adamantane has been researched along with iem 1460 in 39 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 4 (10.26) | 18.2507 |
2000's | 10 (25.64) | 29.6817 |
2010's | 21 (53.85) | 24.3611 |
2020's | 4 (10.26) | 2.80 |
Authors | Studies |
---|---|
Cheng, H; Lakatta, EG; Song, LS; Stern, MD | 1 |
Buldakova, SL; Magazanik, LG; Samoilova, MV; Sharonova, IN; Vorobjev, VS | 2 |
Bol'shakov, KB; Buldakova, SL | 1 |
Buldakova, SL; Gmiro, VE; Magazanik, LG; Samoilova, MV; Tikhonov, DB | 1 |
Bolshakov, KV; Buldakova, SL; Magazanik, LG; Tikhonov, DB | 1 |
Bol'shakov, KB; Buldakova, SL; Gmiro, VE; Magazanik, LG; Samoĭlova, MV; Tikhonov, DB | 1 |
Essin, K; Magazanik, L; Nistri, A | 1 |
Bol'shakov, KV; Buldakova, SL; Gmiro, VE; Magazanik, LG; Samoilova, MV; Tikhonov, DB | 1 |
Bufler, J; Krampfl, K; Schlesinger, F; Tammena, D | 1 |
Buldakova, SL; Kim, KK; Magazanik, LG; Tikhonov, DB | 1 |
Efremov, OM; Gmiro, VE; Serdyuk, SE | 1 |
Asrar, S; Jia, Z; Ren, W; Zhou, Z | 1 |
Gainey, MA; Hurvitz-Wolff, JR; Lambo, ME; Turrigiano, GG | 1 |
Han, TZ; Li, P; Li, YH; Meng, K; Zhang, L | 1 |
Cenci, MA; Crossman, AR; Kobylecki, C; Ravenscroft, P | 1 |
Berke, JD; Fensterheim, BA; Gittis, AH; Kreitzer, AC; Leventhal, DK; Pettibone, JR | 1 |
Baldridge, WH; Daniels, BA; Tremblay, F; Wood, L | 1 |
Derkach, VA; Dwarakanath, D; Fortin, DA; Nygaard, S; Pierre, P; Soderling, TR; Srivastava, T | 1 |
Gittis, A | 1 |
Crossman, AR; Kobylecki, C; Ravenscroft, P | 1 |
Abushik, PA; Antonov, SM; Eaton, MJ; Sibarov, DA; Skatchkov, SN | 1 |
Arai, J; Feig, LA; Jin, SX; Kumar-Singh, R; Tian, X | 1 |
Gmiro, VE; Serdiuk, SE | 1 |
Mareš, P; Szczurowska, E | 1 |
Ambrósio, AF; Castilho, Á; Hartveit, E; Veruki, ML | 1 |
Cheng, LF; Liu, SB; Lu, JS; Shi, J; Zhang, MM; Zhuo, M | 1 |
Amici, M; Bortolotto, ZA; Choi, SL; Collingridge, GL; Kaang, BK; Park, P; Sanderson, TM; Zhuo, M | 1 |
Kim, MH; von Gersdorff, H | 1 |
Chen, Y; Derkach, VA; Smith, PA | 1 |
Balázsfi, D; Biró, L; Ferenczi, S; Haller, J; Klausz, B; Kovács, K; Mikics, É; Miskolczi, C; Sipos, E; Urbán, E; Varga, J; Zelena, D | 1 |
Lee, JK; Leem, YH; Oh, S; Yi, ES | 1 |
Nishikawa, T; Umino, A; Umino, M | 1 |
Bar-Gad, I; Oran, Y | 1 |
Donahue, RR; Doolen, S; Grachen, CM; Morón, JA; Sinha, GP; Taylor, BK | 1 |
Adotevi, N; Dabrowska, N; Joshi, S; Kapur, J; Lewczuk, E; Shan, S; Sun, H; Williamson, J | 1 |
Beck, H; Müller-Komorowska, D; Opitz, T; Pothmann, L; Schmidt, S; Soares da Silva, P | 1 |
Hikosaka, O; Kunimatsu, J; Maeda, K; Yamamoto, S | 1 |
Amakhin, DV; Chizhov, AV; Soboleva, EB; Zaitsev, AV | 1 |
39 other study(ies) available for adamantane and iem 1460
Article | Year |
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Partial depletion of sarcoplasmic reticulum calcium does not prevent calcium sparks in rat ventricular myocytes.
