Page last updated: 2024-08-21

adamantane and sr 142948a

adamantane has been researched along with sr 142948a in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (26.67)18.2507
2000's19 (63.33)29.6817
2010's2 (6.67)24.3611
2020's1 (3.33)2.80

Authors

AuthorsStudies
Bachy, A; Boigegrain, R; Gully, D; Kitabgi, P; Labbé-Jullié, C; Labeeuw, B; Le Fur, G; Maffrand, JP; Oury-Donat, F; Pecceu, F; Poncelet, M; Santucci, V; Soubrié, P; Steinberg, R; Suaud-Chagny, MF; Vita, N1
Heaulme, M; Le Fur, G; Leyris, R; Soubrie, P2
Betancur, C; Burgos, A; Canton, M; Gully, D; Labeeuw, B; Pélaprat, D; Rostène, W1
Bernat, A; Gully, D; Herbert, JM; Laplace, MC; Lespy, L; Prabonnaud, V; Schaeffer, P1
Casellas, P; Combes, T; Gully, D; Maffrand, JP; Portier, M1
Bédard, PJ; Di Paolo, T; Falardeau, P; Goulet, M; Grondin, R; Morissette, M; Rostène, W1
Matthews, RT1
Kruse, CG; Long, SK; Nievelstein, H; Wadman, WJ; Werkman, TR1
Trudeau, LE1
Castagliuolo, I; Matthews, JB; Pothoulakis, C; Riegler, M; Sogukoglu, T; Wang, C; Wenzl, E; Wlk, M1
Belmeguenai, A; Cavelier, F; Leprince, J; Louiset, E; Martinez, J; Vaudry, H; Vivet, B1
Binder, EB; Kilts, CD; Kinkead, B; Nemeroff, CB; Owens, MJ1
Hwang, HM; Li, AH; Tan, PP; Wang, HL; Yeh, TH1
Brun, P; Leonetti, M; Renaud, B; Sotty, F; Soubrié, P; Steinberg, R; Suaud-Chagny, MF1
Binder, EB; Gross, RE; Kilts, CD; Nemeroff, CB1
Bert, L; Brun, P; Leonetti, M; Renaud, B; Sotty, F; Soubrié, P; Steinberg, R; Suaud-Chagny, MF1
Meyer-Spasche, A; Piggins, HD; Reed, HE1
Behbehani, MM; Kreitel, KD; Swisher, CB1
Chen, L; Yung, KK; Yung, WH1
Casti, P; Casu, G; Marchese, G; Pani, L; Ruiu, S1
Binder, EB; Kinkead, B; Nemeroff, CB; Owens, MJ1
Bérod, A; Colussi-Mas, J; Lambás-Señas, L; Panayi, F; Renaud, B; Scarna, H1
Azmi, N; Bennett, GW; Norman, C; Spicer, CH1
Cassaday, HJ; G W, B; Grimond-Billa, SK; Norman, C1
Marie-Claire, C; Noble, F; Palminteri, S; Romualdi, P1
Bennett, GW; Cassaday, HJ; Grimond-Billa, SK; Norman, C1
Kawahara, H; Mitchell, VA; Vaughan, CW1
Binder, EB; Cáceda, R; Kinkead, B; Nemeroff, CB1
Apaijai, N; Chattipakorn, N; Chattipakorn, SC; Chunchai, T; Jaiwongkam, T; Kerdphoo, S; Pratchayasakul, W; Saiyasit, N; Sripetchwandee, J1

Other Studies

30 other study(ies) available for adamantane and sr 142948a

ArticleYear
Biochemical and pharmacological activities of SR 142948A, a new potent neurotensin receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2

    Topics: Adamantane; Animals; Axonal Transport; Binding Sites; Brain; Calcium; Cell Line; Cell Membrane; CHO Cells; Corpus Striatum; Cricetinae; Dopamine; Female; Humans; Imidazoles; Inositol Phosphates; Male; Mice; Mice, Inbred Strains; Neurons; Neurotensin; Nucleus Accumbens; Rats; Rats, Inbred Strains; Rats, Sprague-Dawley; Receptors, Neurotensin; Recombinant Proteins; Stereotyped Behavior; Substantia Nigra; Transfection

