsis; Purines; Pyridoxal Phosphate; Receptors, Purinergic; Receptors, Purinergic P2; Suramin; Thionucleotides

1999
Pharmacological characterization of the human P2Y11 receptor.
    British journal of pharmacology, 1999, Volume: 128, Issue:6

    Topics: Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; CHO Cells; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Humans; Inositol 1,4,5-Trisphosphate; Phosphoadenosine Phosphosulfate; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Recombinant Fusion Proteins; Suramin; Theophylline; Thionucleotides; Time Factors; Triazines; Tumor Cells, Cultured

1999
Characterization of a diadenosine tetraphosphate-receptor distinct from the ATP-purinoceptor in human tracheal gland cells.
    European journal of pharmacology, 1999, Nov-12, Volume: 384, Issue:1

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Binding, Competitive; Calcium; Cells, Cultured; Dinucleoside Phosphates; Dose-Response Relationship, Drug; Humans; Hydrolysis; Proteinase Inhibitory Proteins, Secretory; Proteins; Receptors, Purinergic P2; Secretory Leukocyte Peptidase Inhibitor; Suramin; Thionucleotides; Trachea

1999
Evidence that rat hepatocytes co-express functional P2Y1 and P2Y2 receptors.
    British journal of pharmacology, 2000, Volume: 129, Issue:4

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Calcium; DNA, Complementary; Liver; Male; Pyridoxal Phosphate; Rats; Rats, Wistar; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Suramin; Uridine Diphosphate; Uridine Triphosphate

2000
Complex hippocampal responses to ATP: fade due to nucleotidase inhibition and P2-receptor-mediated adenosine release.
    Brain research, 2000, Mar-31, Volume: 860, Issue:1-2

    Topics: 5'-Nucleotidase; Action Potentials; Adenosine; Adenosine Deaminase; Adenosine Diphosphate; Adenosine Triphosphate; Adenylyl Imidodiphosphate; Animals; Enzyme Inhibitors; Hippocampus; Male; Nerve Tissue Proteins; Rats; Rats, Wistar; Receptors, Purinergic P2; Suramin; Theophylline

2000
Multiple P2Y receptors mediate contraction in guinea pig mesenteric vein.
    General pharmacology, 2000, Volume: 34, Issue:2

    Topics: Adenine Nucleotides; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Guinea Pigs; In Vitro Techniques; Male; Mesenteric Artery, Inferior; Mesenteric Veins; Muscle Contraction; Muscle, Smooth, Vascular; Potassium Chloride; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Pyrimidine Nucleotides; Receptors, Purinergic P2; Receptors, Purinergic P2X; Suramin; Uridine Triphosphate

2000
Coexpression of several types of metabotropic nucleotide receptors in single cerebellar astrocytes.
    Journal of neurochemistry, 2000, Volume: 75, Issue:5

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Astrocytes; Calcium; Cells, Cultured; Cerebellum; Dose-Response Relationship, Drug; Intracellular Fluid; Pertussis Toxin; Protein Kinase C; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P2; Stimulation, Chemical; Suramin; Thionucleotides; Uridine Triphosphate; Virulence Factors, Bordetella

2000
Effects of ATP on intracellular calcium dynamics of the perineurium of peripheral nerve bundles.
    Histochemistry and cell biology, 2000, Volume: 114, Issue:6

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Anesthetics, Local; Animals; Antineoplastic Agents; Calcium; Enzyme Inhibitors; Glyburide; Hypoglycemic Agents; Lidocaine; Male; Microscopy, Confocal; Peripheral Nerves; Rats; Rats, Inbred WKY; Sciatic Nerve; Suramin; Tetraethylammonium; Tetrodotoxin; Thapsigargin; Triazines; Uridine Triphosphate

2000
Nucleotide-evoked relaxation of rat vas deferens--a possible role for endogenous ATP released upon alpha(1)-adrenoceptor stimulation.
    European journal of pharmacology, 2001, Jun-22, Volume: 422, Issue:1-3

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Apyrase; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Relaxation; Norepinephrine; Nucleotides; Potassium; Purinergic P1 Receptor Antagonists; Pyridoxal Phosphate; Pyrophosphatases; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Suramin; Theophylline; Thionucleotides; Triazines; Vas Deferens; Vasoconstrictor Agents

