acetaminophen and warfarin

acetaminophen has been researched along with warfarin in 111 studies

Research

Studies (111)

TimeframeStudies, this research(%)All Research%
pre-199018 (16.22)18.7374
1990's21 (18.92)18.2507
2000's36 (32.43)29.6817
2010's29 (26.13)24.3611
2020's7 (6.31)2.80

Authors

AuthorsStudies
Duffy, EM; Jorgensen, WL1
Topliss, JG; Yoshida, F1
Alvarez-Pedraglio, A; Colmenarejo, G; Lavandera, JL1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Lombardo, F; Obach, RS; Waters, NJ1
He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Sun, Y; Yan, Z1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Botta, M; Dreassi, E; Falchi, F; Maga, G; Santucci, A; Schenone, S; Zizzari, AT1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Avdeef, A; Tam, KY1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1
Bellera, CL; Bruno-Blanch, LE; Castro, EA; Duchowicz, PR; Goodarzi, M; Ortiz, EV; Pesce, G; Talevi, A1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Honda, K; Izumi, T; Miyaji, Y; Nakayama, S; Okazaki, O; Okudaira, N; Shiosakai, K; Sugiyama, D; Suzuki, W; Takakusa, H; Watanabe, A1
Ambroso, JL; Ayrton, AD; Baines, IA; Bloomer, JC; Chen, L; Clarke, SE; Ellens, HM; Harrell, AW; Lovatt, CA; Reese, MJ; Sakatis, MZ; Taylor, MA; Yang, EY1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Andersson, B; Grafström, R; Moldéus, P; Orrenius, S1
Brown, KF; Crooks, MJ1
Assandri, A; Perazzi, A1
Lovering, EG; McGilveray, IJ; McMillan, I; Tostowaryk, W1
Breckenridge, A; Cook, P; Orme, M1
Jones, RV1
Bartle, WR; Blakely, JA1
Justice, JL; Kline, SS1
Jatlow, P1
Coldwell, BB; Grice, HC; Zawidzka, ZZ1
Soloway, HB1
Antlitz, AM; Mead, JA; Tolentino, MA1
Antlitz, AM; Awalt, LF1
Awalt, LF1
Boeijinga, JJ; Boerstra, EE; Breimer, DD; Jeletich-Bastiaanse, A; Ris, P1
Luczynska, C; Wilson, K1
Hawkes, C; Prudden, D; Smith, R1
D'Arcy, PF1
Goldberg, DM1
Bartle, WR; Kwan, D; Walker, SE2
Raiford, DS; Thigpen, MC1
Bartle, WR; Kwan, D1
Buss, DC; Cassidy, SL; Hale, A; Routledge, PA1
Fitzmaurice, DA; Murray, JA1
Heiman, H; Hylek, EM; Sheehan, MA; Singer, DE; Skates, SJ1
Bell, WR1
Brown, D1
Estrada, C1
Gray, CD1
Amato, MG; Bussey, H; Farnett, L; Lyons, R1
Gilroy, C; Hudson, P; McCay, L; Riser, J; Willis, TA1
Pedell, L1
Eliason, BC; Larson, W; Singer, DE; Skates, SJ1
Evans, MF; Gerstein, FH1
Elias, M1
Chan, LN; Nutescu, E; Shek, KL1
Ackermann, BL; Campanale, K; Fisher, MB; VandenBranden, M; Wrighton, SA1
Bates, D; Mintz, M1
Lehmann, DE1
Andrews, FJ1
Evans, IL; Gibbons, AJ; Price, G; Sayers, MS; Snooks, H; Sugar, AW1
Gallus, AS; Gebauer, MG; Henschke, PJ; Nyfort-Hansen, K1
Gadisseur, AP; Rosendaal, FR; Van Der Meer, FJ1
Faulkner, MA; Lenz, NJ; Lenz, TL1
Lesho, EP; Saullo, L; Udvari-Nagy, S1
Hylek, EM1
Claessens, JG; Soute, BA; Thijssen, HH; Vervoort, LM1
Bal dit Sollier, C; Bergmann, JF; Bertrand, N; Caulin, C; Drouet, L; Mahé, I; Mazoyer, E; Simoneau, G2
Ditmer, D; Feldstein, AC; Krall, M; Perrin, N; Platt, R; Simon, SR; Sittig, DF; Smith, DH; Soumerai, SB; Yang, X1
Chaiyakunapruk, N; Jampachaisri, K; Kotirum, S; Rojnuckarin, P; Wattanasombat, S1
Beckey, NP; Parra, D; Stevens, GR1
Ingaszewski, A; Kerr, C; Lynd, L; Richardson, K; Shalansky, S1
Dharmarajan, L; Sajjad, W1
Hersh, EV; Moore, PA; Pinto, A1
Giverhaug, T; Håkonsen, GD; Pettersen, MH; Skurtveit, S1
Launiainen, T; Ojanperä, I; Rasanen, I; Sajantila, A; Vuori, E1
Beyan, C; Beyan, E; Vaizoğlu, SA1
Miller, GP1
Alvarez, JC; Aubourg, R; Bal-dit-Sollier, C; Berge, N; Bergmann, JF; Drouet, L; Mahé, I; Mouly, S; Pruvot, S; Simoneau, G; Zhang, Q1
Gadea, CM; Ruiz, XD1
Berube, C; Lee, R; Wen, A1
Bennett, KP; Bergeron, C; Breneman, CM; Huang, TW; Rydberg, P; Zaretzki, J1
Crowther, MA; Garcia, DA; Horowitz, JD; Hylek, EM; Lopes, RD1
Hughes, GJ; Patel, PN; Saxena, N1
Abobo, CV; Hsiao, C; John, J; John, M; Liang, D; Wu, L1
Beall, JW; Kyle, JA; Pinson, GM1
Dumont, Z; Kosar, L; Mordasiewicz, M; Schuster, B1
Barra, M; Caldeira, D; Costa, J; Ferreira, JJ; Pinto, FJ1
Dalhoff, KP; Naver, SV; Papina, M; Solem, EJ1
Berckmans, P; Covaci, A; Hollanders, K; Maho, W; Peers, B; Remy, S; Verstraelen, S; Witters, H1
Cipolat Mis, T; Del Giudice, R; Nicolì, F; Schiano di Visconte, M1
Li, CJ; Ma, J; Sun, H; Yang, JZ; Zhang, DM1
Cui, J; Fan, L; Hu, H; Kaplowitz, N; Liu, X; Lu, S; Lu, X; Yan, M; Ye, L; Yin, S1
Bell, JS; Farinola, N; Hauta-Aho, M; Huupponen, R; Johns, S; Korhonen, MJ; Shakib, S; Teperi, S1
Leong, D; Wu, PE1
Cheng, D; Gong, X; Lv, Y; Wu, Q; Yuan, J; Yuan, L; Zhang, X1
Dong, JH; Ma, QG; Sang, ZP; Wei, RR1
Jimenez-Solem, E; Nyeland, ME; Odgaard, A; Overgaard, S; Schelde, AB; Sørensen, AMS1
Dai, X; Gao, Z; Huang, J; Jin, ZG; Lan, T; Sun, Y; Tang, J; Wu, X; Xu, S; Yi, W1
Setiawan, A; Vohra, V; Winograd, EJ1

