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adenosine and flumazenil

adenosine has been researched along with flumazenil in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-199015 (55.56)18.7374
1990's4 (14.81)18.2507
2000's4 (14.81)29.6817
2010's4 (14.81)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Dragunow, M1
Greenblatt, DJ; Kaplan, GB; Leduc, BW; Shader, RI; Thompson, ML1
Baldwin, HA; File, SE1
Morgan, PF; Stone, TW1
O'Regan, MH; Phillis, JW1
Stone, TW2
Bender, AS; Hertz, L1
Phillis, JW; Stair, RE1
Hernández, J; Ribeiro, JA; Ruiz, F1
Bortolotto, ZA; Cavalheiro, EA; Ikonomidou, C; Mello, LE; Turski, L; Turski, WA1
Phillis, JW1
Risley, EA; Williams, M1
Lloyd, HG; Morgan, PF; Stone, TW2
Coffin, VL; Phillis, JW; Wu, PH1
Kulkarni, SK; Mehta, AK1
Kanayama, T; Kobayashi, M; Koshikawa, N; Murai, T; Takada, K; Tomiyama, K1
Collins, SW; Porterfield, JG; Porterfield, LM1
Mendelson, WB1
Fidecka, S; Listos, J; Malec, D1

Reviews

3 review(s) available for adenosine and flumazenil

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
The role of adenosine in the central actions of the benzodiazepines.
    Progress in neuro-psychopharmacology & biological psychiatry, 1988, Volume: 12, Issue:4

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Arousal; Benzodiazepinones; Brain; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Neural Inhibition; Neurons; Purkinje Cells; Rats; Receptors, GABA-A

1988
Adenosine's role in the central actions of the benzodiazepines.
    Progress in neuro-psychopharmacology & biological psychiatry, 1984, Volume: 8, Issue:4-6

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Brain; Cats; Cell Line; Cerebral Cortex; Diazepam; Flumazenil; Rats; Synaptosomes; Thioinosine

1984

Other Studies

24 other study(ies) available for adenosine and flumazenil

ArticleYear
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Adenosine receptor antagonism accounts for the seizure-prolonging effects of aminophylline.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:4

    Topics: Adenosine; Aminophylline; Amygdala; Animals; Brain; Carbolines; Diazepam; Flumazenil; Kindling, Neurologic; Male; Picrotoxin; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Purinergic; Rolipram; Seizures; Theophylline; Xanthines

1990
Relationship of plasma and brain concentrations of caffeine and metabolites to benzodiazepine receptor binding and locomotor activity.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3

    Topics: Adenosine; Animals; Brain; Caffeine; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Flumazenil; Male; Mice; Motor Activity; Receptors, GABA-A

1989
Caffeine-induced anxiogenesis: the role of adenosine, benzodiazepine and noradrenergic receptors.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Alprazolam; Anxiety; Caffeine; Chlordiazepoxide; Clonidine; Flumazenil; Motor Activity; Muscle Relaxants, Central; Norepinephrine; Propranolol; Receptors, Adrenergic; Receptors, GABA-A; Receptors, Purinergic; Social Behavior

1989
Inhibition by benzodiazepines and beta-carbolines of brief (5 seconds) synaptosomal accumulation of [3H]-adenosine.
    Biochemical pharmacology, 1986, May-15, Volume: 35, Issue:10

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Benzodiazepinones; Brain; Carbolines; Flumazenil; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Synaptosomes; Time Factors; Tritium

1986
The suppression of hippocampal potentials by the benzodiazepine antagonist Ro 15-1788 may be mediated by purines.
    Brain research, 1986, Aug-20, Volume: 380, Issue:2

    Topics: Adenosine; Animals; Benzodiazepines; Evoked Potentials; Flumazenil; GABA-A Receptor Antagonists; Hippocampus; Male; Neural Inhibition; Purines; Rats; Receptors, GABA-A

1986
Dissimilarities between benzodiazepine-binding sites and adenosine uptake sites in astrocytes and neurons in primary cultures.
    Journal of neuroscience research, 1987, Volume: 17, Issue:2

    Topics: Adenosine; Animals; Astrocytes; Benzodiazepines; Binding Sites; Cells, Cultured; Diazepam; Flumazenil; Isoquinolines; Neurons; Pyrazoles; Receptors, GABA-A

1987
Ro 15-1788 both antagonizes and potentiates adenosine-evoked depression of cerebral cortical neurons.
    European journal of pharmacology, 1987, Apr-14, Volume: 136, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Caffeine; Cerebral Cortex; Evoked Potentials; Flumazenil; Male; Rats; Rats, Inbred Strains