2001
ATP induces Ca(2+) signaling in human chondrons cultured in three-dimensional agarose films.
    Osteoarthritis and cartilage, 2001, Volume: 9, Issue:6

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Antineoplastic Agents; Calcium Signaling; Cells, Cultured; Chondrocytes; Dose-Response Relationship, Drug; Fura-2; Humans; Sepharose; Suramin; Uridine Triphosphate

2001
Suramin inhibits respiration and induces membrane permeability transition in isolated rat liver mitochondria.
    Toxicology, 2001, Dec-01, Volume: 169, Issue:1

    Topics: Adenosine Diphosphate; Animals; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Cell Membrane Permeability; Cell Respiration; Chelating Agents; Cyclosporine; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; Ethylmaleimide; Intracellular Membranes; Magnesium; Membrane Potentials; Mitochondria, Liver; Mitochondrial Swelling; Oxygen Consumption; Rats; Rats, Wistar; Sulfhydryl Reagents; Suramin; Trypanocidal Agents

2001
P2X2 receptor mediates stimulation of parasensory cation absorption by cochlear outer sulcus cells and vestibular transitional cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2001, Dec-01, Volume: 21, Issue:23

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Cations; Cochlea; Diffusion Chambers, Culture; Dose-Response Relationship, Drug; Flufenamic Acid; Gadolinium; Gerbillinae; Hearing; In Vitro Techniques; Ion Channels; Ion Transport; Microelectrodes; Physical Stimulation; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Receptors, Purinergic P2X2; Suramin; Uridine Diphosphate; Uridine Triphosphate; Vestibule, Labyrinth; Vibration

2001
Complementary role of extracellular ATP and adenosine in ischemic preconditioning in the rat heart.
    American journal of physiology. Heart and circulatory physiology, 2002, Volume: 282, Issue:5

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Coloring Agents; Extracellular Space; Ischemic Preconditioning; Male; Microdialysis; Organic Chemicals; Purinergic P1 Receptor Antagonists; Purinergic P2 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Receptors, Purinergic P2; Suramin; Theophylline; Ventricular Function, Left; Ventricular Pressure

2002
Purinergic receptor signaling at the basolateral membrane of macula densa cells.
    Journal of the American Society of Nephrology : JASN, 2002, Volume: 13, Issue:5

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Benzofurans; Calcium; Cytosol; Dose-Response Relationship, Drug; Estrenes; Female; Fura-2; Imidazoles; Kidney Glomerulus; Microscopy, Confocal; Pyrrolidinones; Rabbits; Receptors, Purinergic; Signal Transduction; Suramin; Thionucleotides; Uridine Triphosphate

2002
ATP induces leukemia inhibitory factor mRNA in cultured rat astrocytes.
    Journal of neuroimmunology, 2002, Volume: 129, Issue:1-2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Animals, Newborn; Astrocytes; Cells, Cultured; Central Nervous System; Dose-Response Relationship, Drug; Fetus; Growth Inhibitors; Interleukin-6; Leukemia Inhibitory Factor; Lymphokines; Microglia; Neurons; Neurotransmitter Agents; Pyridoxal Phosphate; Rats; Rats, Sprague-Dawley; Receptors, Neurotransmitter; Receptors, Purinergic; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; RNA, Messenger; Suramin; Uridine Triphosphate

2002
Enzyme kinetics and pharmacological characterization of nucleotidases released from the guinea pig isolated vas deferens during nerve stimulation: evidence for a soluble ecto-nucleoside triphosphate diphosphohydrolase-like ATPase and a soluble ecto-5'-nuc
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 302, Issue:3

    Topics: 5'-Nucleotidase; Adenine Nucleotides; Adenosine; Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Calcium; Chromatography, High Pressure Liquid; Electric Stimulation; Enzyme Inhibitors; Guinea Pigs; In Vitro Techniques; Kinetics; Magnesium; Male; Nucleotidases; Phosphoric Diester Hydrolases; Phosphoric Monoester Hydrolases; Plant Proteins; Pyrophosphatases; Suramin; Sympathetic Nervous System; Vas Deferens

2002
Human Ntera-2/D1 neuronal progenitor cells endogenously express a functional P2Y1 receptor.
    Neuropharmacology, 2002, Volume: 43, Issue:6

