adenosine diphosphate has been researched along with piperidines in 72 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 32 (44.44) | 18.7374 |
1990's | 15 (20.83) | 18.2507 |
2000's | 21 (29.17) | 29.6817 |
2010's | 4 (5.56) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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De Clerck, F; Van Gorp, L; Xhonneux, R | 1 |
Claxton, GP; Grisar, JM; Kariya, T; MacKenzie, RD; Stewart, KT | 1 |
Bond, SE; Dillingham, EO; Feng, Z; Gollamudi, R; Hill, RJ; Korfmacher, WA; Lyman, BA; Purcell, WP | 1 |
Karnovsky, ML; Polanski, M | 1 |
De Clerck, F; Xhonneux, B | 2 |
Bond, SE; Carter-Burks, G; Dillingham, EO; Gollamudi, R; Lasslo, A; Petrusewicz, J | 1 |
Kangasaho, M | 1 |
Bond, SE; Carter-Burks, G; Dillingham, EO; Gollamudi, R; Lasslo, A | 1 |
Arvidsson, S; Bergqvist, D; Haglund, U; Hedner, U; Lindblad, B | 1 |
Affolter, H; Burkard, WP; Pletscher, A | 1 |
Blohm, TR; MacKenzie, RD; Steinbach, JM | 1 |
Bellani, D; Gibelli, A; Montanari, C; Sacchetti, G | 1 |
Brinkhous, KM; Mason, RG; Rodman, NF | 1 |
Gergely, J; Seidel, JC | 1 |
Rozenberg, MC; Walker, CM | 1 |
Prevost, SC; Stone, DB | 1 |
Azzi, A; Bragadin, MA; Santato, M; Tamburro, AM | 1 |
Drott, HR; Santiago, D; Shore, JD | 1 |
Andree, PJ; Zantema, A | 1 |
Blumenfeld, LA; Ignatéva, LG | 1 |
Revina, TA; Ryzhov, AI; Sal'nik, BIu; Saratikov, AS | 1 |
Ackles, KN; Inwood, MJ; Philp, RB; Radomski, MW | 1 |
Lecrubier, C; Samama, M; Uzan, A | 1 |
Belamarich, FA; Simoneit, LW | 1 |
Rifkin, PL; Zucker, MB | 1 |
Claxton, GP; Fleming, RW; Grisar, JM; Roberts, EM | 1 |
Elslager, EF; Haley, NF; McLean, JR; Perricone, SC; Potoczak, D; Veloso, H; Worth, DF | 1 |
Dugdale, M; Johnson, RW; Lasslo, A; Naylor, JL; Quintana, RP | 1 |
Apprill, P; Ashton, J; Buja, LM; Bush, LR; Campbell, WB; Kern, K; Schmitz, J; Tilton, GD; Willerson, JT | 1 |
Bevan, J; Heptinstall, S | 1 |
De Clerck, F; Janssen, PA; Leysen, J; Xhonneux, B | 1 |
De Clerck, F; Van Nueten, JM | 1 |
de Gaetano, G; Lampugnani, MG | 1 |
Bond, SE; Dillingham, EO; Gollamudi, R | 1 |
Heptinstall, S; Lösche, W; Sanderson, HM; Vickers, J | 1 |
Bylund, R; Eriksson, U; Gustafsson, D; Gyzander, E; Teger-Nilsson, AC | 1 |
Chen, PS; Rees, H; Sluka, KA; Tsuruoka, M; Willis, WD | 1 |
Badorc, A; Bernat, A; Bordes, MF; de Cointet, P; Herbert, JM; Lalé, A; Maffrand, JP; Petitou, M; Savi, P | 1 |
Cook, JJ; Ellis, JD; Hand, EL; Holahan, MA; Prueksaritanont, T; Sitko, GR; Stranieri, MT | 1 |
Herbert, JM; Jeske, WP; Savi, P; Walenga, JM | 1 |
Heptinstall, S; Storey, RF; Wilcox, RG | 1 |
Hérault, JP; Herbert, JM; Li, N; Savi, P; Wallén, NH | 1 |
Asano, N; Miwa, I; Taniguchi, S; Tomino, F | 1 |
Goggin, T; Machin, SJ; Mackie, IJ; Timm, U; Wittke, B; Zell, M | 1 |
Bernat, A; Herbert, JM; Hoffmann, P; Lalé, A; Savi, P | 1 |
Ayukawa, O; Kariyazono, H; Moriyama, Y; Nakamura, K; Shinkawa, T; Taira, A; Toyohira, H; Yamada, K; Yamaguchi, T; Yamashita, T; Yotsumoto, G | 1 |
Farkas, B; Literati-Nagy, P; Sumegi, B; Szabados, E | 1 |
Modi, NB; Novotny, W; Reimann, JD | 1 |
Bernat, A; Herbert, JM; Lalé, A; Roque, C; Savi, P; Zamboni, G | 1 |
Asai, F; Iwamura, R; Koike, H; Ogawa, T; Otsuguro, K; Sugidachi, A; Yoneda, K | 1 |
Bari, M; Del Principe, D; Finazzi-Agrò, A; Giuliani, E; MacCarrone, M; Menichelli, A | 1 |
Fareed, J; Herbert, JM; Herring, J; Hoppensteadt, DA; Jeske, W; Orcullo Santillan, MK | 1 |
Kendall, DA; Ralevic, V | 1 |
Ashcroft, FM; Dabrowski, M; Holmes, WE; Wahl, P | 1 |
Boncler, M; Golanski, J; Rozalski, M; Watala, C | 1 |
Bernath, S; Csete, B; Farkas, B; Literáti Nagy, P; Magyarlaki, M; Nemeth, J; Rabloczky, G; Sümegi, B | 1 |