1997
Involvement of potentially distinct neurotensin receptors in neurotensin-induced stimulation of striatal [3H]dopamine release evoked by KCl versus electrical depolarization.
    Neuropharmacology, 1997, Volume: 36, Issue:10

    Topics: Adamantane; Animals; Dopamine; Dose-Response Relationship, Drug; Guinea Pigs; Imidazoles; Male; Neurotensin; Nucleus Accumbens; Potassium; Pyrazoles; Quinolines; Rats; Receptors, Neurotensin; Visual Cortex

1997
Characterization of binding sites of a new neurotensin receptor antagonist, [3H]SR 142948A, in the rat brain.
    European journal of pharmacology, 1998, Feb-05, Volume: 343, Issue:1

    Topics: Adamantane; Animals; Autoradiography; Binding Sites; Brain; Imidazoles; Male; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Tritium

1998
SR142948A is a potent antagonist of the cardiovascular effects of neurotensin.
    Journal of cardiovascular pharmacology, 1998, Volume: 31, Issue:4

    Topics: Adamantane; Administration, Oral; Animals; Blood Pressure; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Endothelium, Vascular; Epoprostenol; Hematocrit; Humans; Imidazoles; Injections, Intradermal; Iodine Radioisotopes; Male; Neurotensin; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Umbilical Veins

1998
Neurotensin type 1 receptor-mediated activation of krox24, c-fos and Elk-1: preventing effect of the neurotensin antagonists SR 48692 and SR 142948.
    FEBS letters, 1998, Jul-31, Volume: 432, Issue:1-2

    Topics: Adamantane; Animals; CHO Cells; Cricetinae; DNA-Binding Proteins; Dose-Response Relationship, Drug; ets-Domain Protein Elk-1; Genes, Reporter; Imidazoles; Neurotensin; Point Mutation; Promoter Regions, Genetic; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-fos; Pyrazoles; Quinolines; Receptors, Neurotensin; Sequence Deletion; Signal Transduction; Transcription Factors

1998
Stimulation by neurotensin of (3H)5-hydroxytryptamine (5HT) release from rat frontal cortex slices.
    Neuropeptides, 1998, Volume: 32, Issue:5

    Topics: Adamantane; Animals; Corpus Striatum; Dizocilpine Maleate; Dopamine Antagonists; Down-Regulation; Frontal Lobe; Hippocampus; Imidazoles; In Vitro Techniques; Inhibitory Concentration 50; Neurotensin; Peptide Fragments; Potassium; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotensin; Serotonin; Tetrodotoxin

1998
Neurotensin receptors and dopamine transporters: effects of MPTP lesioning and chronic dopaminergic treatments in monkeys.
    Synapse (New York, N.Y.), 1999, Jun-01, Volume: 32, Issue:3

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Adamantane; Animals; Autoradiography; Binding Sites; Carrier Proteins; Caudate Nucleus; Denervation; Dopamine; Dopamine Agents; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Down-Regulation; Imidazoles; In Situ Hybridization; Macaca fascicularis; Membrane Glycoproteins; Membrane Transport Proteins; Neostriatum; Nerve Tissue Proteins; Neurotensin; Piperidines; Putamen; Receptors, Dopamine; Receptors, Neurotensin; RNA, Messenger; Substantia Nigra

1999
Neurotensin depolarizes cholinergic and a subset of non-cholinergic septal/diagonal band neurons by stimulating neurotensin-1 receptors.
    Neuroscience, 1999, Volume: 94, Issue:3

    Topics: Action Potentials; Adamantane; Animals; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Male; Membrane Potentials; Neurons; Neurotensin; Patch-Clamp Techniques; Piperidines; Prosencephalon; Receptors, Neurotensin; Tetrodotoxin