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Antineoplastic Agents; Blotting, Western; Calcium; Cell Membrane; Cells, Cultured; Cyclic AMP; Fluorescence; GTP-Binding Protein alpha Subunits, Gq-G11; Heterotrimeric GTP-Binding Proteins; Humans; Membrane Proteins; Mitogen-Activated Protein Kinases; Neurons; Platelet Aggregation Inhibitors; Pyridoxal Phosphate; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Receptors, Purinergic P2Y12; Receptors, Purinergic P2Y2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stem Cells; Suramin; Thionucleotides; Uridine Triphosphate

2002
Presence of diadenosine polyphosphates in the aqueous humor: their effect on intraocular pressure.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 304, Issue:1

    Topics: Adenine Nucleotides; Adenosine Diphosphate; Adenosine Monophosphate; Animals; Aqueous Humor; Chromatography, High Pressure Liquid; Intraocular Pressure; Kinetics; Male; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Rabbits; Structure-Activity Relationship; Suramin; Triazines

2003
Neurotransmitters involved in the fast inhibitory junction potentials in mouse distal colon.
    European journal of pharmacology, 2003, Jan-24, Volume: 460, Issue:2-3

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Apamin; Colon; Dose-Response Relationship, Drug; Male; Membrane Potentials; Mice; Neuromuscular Junction; Neuropeptides; Neurotransmitter Agents; NG-Nitroarginine Methyl Ester; Peptide Fragments; Pituitary Adenylate Cyclase-Activating Polypeptide; Suramin; Tetrodotoxin; Thionucleotides

2003
P2Y receptor specific for diadenosine tetraphosphate in lung: selective inhibition by suramin, PPADS, Ip5I, and not by MRS-2197.
    European journal of pharmacology, 2003, May-02, Volume: 468, Issue:1

    Topics: Adenosine Diphosphate; Animals; Calcium Channel Blockers; Calcium Signaling; Cells, Cultured; Dinucleoside Phosphates; Epithelial Cells; Humans; Lung; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Rats; Suramin

2003
ATP modulates intracellular Ca2+ and firing rate through a P2Y1 purinoceptor in cane toad pacemaker cells.
    The Journal of physiology, 2003, Nov-01, Volume: 552, Issue:Pt 3

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Biological Clocks; Blotting, Western; Bufo marinus; Calcium; Electrophysiology; Heart; Immunohistochemistry; Intracellular Membranes; Myocardium; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Sarcoplasmic Reticulum; Suramin; Thionucleotides; Type C Phospholipases

2003
Expression of P2Y2 purinoceptors in MCG 101 murine sarcoma cells, and HT-29 human colon carcinoma cells.
    Autonomic neuroscience : basic & clinical, 2004, May-31, Volume: 112, Issue:1-2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Antineoplastic Agents; Blotting, Western; Cell Line, Tumor; Colonic Neoplasms; Dose-Response Relationship, Drug; Drug Interactions; Gene Expression Regulation, Neoplastic; HT29 Cells; Humans; Hydrogen-Ion Concentration; Immunohistochemistry; Mice; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Sarcoma; Suramin; Time Factors; Uridine Triphosphate

2004
Adenosine 5'-triphosphate and noradrenaline are excitatory cotransmitters to the fibromuscular stroma of the guinea pig prostate gland.
    European journal of pharmacology, 2004, Sep-24, Volume: 499, Issue:3

    Topics: Actins; Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Atropine; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Immunohistochemistry; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Prazosin; Prostate; Receptors, Purinergic P2; Receptors, Purinergic P2X; Receptors, Purinergic P2X2; Receptors, Purinergic P2X4; Suramin; Tetrodotoxin; Thionucleotides

2004
Characterization of ATP and ADP hydrolysis activity in rat gastric mucosa.
    Cell biology international, 2005, Volume: 29, Issue:7

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Antigens, CD; Apyrase; Calcium; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gastric Mucosa; Hydrogen-Ion Concentration; Hydrolysis; In Vitro Techniques; Magnesium; Male; Rats; Rats, Wistar; Sodium Azide; Substrate Specificity; Suramin; Vanadates

2005
Dual presynaptic control by ATP of glutamate release via facilitatory P2X1, P2X2/3, and P2X3 and inhibitory P2Y1, P2Y2, and/or P2Y4 receptors in the rat hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Jul-06, Volume: 25, Issue:27