Reviews

11 review(s) available for acetaminophen and warfarin

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
The clinical significance of the effects of cigarette smoking on drug disposition.
    Methods and findings in experimental and clinical pharmacology, 1983, Volume: 5, Issue:7

    Topics: Acetaminophen; Antipyrine; Benzodiazepines; Chlorpromazine; Clomipramine; Codeine; Humans; Pharmaceutical Preparations; Phenacetin; Propranolol; Smoking; Theophylline; Warfarin

1983
The expanding role of microsomal enzyme induction, and its implications for clinical chemistry.
    Clinical chemistry, 1980, Volume: 26, Issue:6

    Topics: Acetaminophen; Alcoholism; Animals; Antipyrine; Aryl Hydrocarbon Hydroxylases; Electron Transport; Energy Intake; Enzyme Induction; Epilepsy; Female; Humans; Male; Microsomes, Liver; Pharmacology; Phenobarbital; Phenylbutazone; Phenytoin; Smoking; Tolbutamide; Warfarin

1980
Warfarin-acetaminophen drug interaction revisited.
    Pharmacotherapy, 1999, Volume: 19, Issue:10

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Clinical Trials as Topic; Drug Synergism; Humans; Pharmacogenetics; Warfarin

1999
Phytonadione therapy in a multiple-drug overdose involving warfarin.
    Pharmacotherapy, 2000, Volume: 20, Issue:10

    Topics: Acetaminophen; Acetylcysteine; Aged; Analgesics, Non-Narcotic; Anti-Bacterial Agents; Anticoagulants; Antidotes; Antifibrinolytic Agents; Azabicyclo Compounds; Charcoal; Drug Interactions; Drug Overdose; Female; Gastric Lavage; Humans; Hypnotics and Sedatives; International Normalized Ratio; Piperazines; Vitamin K; Vitamin K 1; Warfarin

2000
Enzymatic shunting: resolving the acetaminophen-warfarin controversy.
    Pharmacotherapy, 2000, Volume: 20, Issue:12

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Animals; Anticoagulants; Binding, Competitive; Cytochrome P-450 Enzyme System; Drug Synergism; Humans; Isoenzymes; Stereoisomerism; Warfarin

2000
Potential interactions between exercise and drug therapy.
    Sports medicine (Auckland, N.Z.), 2004, Volume: 34, Issue:5

    Topics: Absorption; Acetaminophen; Adrenergic beta-Antagonists; Aspirin; Digoxin; Doxycycline; Exercise; Humans; Insulin; Pharmacokinetics; Theophylline; Tissue Distribution; Verapamil; Warfarin

2004
Adverse drug interactions involving common prescription and over-the-counter analgesic agents.
    Clinical therapeutics, 2007, Volume: 29 Suppl

    Topics: Acetaminophen; Analgesics; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Drug Interactions; Ethanol; Health Status; Humans; Lithium Compounds; Methotrexate; Nonprescription Drugs; Selective Serotonin Reuptake Inhibitors; Warfarin

2007
Effect of acetaminophen on international normalized ratio in patients receiving warfarin therapy.
    Pharmacotherapy, 2011, Volume: 31, Issue:6

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Dose-Response Relationship, Drug; Drug Interactions; Drug Monitoring; Humans; International Normalized Ratio; Warfarin

2011
A review of warfarin dosing with concurrent acetaminophen therapy.
    Journal of pharmacy practice, 2013, Volume: 26, Issue:5

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Drug Interactions; Drug Monitoring; Humans; International Normalized Ratio; Practice Guidelines as Topic; Thromboembolism; Warfarin

2013
How safe is acetaminophen use in patients treated with vitamin K antagonists? A systematic review and meta-analysis.
    Thrombosis research, 2015, Volume: 135, Issue:1

    Topics: Acetaminophen; Analgesics; Blood Coagulation; Humans; International Normalized Ratio; Observational Studies as Topic; Randomized Controlled Trials as Topic; Regression Analysis; Treatment Outcome; Vitamin K; Warfarin

2015

Trials

13 trial(s) available for acetaminophen and warfarin

ArticleYear
Potentiation of oral anticoagulant therapy by acetaminophen.
    Current therapeutic research, clinical and experimental, 1968, Volume: 10, Issue:10

    Topics: Acetaminophen; Anticoagulants; Blood Coagulation; Clinical Trials as Topic; Drug Synergism; Humans; Placebos; Prothrombin Time; Warfarin

1968
A double blind study of acetaminophen used in conjunction with oral anticoagulant therapy.
    Current therapeutic research, clinical and experimental, 1969, Volume: 11, Issue:6

    Topics: Acetaminophen; Anticoagulants; Clinical Trials as Topic; Coumarins; Humans; Placebos; Warfarin

1969
Interaction between paracetamol and coumarin anticoagulants.
    Lancet (London, England), 1982, Feb-27, Volume: 1, Issue:8270