Akamatsu, S; Hisamichi, N; Ichihara, M; Inagaki, O; Kaku, S; Kawasaki, T; Matsumoto, Y; Moritani, Y; Nii, T; Sato, K; Shigenaga, T; Suzuki, Ki; Tomioka, K; Yanagisawa, I | 1 |
Bryckaert, M; Contreres, JO; Dupuy, E; Habib, A; Herbert, JM; Job, B; Levy-Toledano, S; Rosa, JP; Savi, P; Simoneau, G | 1 |
Altomare, C; Carotti, A; Carrieri, A; Cellamare, S; de Candia, M; Nardecchia, A; Summo, L | 1 |
Aalto, KT; Aito, H; Raivio, KO | 1 |
Best, D; Jarvis, GE; Watson, SP | 1 |
Ishisaki, A; Kitajima, Y; Kozawa, O; Matsuno, H; Tokuda, H; Zhou, Y | 1 |
Hjemdahl, P; Ostenson, CG; Wallén, NH; Yngen, M | 1 |
Bugert, P; Klüter, H; Schedel, A; Schloss, P | 1 |
Carbery, T; Geddes, JW; Nasr, P | 1 |
Bornstein, JC; Gwynne, RM | 1 |
Naidu, KA; Raghavendra, RH | 1 |
Godbole, MM; Misra, K; Singh, DV | 1 |
Chang, M; Hua, J; Huang, CS; L'Heureux, A; Lam, PY; Lapointe, P; Martel, A; Price, LA; Qiao, JX; Rehfuss, R; Ruel, R; Thibeault, C; Wexler, RR; Wu, Q; Zheng, J | 1 |
Burbury, K; Cole-Sinclair, M; Filshie, R; Horton, L; Kamel, S; Keating, MJ; Khot, A; Levade, M; Nandurkar, H; Reynolds, J; Sandhu, S; Schischka, S; Tam, CS; Tan, S; Ysebaert, L | 1 |
Bergmeier, W; Conley, PB; Lee, RH; Piatt, R | 1 |
6 trial(s) available for adenosine diphosphate and piperidines
Article | Year |
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Effects of decompression on platelets and hemostasis in men and the influence of antiplatelet drugs (RA233 and VK744).
Topics: Adenosine Diphosphate; Adult; Aspartate Aminotransferases; Atmosphere Exposure Chambers; Atmospheric Pressure; Blood Cell Count; Blood Platelets; Cholinesterases; Clinical Trials as Topic; Creatine Kinase; Decompression Sickness; Epinephrine; Ethanolamines; Hematopoiesis; Hemostasis; Humans; L-Lactate Dehydrogenase; Male; Morpholines; Piperidines; Platelet Adhesiveness; Pyrimidines; Thiophenes; Thrombin; Thrombocytopenia; Time Factors | 1974 |
Effect of SR121566A, a potent GP IIb-IIIa antagonist, on the HIT serum/heparin-induced platelet mediated activation of human endothelial cells.
Topics: Adenosine Diphosphate; Antibodies; Benzylamines; Cytokines; Endothelium, Vascular; Heparin; Humans; Membrane Proteins; Piperidines; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Reference Values; Risk Factors; Serotonin; Thiazoles; Thrombocytopenia | 1998 |
Differential effects of glycoprotein IIb/IIIa antagonists on platelet microaggregate and macroaggregate formation and effect of anticoagulant on antagonist potency. Implications for assay methodology and comparison of different antagonists.
Topics: Adenosine Diphosphate; Anticoagulants; Citrates; Collagen; Eptifibatide; Hirudins; Humans; Nephelometry and Turbidimetry; Oligopeptides; Peptides; Peptides, Cyclic; Piperazines; Piperidines; Platelet Aggregation Inhibitors; Platelet Count; Platelet Glycoprotein GPIIb-IIIa Complex; Sodium Citrate; Thiazolidines | 1998 |
Pharmacokinetics and pharmacodynamics of Ro 44-3888 after single ascending oral doses of sibrafiban, an oral platelet aggregation inhibitor, in healthy male volunteers.
Topics: Adenosine Diphosphate; Administration, Oral; Adult; Amidines; Area Under Curve; Contusions; Dose-Response Relationship, Drug; Double-Blind Method; Heterocyclic Compounds; Humans; Male; Oximes; Peptide Fragments; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Prodrugs; Receptors, Thrombin | 1999 |
Pharmacokinetics and pharmacodynamics of sibrafiban, an orally administered GP IIb/IIIa antagonist, following coadministration of aspirin and heparin.