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Adenylyl Imidodiphosphate; Animals; Astrocytoma; Calcium; Cell Line; Cell Line, Tumor; Glutamic Acid; Hippocampus; Kidney; Male; Potassium; Pyramidal Cells; Pyridoxal Phosphate; Rats; Rats, Wistar; Receptors, Presynaptic; Receptors, Purinergic P2; Receptors, Purinergic P2X; Receptors, Purinergic P2X2; Receptors, Purinergic P2X3; Receptors, Purinergic P2Y1; Receptors, Purinergic P2Y2; Recombinant Fusion Proteins; RNA, Messenger; Subcellular Fractions; Suramin; Synaptosomes; Transfection; Triazines; Triazoles; Xanthines

2005
The novel suramin analogue NF864 selectively blocks P2X1 receptors in human platelets with potency in the low nanomolar range.
    Naunyn-Schmiedeberg's archives of pharmacology, 2005, Volume: 372, Issue:1

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Apyrase; Blood Platelets; Calcium; Cell Shape; Dose-Response Relationship, Drug; Humans; Least-Squares Analysis; Linear Models; Phenylmercury Compounds; Platelet Aggregation Inhibitors; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Receptors, Purinergic P2X; Receptors, Purinergic P2Y1; Suramin; Thionucleotides

2005
Changes in purinergic signalling in developing and ageing rat tail artery: importance for temperature control.
    Neuropharmacology, 2006, Volume: 50, Issue:2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Arteries; Dose-Response Relationship, Drug; Electric Stimulation; Immunohistochemistry; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P2; Regional Blood Flow; Signal Transduction; Suramin; Tail; Thionucleotides; Uridine Triphosphate

2006
Ecto-nucleotide pyrophosphatase/phosphodiesterase as part of a multiple system for nucleotide hydrolysis by platelets from rats: kinetic characterization and biochemical properties.
    Platelets, 2006, Volume: 17, Issue:2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Angiotensin II; Animals; Blood Platelets; Gadolinium; Hydrogen-Ion Concentration; Hydrolysis; Kinetics; Male; Nucleotides; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Pyrophosphatases; Rats; Rats, Wistar; Signal Transduction; Sodium Azide; Suramin; Thymidine Monophosphate

2006
Alterations of adenine nucleotide metabolism and function of blood platelets in patients with diabetes.
    Diabetes, 2007, Volume: 56, Issue:2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Amino Acids; Blood Platelets; Diabetes Mellitus; Dose-Response Relationship, Drug; Female; Humans; Hyperglycemia; Male; Middle Aged; Platelet Aggregation; Suramin; Thiobarbituric Acid Reactive Substances; Thrombin

2007
Activation-dependent trafficking of NTPDase2 in Chinese hamster ovary cells.
    The international journal of biochemistry & cell biology, 2007, Volume: 39, Issue:4

    Topics: Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Calcium; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Green Fluorescent Proteins; Hydrolysis; Intracellular Fluid; Microscopy, Confocal; Protein Transport; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Rats; Receptors, Purinergic P2; Recombinant Fusion Proteins; Suramin; Time Factors; Transfection; Uridine Diphosphate; Uridine Triphosphate

2007
Directed molecular screening for RecA ATPase inhibitors.
    Bioorganic & medicinal chemistry letters, 2007, Jun-15, Volume: 17, Issue:12

    Topics: Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Binding Sites; Biological Assay; DNA Gyrase; Drug Evaluation, Preclinical; Enzyme Inhibitors; Escherichia coli; Fluorescent Dyes; Hydrolysis; Nucleotides; Protein-Tyrosine Kinases; Rec A Recombinases; Sensitivity and Specificity; Suramin; Time Factors

2007
Vesicular ATP is the predominant cause of intercellular calcium waves in astrocytes.
    The Journal of general physiology, 2007, Volume: 129, Issue:6

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Aniline Compounds; Animals; Apyrase; Astrocytes; Brefeldin A; Calcium; Calcium Signaling; Cells, Cultured; Cytoplasmic Vesicles; Diffusion; Enzyme Inhibitors; Fluorescent Dyes; Hippocampus; Macrolides; Neurons; Paracrine Communication; Proton-Translocating ATPases; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Suramin; Time Factors; Xanthenes