Topics: Adamantane; Algorithms; Animals; Calcium; Calcium-Transporting ATPases; Enzyme Inhibitors; Fluorescence; Heart Ventricles; In Vitro Techniques; Ion Channels; Microscopy, Confocal; Myocardium; Rats; Rats, Sprague-Dawley; Sarcoplasmic Reticulum; Thapsigargin | 1997 |
Characterization of AMPA receptor populations in rat brain cells by the use of subunit-specific open channel blocking drug, IEM-1460.
Topics: Adamantane; Animals; Brain Chemistry; Cerebellum; Corpus Striatum; Electrophysiology; Excitatory Amino Acid Agonists; Hippocampus; Interneurons; Ion Channel Gating; Kainic Acid; Membrane Potentials; Motor Cortex; Rats; Rats, Wistar; Receptors, AMPA; Somatosensory Cortex | 1999 |
The open channel blocking drug, IEM-1460, reveals functionally distinct alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionate receptors in rat brain neurons.
Topics: Adamantane; Animals; Brain Chemistry; Cerebellum; Corpus Striatum; Excitatory Amino Acid Agonists; Hippocampus; Kainic Acid; Membrane Potentials; Neurons; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA | 1999 |
[Pharmacologic analysis of the subunit composition of AMPA-receptors in the hippocampal neurons].
Topics: Adamantane; Alternative Splicing; Animals; Benzothiadiazines; Dentate Gyrus; Excitatory Amino Acid Agonists; Hippocampus; In Vitro Techniques; Interneurons; Kainic Acid; Neurons; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, AMPA | 1999 |
Voltage-dependent block of native AMPA receptor channels by dicationic compounds.
Topics: Adamantane; Animals; Cations; Diamines; Electrophysiology; Excitatory Amino Acid Agonists; Hippocampus; Kainic Acid; Kinetics; Membrane Potentials; Patch-Clamp Techniques; Pyramidal Cells; Quaternary Ammonium Compounds; Rats; Receptors, AMPA | 2000 |
Ca2+-dependent desensitization of AMPA receptors.
Topics: Adamantane; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Alternative Splicing; Animals; Animals, Newborn; Antihypertensive Agents; Benzothiadiazines; Calcium; Calcium Signaling; Dose-Response Relationship, Drug; Glutamic Acid; Hippocampus; Kainic Acid; Neurons; Nootropic Agents; Pyrrolidinones; Rats; Receptors, AMPA | 2000 |
[Structure of glutamate receptor ion channels and mechanisms of their blockade by organic cations].
Topics: Adamantane; Animals; Brain; Calcium; Cations; Excitatory Amino Acid Antagonists; Hydrophobic and Hydrophilic Interactions; In Vitro Techniques; Ion Channels; Models, Molecular; Neurons; Patch-Clamp Techniques; Quaternary Ammonium Compounds; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate | 2001 |
Evaluation of GluR2 subunit involvement in AMPA receptor function of neonatal rat hypoglossal motoneurons.
Topics: Adamantane; Animals; Animals, Newborn; Calcium; Calcium Signaling; Cell Membrane Permeability; Diamines; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Hippocampus; Hypoglossal Nerve; Interneurons; Male; Medulla Oblongata; Motor Neurons; Neostriatum; Pentobarbital; Pyramidal Cells; Quaternary Ammonium Compounds; Rats; Rats, Wistar; Receptors, AMPA; Spermine; Synaptic Transmission | 2002 |
Studies of the structure of glutamate receptor ion channels and the mechanisms of their blockade by organic cations.
Topics: Adamantane; Amantadine; Animals; Animals, Newborn; Brain; Cations; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; In Vitro Techniques; Ion Channels; Models, Biological; Models, Molecular; Neurons; Patch-Clamp Techniques; Quaternary Ammonium Compounds; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate | 2003 |
Two mechanisms of action of the adamantane derivative IEM-1460 at human AMPA-type glutamate receptors.
Topics: Adamantane; Animals; Binding, Competitive; Cell Line; Dose-Response Relationship, Drug; Electrophysiology; Excitatory Amino Acid Antagonists; Humans; Membrane Potentials; Patch-Clamp Techniques; Rats; Receptors, AMPA | 2005 |
Selective blockade of Ca2+ permeable AMPA receptors in CA1 area of rat hippocampus.
Topics: Adamantane; Animals; Bicuculline; Calcium; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Interneurons; Pyramidal Cells; Rats; Receptors, AMPA; Synapses | 2007 |
Peripheral and central routes of administration of quaternary ammonium compound IEM-1460 are equally potent in reducing the severity of nicotine-induced seizures in mice.