1999
Neurotensin attenuates the quinpirole-induced inhibition of the firing rate of dopamine neurons in the rat substantia nigra pars compacta and the ventral tegmental area.
    Neuroscience, 2000, Volume: 95, Issue:2

    Topics: Action Potentials; Adamantane; Animals; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; Electrophysiology; Imidazoles; In Vitro Techniques; Logistic Models; Male; Neurons; Neurotensin; Peptide Fragments; Quinpirole; Rats; Rats, Wistar; Receptors, Neurotensin; Substantia Nigra; Ventral Tegmental Area

2000
Neurotensin regulates intracellular calcium in ventral tegmental area astrocytes: evidence for the involvement of multiple receptors.
    Neuroscience, 2000, Volume: 97, Issue:2

    Topics: Adamantane; Animals; Animals, Newborn; Astrocytes; Calcium; Cells, Cultured; Estrenes; Gadolinium; Imidazoles; Neurotensin; Peptide Fragments; Piperidines; Pyrrolidinones; Rats; Receptors, Neurotensin; Thapsigargin; Type C Phospholipases; Ventral Tegmental Area

2000
Neurotensin stimulates Cl(-) secretion in human colonic mucosa In vitro: role of adenosine.
    Gastroenterology, 2000, Volume: 119, Issue:2

    Topics: Adamantane; Adenosine; Adenosine Deaminase Inhibitors; Affinity Labels; Anti-Inflammatory Agents, Non-Steroidal; Cells, Cultured; Chlorides; Colon; Electrophysiology; Enteric Nervous System; Enzyme Inhibitors; Guanosine; Histamine; Humans; Imidazoles; In Vitro Techniques; Indomethacin; Intestinal Mucosa; Mast Cells; Membrane Potentials; Neurotensin; Pentostatin; Pyrazoles; Quinolines; Receptors, Neurotensin; Tetrodotoxin; Thioinosine; Thionucleosides

2000
Neurotensin modulates the electrical activity of frog pituitary melanotropes via activation of a G-protein-coupled receptor pharmacologically related to both the NTS1 and nts2 receptors of mammals.
    Neuroendocrinology, 2000, Volume: 72, Issue:6

    Topics: Adamantane; Animals; Cells, Cultured; GTP-Binding Protein alpha Subunits, Gq-G11; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Heterotrimeric GTP-Binding Proteins; Imidazoles; Ligands; Male; Mammals; Melanocytes; Membrane Potentials; Neurotensin; Patch-Clamp Techniques; Peptide Fragments; Pituitary Gland; Pyrazoles; Quinolines; Rana ridibunda; Receptors, Neurotensin; Signal Transduction; Thionucleotides

2000
Enhanced neurotensin neurotransmission is involved in the clinically relevant behavioral effects of antipsychotic drugs: evidence from animal models of sensorimotor gating.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2001, Jan-15, Volume: 21, Issue:2

    Topics: Acoustic Stimulation; Adamantane; Animals; Antipsychotic Agents; Behavior, Animal; Brain; Conditioning, Classical; Dibenzothiazepines; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Female; Haloperidol; Imidazoles; Inhibition, Psychological; Neurotensin; Photic Stimulation; Psychomotor Performance; Quetiapine Fumarate; Rats; Rats, Long-Evans; Reaction Time; Receptors, Neurotensin; Reflex, Startle; RNA, Messenger; Schizophrenia; Social Isolation; Synaptic Transmission

2001
Neurotensin excitation of serotonergic neurons in the rat nucleus raphe magnus: ionic and molecular mechanisms.
    Neuropharmacology, 2001, Volume: 40, Issue:8

    Topics: Adamantane; Animals; Calcium; Calcium Channels; Guanosine Diphosphate; Imidazoles; Inositol 1,4,5-Trisphosphate Receptors; Ion Channels; Neurons; Neurotensin; Pyrazoles; Quinolines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Cytoplasmic and Nuclear; Receptors, Neurotensin; Serotonin; Thionucleotides

2001
Endogenous neurotensin down-regulates dopamine efflux in the nucleus accumbens as revealed by SR-142948A, a selective neurotensin receptor antagonist.
    Journal of neurochemistry, 2001, Volume: 77, Issue:6