Topics: Adenosine Diphosphate; Administration, Oral; Adult; Anticoagulants; Area Under Curve; Aspirin; Bleeding Time; Cross-Over Studies; Drug Interactions; Female; Heparin; Humans; Male; Middle Aged; Oximes; Partial Thromboplastin Time; Peptide Fragments; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Prodrugs; Prothrombin Time; Receptors, Thrombin | 2000 |
Meal-induced platelet activation in Type 2 diabetes mellitus: effects of treatment with repaglinide and glibenclamide.
Topics: Adenosine Diphosphate; Blood Glucose; C-Reactive Protein; Carbamates; Cross-Over Studies; Diabetes Mellitus, Type 2; Eating; Fasting; Female; Glyburide; Humans; Hypoglycemic Agents; Insulin; Intercellular Adhesion Molecule-1; Male; Middle Aged; P-Selectin; Piperidines; Platelet Activation; Platelet Function Tests; Postprandial Period; Treatment Outcome; von Willebrand Factor | 2006 |
66 other study(ies) available for adenosine diphosphate and piperidines
Article | Year |
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Effect of lorcainide, a new antiarrhythmic compound, on the changes in heart rhythm induced by intravenous injection of adenosine-5'-diphosphate in rats.
Topics: Acetamides; Adenosine Diphosphate; Animals; Anti-Arrhythmia Agents; Aprindine; Arrhythmias, Cardiac; Benzeneacetamides; Drug Interactions; Heart Rate; Lidocaine; Male; Piperidines; Procaine; Propanolamines; Rats; Thrombocytopenia; Time Factors | 1978 |
(2-Piperidine)- and (2-pyrrolidine)ethanones and -ethanols as inhibitors of blood platelet aggregation.
Topics: Adenosine Diphosphate; Animals; Blood Platelets; Cholestadienols; Cholesterol; Depression, Chemical; Dogs; Ethanol; Guinea Pigs; Humans; In Vitro Techniques; Male; Piperidines; Platelet Aggregation; Platelet Factor 3; Pyrrolidines; Rats; Structure-Activity Relationship | 1976 |
Molecular determinants of the platelet aggregation inhibitory activity of carbamoylpiperidines.
Topics: Adenosine Diphosphate; Carbamates; Chromatography, High Pressure Liquid; Collagen; Models, Molecular; Piperidines; Platelet Aggregation Inhibitors; Stereoisomerism; Structure-Activity Relationship | 1992 |
Serotonergic aspects of the response of human platelets to immune-adjuvant muramyl dipeptide.
Topics: Acetylmuramyl-Alanyl-Isoglutamine; Adenosine Diphosphate; Adjuvants, Immunologic; Blood Platelets; Carrier Proteins; Humans; Imipramine; Ketanserin; Lysergic Acid Diethylamide; Paroxetine; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1992 |
Continuous inhibition of platelet S2-serotonergic receptors during chronic administration of ketanserin in humans.
Topics: Adenosine Diphosphate; Blood Platelets; Collagen; Epinephrine; Female; Humans; Ketanserin; Male; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin Antagonists; Time Factors | 1985 |
Relationships between chemical structure and inhibition of epinephrine-induced human blood platelet aggregation.
Topics: Adenosine Diphosphate; Epinephrine; Humans; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Structure-Activity Relationship; Yohimbine | 1989 |
Effects of lidocaine, codeine and vadocaine hydrochloride on platelet aggregation in human platelet-rich plasma.
Topics: Adenosine Diphosphate; Alprostadil; Antitussive Agents; Bucladesine; Codeine; Female; Humans; In Vitro Techniques; Lidocaine; Male; Piperidines; Platelet Aggregation; Thromboxane B2 | 1988 |
Relationships between chemical structure and inhibition of ADP-stimulated human thrombocyte release of serotonin and platelet factor 4.
Topics: Adenosine Diphosphate; Blood Platelets; Humans; Molecular Probes; Piperazines; Piperidines; Platelet Aggregation; Platelet Factor 4; Serotonin; Structure-Activity Relationship | 1989 |
Effects of ketanserin, a selective 5-HT2 serotonergic antagonist, on the secondary recruitment of human platelets in vitro.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Blood Platelets; Collagen; Epinephrine; Humans; Ketanserin; Kinetics; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1986 |
The influence of ketanserin on hemostasis in vitro.
Topics: Adenosine Diphosphate; Adult; Blood Coagulation; Collagen; Epinephrine; Female; Fibrinolysis; Hemostasis; Humans; In Vitro Techniques; Ketanserin; Male; Piperidines; Platelet Aggregation; Serotonin Antagonists | 1986 |
Verapamil, an antagonist at 5-hydroxytryptamine receptors of human blood platelets.
Topics: Adenosine Diphosphate; Binding, Competitive; Blood Platelets; Cerebral Cortex; Gallopamil; Humans; In Vitro Techniques; Ketanserin; Membranes; Piperidines; Receptors, Serotonin; Spiperone; Verapamil | 1985 |
Effects in vivo of -(p-(fluoren-9-ylidenemethyl)phenyl)-2-piperidineethanol (RMI 10,393) on platelet aggregation and blood coagulation.
Topics: Adenosine Diphosphate; Animals; Blood Coagulation; Blood Coagulation Tests; Collagen; Dicumarol; Epinephrine; Ethanol; Fluorenes; Guinea Pigs; Male; Phenylbutazone; Piperidines; Platelet Adhesiveness; Rats; Serotonin Antagonists; Thrombin | 1972 |
Effects "in vitro" of some cardiovascular drugs and other agents on human platelet aggregation.