Topics: Adamantane; Animals; Biguanides; Male; Mice; Nicotine; Receptors, AMPA; Receptors, Nicotinic; Seizures | 2008 |
Ca(2+) permeable AMPA receptor induced long-term potentiation requires PI3/MAP kinases but not Ca/CaM-dependent kinase II.
Topics: Adamantane; Animals; Calcium; Calcium Signaling; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Hippocampus; Ions; Long-Term Potentiation; MAP Kinase Signaling System; Mice; Mice, Knockout; Mitogen-Activated Protein Kinases; Permeability; Phosphatidylinositol 3-Kinases; Protein Biosynthesis; Protein Transport; Receptors, AMPA; Synapses | 2009 |
Synaptic scaling requires the GluR2 subunit of the AMPA receptor.
Topics: Adamantane; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analysis of Variance; Animals; Animals, Newborn; Biophysics; Cells, Cultured; Disks Large Homolog 4 Protein; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Long-Term Potentiation; Membrane Proteins; Neurons; Patch-Clamp Techniques; Rats; Rats, Long-Evans; Receptors, AMPA; RNA Interference; RNA, Small Interfering; Sodium Channel Blockers; Synapses; Tetrodotoxin; Transfection; Visual Cortex | 2009 |
Ca2+-permeable AMPA receptors mediate induction of test pulse depression of naive synapses in rat visual cortical slices at early postnatal stage.
Topics: 2-Amino-5-phosphonovalerate; Adamantane; Aging; Animals; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Neural Inhibition; Patch-Clamp Techniques; Presynaptic Terminals; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Spermine; Synapses; Synaptic Transmission; Visual Cortex | 2010 |
Calcium-permeable AMPA receptors are involved in the induction and expression of l-DOPA-induced dyskinesia in Parkinson's disease.
Topics: Adamantane; Animals; Antiparkinson Agents; Behavior, Animal; Benserazide; Brain; Calcium; Callithrix; Dyskinesia, Drug-Induced; Enkephalins; Levodopa; Male; Motor Activity; Oxidopamine; Parkinson Disease; Protein Precursors; Rats; Rats, Sprague-Dawley; Receptors, AMPA | 2010 |
Selective inhibition of striatal fast-spiking interneurons causes dyskinesias.
Topics: Action Potentials; Adamantane; Analysis of Variance; Animals; Area Under Curve; Cholinergic Antagonists; Corpus Striatum; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Dyskinesias; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Functional Laterality; Green Fluorescent Proteins; Interneurons; LIM-Homeodomain Proteins; Male; Mecamylamine; Mice; Mice, Transgenic; N-Methylaspartate; Nerve Tissue Proteins; Scopolamine; Transcription Factors | 2011 |
Functional evidence for D-serine inhibition of non-N-methyl-D-aspartate ionotropic glutamate receptors in retinal neurons.
Topics: Adamantane; Animals; Calcium; Guinea Pigs; Kainic Acid; Patch-Clamp Techniques; Rats; Rats, Long-Evans; Receptors, AMPA; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Retinal Neurons; Serine | 2012 |
Brain-derived neurotrophic factor activation of CaM-kinase kinase via transient receptor potential canonical channels induces the translation and synaptic incorporation of GluA1-containing calcium-permeable AMPA receptors.
Topics: 2-Amino-5-phosphonovalerate; Adamantane; Animals; Benzimidazoles; Brain-Derived Neurotrophic Factor; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinase Kinase; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Female; Gene Knockdown Techniques; Hippocampus; Imidazoles; Male; Miniature Postsynaptic Potentials; Naphthalimides; Neurons; Primary Cell Culture; Rats; Rats, Sprague-Dawley; Receptors, AMPA; RNA, Small Interfering; TOR Serine-Threonine Kinases; TRPC Cation Channels | 2012 |
Eppendorf finalist. Striatal interneurons: causes of or cures for movement disorders?
Topics: Adamantane; Adrenergic Agents; Animals; Antiparkinson Agents; Corpus Striatum; Dopamine; Humans; Interneurons; Levodopa; Mice; Mice, Transgenic; Movement Disorders; Neural Pathways; Oxidopamine; Parkinsonian Disorders; Receptors, AMPA; Receptors, Kainic Acid; Treatment Failure | 2012 |
Alternative splicing of AMPA receptor subunits in the 6-OHDA-lesioned rat model of Parkinson's disease and L-DOPA-induced dyskinesia.