    Topics: Acetaminophen; Blood Coagulation; Clinical Trials as Topic; Double-Blind Method; Drug Interactions; Humans; Random Allocation; Warfarin

1982
The effects of acetaminophen on pharmacokinetics and pharmacodynamics of warfarin.
    Journal of clinical pharmacology, 1999, Volume: 39, Issue:1

    Topics: Acetaminophen; Administration, Oral; Adolescent; Alanine Transaminase; Analgesics, Non-Narcotic; Analysis of Variance; Anticoagulants; Aspartate Aminotransferases; Cross-Over Studies; Dose-Response Relationship, Drug; Drug Interactions; Factor VII; Humans; Male; Middle Aged; Prothrombin Time; Stereoisomerism; Time Factors; Warfarin

1999
Can warfarin be continued during dental extraction? Results of a randomized controlled trial.
    The British journal of oral & maxillofacial surgery, 2002, Volume: 40, Issue:3

    Topics: Acetaminophen; Adult; Aged; Aged, 80 and over; Analgesics, Non-Narcotic; Anesthetics, Local; Anticoagulants; Chi-Square Distribution; Confidence Intervals; Female; Follow-Up Studies; Hemostasis, Surgical; Humans; International Normalized Ratio; Lidocaine; Male; Middle Aged; Oral Hemorrhage; Postoperative Hemorrhage; Risk Factors; Statistics as Topic; Tooth Extraction; Warfarin

2002
Sustained intake of paracetamol (acetaminophen) during oral anticoagulant therapy with coumarins does not cause clinically important INR changes: a randomized double-blind clinical trial.
    Journal of thrombosis and haemostasis : JTH, 2003, Volume: 1, Issue:4

    Topics: Acetaminophen; Adult; Aged; Anticoagulants; Coumarins; Dose-Response Relationship, Drug; Double-Blind Method; Drug Interactions; Drug Therapy, Combination; Female; Humans; International Normalized Ratio; Male; Middle Aged; Prothrombin Time

2003
Paracetamol: a haemorrhagic risk factor in patients on warfarin.
    British journal of clinical pharmacology, 2005, Volume: 59, Issue:3

    Topics: Acetaminophen; Adult; Aged; Aged, 80 and over; Analgesics, Non-Narcotic; Anticoagulants; Contraindications; Cross-Over Studies; Double-Blind Method; Drug Synergism; Drug Therapy, Combination; Hemorrhage; Humans; International Normalized Ratio; Middle Aged; Prospective Studies; Risk Factors; Warfarin

2005
Reducing warfarin medication interactions: an interrupted time series evaluation.
    Archives of internal medicine, 2006, May-08, Volume: 166, Issue:9

    Topics: Acetaminophen; Adult; Aged; Aged, 80 and over; Anti-Infective Agents; Anti-Inflammatory Agents, Non-Steroidal; Anticoagulants; Drug Interactions; Drug Prescriptions; Education, Medical, Continuing; Female; Fluconazole; Health Maintenance Organizations; Humans; Male; Medical Records Systems, Computerized; Metronidazole; Middle Aged; Sulfamethoxazole; Warfarin

2006
Interaction between paracetamol and warfarin in patients: a double-blind, placebo-controlled, randomized study.
    Haematologica, 2006, Volume: 91, Issue:12

    Topics: Acetaminophen; Adult; Aged; Aged, 80 and over; Cross-Over Studies; Double-Blind Method; Drug Interactions; Female; Humans; International Normalized Ratio; Male; Middle Aged; Prospective Studies; Warfarin

2006
The effect of acetaminophen on the international normalized ratio in patients stabilized on warfarin therapy.
    Pharmacotherapy, 2007, Volume: 27, Issue:5

    Topics: Acetaminophen; Aged; Alanine Transaminase; Analgesics, Non-Narcotic; Anticoagulants; Aspartate Aminotransferases; Double-Blind Method; Drug Interactions; Drug Monitoring; Female; Humans; International Normalized Ratio; Male; Middle Aged; Prospective Studies; Warfarin

2007
Risk of warfarin-related bleeding events and supratherapeutic international normalized ratios associated with complementary and alternative medicine: a longitudinal analysis.
    Pharmacotherapy, 2007, Volume: 27, Issue:9

    Topics: Acetaminophen; Adult; Age Factors; Aged; Aged, 80 and over; Anticoagulants; Canada; Coenzymes; Complementary Therapies; Diarrhea; Dietary Supplements; Drug Interactions; Ethanol; Female; Hemorrhage; Herb-Drug Interactions; Humans; International Normalized Ratio; Longitudinal Studies; Male; Middle Aged; Phytotherapy; Plants, Medicinal; Prospective Studies; Risk Factors; Ubiquinone; Vitamins; Warfarin; Zingiber officinale

2007
Interaction between acetaminophen and warfarin in adults receiving long-term oral anticoagulants: a randomized controlled trial.
    European journal of clinical pharmacology, 2011, Volume: 67, Issue:3

    Topics: Acetaminophen; Administration, Oral; Adult; Aged; Aged, 80 and over; Analgesics, Non-Narcotic; Anticoagulants; Dose-Response Relationship, Drug; Double-Blind Method; Drug Interactions; Drug Monitoring; Female; Humans; International Normalized Ratio; Male; Middle Aged; Prospective Studies; Warfarin; Young Adult

2011
Effect of a mixture of diosmin, coumarin glycosides, and triterpenes on bleeding, thrombosis, and pain after stapled anopexy: a prospective, randomized, placebo-controlled clinical trial.
    International journal of colorectal disease, 2017, Volume: 32, Issue:3

    Topics: Acetaminophen; Adult; Aged; Blood Loss, Surgical; Coumarins; Demography; Digestive System Surgical Procedures; Diosmin; Female; Glycosides; Hemorrhoids; Humans; Male; Middle Aged; Pain Measurement; Pain, Postoperative; Placebos; Prospective Studies; Surgical Stapling; Thrombosis; Triterpenes

