Page last updated: 2024-09-03

adenosine amine congener and cgs 15943

adenosine amine congener has been researched along with cgs 15943 in 2 studies

Compound Research Comparison

Studies
(adenosine amine congener)
Trials
(adenosine amine congener)
Recent Studies (post-2010)
(adenosine amine congener)
Studies
(cgs 15943)
Trials
(cgs 15943)
Recent Studies (post-2010) (cgs 15943)
2905139028

Protein Interaction Comparison

ProteinTaxonomyadenosine amine congener (IC50)cgs 15943 (IC50)
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)0.97
Adenosine receptor A3Homo sapiens (human)0.406
Adenosine receptor A1Rattus norvegicus (Norway rat)0.006
Adenosine receptor A3Rattus norvegicus (Norway rat)0.0607
Adenosine receptor A2aHomo sapiens (human)0.012
Adenosine receptor A2bHomo sapiens (human)0.6304
Adenosine receptor A2bRattus norvegicus (Norway rat)0.0028
Adenosine receptor A2aRattus norvegicus (Norway rat)0.0029
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformHomo sapiens (human)1.28
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)8.48
Casein kinase I isoform alphaHomo sapiens (human)0.82
Casein kinase I isoform deltaHomo sapiens (human)0.24
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)0.11
Casein kinase I isoform epsilonHomo sapiens (human)0.49
DNA-dependent protein kinase catalytic subunitHomo sapiens (human)0.14

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Jacobson, KA; van Galen, PJ; Williams, M1
Bivalacqua, TJ; Champion, HC; Kadowitz, PJ; Lambert, DG1

Reviews

1 review(s) available for adenosine amine congener and cgs 15943

ArticleYear
Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.
    Journal of medicinal chemistry, 1992, Feb-07, Volume: 35, Issue:3

    Topics: Adenosine; Animals; Humans; Models, Chemical; Receptors, Purinergic; Second Messenger Systems; Structure-Activity Relationship

1992

Other Studies

1 other study(ies) available for adenosine amine congener and cgs 15943

ArticleYear
Vasodilator responses to adenosine and hyperemia are mediated by A(1) and A(2) receptors in the cat vascular bed.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2002, Volume: 282, Issue:6

    Topics: Adenosine; Adenosine Triphosphate; Animals; Cats; Dose-Response Relationship, Drug; Female; Hemodynamics; Hindlimb; Hyperemia; Male; Perfusion; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Quinazolines; Receptors, Purinergic P1; Triazoles; Vascular Resistance; Vasodilation; Xanthines

2002