1987
Theophylline antagonizes the effect of diazepam on ventricular automaticity.
    European journal of pharmacology, 1988, Oct-18, Volume: 155, Issue:3

    Topics: Adenosine; Animals; Diazepam; Female; Flumazenil; Heart Rate; Heart Ventricles; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Theophylline; Ventricular Function

1988
Effects of aminophylline and 2-chloroadenosine on seizures produced by pilocarpine in rats: morphological and electroencephalographic correlates.
    Brain research, 1985, Dec-30, Volume: 361, Issue:1-2

    Topics: 2-Chloroadenosine; Adenosine; Aminophylline; Animals; Benzodiazepinones; Bicuculline; Brain; Carbolines; Convulsants; Electroencephalography; Flumazenil; Male; Motor Activity; Pilocarpine; Rats; Rats, Inbred Strains; Seizures

1985
Interaction of the benzodiazepine antagonists, CGS 8216 and Ro 15-1788, with central adenosine A-1 receptors.
    Archives internationales de pharmacodynamie et de therapie, 1982, Volume: 260, Issue:1

    Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Brain; Flumazenil; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, Purinergic

1982
Benzodiazepine inhibition of adenosine uptake is not prevented by benzodiazepine antagonists.
    European journal of pharmacology, 1983, Jan-28, Volume: 87, Issue:1

    Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Brain; Diazepam; Flumazenil; Flurazepam; Hexobendine; In Vitro Techniques; Pyrazoles; Rats; Rats, Inbred Strains; Synaptosomes; Temperature

1983
Inhibition of adenosine uptake into rat brain synaptosomes by prostaglandins, benzodiazepines and other centrally active compounds.
    General pharmacology, 1983, Volume: 14, Issue:5

    Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Brain; Calmodulin; Carbolines; Flumazenil; Hydroxyzine; Imidazoles; Male; Prostaglandins; Pyrazoles; Rats; Rats, Inbred Strains; Sulfonamides; Synaptosomes

1983
Inhibition of adenosine accumulation by a CNS benzodiazepine antagonist (Ro 15-1788) and a peripheral benzodiazepine receptor ligand (Ro 05-4864).
    Neuroscience letters, 1983, Oct-31, Volume: 41, Issue:1-2

    Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Central Nervous System; Diazepam; Flumazenil; Flurazepam; Hexobendine; Male; Rats; Synaptosomes; Time Factors

1983
Mechanism of potentiation by diazepam of adenosine response.
    Life sciences, 1984, Jan-02, Volume: 34, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Animals; Benzodiazepinones; Cecum; Diazepam; Dipyridamole; Dose-Response Relationship, Drug; Drug Synergism; Female; Flumazenil; Hypoxanthine; Hypoxanthines; Inosine; Male; Rats; Rats, Inbred Strains

1984
Opposite effects of midazolam and beta-carboline-3-carboxylate ethyl ester on the release of dopamine from rat nucleus accumbens measured by in vivo microdialysis.
    European journal of pharmacology, 1994, Aug-11, Volume: 261, Issue:1-2

    Topics: Adenosine; Animals; Carbolines; Dopamine; Dose-Response Relationship, Drug; Flumazenil; Ligands; Male; Microdialysis; Midazolam; Nucleus Accumbens; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Tetrodotoxin; Theobromine; Xanthines

1994
The cutting edge in arrhythmias.
    Critical care nurse, 1993, Volume: 13, Issue:3 Suppl

    Topics: Adenosine; Arrhythmias, Cardiac; Defibrillators, Implantable; Flumazenil; Humans; Pacemaker, Artificial

1993
Actions of benzodiazepines and the benzodiazepine antagonist flumazenil may involve adenosine.
    Journal of the neurological sciences, 1999, Mar-01, Volume: 163, Issue:2

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Antidotes; Brain; Flumazenil; Neurons

1999
Sleep-inducing effects of adenosine microinjections into the medial preoptic area are blocked by flumazenil.
    Brain research, 2000, Jan-10, Volume: 852, Issue:2

    Topics: Adenosine; Analgesics; Animals; Drug Interactions; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Male; Microinjections; Preoptic Area; Rats; Rats, Sprague-Dawley; Sleep

2000
Influence of adenosine receptor agonists on benzodiazepine withdrawal signs in mice.
    European journal of pharmacology, 2005, Oct-31, Volume: 523, Issue:1-3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Mice; Pentylenetetrazole; Phenethylamines; Purinergic Agonists; Purinergic P1 Receptor Agonists; Purinergic P2 Receptor Agonists; Seizures; Substance Withdrawal Syndrome; Temazepam

2005