Topics: Adenosine Diphosphate; Adrenergic beta-Antagonists; Aniline Compounds; Humans; In Vitro Techniques; Indoles; Isoproterenol; Male; Norepinephrine; Papaverine; Phentolamine; Piperidines; Platelet Adhesiveness | 1973 |
Effect of a new antiaggregating chemical on the structure and function of the human platelet.
Topics: Adenosine Diphosphate; Adenosine Triphosphatases; Adenylyl Cyclases; Blood Platelets; Cell Aggregation; Cholinesterases; Clot Retraction; Collagen; Electrophoresis; Epinephrine; Ethanol; Humans; In Vitro Techniques; Microscopy, Electron; Piperidines; Thrombin | 1971 |
The conformation of myosin during the steady state of ATP hydrolysis: studies with myosin spin labeled at the S 1 thiol groups.
Topics: Acetamides; Adenosine Diphosphate; Adenosine Triphosphate; Chlorides; Cyclic N-Oxides; Electron Spin Resonance Spectroscopy; Hydrolysis; Iodoacetates; Kinetics; Magnesium; Muscle Proteins; Myosins; Piperidines; Protein Binding; Protein Conformation; Sulfhydryl Compounds | 1971 |
The effect of pyrimidine compounds on the potentiation of adenosine inhibition of aggregation, on adenosine phosphorylation and phosphodiesterase activity of blood platelets.
Topics: Adenosine; Adenosine Diphosphate; Adenosine Monophosphate; Blood Platelets; Carbon Isotopes; Cyclic AMP; Dipyridamole; Ethanolamines; Ethylamines; Humans; In Vitro Techniques; Morpholines; Phosphoric Diester Hydrolases; Piperidines; Platelet Adhesiveness; Pyrimidines; Thiophenes | 1973 |
Characterization of modified myosin at low ionic strength. Enzymatic and spin-label studies.
Topics: Actins; Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Butanols; Chloromercuribenzoates; Cyclic N-Oxides; Electron Spin Resonance Spectroscopy; Enzyme Activation; Hydrogen-Ion Concentration; Hydrolysis; Inosine Nucleotides; Iodoacetates; Magnesium; Muscle Contraction; Myosin Subfragments; Myosins; Osmolar Concentration; Piperidines; Protein Conformation; Rabbits; Spectrophotometry; Spin Labels; Sulfhydryl Reagents | 1973 |
Site-directed spin labeling of the mitochondrial membrane. Synthesis and utilization of the adenosine triphosphatase inhibitor (N-(2, 2, 6, 6-tetramethyl-piperidyl-1-oxyl)-N'-(cyclohexyl)-carbodiimide).
Topics: Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Binding Sites; Carbodiimides; Cattle; Cyclic N-Oxides; Electron Spin Resonance Spectroscopy; Hydrogen-Ion Concentration; Kinetics; Manganese; Mathematics; Membranes; Mitochondria, Muscle; Myocardium; Piperidines; Protein Binding; Spectrophotometry, Infrared; Spin Labels; Temperature; Time Factors | 1973 |
Electron paramagnetic resonance study of the interaction of a spin-labeled analog of adenosine diphosphoribose with paramagnetic cobalt(II) liver alcohol dehydrogenase.
Topics: Adenosine Diphosphate; Alcohol Oxidoreductases; Animals; Binding Sites; Cobalt; Electron Spin Resonance Spectroscopy; Liver; Mathematics; NAD; Nucleoside Diphosphate Sugars; Oxidation-Reduction; Piperidines; Protein Binding; Protein Conformation; Pyrazoles; Ribose; Spectrometry, Fluorescence; Spectrophotometry, Atomic; Spectrophotometry, Ultraviolet; Spin Labels; Temperature; Time Factors; Zinc | 1974 |
Magnetic resonance studies on glutamate dehydrogenase.
Topics: Adenosine Diphosphate; Binding Sites; Deuterium; Electron Spin Resonance Spectroscopy; Glutamate Dehydrogenase; Guanine Nucleotides; Iodoacetates; Ketoglutaric Acids; Kinetics; Magnetic Resonance Spectroscopy; Molecular Conformation; NAD; Oxidation-Reduction; Piperidines; Protein Binding; Protein Conformation; Spin Labels | 1974 |
Conformational changes in myosin under ATP hydrolysis.
Topics: Acetates; Adenosine Diphosphate; Adenosine Triphosphate; Binding Sites; Electron Spin Resonance Spectroscopy; Hydrolysis; Kinetics; Myosins; Piperidines; Protein Conformation; Spin Labels; Sulfhydryl Compounds | 1974 |
[Effect of pyridrol on energy metabolism in the brain during prolonged muscular activity].
Topics: Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Brain; Cytochromes; Glucose; Glycogen; Hexokinase; Lactates; Mitochondria; Oxidative Phosphorylation; Oxidoreductases; Phosphocreatine; Physical Exertion; Piperidines; Rats; Succinate Dehydrogenase | 1971 |
[Effect of a new cerebral vasodilator agent, viquidil, on the aggregation of blood platelets].
