Page last updated: 2024-09-02

acetylleucyl-leucyl-norleucinal and carfilzomib

acetylleucyl-leucyl-norleucinal has been researched along with carfilzomib in 2 studies

Compound Research Comparison

Studies
(acetylleucyl-leucyl-norleucinal)
Trials
(acetylleucyl-leucyl-norleucinal)
Recent Studies (post-2010)
(acetylleucyl-leucyl-norleucinal)
Studies
(carfilzomib)
Trials
(carfilzomib)
Recent Studies (post-2010) (carfilzomib)
321053748121716

Protein Interaction Comparison

ProteinTaxonomyacetylleucyl-leucyl-norleucinal (IC50)carfilzomib (IC50)
Proteasome subunit beta type-11Homo sapiens (human)0.0608
26S proteasome non-ATPase regulatory subunit 11Homo sapiens (human)0.0086
26S proteasome non-ATPase regulatory subunit 12Homo sapiens (human)0.0086
26S proteasome non-ATPase regulatory subunit 14Homo sapiens (human)0.0086
Proteasome subunit alpha type-7Homo sapiens (human)0.0608
26S proteasome non-ATPase regulatory subunit 3Homo sapiens (human)0.0086
26S proteasome regulatory subunit 6AHomo sapiens (human)0.0086
Proteasome subunit beta type-1Homo sapiens (human)0.5937
Proteasome subunit alpha type-1Homo sapiens (human)0.0608
Proteasome subunit alpha type-2Homo sapiens (human)0.0608
Proteasome subunit alpha type-3Homo sapiens (human)0.0608
Proteasome subunit alpha type-4Homo sapiens (human)0.0608
Proteasome subunit beta type-8Homo sapiens (human)0.0407
Proteasome subunit beta type-9Homo sapiens (human)0.7166
Proteasome subunit alpha type-5Homo sapiens (human)0.0608
Proteasome subunit beta type-4Homo sapiens (human)0.0608
Proteasome subunit beta type-6Homo sapiens (human)0.199
Proteasome subunit beta type-5Homo sapiens (human)0.0237
26S proteasome regulatory subunit 7Homo sapiens (human)0.0086
Proteasome subunit beta type-10Homo sapiens (human)0.1339
26S proteasome regulatory subunit 6BHomo sapiens (human)0.0086
26S proteasome non-ATPase regulatory subunit 8Homo sapiens (human)0.0086
Proteasome subunit beta type-3Homo sapiens (human)0.0608
Proteasome subunit beta type-2Homo sapiens (human)0.7493
26S proteasome non-ATPase regulatory subunit 7Homo sapiens (human)0.0086
26S proteasome non-ATPase regulatory subunit 4Homo sapiens (human)0.0086
26S proteasome complex subunit SEM1Homo sapiens (human)0.0086
Proteasome subunit alpha type-6Homo sapiens (human)0.0608
26S proteasome regulatory subunit 4Homo sapiens (human)0.0086
26S proteasome regulatory subunit 8Homo sapiens (human)0.0086
26S proteasome regulatory subunit 10BHomo sapiens (human)0.0086
Glutathione S-transferase omega-1Homo sapiens (human)0.15
26S proteasome non-ATPase regulatory subunit 2Homo sapiens (human)0.0086
26S proteasome non-ATPase regulatory subunit 6Homo sapiens (human)0.0086
Proteasomal ubiquitin receptor ADRM1Homo sapiens (human)0.0086
Proteasome subunit alpha-type 8Homo sapiens (human)0.0608
Proteasome subunit beta type-7Homo sapiens (human)0.0578
26S proteasome non-ATPase regulatory subunit 1Homo sapiens (human)0.0086
26S proteasome non-ATPase regulatory subunit 13Homo sapiens (human)0.0086

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's2 (100.00)2.80

Authors

AuthorsStudies
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1
Fan, Y; You, G1

Other Studies

2 other study(ies) available for acetylleucyl-leucyl-norleucinal and carfilzomib

ArticleYear
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023
Proteasome Inhibitors Bortezomib and Carfilzomib Stimulate the Transport Activity of Human Organic Anion Transporter 1.
    Molecular pharmacology, 2020, Volume: 97, Issue:6

    Topics: Antineoplastic Agents; Biological Transport, Active; Bortezomib; HEK293 Cells; Humans; Leupeptins; Oligopeptides; Organic Anion Transport Protein 1; p-Aminohippuric Acid; Proteasome Endopeptidase Complex; Proteasome Inhibitors; Proteolysis; Ubiquitination

2020