Page last updated: 2024-09-02

acetylleucyl-leucyl-norleucinal and epoxomicin

acetylleucyl-leucyl-norleucinal has been researched along with epoxomicin in 3 studies

Compound Research Comparison

Studies
(acetylleucyl-leucyl-norleucinal)
Trials
(acetylleucyl-leucyl-norleucinal)
Recent Studies (post-2010)
(acetylleucyl-leucyl-norleucinal)
Studies
(epoxomicin)
Trials
(epoxomicin)
Recent Studies (post-2010) (epoxomicin)
3210532510111

Protein Interaction Comparison

ProteinTaxonomyacetylleucyl-leucyl-norleucinal (IC50)epoxomicin (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.98
Proteasome subunit beta type-1Homo sapiens (human)1.25
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.98
Proteasome subunit beta type-5Homo sapiens (human)0.0256
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.98
Proteasome subunit beta type-2Homo sapiens (human)0.57
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.98
GABA theta subunitRattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.98

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's1 (33.33)24.3611
2020's1 (33.33)2.80

Authors

AuthorsStudies
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1
Dolcet, X; Encinas, M; Eritja, N; Llobet, D; Llombart-Cussac, A; Marti, RM; Matias-Guiu, X; Schoenenberger, JA; Sorolla, A; Yeramian, A1
Harada, M; Honma, Y; Shimizu, S; Takehara, T1

Other Studies

3 other study(ies) available for acetylleucyl-leucyl-norleucinal and epoxomicin

ArticleYear
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023
Antioxidants block proteasome inhibitor function in endometrial carcinoma cells.
    Anti-cancer drugs, 2008, Volume: 19, Issue:2

    Topics: Antioxidants; Antipyrine; Apoptosis; Ascorbic Acid; Blotting, Western; Boronic Acids; Bortezomib; Butylated Hydroxyanisole; Caspase 3; Caspase 9; Caspase Inhibitors; Cell Line, Tumor; Cell Survival; Coumarins; Cysteine Proteinase Inhibitors; Dose-Response Relationship, Drug; Edaravone; Endometrial Neoplasms; Ergothioneine; Female; Humans; Leupeptins; Oligopeptides; Proteasome Inhibitors; Pyrazines; Ubiquitin; Vitamin E; Vitamins

2008
Sorafenib enhances proteasome inhibitor-induced cell death via inactivation of Akt and stress-activated protein kinases.
    Journal of gastroenterology, 2014, Volume: 49, Issue:3

    Topics: Antineoplastic Agents; Apoptosis; Carcinoma, Hepatocellular; Cell Death; Cell Line, Tumor; Down-Regulation; Drug Synergism; Humans; Leupeptins; Liver Neoplasms; Molecular Targeted Therapy; Niacinamide; Oligopeptides; Phenylurea Compounds; Proteasome Inhibitors; Protein Kinase Inhibitors; Protein Kinases; Proto-Oncogene Proteins c-akt; Signal Transduction; Sorafenib

2014