2017

Other Studies

87 other study(ies) available for acetaminophen and warfarin

ArticleYear
Prediction of drug solubility from Monte Carlo simulations.
    Bioorganic & medicinal chemistry letters, 2000, Jun-05, Volume: 10, Issue:11

    Topics: Monte Carlo Method; Pharmaceutical Preparations; Solubility

2000
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Cheminformatic models to predict binding affinities to human serum albumin.
    Journal of medicinal chemistry, 2001, Dec-06, Volume: 44, Issue:25

    Topics: Adrenergic beta-Antagonists; Antidepressive Agents, Tricyclic; Chromatography, Affinity; Cyclooxygenase Inhibitors; Databases, Factual; Humans; Hydrophobic and Hydrophilic Interactions; Penicillins; Pharmaceutical Preparations; Protein Binding; Quantitative Structure-Activity Relationship; Reproducibility of Results; Serum Albumin; Steroids

2001
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
First-principle, structure-based prediction of hepatic metabolic clearance values in human.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:4

    Topics: Computational Biology; Drug Discovery; Hepatocytes; Humans; Hydrogen-Ion Concentration; Liver; Metabolic Clearance Rate; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship; Sensitivity and Specificity; Software

2009
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Determination of permeability and lipophilicity of pyrazolo-pyrimidine tyrosine kinase inhibitors and correlation with biological data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:9

    Topics: Humans; Lipids; Membranes, Artificial; Permeability; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-abl; Pyrazoles; Pyrimidines

2009
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
How well can the Caco-2/Madin-Darby canine kidney models predict effective human jejunal permeability?
    Journal of medicinal chemistry, 2010, May-13, Volume: 53, Issue:9

    Topics: Animals; Disease Models, Animal; Dogs; Humans; Jejunal Diseases; Kidney Diseases; Models, Biological; Permeability; Porosity; Regression Analysis

2010
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Prediction of drug intestinal absorption by new linear and non-linear QSPR.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:1

    Topics: Humans; Intestinal Absorption; Linear Models; Molecular Conformation; Nonlinear Dynamics; Permeability; Pharmaceutical Preparations; Probability; Quantitative Structure-Activity Relationship; Thermodynamics

2011
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Combination of GSH trapping and time-dependent inhibition assays as a predictive method of drugs generating highly reactive metabolites.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:7

    Topics: Glutathione; Pharmacology; Sulfur Radioisotopes

2011
Preclinical strategy to reduce clinical hepatotoxicity using in vitro bioactivation data for >200 compounds.
    Chemical research in toxicology, 2012, Oct-15, Volume: 25, Issue:10

    Topics: Chemical and Drug Induced Liver Injury; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Decision Trees; Drug Evaluation, Preclinical; Drug-Related Side Effects and Adverse Reactions; Glutathione; Humans; Liver; Pharmaceutical Preparations; Protein Binding

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Xenobiotic metabolism by isolated rat small intestinal cells.
    Medical biology, 1979, Volume: 57, Issue:5

    Topics: Acetaminophen; Animals; Benzopyrenes; Biotransformation; Cell Separation; Coumarins; Cytochrome P-450 Enzyme System; Glucuronates; Harmine; Intestine, Small; Male; Methylcholanthrene; Oxazines; Rats

1979
Displacement of tolbutamide, glibencalmide and chlorpropamide from serum albumin by anionic drugs.
    Biochemical pharmacology, 1976, May-15, Volume: 25, Issue:10

    Topics: Acetaminophen; Animals; Cattle; Chlorpropamide; Dialysis; Glyburide; Humans; Phenylbutazone; Protein Binding; Salicylates; Serum Albumin; Serum Albumin, Bovine; Sulfaphenazole; Tolbutamide; Warfarin

1976
Competition between diftalone and other drugs for the binding site(s) on human serum albumin.
    Medical biology, 1976, Volume: 54, Issue:3

    Topics: Acetaminophen; Aspirin; Binding Sites; Dexamethasone; Drug Interactions; Humans; Indomethacin; Phenobarbital; Phenylbutazone; Phthalazines; Protein Binding; Pyridazines; Serum Albumin; Temperature; Tolbutamide; Warfarin

1976
Comparative bioavailabilities from truncated blood level curves.
    Journal of pharmaceutical sciences, 1975, Volume: 64, Issue:9

    Topics: Acetaminophen; Aminosalicylic Acids; Biological Availability; Biopharmaceutics; Chloramphenicol; Chlordiazepoxide; Digoxin; Humans; Isoniazid; Kinetics; Pharmaceutical Preparations; Phenylbutazone; Sulfamethizole; Tetracycline; Time Factors; Warfarin

1975
Warfarin and Distalgesic interaction.
    British medical journal, 1976, Jan-24, Volume: 1, Issue:6003

    Topics: Acetaminophen; Aged; Animals; Dextropropoxyphene; Drug Interactions; Female; Hematuria; Humans; Male; Middle Aged; Rats; Warfarin

1976
Letter: Warfarin and distalgesic interaction.
    British medical journal, 1976, Feb-21, Volume: 1, Issue:6007

    Topics: Acetaminophen; Adult; Dextropropoxyphene; Drug Combinations; Drug Interactions; Female; Hematuria; Humans; Warfarin

1976
Potentiation of warfarin anticoagulation by acetaminophen.
    JAMA, 1991, Mar-13, Volume: 265, Issue:10

    Topics: Acetaminophen; Aged; Blood Coagulation; Drug Interactions; Drug Synergism; Female; Humans; Warfarin

1991
Analgesics and warfarin. A case that brings up questions and cautions.
    Postgraduate medicine, 1988, Volume: 83, Issue:5

    Topics: Acetaminophen; Adult; Analgesics; Blood Coagulation; Dextropropoxyphene; Drug Combinations; Drug Interactions; Humans; Male; Partial Thromboplastin Time; Prothrombin Time; Self Medication; Warfarin

1988
Ultraviolet spectrophotometric analysis of barbiturates: evaluation of potential interferences.
    American journal of clinical pathology, 1973, Volume: 59, Issue:2

