Page last updated: 2024-09-02

acetylleucyl-leucyl-norleucinal and valinomycin

acetylleucyl-leucyl-norleucinal has been researched along with valinomycin in 2 studies

Compound Research Comparison

Studies
(acetylleucyl-leucyl-norleucinal)
Trials
(acetylleucyl-leucyl-norleucinal)
Recent Studies (post-2010)
(acetylleucyl-leucyl-norleucinal)
Studies
(valinomycin)
Trials
(valinomycin)
Recent Studies (post-2010) (valinomycin)
3210532,6670144

Protein Interaction Comparison

ProteinTaxonomyacetylleucyl-leucyl-norleucinal (IC50)valinomycin (IC50)
Bile salt export pumpHomo sapiens (human)3.4533
ATP-dependent translocase ABCB1Homo sapiens (human)3.2

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Assaraf, YG; Borgnia, MJ; Eytan, GD1
Broxterman, HJ; de Jong, MC; Dinkelberg, R; Kool, M; Meloen, RH; Puijk, WC; Scheffer, GL; Scheper, RJ; Schroeijers, AB; Slootstra, JW1

Other Studies

2 other study(ies) available for acetylleucyl-leucyl-norleucinal and valinomycin

ArticleYear
Competition of hydrophobic peptides, cytotoxic drugs, and chemosensitizers on a common P-glycoprotein pharmacophore as revealed by its ATPase activity.
    The Journal of biological chemistry, 1996, Feb-09, Volume: 271, Issue:6

    Topics: Adenosine Triphosphatases; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; CHO Cells; Clone Cells; Computer Simulation; Cricetinae; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Emetine; Gramicidin; Ionophores; Kinetics; Mathematics; Models, Theoretical; N-Formylmethionine Leucyl-Phenylalanine; Oligopeptides; Valinomycin

1996
Peptide transport by the multidrug resistance protein MRP1.
    Cancer research, 2001, Mar-15, Volume: 61, Issue:6

    Topics: Anti-Bacterial Agents; Antimetabolites, Antineoplastic; ATP-Binding Cassette Transporters; Biological Transport; Buthionine Sulfoximine; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; HL-60 Cells; Humans; Leupeptins; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Oligopeptides; Tumor Cells, Cultured; Valinomycin

2001