    Topics: Adamantane; Animals; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Electrochemistry; Haloperidol; Imidazoles; Male; Neurotensin; Nucleus Accumbens; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Stimulation, Chemical

2001
Effects of neurotensin receptor antagonism on latent inhibition in Sprague-Dawley rats.
    Psychopharmacology, 2002, Volume: 161, Issue:3

    Topics: Adamantane; Analysis of Variance; Animals; Association Learning; Conditioning, Operant; Dopamine Antagonists; Dose-Response Relationship, Drug; Imidazoles; Inhibition, Psychological; Male; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Sulpiride

2002
The neurotensin receptor antagonist SR 142948A blocks the efflux of dopamine evoked in nucleus accumbens by neurotensin ejection into the ventral tegmental area.
    Naunyn-Schmiedeberg's archives of pharmacology, 2002, Volume: 365, Issue:6

    Topics: Adamantane; Animals; Dopamine; Imidazoles; Male; N-Methylaspartate; Neurotensin; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Ventral Tegmental Area

2002
Neurotensin phase-shifts the firing rate rhythm of neurons in the rat suprachiasmatic nuclei in vitro.
    The European journal of neuroscience, 2002, Volume: 16, Issue:2

    Topics: Action Potentials; Adamantane; Animals; Circadian Rhythm; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Imidazoles; Male; Neurons; Neurotensin; Pyrazoles; Quinolines; Rats; Rats, Wistar; Receptors, Neurotensin; Suprachiasmatic Nucleus; Type C Phospholipases

2002
The effects of diphenhydramine and SR142948A on periaqueductal gray neurons and on the interactions between the medial preoptic nucleus and the periaqueductal gray.
    Neuroscience, 2002, Volume: 114, Issue:4

    Topics: Adamantane; Anesthetics, Local; Animals; Diphenhydramine; Electrophysiology; Imidazoles; Male; Membrane Potentials; Neural Pathways; Neurons; Periaqueductal Gray; Preoptic Area; Rats; Rats, Sprague-Dawley; Stimulation, Chemical

2002
Neurotensin depolarizes globus pallidus neurons in rats via neurotensin type-1 receptor.
    Neuroscience, 2004, Volume: 125, Issue:4

    Topics: Action Potentials; Adamantane; Anesthetics, Local; Animals; Electrophysiology; Globus Pallidus; Imidazoles; Neurons; Neurotensin; Organ Culture Techniques; Patch-Clamp Techniques; Peptide Fragments; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Synaptic Transmission; Tetrodotoxin

2004
Blockade of neurotensin receptors affects differently hypo-locomotion and catalepsy induced by haloperidol in mice.
    Neuropharmacology, 2004, Volume: 47, Issue:1

    Topics: Adamantane; Analysis of Variance; Animals; Catalepsy; Dopamine Antagonists; Haloperidol; Imidazoles; Injections, Intraperitoneal; Male; Mice; Motor Activity; Pyrazoles; Quinolines; Receptors, Neurotensin

2004
Neurotensin receptor antagonist SR 142948A alters Fos expression and extrapyramidal side effect profile of typical and atypical antipsychotic drugs.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2004, Volume: 29, Issue:12

    Topics: Adamantane; Analysis of Variance; Animals; Antipsychotic Agents; Behavior, Animal; Catalepsy; Cell Count; Dose-Response Relationship, Drug; Drug Interactions; Imidazoles; Immunohistochemistry; Male; Neostriatum; Oncogene Proteins v-fos; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Time Factors

2004
Endogenous neurotensin in the ventral tegmental area contributes to amphetamine behavioral sensitization.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2005, Volume: 30, Issue:5

    Topics: Adamantane; Amphetamine; Animals; Behavior, Animal; Central Nervous System Stimulants; Imidazoles; Injections, Subcutaneous; Male; Microinjections; Motor Activity; Neurotensin; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Ventral Tegmental Area