    Topics: Acetaminophen; Barbiturates; Chlorothiazide; Chlorpropamide; Dicumarol; Humans; Methods; Nicotinic Acids; Oxyphenbutazone; Phenacetin; Phenindione; Phenobarbital; Phenylbutazone; Phenytoin; Salicylates; Spectrophotometry, Ultraviolet; Sulfamethoxazole; Sulfinpyrazone; Sulfisoxazole; Theobromine; Theophylline; Warfarin

1973
Effect of non-narcotic analgesics on anticoagulant-induced hypoprothrombinemia in rats.
    Experientia, 1972, Dec-15, Volume: 28, Issue:12

    Topics: Acetaminophen; Acetanilides; Administration, Oral; Animals; Antipyrine; Aspirin; Blood Coagulation; Dicumarol; Female; Hypoprothrombinemias; Injections, Intraperitoneal; Male; Phenacetin; Phenindione; Phenylbutazone; Rats; Salicylamides; Sodium Salicylate; Species Specificity; Time Factors; Warfarin

1972
Drug-induced bleeding.
    American journal of clinical pathology, 1974, Volume: 61, Issue:5

    Topics: Acetaminophen; Anemia, Aplastic; Anticoagulants; Aspirin; Blood Platelets; Bone Marrow; Capillary Fragility; Drug Hypersensitivity; Drug Synergism; Hemorrhagic Disorders; Hemostasis; Heparin; Heparin Antagonists; Humans; Indenes; Platelet Adhesiveness; Purpura; Thrombocytopenia; Vascular Diseases; Warfarin

1974
Effect of other drugs on oral anticoagulants.
    Maryland state medical journal, 1969, Volume: 18, Issue:10

    Topics: Acetaminophen; Anticoagulants; Coumarins; Drug Antagonism; Drug Synergism; Heparin; Humans; Oxyphenbutazone; Phenylbutazone; Prothrombin Time; Quinidine; Thromboembolism; Vitamin K; Warfarin

1969
Propoxyphene and warfarin interaction.
    Drug intelligence & clinical pharmacy, 1984, Volume: 18, Issue:10

    Topics: Acetaminophen; Dextropropoxyphene; Drug Therapy, Combination; Humans; Prothrombin Time; Warfarin

1984
Early reports on drug interactions.
    Drug intelligence & clinical pharmacy, 1983, Volume: 17, Issue:2

    Topics: Acetaminophen; Amiodarone; Apazone; Aspirin; Carbamazepine; Chlordiazepoxide; Cimetidine; Coumarins; Drug Interactions; Erythromycin; Ethanol; Furosemide; Gentamicins; Humans; Levodopa; Lidocaine; Phenytoin; Prenylamine; Quinidine

1983
Abnormal serum transaminases following therapeutic doses of acetaminophen in the absence of known risk factors.
    Digestive diseases and sciences, 1995, Volume: 40, Issue:9

    Topics: Acetaminophen; Adult; Alanine Transaminase; Analgesics, Non-Narcotic; Aspartate Aminotransferases; Chemical and Drug Induced Liver Injury; Drug Administration Schedule; Humans; Liver Function Tests; Male; Risk Factors; Time Factors; Warfarin

1995
Kupffer cell stimulation with Corynebacterium parvum reduces some cytochrome P450-dependent activities and diminishes acetaminophen and carbon tetrachloride-induced liver injury in the rat.
    Toxicology and applied pharmacology, 1994, Volume: 129, Issue:1

    Topics: Acetaminophen; Alanine Transaminase; Animals; Biotransformation; Carbon Tetrachloride; Cells, Cultured; Coumarins; Cytochrome P-450 CYP2E1; Cytochrome P-450 Enzyme System; Galactosamine; Glutathione; Immunization; Kupffer Cells; Liver; Male; Microsomes, Liver; Nitrophenols; Oxidation-Reduction; Oxidoreductases, N-Demethylating; Propionibacterium acnes; Rats; Rats, Sprague-Dawley; Spectrometry, Fluorescence

1994
Drug interactions with warfarin.
    The Medical journal of Australia, 1993, Apr-19, Volume: 158, Issue:8

    Topics: Acetaminophen; Aged; Drug Interactions; Female; Humans; Prothrombin Time; Warfarin

1993
In vitro drug adsorption to charcoal, silicas, acrylate copolymer and silicone oil with charcoal and with acrylate copolymer.
    Human & experimental toxicology, 1997, Volume: 16, Issue:1

    Topics: Acetaminophen; Acrylates; Adsorption; Antipyrine; Binding Sites; Charcoal; Metoclopramide; Pharmaceutical Preparations; Silicon Dioxide; Silicone Oils; Warfarin

1997
Potentiation of the anticoagulant effect of warfarin.
    Postgraduate medical journal, 1997, Volume: 73, Issue:861

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Blood Coagulation; Drug Synergism; Female; Humans; Middle Aged; Warfarin

1997
Acetaminophen and other risk factors for excessive warfarin anticoagulation.
    JAMA, 1998, Mar-04, Volume: 279, Issue:9

    Topics: Acetaminophen; Adult; Aged; Aged, 80 and over; Alcohol Drinking; Analgesics, Non-Narcotic; Anticoagulants; Case-Control Studies; Diet; Dose-Response Relationship, Drug; Drug Interactions; Female; Hemorrhage; Humans; Logistic Models; Male; Middle Aged; Multivariate Analysis; Risk Factors; Statistics, Nonparametric; Thromboembolism; Warfarin

1998
Acetaminophen and warfarin: undesirable synergy.
    JAMA, 1998, Mar-04, Volume: 279, Issue:9

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Drug Synergism; Hemorrhage; Humans; Risk; Warfarin

1998
Acetaminophen and warfarin.
    Harvard health letter, 1998, Volume: 23, Issue:7

    Topics: Acetaminophen; Anticoagulants; Drug Interactions; Hemorrhage; Humans; International Normalized Ratio; Warfarin