Topics: Adenosine Diphosphate; Animals; Blood Platelets; Cell Aggregation; Collagen; Dogs; Epinephrine; Humans; Ketones; Male; Papaverine; Piperidines; Quinolines; Vasodilator Agents; Vinyl Compounds | 1972 |
Aggregation of duck thrombocytes by 5-hydroxytryptamine.
Topics: Adenosine; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Blood Platelets; Dose-Response Relationship, Drug; Ducks; Methysergide; Piperidines; Platelet Adhesiveness; Prostaglandins; Pyrimidines; Serotonin | 1973 |
The effect of dipyridamole and RA 233 on human platelet function in vitro.
Topics: Adenosine; Adenosine Diphosphate; Blood Platelets; Dipyridamole; Erythrocytes; Ethanolamines; Humans; Piperidines; Platelet Adhesiveness; Pyrimidines | 1973 |
Synthesis of -(p-(fluoren-9-ylidenemethyl)phenyl)-2-piperidineethanol, an inhibitor of platelet aggregation.
Topics: Adenosine Diphosphate; Animals; Blood Coagulation; Collagen; Depression, Chemical; Ethanol; Fluorenes; Guinea Pigs; Humans; Infrared Rays; Piperidines; Platelet Adhesiveness; Spectrum Analysis; Stereoisomerism; Structure-Activity Relationship; Thrombin; Ultraviolet Rays | 1972 |
Inhibitors of platelet aggregation. 2. 9-((Dialkylamino)alkyl)thio-3-(dimethylamino)acridines and related acridine derivatives.
Topics: Acridines; Adenosine Diphosphate; Aniline Compounds; Animals; Anticoagulants; Blood Coagulation; Drug Antagonism; In Vitro Techniques; Mesentery; Methylamines; Morpholines; Piperidines; Platelet Adhesiveness; Pyridines; Pyrrolidines; Quinolines; Rabbits; Structure-Activity Relationship; Sulfides | 1971 |
Relationships between the chemical constitution of aggregation inhibitors and human blood platelet response profile.
Topics: Adenosine Diphosphate; Arachidonic Acid; Arachidonic Acids; Aspirin; Calcimycin; Calcium; Calcium Channel Blockers; Carbamates; Chlorpromazine; Gallic Acid; Humans; In Vitro Techniques; Piperidines; Platelet Aggregation; Propranolol; Thrombin | 1984 |
The effects of alpha 2-adrenergic and serotonergic receptor antagonists on cyclic blood flow alterations in stenosed canine coronary arteries.
Topics: Adenosine Diphosphate; Animals; Blood Flow Velocity; Coronary Circulation; Coronary Disease; Dogs; Female; Heart Rate; Hemodynamics; Ketanserin; Male; Piperidines; Platelet Aggregation; Prazosin; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Yohimbine | 1984 |
Effects of ketanserin and mepyramine on platelet aggregation and on the uptake of 5-hydroxytryptamine into platelets.
Topics: Adenosine Diphosphate; Aminopyridines; Blood Platelets; Humans; Ketanserin; Piperidines; Platelet Aggregation; Pyrilamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1983 |
The involvement of 5-HT2-receptor sites in the activation of cat platelets.
Topics: Adenosine Diphosphate; Animals; Blood Platelets; Cats; Collagen; Dose-Response Relationship, Drug; Ketanserin; Kinetics; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin | 1984 |
Platelet-mediated vascular contractions: inhibition of the serotonergic component by ketanserin.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Depression, Chemical; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Suprofen; Thrombin | 1982 |
Comparative effects of ketanserin, a novel serotonergic receptor antagonist, on 5HT-induced shape change and 5HT uptake in rat and human platelets.
Topics: Adenosine Diphosphate; Animals; Blood Platelets; Clomipramine; Female; Humans; In Vitro Techniques; Ketanserin; Kinetics; Male; Methysergide; Piperidines; Rats; Serotonin; Serotonin Antagonists | 1982 |
Inhibition of agonist-induced rise in platelet Ca2+ by antithrombotic nipecotamides.
Topics: Adenosine Diphosphate; Adult; Blood Platelets; Calcium; Collagen; Egtazic Acid; Female; Fibrinolytic Agents; Humans; Male; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Stereoisomerism | 1994 |
Studies on the effects of agonists and antagonists on platelet shape change and platelet aggregation in whole blood.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adenosine Diphosphate; Adenosine Triphosphate; Azepines; Blood Platelets; Humans; In Vitro Techniques; Piperazines; Piperidines; Platelet Activating Factor; Platelet Aggregation; Platelet Aggregation Inhibitors; Prostaglandin Endoperoxides, Synthetic; Serotonin; Succinates; Sulfonamides; Thromboxane A2; Triazoles; Vasoconstrictor Agents | 1996 |
In vitro effects of inogatran, a selective low molecular weight thrombin inhibitor.
