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acetylleucyl-leucyl-norleucinal and brefeldin a

acetylleucyl-leucyl-norleucinal has been researched along with brefeldin a in 10 studies

Compound Research Comparison

Studies
(acetylleucyl-leucyl-norleucinal)
Trials
(acetylleucyl-leucyl-norleucinal)
Recent Studies (post-2010)
(acetylleucyl-leucyl-norleucinal)
Studies
(brefeldin a)
Trials
(brefeldin a)
Recent Studies (post-2010) (brefeldin a)
3210532,6001456

Protein Interaction Comparison

ProteinTaxonomyacetylleucyl-leucyl-norleucinal (IC50)brefeldin a (IC50)
major prion protein preproprotein Prp precursorHomo sapiens (human)3.505
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)0.1343

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (50.00)18.2507
2000's5 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bilter, GK; Dias, J; Huang, Z; Keon, BH; Lamerdin, J; MacDonald, ML; Michnick, SW; Minami, T; Owens, S; Shang, Z; Westwick, JK; Yu, H1
Getz, GS; Reardon, CA; Ye, SQ1
Davis, EC; Mecham, RP1
Ginsberg, HN; Jiang, H; Lele, KM; Sakata, N; Wu, X; Zhou, M1
Broekelmann, TJ; Davis, EC; Mecham, RP; Ozawa, Y1
Asakura, T; Hashizume, Y; Ohkawa, K; Okawa, Y; Sawai, T; Takada, K; Yanaihara, N1
Franco, AV; Gray, CP; Hersey, P; Nguyen, T; Zhang, XD1
Horonchik, L; Taraboulos, A; Tzaban, S; Yanai, A; Yedidia, Y1
Alderson, MR; Grotzke, JE; Heinzel, AS; Johnson, M; Lewinsohn, DM; Ovendale, PJ; Zhu, L1
Amano, T; Kameyama, N; Mochizuki, H; Nobukuni, M; Okada, S; Sakai, N; Seki, T; Tanaka, A; Yamamoto, H1

Other Studies

10 other study(ies) available for acetylleucyl-leucyl-norleucinal and brefeldin a

ArticleYear
Identifying off-target effects and hidden phenotypes of drugs in human cells.
    Nature chemical biology, 2006, Volume: 2, Issue:6

    Topics: Bacterial Proteins; Cell Line; Cell Proliferation; Cluster Analysis; Drug Design; Drug Evaluation, Preclinical; Genetics; Humans; Luminescent Proteins; Molecular Structure; Phenotype; Recombinant Fusion Proteins; Signal Transduction; Structure-Activity Relationship

2006
Inhibition of apolipoprotein E degradation in a post-Golgi compartment by a cysteine protease inhibitor.
    The Journal of biological chemistry, 1993, Apr-25, Volume: 268, Issue:12

    Topics: Albumins; Ammonium Chloride; Animals; Apolipoproteins E; Brefeldin A; Calcium; Cathepsin B; Cathepsin L; Cathepsins; Chloroquine; CHO Cells; Cricetinae; Cyclopentanes; Cysteine Endopeptidases; Cysteine Proteinase Inhibitors; Endopeptidases; Golgi Apparatus; Humans; Kinetics; Leupeptins; Molecular Sequence Data; Transfection; Tumor Cells, Cultured

1993
Selective degradation of accumulated secretory proteins in the endoplasmic reticulum. A possible clearance pathway for abnormal tropoelastin.
    The Journal of biological chemistry, 1996, Feb-16, Volume: 271, Issue:7

    Topics: Ammonium Chloride; Animals; Blotting, Northern; Brefeldin A; Cattle; Cells, Cultured; Cycloheximide; Cyclopentanes; Endoplasmic Reticulum; Leucine; Leupeptins; Ligaments; Microscopy, Electron; Nocodazole; Organelles; Protein Synthesis Inhibitors; RNA, Messenger; Serine Proteinase Inhibitors; Transcription, Genetic; Tropoelastin

1996
A two-site model for ApoB degradation in HepG2 cells.
    The Journal of biological chemistry, 1997, Apr-25, Volume: 272, Issue:17

    Topics: Apolipoproteins B; Biological Transport; Brefeldin A; Cyclopentanes; Cysteine Proteinase Inhibitors; Dithiothreitol; Endoplasmic Reticulum; Humans; Leupeptins; Liver; Models, Biological; Oleic Acid; Peptide Fragments; Protein Synthesis Inhibitors