1998
Potentiation of warfarin by acetaminophen.
    The Journal of family practice, 1998, Volume: 46, Issue:6

    Topics: Acetaminophen; Aged; Analgesics, Non-Narcotic; Anticoagulants; Blood Coagulation; Case-Control Studies; Dose-Response Relationship, Drug; Drug Synergism; Female; Humans; International Normalized Ratio; Male; Reproducibility of Results; Risk Factors; Warfarin

1998
Taking blood thinners safely.
    Harvard heart letter : from Harvard Medical School, 1998, Volume: 8, Issue:11

    Topics: Acetaminophen; Anticoagulants; Drug Interactions; Humans; International Normalized Ratio; Warfarin

1998
Acetaminophen and risk factors for excess anticoagulation with warfarin.
    JAMA, 1998, Aug-26, Volume: 280, Issue:8

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Drug Interactions; Humans; Risk Factors; Warfarin

1998
Acetaminophen and risk factors for excess anticoagulation with warfarin.
    JAMA, 1998, Aug-26, Volume: 280, Issue:8

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Drug Interactions; Humans; Risk Factors; Warfarin

1998
Acetaminophen and risk factors for excess anticoagulation with warfarin.
    JAMA, 1998, Aug-26, Volume: 280, Issue:8

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Drug Interactions; Humans; Risk Factors; Warfarin

1998
Acetaminophen and risk factors for excess anticoagulation with warfarin.
    JAMA, 1998, Aug-26, Volume: 280, Issue:8

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Drug Interactions; Humans; Risk Factors; Warfarin

1998
Acetaminophen and risk factors for excess anticoagulation with warfarin.
    JAMA, 1998, Aug-26, Volume: 280, Issue:8

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Drug Interactions; Humans; Risk Factors; Warfarin

1998
Acetaminophen and risk factors for excess anticoagulation with warfarin.
    JAMA, 1998, Aug-26, Volume: 280, Issue:8

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Drug Interactions; Humans; Risk Factors; Vitamin K; Warfarin

1998
When the INR comes back too high.
    Canadian family physician Medecin de famille canadien, 1998, Volume: 44

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Drug Monitoring; Drug Synergism; Humans; International Normalized Ratio; Research Design; Risk Factors; Warfarin

1998
Postoperative acetaminophen and warfarin. Undesirable combination.
    Anesthesiology, 1998, Volume: 89, Issue:5

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Drug Interactions; Humans; Postoperative Complications; Warfarin

1998
In vitro glucuronidation using human liver microsomes and the pore-forming peptide alamethicin.
    Drug metabolism and disposition: the biological fate of chemicals, 2000, Volume: 28, Issue:5

    Topics: Acetaminophen; Alamethicin; Analgesics, Non-Narcotic; Analgesics, Opioid; Anti-Bacterial Agents; Coumarins; Estradiol; Glucuronides; Glucuronosyltransferase; Humans; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Microsomes, Liver; Morphine; Oxidation-Reduction; Testosterone

2000
Retroperitoneal haematoma after paracetamol increased anticoagulation.
    Emergency medicine journal : EMJ, 2002, Volume: 19, Issue:1

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Drug Synergism; Female; Femoral Neuropathy; Hematoma; Humans; International Normalized Ratio; Middle Aged; Retroperitoneal Space; Warfarin

2002
Warfarin and acetaminophen interaction.
    Pharmacotherapy, 2003, Volume: 23, Issue:1

    Topics: Acetaminophen; Aged; Analgesics, Non-Narcotic; Anticoagulants; Atrial Fibrillation; Drug Synergism; Humans; International Normalized Ratio; Male; Warfarin

2003
Pharmaceutical drug overdose case reports. From the World Literature.
    Toxicological reviews, 2003, Volume: 22, Issue:3

    Topics: Acetaminophen; Adolescent; Adult; Aged; Amlodipine; Child, Preschool; Diphenhydramine; Dizocilpine Maleate; Drug Overdose; Female; Humans; International Normalized Ratio; Lithium; Male; Middle Aged; Paroxetine; Salicylates; Valproic Acid; Warfarin

2003
A 76-year-old woman with erratic anticoagulation.
    Cleveland Clinic journal of medicine, 2004, Volume: 71, Issue:8

    Topics: Acetaminophen; Aged; Analgesics, Non-Narcotic; Anticoagulants; Drug Interactions; Female; Gingival Hemorrhage; Hematuria; Humans; International Normalized Ratio; Phytotherapy; Warfarin; Zingiber officinale

2004
Paracetamol (acetaminophen) and warfarin interaction: unraveling the pivotal role of the vitamin K cycle.
    Thrombosis and haemostasis, 2004, Volume: 92, Issue:4

    Topics: Acetaminophen; Blood Coagulation Factors; Carboxylic Acids; Dissent and Disputes; Drug Interactions; Humans; Vitamin K; Warfarin

2004
Paracetamol (acetaminophen) warfarin interaction: NAPQI, the toxic metabolite of paracetamol, is an inhibitor of enzymes in the vitamin K cycle.
    Thrombosis and haemostasis, 2004, Volume: 92, Issue:4

    Topics: Acetaminophen; Aged; Benzoquinones; Carbon-Carbon Ligases; Drug Interactions; Enzyme Inhibitors; Female; Humans; Imines; Kinetics; Mixed Function Oxygenases; Vitamin K; Vitamin K Epoxide Reductases; Warfarin

2004
Medical mystery. A woman with too-thin blood. Why was the patient bleeding? What's her case mean to you?
    Heart advisor, 2004, Volume: 7, Issue:12

    Topics: Acetaminophen; Aged; Analgesics, Non-Narcotic; Anticoagulants; Blood Coagulation; Female; Herb-Drug Interactions; Humans; Phytotherapy; Warfarin; Zingiber officinale

2004
Utilization review of concomitant use of potentially interacting drugs in Thai patients using warfarin therapy.
    Pharmacoepidemiology and drug safety, 2007, Volume: 16, Issue:2

    Topics: Acetaminophen; Adult; Ambulatory Care; Analgesics, Non-Narcotic; Anticoagulants; Antithyroid Agents; Aspirin; Diclofenac; Drug Interactions; Drug Monitoring; Drug Prescriptions; Drug Utilization Review; Female; Follow-Up Studies; Humans; International Normalized Ratio; Male; Middle Aged; Polypharmacy; Propylthiouracil; Retrospective Studies; Thailand; Warfarin