2007
Inhibition of human and mouse plasma membrane bound NTPDases by P2 receptor antagonists.
    Biochemical pharmacology, 2007, Nov-15, Volume: 74, Issue:10

    Topics: Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Antigens, CD; Aorta, Thoracic; Apyrase; Benzenesulfonates; Cell Membrane; Chlorocebus aethiops; COS Cells; Humans; Hydrolysis; Mice; Mice, Knockout; Purinergic P2 Receptor Antagonists; Recombinant Proteins; Suramin; Transfection; Triazines

2007
E-NTPDases and ecto-5'-nucleotidase expression profile in rat heart left ventricle and the extracellular nucleotide hydrolysis by their nerve terminal endings.
    Life sciences, 2008, Feb-27, Volume: 82, Issue:9-10

    Topics: 5'-Nucleotidase; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Dose-Response Relationship, Drug; Extracellular Space; Gene Expression Profiling; Heart Ventricles; Hydrogen-Ion Concentration; Hydrolysis; Isoenzymes; Kinetics; Male; Myocardium; Nerve Endings; Nucleotides; Ouabain; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Sodium Azide; Suramin; Synaptosomes

2008
Ca2+ signaling in injured in situ endothelium of rat aorta.
    Cell calcium, 2008, Volume: 44, Issue:3

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Aorta, Abdominal; Aorta, Thoracic; Calcium Signaling; Endothelium, Vascular; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Rats; Receptors, Purinergic P2; Suramin

2008
Dinucleotide polyphosphates contribute to purinergic signalling via inhibition of adenylate kinase activity.
    Bioscience reports, 2008, Volume: 28, Issue:4

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Adenylate Kinase; Cells, Cultured; Dinucleoside Phosphates; Humans; Nucleotides; Signal Transduction; Suramin

2008
Adenine nucleotide changes in the remnant liver: An early signal for regeneration after partial hepatectomy.
    Hepatology (Baltimore, Md.), 2008, Volume: 48, Issue:3

    Topics: Adenine Nucleotides; Adenosine Diphosphate; Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Biomarkers; Blood Glucose; Hepatectomy; Liver; Liver Regeneration; Male; Mitochondria, Liver; Phentolamine; Proto-Oncogene Proteins c-fos; Purinergic Antagonists; Rats; Rats, Sprague-Dawley; Signal Transduction; Suramin

2008
P2Y receptors mediate Ca2+ signaling in duodenocytes and contribute to duodenal mucosal bicarbonate secretion.
    American journal of physiology. Gastrointestinal and liver physiology, 2009, Volume: 296, Issue:2

    Topics: Adenosine Diphosphate; Aminoquinolines; Animals; Bicarbonates; Boron Compounds; Calcium Channel Blockers; Calcium Signaling; Cell Line; Dogs; Duodenum; Epithelial Cells; Estrenes; Female; Hydrogen-Ion Concentration; Intestinal Mucosa; Intestinal Secretions; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Nifedipine; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Pyrrolidinones; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Suramin; Time Factors; Uridine Triphosphate

2009
CrATP as a new inhibitor of ecto-ATPases of trypanosomatids.
    Parasitology, 2009, Volume: 136, Issue:1

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Enzyme Inhibitors; Suramin; Time Factors; Trypanosomatina

2009
Investigation of the role of adrenergic and non-nitrergic, non-adrenergic neurotransmission in the sheep isolated internal anal sphincter.
    Neurogastroenterology and motility, 2009, Volume: 21, Issue:3

    Topics: Adenosine Diphosphate; Adrenergic alpha-Antagonists; Anal Canal; Animals; Anti-Arrhythmia Agents; Apamin; Bretylium Compounds; Electric Stimulation; Enzyme Inhibitors; Epinephrine; Humans; Muscle Contraction; Muscle Tonus; Neurotransmitter Agents; NG-Nitroarginine Methyl Ester; Nitric Oxide; Norepinephrine; Prazosin; Sheep; Stress, Mechanical; Suramin; Synaptic Transmission

2009
Activation of purinergic receptors by ATP induces ventricular tachycardia by membrane depolarization and modifications of Ca2+ homeostasis.
    Journal of molecular and cellular cardiology, 2009, Volume: 47, Issue:5