Topics: Adamantane; Alternative Splicing; Animals; Antiparkinson Agents; Cocaine; Corpus Striatum; Disease Models, Animal; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Iodine Isotopes; Levodopa; Male; Motor Activity; Oxidopamine; Parkinson Disease; Rats; Rats, Sprague-Dawley; Receptors, AMPA; RNA, Messenger; Sympatholytics | 2013 |
Kainate-induced calcium overload of cortical neurons in vitro: Dependence on expression of AMPAR GluA2-subunit and down-regulation by subnanomolar ouabain.
Topics: Adamantane; Animals; Calcium; Calcium Signaling; Cells, Cultured; Cerebral Cortex; Disease Models, Animal; Down-Regulation; Enzyme Inhibitors; Female; In Vitro Techniques; Kainic Acid; Nerve Degeneration; Neurons; Ouabain; Patch-Clamp Techniques; Piperidines; Pregnancy; Rats; Rats, Wistar; Receptors, AMPA | 2013 |
Acquisition of contextual discrimination involves the appearance of a RAS-GRF1/p38 mitogen-activated protein (MAP) kinase-mediated signaling pathway that promotes long term potentiation (LTP).
Topics: Adamantane; Animals; Butadienes; CA1 Region, Hippocampal; Calcium; Discrimination, Psychological; Extracellular Signal-Regulated MAP Kinases; Imidazoles; Long-Term Potentiation; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Nitriles; p38 Mitogen-Activated Protein Kinases; Pyridines; ras-GRF1; Receptors, AMPA; RNA Interference; Signal Transduction; Time Factors | 2013 |
[IEM-1460 and spermine potentiate analgesic effect of fentanyl and dipyrone in rats].
Topics: Adamantane; Anesthetics, Intravenous; Animals; Anti-Inflammatory Agents, Non-Steroidal; Dipyrone; Drug Synergism; Fentanyl; Male; Rats; Spermine | 2013 |
An antagonist of calcium permeable AMPA receptors, IEM1460: Anticonvulsant action in immature rats?
Topics: Adamantane; Animals; Anticonvulsants; Brain; Disease Models, Animal; Dose-Response Relationship, Drug; Electrodes, Implanted; Electroencephalography; Male; Pentylenetetrazole; Rats, Wistar; Receptors, AMPA; Seizures | 2015 |
Disruption of a neural microcircuit in the rod pathway of the mammalian retina by diabetes mellitus.
Topics: Adamantane; Amacrine Cells; Animals; Calcium; Diabetes Mellitus, Experimental; Excitatory Postsynaptic Potentials; Female; gamma-Aminobutyric Acid; Glutamic Acid; Neural Pathways; Rats; Receptors, AMPA; Retinal Bipolar Cells; Retinal Rod Photoreceptor Cells; Up-Regulation | 2015 |
Long-term upregulation of cortical glutamatergic AMPA receptors in a mouse model of chronic visceral pain.
Topics: Adamantane; Adenylyl Cyclases; Animals; Behavior, Animal; Calcium; Cell Membrane; Chronic Pain; Disease Models, Animal; Excitatory Postsynaptic Potentials; Gene Deletion; Glutamates; Gyrus Cinguli; Injections; Irritable Bowel Syndrome; Mice; Models, Biological; Phosphorylation; Phosphoserine; Protein Transport; Receptors, AMPA; Synaptic Transmission; Time Factors; Up-Regulation; Visceral Pain; Zymosan | 2015 |
Calcium-Permeable AMPA Receptors Mediate the Induction of the Protein Kinase A-Dependent Component of Long-Term Potentiation in the Hippocampus.
Topics: Adamantane; Analysis of Variance; Animals; Biophysics; Calcium; Cyclic AMP-Dependent Protein Kinases; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Polyamines; Rats; Receptors, AMPA; Rolipram | 2016 |
Postsynaptic Plasticity Triggered by Ca²⁺-Permeable AMPA Receptor Activation in Retinal Amacrine Cells.
Topics: Adamantane; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amacrine Cells; Animals; Calcium; Egtazic Acid; Excitatory Postsynaptic Potentials; Glutamic Acid; Goldfish; Membrane Potentials; Neuronal Plasticity; Receptors, AMPA; Retinal Bipolar Cells | 2016 |
Loss of Ca(2+)-permeable AMPA receptors in synapses of tonic firing substantia gelatinosa neurons in the chronic constriction injury model of neuropathic pain.