2007
I have osteoarthritis in my knees. I also have a blood-clotting disorder and have been put on Coumadin, which means I can't take NSAIDs. I take a daily dose of Tylenol, but it doesn't have much effect. What do you suggest?
    DukeMedicine healthnews, 2007, Volume: 13, Issue:8

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anti-Inflammatory Agents, Non-Steroidal; Anticoagulants; Blood Coagulation Disorders; Capsaicin; Contraindications; Humans; Osteoarthritis, Knee; Warfarin

2007
Potentially lethal acetaminophen-warfarin interaction in an older adult: an under-recognized phenomenon?
    Journal of the American Medical Directors Association, 2007, Volume: 8, Issue:8

    Topics: Acetaminophen; Aged, 80 and over; Analgesics, Non-Narcotic; Anticoagulants; Drug Synergism; Female; Humans; Warfarin

2007
Warfarin-acetaminophen interaction.
    The Medical letter on drugs and therapeutics, 2008, Jun-16, Volume: 50, Issue:1288

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Blood Coagulation; Drug Interactions; Drug Monitoring; Humans; International Normalized Ratio; Pharmacogenetics; Warfarin

2008
[Concomitant use of warfarin, analgesics and anti-inflammatory agents].
    Tidsskrift for den Norske laegeforening : tidsskrift for praktisk medicin, ny raekke, 2009, Jun-11, Volume: 129, Issue:12

    Topics: Acetaminophen; Aged; Analgesics, Non-Narcotic; Analgesics, Opioid; Anti-Inflammatory Agents, Non-Steroidal; Anticoagulants; Cyclooxygenase Inhibitors; Drug Interactions; Drug Prescriptions; Drug Therapy, Combination; Female; Hemorrhage; Humans; Male; Middle Aged; Norway; Risk Factors; Warfarin

2009
Adverse interaction of warfarin and paracetamol: evidence from a post-mortem study.
    European journal of clinical pharmacology, 2010, Volume: 66, Issue:1

    Topics: Acetaminophen; Adverse Drug Reaction Reporting Systems; Aged; Analgesics, Non-Narcotic; Analgesics, Opioid; Anticoagulants; Autopsy; Cause of Death; Databases, Factual; Drug Interactions; Drug Therapy, Combination; Female; Hemorrhage; Humans; Male; Middle Aged; Tramadol; Warfarin

2010
Adverse interaction of warfarin and paracetamol: evidence from a post-mortem study.
    European journal of clinical pharmacology, 2010, Volume: 66, Issue:2

    Topics: Acetaminophen; Anti-Inflammatory Agents, Non-Steroidal; Anticoagulants; Drug Interactions; Emergency Service, Hospital; Hemorrhage; Humans; Nonprescription Drugs; Patient Education as Topic; Turkey; Warfarin

2010
I've read where people on coumadin shouldn't take acetaminophen (Tylenol), but I've also been told that it's a safe alternative to aspirin, which warfarin (Coumadin) takers are not supposed to take. Can you clear up the confusion?
    Heart advisor, 2009, Volume: 12, Issue:4

    Topics: Acetaminophen; Anticoagulants; Aspirin; Drug Interactions; Drug Therapy, Combination; Fibrinolytic Agents; Health Knowledge, Attitudes, Practice; Humans; Platelet Aggregation Inhibitors; Thromboembolism; Warfarin

2009
Warfarin therapy: how the less interesting half just got interesting.
    Journal of thrombosis and haemostasis : JTH, 2010, Volume: 8, Issue:12

    Topics: Acetaminophen; Anticoagulants; Azithromycin; Cimetidine; Cytochrome P-450 Enzyme System; Drug Interactions; Gefitinib; Humans; Omeprazole; Quinazolines; Stereoisomerism; Substrate Specificity; Warfarin

2010
Familial Mediterranean fever presenting with pulmonary embolism.
    Connecticut medicine, 2011, Volume: 75, Issue:1

    Topics: Acetaminophen; Adult; Analgesics, Non-Narcotic; Anticoagulants; Chest Pain; Colchicine; Diagnosis, Differential; Familial Mediterranean Fever; Follow-Up Studies; Heparin; Humans; Male; Pulmonary Embolism; Serositis; Tubulin Modulators; Turkey; Warfarin

2011
Moxifloxacin-acetaminophen-warfarin interaction during bacille Calmette-Guerin treatment for bladder cancer.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2011, May-01, Volume: 68, Issue:9

    Topics: Acetaminophen; Adjuvants, Immunologic; Aged, 80 and over; Analgesics, Non-Narcotic; Anti-Infective Agents; Anticoagulants; Antifibrinolytic Agents; Aza Compounds; BCG Vaccine; Drug Interactions; Fluoroquinolones; Humans; International Normalized Ratio; Male; Moxifloxacin; Quinolines; Urinary Bladder Neoplasms; Vitamin K 1; Warfarin

2011
RS-predictor: a new tool for predicting sites of cytochrome P450-mediated metabolism applied to CYP 3A4.
    Journal of chemical information and modeling, 2011, Jul-25, Volume: 51, Issue:7

    Topics: Acetaminophen; Binding Sites; Cytochrome P-450 CYP3A; Models, Molecular; Molecular Structure; Stereoisomerism; Warfarin

2011
Warfarin and acetaminophen interaction: a summary of the evidence and biologic plausibility.
    Blood, 2011, Dec-08, Volume: 118, Issue:24

    Topics: Acetaminophen; Aged; Analgesics, Non-Narcotic; Anticoagulants; Atrial Fibrillation; Back Pain; Biotransformation; Diabetes Complications; Drug Interactions; Drug Monitoring; Embolism; Female; Humans; Hypertension; International Normalized Ratio; Vitamin K; Warfarin

2011
Effects of etravirine on the pharmacokinetics and pharmacodynamics of warfarin in rats.
    British journal of pharmacology, 2013, Volume: 168, Issue:8