    Topics: Action Potentials; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Arrhythmias, Cardiac; Calcium; In Vitro Techniques; Membrane Potentials; Mice; Microscopy, Confocal; Myocytes, Cardiac; Patch-Clamp Techniques; Purinergic Agonists; Pyridoxal Phosphate; Receptors, Purinergic; Suramin; Tachycardia, Ventricular

2009
Interaction of new, very potent non-nucleotide antagonists with Arg256 of the human platelet P2Y12 receptor.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 331, Issue:2

    Topics: Adenosine Diphosphate; Animals; Arginine; Binding, Competitive; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cyclic AMP Response Element Modulator; Humans; Isomerism; Luciferases; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Receptors, Purinergic P2Y12; Sulfonic Acids; Suramin; Thionucleotides; Triazines

2009
Assessment and characterization of purinergic contractions and relaxations in the rat urinary bladder.
    Basic & clinical pharmacology & toxicology, 2010, Volume: 107, Issue:1

    Topics: Adenine Nucleotides; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Drug Antagonism; Electric Stimulation; Glyburide; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P2; Suramin; Theophylline; Uracil Nucleotides; Urinary Bladder; Xanthines

2010
Purine receptors modulate chondrocyte extracellular inorganic pyrophosphate production.
    Osteoarthritis and cartilage, 2010, Volume: 18, Issue:11

    Topics: Adenosine Diphosphate; Animals; Cartilage, Articular; Cells, Cultured; Chondrocytes; Cyclic AMP; Diphosphates; Purinergic P1 Receptor Agonists; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Receptors, Purinergic; RNA, Messenger; Suramin; Swine

2010
Mechanical stress-induced interleukin-1beta expression through adenosine triphosphate/P2X7 receptor activation in human periodontal ligament cells.
    Journal of periodontal research, 2013, Volume: 48, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Diphosphate; Adenosine Triphosphate; Apyrase; Benzenesulfonates; Calcium Channel Blockers; Calcium Signaling; Cell Culture Techniques; Cell Survival; Cells, Cultured; Coloring Agents; Dactinomycin; Homeostasis; Humans; Interleukin-1beta; Luminescent Measurements; Periodontal Ligament; Purinergic P2X Receptor Antagonists; Receptors, Purinergic P2X7; RNA, Small Interfering; Signal Transduction; Stress, Mechanical; Suramin; Tetrazolium Salts; Thiazoles; Time Factors; Up-Regulation

2013
A new family of covalent inhibitors block nucleotide binding to the active site of pyruvate kinase.
    The Biochemical journal, 2012, Nov-15, Volume: 448, Issue:1

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Arginine; Benzoates; Catalytic Domain; Conserved Sequence; Crystallography, X-Ray; Enzyme Inhibitors; High-Throughput Screening Assays; Humans; Isoenzymes; Leishmania mexicana; Lysine; Models, Molecular; Protein Binding; Protein Conformation; Pyruvate Kinase; Recombinant Proteins; Saccharin; Species Specificity; Structure-Activity Relationship; Suramin

2012
Characterization of ecto-ATPase activity in the surface of LLC-PK1 cells and its modulation by ischemic conditions.
    Biochimica et biophysica acta, 2012, Volume: 1820, Issue:12

    Topics: Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Antineoplastic Agents; Cells, Cultured; Hydrogen-Ion Concentration; Hydrolysis; Ischemia; Kidney Tubules, Proximal; Kinetics; L-Lactate Dehydrogenase; LLC-PK1 Cells; Suramin; Swine

2012
ADP is a vasodilator component from Lasiodora sp. mygalomorph spider venom.
    Toxicon : official journal of the International Society on Toxinology, 2013, Volume: 72

    Topics: Adenosine Diphosphate; Adenosine Monophosphate; Animals; Blotting, Western; Chemical Fractionation; Endothelium; In Vitro Techniques; Mass Spectrometry; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Nuclear Magnetic Resonance, Biomolecular; Phosphorylation; Rats; Spider Venoms; Spiders; Suramin; Vasodilation; Vasodilator Agents

2013
Gravity loading induces adenosine triphosphate release and phosphorylation of extracellular signal-regulated kinases in human periodontal ligament cells.
    Journal of investigative and clinical dentistry, 2014, Volume: 5, Issue:4