1997
Identification of tropoelastin as a ligand for the 65-kD FK506-binding protein, FKBP65, in the secretory pathway.
    The Journal of cell biology, 1998, Jan-26, Volume: 140, Issue:2

    Topics: Amino Acid Isomerases; Animals; Brefeldin A; Carrier Proteins; Cattle; Cell Compartmentation; Centrifugation, Density Gradient; Cyclopentanes; Cysteine; DNA-Binding Proteins; Heat-Shock Proteins; Leupeptins; Ligands; Methionine; Molecular Weight; Protein Folding; Protein Synthesis Inhibitors; Tacrolimus; Tacrolimus Binding Proteins; Tropoelastin

1998
Calpain inhibitor causes accumulation of ubiquitinated P-glycoprotein at the cell surface: possible role of calpain in P-glycoprotein turnover.
    International journal of oncology, 1999, Volume: 15, Issue:4

    Topics: Acetylcysteine; Ammonium Chloride; ATP Binding Cassette Transporter, Subfamily B; Blotting, Western; Brefeldin A; Calpain; Cell Membrane; Cysteine Proteinase Inhibitors; Dipeptides; Doxorubicin; Enzyme-Linked Immunosorbent Assay; Glycoproteins; Humans; K562 Cells; Leucine; Leupeptins; Membrane Proteins; Protein Synthesis Inhibitors; Time Factors; Ubiquitins

1999
Differential localization and regulation of death and decoy receptors for TNF-related apoptosis-inducing ligand (TRAIL) in human melanoma cells.
    Journal of immunology (Baltimore, Md. : 1950), 2000, Apr-15, Volume: 164, Issue:8

    Topics: Amino Acid Chloromethyl Ketones; Apoptosis; Apoptosis Regulatory Proteins; Brefeldin A; Cell Nucleus; Cysteine Proteinase Inhibitors; DNA, Complementary; GPI-Linked Proteins; Humans; Leupeptins; Ligands; Melanoma; Membrane Glycoproteins; Protein Synthesis Inhibitors; Receptors, TNF-Related Apoptosis-Inducing Ligand; Receptors, Tumor Necrosis Factor; Receptors, Tumor Necrosis Factor, Member 10c; Signal Transduction; Subcellular Fractions; TNF-Related Apoptosis-Inducing Ligand; Transfection; Tumor Cells, Cultured; Tumor Necrosis Factor Decoy Receptors; Tumor Necrosis Factor-alpha

2000
Proteasomes and ubiquitin are involved in the turnover of the wild-type prion protein.
    The EMBO journal, 2001, Oct-01, Volume: 20, Issue:19

    Topics: Animals; Brefeldin A; CHO Cells; Cricetinae; Cysteine Endopeptidases; Cytoplasm; Endoplasmic Reticulum; Leupeptins; Membrane Proteins; Mice; Multienzyme Complexes; Protease Inhibitors; Proteasome Endopeptidase Complex; Protein Processing, Post-Translational; PrPC Proteins; Solubility; Tumor Cells, Cultured; Ubiquitin

2001
Secreted proteins from Mycobacterium tuberculosis gain access to the cytosolic MHC class-I antigen-processing pathway.
    Journal of immunology (Baltimore, Md. : 1950), 2006, Jul-01, Volume: 177, Issue:1

    Topics: Adenoviruses, Human; Amino Acid Sequence; Antigen Presentation; ATP-Binding Cassette Transporters; Bacterial Proteins; Brefeldin A; Cell Line; Cell Line, Transformed; Clone Cells; Cytosol; Histocompatibility Antigens Class I; Humans; Immediate-Early Proteins; Lactic Acid; Leupeptins; Microspheres; Molecular Sequence Data; Mycobacterium tuberculosis; Polyglycolic Acid; Polylactic Acid-Polyglycolic Acid Copolymer; Polymers; Proteasome Inhibitors; Signal Transduction; Viral Proteins

2006
The C-terminal region of serotonin transporter is important for its trafficking and glycosylation.
    Journal of pharmacological sciences, 2009, Volume: 111, Issue:4

    Topics: Acetylcysteine; Animals; Binding Sites; Brefeldin A; Chlorocebus aethiops; COS Cells; Cysteine Proteinase Inhibitors; Endoplasmic Reticulum; Glycosylation; Leupeptins; Membrane Transport Modulators; Protein Structure, Tertiary; Protein Transport; Quinones; Sequence Deletion; Serotonin; Serotonin Plasma Membrane Transport Proteins; Sesquiterpenes; Structure-Activity Relationship; Transfection

2009