Topics: Adamantane; Animals; Calcium; Constriction, Pathologic; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Male; Neuralgia; Neurons; Rats; Receptors, AMPA; Spinal Cord; Substantia Gelatinosa; Synapses | 2016 |
Enduring abolishment of remote but not recent expression of conditioned fear by the blockade of calcium-permeable AMPA receptors before extinction training.
Topics: Adamantane; Amygdala; Animals; Calcium; Conditioning, Psychological; Extinction, Psychological; Fear; Hormones; Male; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, AMPA; RNA, Messenger | 2016 |
Chronic stress-induced dendritic reorganization and abundance of synaptosomal PKA-dependent CP-AMPA receptor in the basolateral amygdala in a mouse model of depression.
Topics: Adamantane; Animals; Antidepressive Agents; Basolateral Nuclear Complex; Cyclic AMP-Dependent Protein Kinases; Depression; Disease Models, Animal; Disks Large Homolog 4 Protein; Fluoxetine; Gene Expression Regulation; Guanylate Kinases; Male; Membrane Proteins; Mice; Mice, Inbred C57BL; Neurons; Phosphorylation; Post-Synaptic Density; Receptors, AMPA; Signal Transduction; Stress, Psychological; Synapses; Synaptophysin; Synaptosomes | 2017 |
Effects of selective calcium-permeable AMPA receptor blockade by IEM 1460 on psychotomimetic-induced hyperactivity in the mouse.
Topics: Adamantane; Animals; Behavior, Animal; Excitatory Amino Acid Antagonists; Hyperkinesis; Male; Mice; Mice, Inbred C57BL; Phencyclidine; Receptors, AMPA; Schizophrenia | 2018 |
Loss of Balance between Striatal Feedforward Inhibition and Corticostriatal Excitation Leads to Tremor.
Topics: Adamantane; Animals; Basal Ganglia Diseases; Cerebral Cortex; Corpus Striatum; Evoked Potentials; Female; Globus Pallidus; Interneurons; Microinjections; Motor Cortex; Muscimol; Rats; Rats, Long-Evans; Tremor | 2018 |
Opioid receptors inhibit the spinal AMPA receptor Ca
Topics: Adamantane; Animals; Calcium; Chronic Pain; Excitatory Postsynaptic Potentials; Freund's Adjuvant; Male; Mice; Mice, Inbred C57BL; Naltrexone; Narcotic Antagonists; Nerve Fibers, Unmyelinated; Nociception; Posterior Horn Cells; Receptors, AMPA; Receptors, Glutamate; Receptors, Opioid; Spinal Cord; Synapses | 2019 |
α-Amino-3-Hydroxy-5-Methyl-4-Isoxazolepropionic Acid Receptor Plasticity Sustains Severe, Fatal Status Epilepticus.
Topics: Adamantane; Amantadine; Animals; Atropine; CA1 Region, Hippocampal; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gene Knockdown Techniques; Hippocampus; Male; Mice; Mice, Knockout; Neuronal Plasticity; Receptors, AMPA; Status Epilepticus; Synaptic Transmission | 2020 |
Complex effects of eslicarbazepine on inhibitory micro networks in chronic experimental epilepsy.
Topics: Adamantane; Animals; Anticonvulsants; CA1 Region, Hippocampal; Calcium; Dibenzazepines; Disease Models, Animal; Dose-Response Relationship, Drug; Epilepsy; Feedback, Physiological; Hippocampus; Inhibitory Postsynaptic Potentials; Interneurons; Long-Term Potentiation; Muscarinic Agonists; Neural Inhibition; Neuronal Plasticity; Neurons; Pilocarpine; Pyramidal Cells; Rats; Receptors, AMPA | 2021 |
Environment-based object values learned by local network in the striatum tail.
Topics: Adamantane; Animals; Basal Ganglia; Corpus Striatum; Environment; Humans; Interneurons; Learning; Macaca mulatta; Male; Primates; Saccades | 2021 |
Insertion of Calcium-Permeable AMPA Receptors during Epileptiform Activity In Vitro Modulates Excitability of Principal Neurons in the Rat Entorhinal Cortex.
Topics: Adamantane; Animals; Calcium; Computer Simulation; Dizocilpine Maleate; Entorhinal Cortex; Epilepsy; GABA-B Receptor Antagonists; In Vitro Techniques; Male; Membranes; Models, Theoretical; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Rats, Wistar; Receptors, AMPA; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate | 2021 |