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Apyrase; Calcium; Cell Culture Techniques; Cells, Cultured; Centrifugation; Extracellular Signal-Regulated MAP Kinases; Fibroblasts; Gingiva; Gravitation; Humans; Periodontal Ligament; Phosphorylation; Purinergic Agonists; Purinergic Antagonists; Purinergic P2X Receptor Antagonists; Purinergic P2Y Receptor Antagonists; Receptors, Purinergic P2; Signal Transduction; Stress, Mechanical; Suramin

2014
Plasma ATP is required for neutrophil activation in a mouse sepsis model.
    Shock (Augusta, Ga.), 2014, Volume: 42, Issue:2

    Topics: Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Disease Models, Animal; Male; Mice, Inbred C57BL; Neutrophil Activation; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Sepsis; Suramin

2014
Uridine adenosine tetraphosphate is a novel neurogenic P2Y1 receptor activator in the gut.
    Proceedings of the National Academy of Sciences of the United States of America, 2014, Nov-04, Volume: 111, Issue:44

    Topics: Adenosine Diphosphate; Animals; Antineoplastic Agents; Colon; Deoxyadenine Nucleotides; Dinucleoside Phosphates; Gastrointestinal Motility; Humans; Mice; Mice, Knockout; Muscle Relaxation; Muscle, Smooth; Purinergic P2Y Receptor Agonists; Receptors, Purinergic P2Y1; Small-Conductance Calcium-Activated Potassium Channels; Suramin; Uridine Diphosphate

2014
Enhancement of acid-sensing ion channel activity by metabotropic P2Y UTP receptors in primary sensory neurons.
    Purinergic signalling, 2016, Volume: 12, Issue:1

    Topics: Acid Sensing Ion Channels; Acidosis; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Dose-Response Relationship, Drug; Ganglia, Spinal; Male; Membrane Potentials; Pain; Pain Measurement; Protons; Purinergic P2Y Receptor Agonists; Purinergic P2Y Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P2Y1; Sensory Receptor Cells; Signal Transduction; Suramin; Uridine Triphosphate

2016
Characterization of E-NTPDase (EC 3.6.1.5) activity in hepatic lymphocytes: A different activity profile from peripheral lymphocytes.
    Cell biochemistry and function, 2017, Volume: 35, Issue:2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Antigens, CD; Apyrase; Blood Cells; Calcium; Cations, Divalent; Cell Separation; Enzyme Assays; Enzyme Inhibitors; Gene Expression; Hydrogen-Ion Concentration; Kinetics; Liver; Lymphocytes; Male; Organ Specificity; Ouabain; Rats; Rats, Wistar; Sodium Azide; Substrate Specificity; Suramin; Vanadates

2017
Nucleotide transmitters ATP and ADP mediate intercellular calcium wave communication via P2Y12/13 receptors among BV-2 microglia.
    PloS one, 2017, Volume: 12, Issue:8

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Apyrase; Biomechanical Phenomena; Boron Compounds; Calcium; Calcium Signaling; Cell Communication; Cell Line, Transformed; Gene Expression; Inositol Phosphates; Mechanotransduction, Cellular; Mice; Microglia; Molecular Imaging; Receptors, Purinergic P2; Receptors, Purinergic P2Y12; Suramin; Thapsigargin

2017
Activation of retinal glial (Müller) cells by extracellular ATP induces pronounced increases in extracellular H+ flux.
    PloS one, 2018, Volume: 13, Issue:2

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adenosine Diphosphate; Adenosine Triphosphate; Ambystoma; Animals; Ependymoglial Cells; Extracellular Fluid; Humans; Hydrogen-Ion Concentration; Ictaluridae; In Vitro Techniques; Ion Transport; Lampreys; Macaca fascicularis; Macaca mulatta; Pyridoxal Phosphate; Rats; Receptors, Purinergic P2Y; Retina; Signal Transduction; Skates, Fish; Suramin

2018
Contribution of ATP-Mediated Positive Feedback to Sympathetic Nerve-Induced Positive Inotropy in Guinea Pig Ventricular Myocardium.
    Biological & pharmaceutical bulletin, 2021, Volume: 44, Issue:3

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Feedback, Physiological; Guinea Pigs; Heart Ventricles; Male; Muscle Contraction; Norepinephrine; Papillary Muscles; Prazosin; Propranolol; Pyridoxal Phosphate; Suramin; Sympathetic Nervous System; Ventricular Function

2021