Topics: Adenosine Diphosphate; Animals; Antithrombins; Collagen; Dogs; Fibrinolysis; Glycine; Humans; Kinetics; Male; Piperidines; Platelet Aggregation; Rats; Rats, Sprague-Dawley; Serine Endopeptidases; Thrombin; Thrombin Time | 1997 |
Inhibitors of G-proteins and protein kinases reduce the sensitization to mechanical stimulation and the desensitization to heat of spinothalamic tract neurons induced by intradermal injection of capsaicin in the primate.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Diphosphate; Animals; Capsaicin; Enzyme Inhibitors; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Haplorhini; Hot Temperature; Injections, Intradermal; Isoquinolines; Microdialysis; Nerve Fibers; Neural Pathways; Physical Stimulation; Piperidines; Protein Kinase Inhibitors; Spinal Cord; Sulfonamides; Thalamus; Thionucleotides | 1997 |
New orally active non-peptide fibrinogen receptor (GpIIb-IIIa) antagonists: identification of ethyl 3-[N-[4-[4-[amino[(ethoxycarbonyl) imino]methyl]phenyl]-1,3-thiazol-2-yl]-N-[1-[(ethoxycarbonyl)methyl]pip erid -4-yl]amino]propionate (SR 121787) as a pot
Topics: Adenosine Diphosphate; Administration, Oral; Animals; Benzylamines; Fibrinogen; Fibrinolytic Agents; Humans; Molecular Structure; Papio; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Protein Binding; Thiazoles | 1997 |
Effects of pentobarbital on pharmacokinetics and pharmacodynamics of a potent fibrinogen receptor antagonist, L-734,217, in dogs.
Topics: Adenosine Diphosphate; Adjuvants, Anesthesia; Animals; Area Under Curve; beta-Alanine; Collagen; Cross-Over Studies; Dogs; Dose-Response Relationship, Drug; Half-Life; Injections, Intravenous; Male; Pentobarbital; Piperidines; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Radioimmunoassay | 1997 |
Effects of a new platelet glycoprotein IIb/IIIa antagonist, SR121566, on platelet activation, platelet-leukocyte interaction and thrombin generation.
Topics: Adenosine Diphosphate; Adult; Aged; Benzylamines; Blood Platelets; Cell Aggregation; Female; Fibrinogen; Flow Cytometry; Humans; Iodine Radioisotopes; Leukocytes; Male; Middle Aged; Piperidines; Platelet Activation; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Thiazoles; Thrombin | 1998 |
Potentiation of glucose-induced insulin secretion by fagomine, a pseudo-sugar isolated from mulberry leaves.
Topics: Acetyl Coenzyme A; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Drug Synergism; Enzyme Inhibitors; Female; Glucose; Glyceraldehyde; Glyceraldehyde 3-Phosphate; Glycolysis; Imino Pyranoses; Insulin; Insulin Secretion; Islets of Langerhans; Lactic Acid; Oligo-1,6-Glucosidase; Piperidines; Rats; Rats, Wistar | 1998 |
Interspecies comparison of the antiplatelet, antithrombotic, and hemorrhagic effects of SR 121566A, a novel nonpeptide GP IIb/IIIa antagonist.
Topics: Adenosine Diphosphate; Animals; Arteriovenous Shunt, Surgical; Benzylamines; Dogs; Fibrinolytic Agents; Guinea Pigs; Hemorrhage; Humans; In Vitro Techniques; Male; Mice; Papio; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Rabbits; Rats; Species Specificity; Thiazoles | 1999 |
Inhibitory effects of H2-receptor antagonists on platelet function in vitro.
Topics: Adenosine Diphosphate; Adult; Arachidonic Acid; Aspirin; Blood Platelets; Cimetidine; Collagen; Famotidine; Female; Heterocyclic Compounds, 1-Ring; Histamine H2 Antagonists; Humans; In Vitro Techniques; Male; Middle Aged; P-Selectin; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Ranitidine; Structure-Activity Relationship | 1999 |
BGP-15, a nicotinic amidoxime derivate protecting heart from ischemia reperfusion injury through modulation of poly(ADP-ribose) polymerase.
Topics: Adenosine Diphosphate; ADP Ribose Transferases; Animals; Carrier Proteins; Cell Nucleus; Cytoplasm; DNA Damage; Endoplasmic Reticulum Chaperone BiP; Heat-Shock Proteins; In Vitro Techniques; Lipid Peroxidation; Male; Molecular Chaperones; NAD; Oximes; Perfusion; Piperidines; Poly (ADP-Ribose) Polymerase-1; Poly(ADP-ribose) Polymerase Inhibitors; Poly(ADP-ribose) Polymerases; Protective Agents; Proteins; Rats; Rats, Wistar; Reactive Oxygen Species; Reperfusion Injury | 2000 |
Effect of aspirin on platelet desaggregation induced by SR121566, a potent GP-IIb/IIIa antagonist.
Topics: Adenosine Diphosphate; Animals; Arachidonic Acid; Aspirin; Benzylamines; Blood Flow Velocity; Blood Platelets; Carotid Arteries; Disease Models, Animal; Electric Stimulation; Female; Fibrinolytic Agents; Humans; Male; Oligopeptides; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Rabbits; Recombinant Proteins; Thiazoles; Thrombosis; Thrombospondins; Tissue Plasminogen Activator | 2000 |
Antiplatelet action of R-99224, an active metabolite of a novel thienopyridine-type G(i)-linked P2T antagonist, CS-747.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Calcium; Cyclic AMP; Cyclopropanes; Fibrinogen; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; In Vitro Techniques; Male; Membrane Proteins; Piperazines; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Prasugrel Hydrochloride; Purinergic P2 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P2; Receptors, Purinergic P2Y12; Thionucleotides; Thiophenes | 2001 |
Human platelets bind and degrade 2-arachidonoylglycerol, which activates these cells through a cannabinoid receptor.
