Page last updated: 2024-09-02

acetylleucyl-leucyl-norleucinal and calpain inhibitor iii

acetylleucyl-leucyl-norleucinal has been researched along with calpain inhibitor iii in 4 studies

Compound Research Comparison

Studies
(acetylleucyl-leucyl-norleucinal)
Trials
(acetylleucyl-leucyl-norleucinal)
Recent Studies (post-2010)
(acetylleucyl-leucyl-norleucinal)
Studies
(calpain inhibitor iii)
Trials
(calpain inhibitor iii)
Recent Studies (post-2010) (calpain inhibitor iii)
321053187076

Protein Interaction Comparison

ProteinTaxonomyacetylleucyl-leucyl-norleucinal (IC50)calpain inhibitor iii (IC50)
Calpain-9Homo sapiens (human)1.61
Calpain-1 catalytic subunitHomo sapiens (human)0.183
Procathepsin LHomo sapiens (human)0.6365
Cathepsin BHomo sapiens (human)0.5186
Calpain-2 catalytic subunitHomo sapiens (human)0.35
Calpain-1 catalytic subunitSus scrofa (pig)0.02
Vascular endothelial growth factor receptor 2Homo sapiens (human)0.1
Falcipain 2B Plasmodium falciparum (malaria parasite P. falciparum)5
Cysteine proteinase falcipain 2a Plasmodium falciparum (malaria parasite P. falciparum)5

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Inomata, M; Nakamura, M; Ohno, H; Shintani-Ishida, K; Uemura, K; Yoshida, K1
Endo, S; Kondo, M; Mourin, R; Nakazawa, T; Nishida, K; Saido, TC; Shimura, M; Yokokura, S1
Ali, MA; Fan, X; Holt, A; Schulz, R; Stepanko, A1
Duregotti, E; Montecucco, C; Rigoni, M; Tedesco, E1

Other Studies

4 other study(ies) available for acetylleucyl-leucyl-norleucinal and calpain inhibitor iii

ArticleYear
Ischemia promotes calpain-mediated degradation of p120-catenin in SH-SY5Y cells.
    Biochemical and biophysical research communications, 2007, Feb-16, Volume: 353, Issue:3

    Topics: Acetylcysteine; Calpain; Catenins; Cell Adhesion Molecules; Cell Aggregation; Cell Death; Cell Line, Tumor; Delta Catenin; Dipeptides; Humans; Ischemia; Leupeptins; Neuroblastoma; Phosphoproteins

2007
Calpain-mediated degradation of G-substrate plays a critical role in retinal excitotoxicity for amacrine cells.
    Journal of neuroscience research, 2009, May-01, Volume: 87, Issue:6

    Topics: Amacrine Cells; Analysis of Variance; Animals; Blotting, Western; Calpain; Cell Death; Cysteine Proteinase Inhibitors; Dipeptides; Immunohistochemistry; In Situ Nick-End Labeling; Leupeptins; Mice; Mice, Inbred C57BL; Mice, Knockout; N-Methylaspartate; Nerve Tissue Proteins; Proto-Oncogene Proteins c-akt; Rats; Rats, Sprague-Dawley; Retina

2009
Calpain inhibitors exhibit matrix metalloproteinase-2 inhibitory activity.
    Biochemical and biophysical research communications, 2012, Jun-22, Volume: 423, Issue:1

    Topics: Acrylates; Calpain; Catalysis; Cell Line; Cysteine Proteinase Inhibitors; Dipeptides; Gelatin; Humans; Inhibitory Concentration 50; Leupeptins; Matrix Metalloproteinase 2; Matrix Metalloproteinase Inhibitors; Oligopeptides; Phenyl Ethers; Troponin I

2012
Calpains participate in nerve terminal degeneration induced by spider and snake presynaptic neurotoxins.
    Toxicon : official journal of the International Society on Toxinology, 2013, Mar-15, Volume: 64

    Topics: Acrylates; Animals; Animals, Newborn; Calcium Signaling; Calpain; Cell Membrane Permeability; Cells, Cultured; Cytoskeleton; Dipeptides; Leupeptins; Nerve Degeneration; Neurofilament Proteins; Neurons; Neurotoxins; Phospholipases A2; Presynaptic Terminals; Rats; Rats, Wistar; Snake Venoms; Spectrin; Spider Venoms

2013