Page last updated: 2024-08-21

adamantane and az10606120

adamantane has been researched along with az10606120 in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's9 (64.29)24.3611
2020's5 (35.71)2.80

Authors

AuthorsStudies
Khadra, A; Li, S; Sherman, A; Stojilkovic, SS; Tomic, M; Yan, Z1
Marks, DC; Mullany, PR; Sluyter, R; Sophocleous, RA; Winter, KM1
Giannuzzo, A; Novak, I; Pedersen, SF1
Araújo, MGL; Fernandes, MJS; Franke, H; Gao, P; Illes, P; Khan, MT; Krügel, U; Liu, J; Rong, W; Rozmer, K; Tang, Y1
Alves, F; Ellegaard, M; Giannuzzo, A; Napp, J; Novak, I; Saccomano, M1
Sluyter, R; Vine, KL1
Allsopp, RC; Dayl, S; Evans, RJ; Schmid, R1
da Cunha-Bang, S; Dam, VH; Hjordt, LV; Knudsen, GM; Sestoft, D; Stenbæk, DS1
Ettrup, A; Farde, L; Finnema, SJ; Halldin, C; Knudsen, GM; Martinsson, S; Stepanov, V; Takano, A; Yang, KC1
Negulyaev, Y; Pugovkina, N; Semenova, S; Shamatova, M; Shatrova, A; Vassilieva, I1
Dunay, IR; Hörauf, JA; Janicova, A; Kany, S; Martin, L; Relja, B; Sturm, R; Vrdoljak, T; Xu, B1
Drummond, KJ; Kan, LK; Monif, M; O'Brien, TJ; Seneviratne, S; Williams, DA1
Drill, M; Hamilton, JA; Jones, NC; Kan, LK; Monif, M; O'Brien, TJ; Powell, KL1
Drill, M; Drummond, KJ; Galea, E; Hunn, M; Jayakrishnan, PC; Kan, LK; Monif, M; O'Brien, TJ; Sanfilippo, PG; Sequeira, RP; Todaro, M; Williams, DA1

Other Studies

14 other study(ies) available for adamantane and az10606120

ArticleYear
Experimental characterization and mathematical modeling of P2X7 receptor channel gating.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Oct-20, Volume: 30, Issue:42

    Topics: Adamantane; Algorithms; Aminoquinolines; Animals; Calcium; Cells, Cultured; Electrophysiology; Humans; Ion Channel Gating; Kinetics; Markov Chains; Models, Neurological; Models, Statistical; Nonlinear Dynamics; Patch-Clamp Techniques; Purinergic P2 Receptor Agonists; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Transfection

2010
Propensity of red blood cells to undergo P2X7 receptor-mediated phosphatidylserine exposure does not alter during in vivo or ex vivo aging.
    Transfusion, 2015, Volume: 55, Issue:8

    Topics: Adamantane; Adenosine Triphosphate; Aminoquinolines; Annexin A5; Azo Compounds; Benzenesulfonates; Blood Preservation; Cellular Senescence; Erythrocyte Membrane; Humans; Membrane Lipids; Osmotic Fragility; Phosphatidylserines; Purinergic P2X Receptor Antagonists; Pyridines; Pyridoxal Phosphate; Receptors, Purinergic P2X1; Receptors, Purinergic P2X7; Tetrazoles

2015
The P2X7 receptor regulates cell survival, migration and invasion of pancreatic ductal adenocarcinoma cells.
    Molecular cancer, 2015, Nov-25, Volume: 14

    Topics: Adamantane; Adenosine Triphosphate; Aminoquinolines; Apoptosis; Carcinoma, Pancreatic Ductal; Caspase 3; Caspase 7; Cell Line, Tumor; Cell Movement; Cell Survival; Humans; Neoplasm Invasiveness; Pancreatic Neoplasms; Purinergic P2X Receptor Agonists; Purinergic P2X Receptor Antagonists; Pyridines; Receptors, Purinergic P2X7; Tetrazoles

2015
Pilocarpine-Induced Status Epilepticus Increases the Sensitivity of P2X7 and P2Y1 Receptors to Nucleotides at Neural Progenitor Cells of the Juvenile Rodent Hippocampus.
    Cerebral cortex (New York, N.Y. : 1991), 2017, 07-01, Volume: 27, Issue:7

    Topics: Adamantane; Adenosine Triphosphate; Aminoquinolines; Animals; Disease Models, Animal; Excitatory Amino Acid Agents; Female; Gene Expression Regulation; Green Fluorescent Proteins; Hippocampus; Male; Membrane Potentials; Mice; Mice, Transgenic; Muscarinic Agonists; Neural Stem Cells; Nucleotides; Pilocarpine; Purinergic P2X Receptor Antagonists; Receptors, Purinergic P2X7; Receptors, Purinergic P2Y1; Status Epilepticus

2017
Targeting of the P2X7 receptor in pancreatic cancer and stellate cells.
    International journal of cancer, 2016, 12-01, Volume: 139, Issue:11