Topics: Adenosine Diphosphate; Amidohydrolases; Arachidonic Acids; Aspirin; Biological Transport; Blood Platelets; Calcium Channel Blockers; Camphanes; Cannabinoid Receptor Modulators; Collagen; Cyclic AMP; Endocannabinoids; Glycerides; Humans; Hydrolysis; Inositol 1,4,5-Trisphosphate; Kinetics; Piperidines; Platelet Activation; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Serotonin; Time Factors | 2001 |
The effect of a novel glycoprotein IIb/IIIa antagonist, SR 121566A, on platelet aggregation and activation in rhesus monkeys.
Topics: Adenosine Diphosphate; Animals; Benzylamines; Drug Administration Routes; Drug Evaluation, Preclinical; Macaca mulatta; Male; P-Selectin; Piperidines; Platelet Activation; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Thiazoles; Time Factors | 2001 |
Cannabinoid inhibition of capsaicin-sensitive sensory neurotransmission in the rat mesenteric arterial bed.
Topics: Adenosine Diphosphate; Animals; Benzofurans; Calcitonin Gene-Related Peptide; Camphanes; Cannabinoids; Capsaicin; Dose-Response Relationship, Drug; Dronabinol; Electric Stimulation; Electrophysiology; Male; Mesenteric Arteries; Neurons, Afferent; Nitroprusside; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Synaptic Transmission; Time Factors; Vasodilation; Vasodilator Agents | 2001 |
Effect of repaglinide on cloned beta cell, cardiac and smooth muscle types of ATP-sensitive potassium channels.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Carbamates; Cell Line; Cloning, Molecular; Drug Synergism; Electric Conductivity; Female; Humans; Islets of Langerhans; Mice; Muscle, Smooth; Myocardium; Oocytes; Piperidines; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Sulfonylurea Receptors; Xenopus laevis | 2001 |
Effects of fibrinogen receptor antagonist GR144053F and aurintricarboxylic acid on platelet activation and degranulation.
Topics: Adenosine Diphosphate; Adult; Aurintricarboxylic Acid; Cell Degranulation; Collagen Type I; Female; Flow Cytometry; Hemostasis; Humans; Male; Middle Aged; Piperazines; Piperidines; Platelet Activation; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex | 2001 |
Reduction of acute photodamage in skin by topical application of a novel PARP inhibitor.
Topics: Adenosine Diphosphate; Administration, Topical; Animals; DNA Damage; DNA, Single-Stranded; Epidermis; Interleukin-10; Mice; Mice, Nude; Oximes; Piperidines; Poly(ADP-ribose) Polymerase Inhibitors; Protective Agents; Radiodermatitis; Sunburn; Tumor Necrosis Factor-alpha; Ultraviolet Rays | 2002 |
Pharmacological properties of YM-57029, a novel platelet glycoprotein IIb/IIIa antagonist.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Benzamidines; Biotinylation; Bleeding Time; Blood Platelets; Collagen; Cricetinae; Dogs; Dose-Response Relationship, Drug; Fibrinogen; Fibrinolytic Agents; Guinea Pigs; Haplorhini; Humans; Mice; Microspheres; Oligopeptides; Piperazines; Piperidines; Platelet Adhesiveness; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Protein Binding; Rabbits; Rats; Stress, Mechanical | 2002 |
Effect of clopidogrel administration to healthy volunteers on platelet phosphorylation events triggered by ADP.
Topics: Adenosine Diphosphate; Adolescent; Adult; Benzylamines; Blood Platelets; Clopidogrel; Electrophoresis, Polyacrylamide Gel; Humans; Male; Membrane Proteins; Phosphorylation; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Receptors, Purinergic P2Y12; Serine; Signal Transduction; Thiazoles; Thionucleotides; Threonine; Ticlopidine; Tyrosine | 2003 |
Investigation of platelet aggregation inhibitory activity by phenyl amides and esters of piperidinecarboxylic acids.
Topics: Adenosine Diphosphate; Amides; Buffers; Carboxylic Acids; Chemical Phenomena; Chemistry, Physical; Drug Evaluation, Preclinical; Epinephrine; Esters; Half-Life; Humans; In Vitro Techniques; Indicators and Reagents; Magnetic Resonance Spectroscopy; Models, Molecular; Nipecotic Acids; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Quantitative Structure-Activity Relationship | 2003 |
Adenine nucleotide metabolism and cell fate after oxidant exposure of rat cortical neurons: effects of inhibition of poly(ADP-ribose) polymerase.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Cell Count; Cells, Cultured; Cerebral Cortex; Embryo, Mammalian; Enzyme Inhibitors; Isoquinolines; Neurons; Oxidants; Piperidines; Poly(ADP-ribose) Polymerase Inhibitors; Poly(ADP-ribose) Polymerases; Rats | 2004 |
Differential roles of integrins alpha2beta1 and alphaIIbbeta3 in collagen and CRP-induced platelet activation.