    Topics: Acetaminophen; Animals; Anticoagulants; Blood Coagulation; Drug Synergism; Male; Nitriles; Pyridazines; Pyrimidines; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Inhibitors; Warfarin

2013
Warfarin: its highs and lows.
    Canadian family physician Medecin de famille canadien, 2013, Volume: 59, Issue:8

    Topics: Acetaminophen; Aged, 80 and over; Analgesics, Non-Narcotic; Anticoagulants; Atrial Fibrillation; Chondroitin; Dietary Supplements; Drug Interactions; Drug Monitoring; Glucosamine; Humans; International Normalized Ratio; Male; Nomograms; Stroke; Warfarin

2013
[Fatal intracerebral haemorrhage possibly caused by interaction between paracetamol and warfarin].
    Ugeskrift for laeger, 2015, Jun-01, Volume: 177, Issue:23

    Topics: Acetaminophen; Aged, 80 and over; Analgesics, Non-Narcotic; Anticoagulants; Cerebral Hemorrhage; Drug Interactions; Fatal Outcome; Humans; Male; Tomography, X-Ray Computed; Warfarin

2015
Phenotypic and biomarker evaluation of zebrafish larvae as an alternative model to predict mammalian hepatotoxicity.
    Journal of applied toxicology : JAT, 2016, Volume: 36, Issue:9

    Topics: Acetaminophen; Amiodarone; Animals; Apoptosis; Aryl Hydrocarbon Hydroxylases; Ceruloplasmin; Coumarins; Female; Gene Expression Regulation; Genetic Markers; Genome-Wide Association Study; Humans; In Situ Hybridization; Larva; Liver; Male; Methapyrilene; Nitriles; Oxidoreductases, N-Demethylating; Phenotype; Toxicity Tests; Transferrin; Triazoles; Zebrafish; Zebrafish Proteins

2016
New Phenylpropanoid and Coumarin Glycosides from the Stems of Hydrangea paniculata Sieb.
    Molecules (Basel, Switzerland), 2017, Jan-18, Volume: 22, Issue:1

    Topics: Acetaminophen; Antipyretics; Coumarins; Glycosides; Hep G2 Cells; Humans; Hydrangea; Molecular Structure; Plant Stems; Propanols; Protective Agents; Structure-Activity Relationship

2017
Glycycoumarin protects mice against acetaminophen-induced liver injury predominantly via activating sustained autophagy.
    British journal of pharmacology, 2018, Volume: 175, Issue:19

    Topics: Acetaminophen; Animals; Autophagy; Chemical and Drug Induced Liver Injury; Coumarins; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Male; Mice; Mice, Inbred C57BL; Protective Agents; Structure-Activity Relationship

2018
Frailty and Co-Prescribing of Potentially Interacting Drugs in New Users of Warfarin.
    Drugs & aging, 2020, Volume: 37, Issue:5

    Topics: Acetaminophen; Aged; Aged, 80 and over; Anti-Inflammatory Agents, Non-Steroidal; Anticoagulants; Clopidogrel; Drug Interactions; Drug Prescriptions; Drug Utilization Review; Female; Frail Elderly; Frailty; Hemorrhage; Humans; Male; Platelet Aggregation Inhibitors; Warfarin

2020
Warfarin and acetaminophen interaction in a 47-year-old woman.
    CMAJ : Canadian Medical Association journal = journal de l'Association medicale canadienne, 2020, 05-11, Volume: 192, Issue:19

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Anticoagulants; Diagnosis, Differential; Drug Interactions; Female; Heart Valve Prosthesis Implantation; Humans; Middle Aged; Mitral Valve; Warfarin

2020
High-Selectivity Fluorescent Reporter toward Peroxynitrite in a Coexisting Nonalcoholic Fatty Liver and Drug-Induced Liver Diseases Model.
    Analytical chemistry, 2020, 08-18, Volume: 92, Issue:16

    Topics: Acetaminophen; Animals; Chemical and Drug Induced Liver Injury; Coumarins; Cytochrome P-450 CYP2E1; Diet, High-Fat; Fatty Acids; Fluorescent Dyes; Hep G2 Cells; Humans; Limit of Detection; Liver; Mice; Microscopy, Fluorescence; Mitochondria; Non-alcoholic Fatty Liver Disease; Peroxynitrous Acid

2020
Structurally diverse coumarin-homoisoflavonoid derivatives with hepatoprotective activities from the fruits of Cucumis bisexualis.
    Fitoterapia, 2021, Volume: 149

    Topics: Acetaminophen; China; Coumarins; Cucumis; Flavonoids; Fruit; Hep G2 Cells; Humans; Molecular Structure; Phytochemicals; Protective Agents

2021
Drug-related challenges following primary total hip and knee arthroplasty.
    Basic & clinical pharmacology & toxicology, 2021, Volume: 129, Issue:2

    Topics: Acetaminophen; Adult; Aged; Aged, 80 and over; Analgesics; Analgesics, Opioid; Angiotensins; Arthroplasty, Replacement, Hip; Arthroplasty, Replacement, Knee; Diuretics; Drug Interactions; Female; Hospitals; Humans; Male; Middle Aged; Patient Readmission; Postoperative Complications; Risk Factors; Warfarin

2021
Urolithin A protects against acetaminophen-induced liver injury in mice via sustained activation of Nrf2.
    International journal of biological sciences, 2022, Volume: 18, Issue:5

    Topics: Acetaminophen; Animals; Chemical and Drug Induced Liver Injury; Coumarins; Kelch-Like ECH-Associated Protein 1; Liver; Mice; Molecular Docking Simulation; NF-E2-Related Factor 2; Oxidative Stress

2022
Massive warfarin overdose management in an adolescent patient.
    Clinical toxicology (Philadelphia, Pa.), 2022, Volume: 60, Issue:10

    Topics: Acetaminophen; Adolescent; Anticoagulants; Child; Ethanol; Hemorrhage; Humans; International Normalized Ratio; Male; Poisons; Salicylates; Vitamin K; Warfarin

2022
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