2005
Effects of a neurotensin analogue (PD149163) and antagonist (SR142948A) on the scopolamine-induced deficits in a novel object discrimination task.
    Behavioural pharmacology, 2006, Volume: 17, Issue:4

    Topics: Adamantane; Animals; Brain; Depression, Chemical; Discrimination, Psychological; Dose-Response Relationship, Drug; Form Perception; Imidazoles; Injections, Intraventricular; Male; Memory, Short-Term; Muscarinic Antagonists; Neurotensin; Rats; Receptors, Neurotensin; Scopolamine; Space Perception

2006
Selectively increased trace conditioning under the neurotensin agonist PD 149163 in an aversive procedure in which SR 142948A was without intrinsic effect.
    Journal of psychopharmacology (Oxford, England), 2008, Volume: 22, Issue:3

    Topics: Adamantane; Animals; Association Learning; Avoidance Learning; Cognition; Conditioning, Operant; Cues; Dopamine Agonists; Dose-Response Relationship, Drug; Electroshock; Imidazoles; Male; Neurotensin; Rats; Rats, Wistar; Reinforcement, Psychology; Stimulation, Chemical

2008
Effects of the selective neurotensin antagonist SR 142948A on 3,4-methylenedioxymethamphetamine-induced behaviours in mice.
    Neuropharmacology, 2008, Volume: 54, Issue:7

    Topics: 3,4-Methylenedioxyamphetamine; Adamantane; Analysis of Variance; Animals; Behavior, Animal; Conditioning, Operant; Corpus Striatum; Drug Interactions; Gene Expression Regulation; Hallucinogens; Imidazoles; Male; Mice; Motor Activity; Neurotensin; Receptors, Neurotensin; Time Factors

2008
A neurotensin agonist and antagonist decrease and increase activity, respectively, but do not preclude discrete cue conditioning.
    Journal of psychopharmacology (Oxford, England), 2010, Volume: 24, Issue:3

    Topics: Adamantane; Animals; Appetitive Behavior; Association Learning; Dose-Response Relationship, Drug; Imidazoles; Male; Neurotensin; Rats; Rats, Wistar; Receptors, Neurotensin

2010
Neurotensin inhibition of GABAergic transmission via mGluR-induced endocannabinoid signalling in rat periaqueductal grey.
    The Journal of physiology, 2009, Jun-01, Volume: 587, Issue:Pt 11

    Topics: Adamantane; Animals; Cannabinoid Receptor Modulators; Endocannabinoids; Excitatory Amino Acid Antagonists; Female; gamma-Aminobutyric Acid; Imidazoles; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Miniature Postsynaptic Potentials; Neural Inhibition; Neurons; Neurotensin; Pain; Periaqueductal Gray; Piperidines; Presynaptic Terminals; Pyrazoles; Pyridines; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, Neurotensin; Synaptic Transmission; Tetrodotoxin; Time Factors

2009
The role of endogenous neurotensin in psychostimulant-induced disruption of prepulse inhibition and locomotion.
    Schizophrenia research, 2012, Volume: 136, Issue:1-3

    Topics: Acoustic Stimulation; Adamantane; Amphetamine; Analysis of Variance; Animals; Apomorphine; Behavior, Animal; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Gait Disorders, Neurologic; Gene Expression Regulation; Imidazoles; Male; Neurotensin; Proto-Oncogene Proteins c-fos; Psychomotor Performance; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Reflex, Startle; RNA, Messenger

2012
Neurotensin receptor 1 agonist provides neuroprotection in pre-diabetic rats.
    The Journal of endocrinology, 2021, Volume: 248, Issue:1

    Topics: Adamantane; Animals; Cognitive Dysfunction; Diet, High-Fat; Drug Evaluation, Preclinical; Drug Therapy, Combination; Hippocampus; Ileum; Imidazoles; Insulin Resistance; Male; Neuronal Plasticity; Obesity; Oligopeptides; Oxidative Stress; Prediabetic State; Random Allocation; Rats, Wistar; Receptors, Neurotensin

2021