Topics: Adenosine Diphosphate; Benzodiazepines; Carrier Proteins; Collagen; Cytoplasmic Granules; Dual Specificity Phosphatase 2; Humans; Integrin alpha2beta1; P-Selectin; Peptides; Piperidines; Platelet Activation; Platelet Aggregation; Platelet Glycoprotein GPIIb-IIIa Complex; Platelet Membrane Glycoproteins; Protein Phosphatase 2; Protein Tyrosine Phosphatases; Thromboxane A2 | 2004 |
P2Y12 receptors play a significant role in the development of platelet microaggregation in patients with diabetes.
Topics: Adenosine Diphosphate; Adenosine Monophosphate; Aged; Diabetes Mellitus, Type 2; Female; Humans; Male; Membrane Proteins; Middle Aged; Piperazines; Piperidines; Platelet Aggregation; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Receptors, Purinergic P2Y12; Reference Values | 2005 |
The dopamine agonism on ADP-stimulated platelets is mediated through D2-like but not D1-like dopamine receptors.
Topics: Adenosine Diphosphate; Antigens, CD; Benzazepines; Clozapine; Collagen Type IV; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Epinephrine; Flow Cytometry; Humans; Indoles; Methylphenidate; P-Selectin; Piperidines; Platelet Activation; Platelet Adhesiveness; Platelet Aggregation; Platelet Membrane Glycoproteins; Platelet-Rich Plasma; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2; Tetraspanin 30 | 2008 |
N-methyl-D-aspartate receptor antagonists have variable affect in 3-nitropropionic acid toxicity.
Topics: Adenosine Diphosphate; Animals; Corpus Striatum; Dizocilpine Maleate; Drug Interactions; Male; Memantine; Motor Activity; Nerve Degeneration; Neuroprotective Agents; Nitro Compounds; Piperidines; Poly (ADP-Ribose) Polymerase-1; Poly(ADP-ribose) Polymerases; Propionates; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Tyrosine | 2009 |
Electrical stimulation of the mucosa evokes slow EPSPs mediated by NK1 tachykinin receptors and by P2Y1 purinoceptors in different myenteric neurons.
Topics: Adenosine Diphosphate; Animals; Electric Stimulation; Evoked Potentials; Excitatory Postsynaptic Potentials; Female; Guinea Pigs; Ileum; Immunohistochemistry; In Vitro Techniques; Intestinal Mucosa; Jejunum; Kinetics; Male; Myenteric Plexus; Neurokinin-1 Receptor Antagonists; Nitrergic Neurons; Nitric Oxide Synthase Type I; Piperidines; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Quinuclidines; Receptors, Neurokinin-1; Receptors, Purinergic P2; Receptors, Purinergic P2Y1 | 2009 |
Spice active principles as the inhibitors of human platelet aggregation and thromboxane biosynthesis.
Topics: Acrolein; Adenosine Diphosphate; Alkaloids; Allyl Compounds; Arachidonic Acid; Benzodioxoles; Calcimycin; Capsaicin; Collagen Type III; Curcumin; Eugenol; Humans; Malondialdehyde; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Polyunsaturated Alkamides; Quercetin; Spices; Sulfides; Thromboxanes | 2009 |
A plausible explanation for enhanced bioavailability of P-gp substrates in presence of piperine: simulation for next generation of P-gp inhibitors.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Adenylyl Imidodiphosphate; Alkaloids; Amino Acids; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzodioxoles; Binding Sites; Biological Availability; Cell Survival; Computer Simulation; Dogs; Flow Cytometry; Humans; Madin Darby Canine Kidney Cells; Models, Molecular; Piperidines; Polyunsaturated Alkamides; Protein Structure, Tertiary; Rhodamines; Structural Homology, Protein; Substrate Specificity | 2013 |
Potent P2Y1 urea antagonists bearing various cyclic amine scaffolds.
Topics: Adenosine Diphosphate; Amines; Animals; Blood Platelets; Half-Life; Humans; Microsomes, Liver; Piperidines; Platelet Aggregation Inhibitors; Protein Binding; Purinergic P2Y Receptor Agonists; Rats; Receptors, Purinergic P2Y1; Structure-Activity Relationship; Urea | 2013 |
Ibrutinib inhibits collagen-mediated but not ADP-mediated platelet aggregation.
Topics: Adenine; Adenosine Diphosphate; Aged; Aged, 80 and over; Antineoplastic Agents; Blood Platelets; Cells, Cultured; Collagen; Female; Hemorrhage; Humans; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, Mantle-Cell; Male; Middle Aged; Piperidines; Platelet Aggregation; Pyrazoles; Pyrimidines; Severity of Illness Index | 2015 |
Effects of ibrutinib treatment on murine platelet function during inflammation and in primary hemostasis.
Topics: Adenine; Adenosine Diphosphate; Animals; Blood Platelets; Collagen; Crotalid Venoms; Gene Expression Regulation; Hemorrhage; Hemostasis; Inflammation; Lectins, C-Type; Lipopolysaccharides; Lung; Membrane Glycoproteins; Mice; Oligopeptides; Piperidines; Platelet Aggregation; Platelet Membrane Glycoproteins; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Receptors, Purinergic P2Y12; Skin | 2017 |