    Topics: Adamantane; Aminoquinolines; Animals; Carcinoma, Pancreatic Ductal; Cell Growth Processes; Cell Line, Tumor; Heterografts; Humans; Luminescent Measurements; Male; Mice; Mice, Inbred BALB C; Molecular Targeted Therapy; Pancreatic Neoplasms; Pancreatic Stellate Cells; Receptors, Purinergic P2X7

2016
N-Alkyl-Substituted Isatins Enhance P2X7 Receptor-Induced Interleukin-1β Release from Murine Macrophages.
    Mediators of inflammation, 2016, Volume: 2016

    Topics: Adamantane; Aminoquinolines; Animals; Cell Line; Interleukin-1beta; Isatin; Macrophages; Mice; Purinergic P2X Receptor Antagonists; Receptors, Purinergic P2X7

2016
Unique residues in the ATP gated human P2X7 receptor define a novel allosteric binding pocket for the selective antagonist AZ10606120.
    Scientific reports, 2017, 04-07, Volume: 7, Issue:1

    Topics: Adamantane; Adenosine Triphosphate; Alleles; Allosteric Regulation; Allosteric Site; Amino Acid Sequence; Amino Acid Substitution; Aminoquinolines; Binding Sites; Humans; Ion Channel Gating; Lignans; Models, Molecular; Molecular Conformation; Mutation; Protein Binding; Protein Interaction Domains and Motifs; Purinergic P2X Receptor Antagonists; Receptors, Purinergic P2X7; Structure-Activity Relationship

2017
Anterior cingulate serotonin 1B receptor binding is associated with emotional response inhibition.
    Journal of psychiatric research, 2017, Volume: 92

    Topics: Adamantane; Adult; Aminoquinolines; Emotions; Gyrus Cinguli; Humans; Image Processing, Computer-Assisted; Iodine Isotopes; Magnetic Resonance Imaging; Male; Neuropsychological Tests; Personality Disorders; Photic Stimulation; Positron-Emission Tomography; Protein Binding; Receptor, Serotonin, 5-HT1B; Violence; Young Adult

2017
Fenfluramine Reduces [11C]Cimbi-36 Binding to the 5-HT2A Receptor in the Nonhuman Primate Brain.
    The international journal of neuropsychopharmacology, 2017, 09-01, Volume: 20, Issue:9

    Topics: Adamantane; Aminoquinolines; Animals; Benzylamines; Brain; Brain Mapping; Dose-Response Relationship, Drug; Female; Fenfluramine; Fluorobenzenes; Macaca mulatta; Magnetic Resonance Imaging; Phenethylamines; Piperidines; Positron-Emission Tomography; Protein Binding; Purinergic P2X Receptor Antagonists; Receptor, Serotonin, 5-HT2A; Serotonin Agents

2017
Adenosine-5'-triphosphate suppresses proliferation and migration capacity of human endometrial stem cells.
    Journal of cellular and molecular medicine, 2020, Volume: 24, Issue:8

    Topics: Adamantane; Adenosine Triphosphate; Aminoquinolines; Cell Movement; Cell Proliferation; Endometrium; Female; Gene Expression Regulation, Developmental; Humans; Mesenchymal Stem Cells; Purinergic P2X Receptor Agonists; Purinergic P2X Receptor Antagonists; Receptors, Purinergic P2X7; Receptors, Purinergic P2Y; Regeneration

2020
Short Exposure to Ethanol Diminishes Caspase-1 and ASC Activation in Human HepG2 Cells In Vitro.
    International journal of molecular sciences, 2020, Apr-30, Volume: 21, Issue:9

    Topics: Adamantane; Amino Acid Chloromethyl Ketones; Aminoquinolines; Caspase 1; Ethanol; Hep G2 Cells; Humans; Inflammasomes; Lipopolysaccharides; Liver; Reactive Oxygen Species; Vanadates

2020
P2X7 receptor antagonism inhibits tumour growth in human high-grade gliomas.
    Purinergic signalling, 2020, Volume: 16, Issue:3

    Topics: Adamantane; Aminoquinolines; Brain Neoplasms; Cell Line, Tumor; Cell Proliferation; Glioma; Humans; Microglia; Microscopy, Confocal; Purinergic P2X Receptor Antagonists; Receptors, Purinergic P2X7; Rosaniline Dyes; Signal Transduction; Tumor Microenvironment

2020
Inhibition of purinergic P2X receptor 7 (P2X7R) decreases granulocyte-macrophage colony-stimulating factor (GM-CSF) expression in U251 glioblastoma cells.
    Scientific reports, 2020, 09-09, Volume: 10, Issue:1

    Topics: Adamantane; Aminoquinolines; Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Gene Expression Regulation, Neoplastic; Glioblastoma; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Purinergic P2X Receptor Antagonists; Receptors, Purinergic P2X7

2020
P2X7 receptor antagonism by AZ10606120 significantly reduced in vitro tumour growth in human glioblastoma.
    Scientific reports, 2023, 05-24, Volume: 13, Issue:1

    Topics: Adamantane; Aminoquinolines; Glioblastoma; Humans; Purinergic P2X Receptor Antagonists; Receptors, Purinergic P2X7; Temozolomide; Tumor Microenvironment

2023